NOVEL IMIDAZOLE DERIVATIVES
    4.
    发明申请
    NOVEL IMIDAZOLE DERIVATIVES 审中-公开
    新咪唑衍生物

    公开(公告)号:US20110224252A1

    公开(公告)日:2011-09-15

    申请号:US12739863

    申请日:2008-10-24

    摘要: The present invention relates to novel imidazole derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is halogen, C1-C4alkyl or C1-C4haloalkyl; R2 is an optionally substituted aryl or heteroaryl; R3 is halogen; R4 is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy or cyano; R5 is halogen; X is N or C(R); and R is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy or cyano; or an agrochemically usable salt form thereof; provided that when X is C(R), R2 cannot be an optionally substituted aryl.

    摘要翻译: 本发明涉及式(I)的新咪唑衍生物作为具有杀微生物活性,特别是杀真菌活性的活性成分:其中R1是卤素,C1-C4烷基或C1-C4卤代烷基; R2是任选取代的芳基或杂芳基; R3是卤素; R4是氢,卤素,C1-C4烷基,C1-C4卤代烷基,C1-C4烷氧基,C1-C4卤代烷氧基或氰基; R5是卤素; X是N或C(R); 且R为氢,卤素,C 1 -C 4烷基,C 1 -C 4卤代烷基,C 1 -C 4烷氧基,C 1 -C 4卤代烷氧基或氰基; 或其农业化学可用的盐形式; 条件是当X是C(R)时,R 2不能是任选取代的芳基。

    PYRIDAZINE DERIVATIVES
    6.
    发明申请
    PYRIDAZINE DERIVATIVES 审中-公开
    吡啶衍生物

    公开(公告)号:US20100144674A1

    公开(公告)日:2010-06-10

    申请号:US12447028

    申请日:2007-10-23

    摘要: The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is hydrogen, C1-C6alkyl, C1-C8haloalkyl or C3-C6cycloalkyl; R2 is cycloalkyl, cycloalkylalkyl, halocycloalkyl, cycloalkoxy, halocycloalkoxy, cycloalkylalkoxy, halocycloalkylalkoxy, alkoxyalkyl, cycloalkoxyalkoxyalkyl, haloalkoxyalkyl, trialkylsilyl, alkylthioalkyl, haloalkylthioalkyl, cycloalkylthio, halocycloalkylthio, cycloalkylalkylthio, halocycloalkylalkylthio, alkylsulfinylalkyl, alkylsulfonylalkyl, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, C2-C6alkenyl, C2-C6alkynyl, optionally substituted arylsulfonyl, optionally substituted aryloxy, optionally optionally substituted heteroaryloxy, optionally substituted arylthio, optionally substituted heteroarylthio; or R2 together with an adjacent carbon atom forms an optionally substituted fused ring; R3 is an optionally substituted aryl; R4 is hydrogen, halogen, C1-C6alkyl, C1-C6haloalkyl, C1-C8alkoxy, C1-C6haloalkoxy, hydroxy or cyano; and n is a whole number from 1 to 4; or an agrochemically usable salt form thereof.

    摘要翻译: 本发明涉及具有杀微生物活性,特别是杀真菌活性的活性成分的式(I)的新哒嗪衍生物,其中R1是氢,C1-C6烷基,C1-C8卤代烷基或C3-C6环烷基; R 2是环烷基,环烷基烷基,卤代环烷基,环烷氧基,卤代环烷氧基,环烷基烷氧基,卤代环烷基烷氧基,烷氧基烷基,环烷氧基烷氧基烷基,卤代烷氧基烷基,三烷基甲硅烷基,烷硫基烷基,卤代烷硫基烷基,环烷硫基,卤代环烷硫基,环烷基烷硫基,卤代环烷基烷硫基,烷基亚磺酰基烷基,烷基磺酰基烷基,烷基亚磺酰基,卤代烷基亚磺酰基,烷基磺酰基,卤代烷基磺酰基, C 6链烯基,C 2 -C 6炔基,任选取代的芳基磺酰基,任选取代的芳氧基,任选任选取代的杂芳氧基,任选取代的芳硫基,任选取代的杂芳硫基; 或R 2与相邻的碳原子一起形成任选取代的稠环; R3是任选取代的芳基; R4是氢,卤素,C1-C6烷基,C1-C6卤代烷基,C1-C8烷氧基,C1-C6卤代烷氧基,羟基或氰基; n为1〜4的整数; 或其农业化学上可用的盐形式。

    NOVEL PYRIDAZINE DERIVATIVES
    10.
    发明申请
    NOVEL PYRIDAZINE DERIVATIVES 审中-公开
    新的吡咯烷酮衍生物

    公开(公告)号:US20100113457A1

    公开(公告)日:2010-05-06

    申请号:US12447025

    申请日:2007-10-23

    摘要: The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is hydrogen, C1-C6alkyl, C1-C6haloalkyl or C3-C6cycloalkyl; R2 is halogen, nitro, cyano, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy, C1-C4alkylthio or C1-C4haloalkylthio; R3 is an optionally substituted aryl; R4 is fluoro, cyano, C1-C6haloalkyl, C3-C6cycloalkyl, C1-C6haloalkoxy, C1-C6alkylthio or C1-C6haloalkylthio; and n is a whole number from 1 to 4; or an agrochemically usable salt form thereof.

    摘要翻译: 本发明涉及具有杀微生物活性,特别是杀真菌活性的活性成分的式(I)的新哒嗪衍生物,其中R1是氢,C1-C6烷基,C1-C6卤代烷基或C3-C6环烷基; R 2是卤素,硝基,氰基,C 1 -C 4烷基,C 1 -C 4卤代烷基,C 1 -C 4烷氧基,C 1 -C 4卤代烷氧基,C 1 -C 4烷硫基或C 1 -C 4卤代烷硫基; R3是任选取代的芳基; R 4是氟,氰基,C 1 -C 6卤代烷基,C 3 -C 6环烷基,C 1 -C 6卤代烷氧基,C 1 -C 6烷硫基或C 1 -C 6卤代烷硫基; n为1〜4的整数; 或其农业化学上可用的盐形式。