公开(公告)号：US07943642B2

公开(公告)日：2011-05-17

申请号：US11577664

申请日：2005-10-27

申请人： David M. Roush ,  John F. Chiarello ,  George Theodoridis ,  Hongyan Qi

发明人： David M. Roush ,  John F. Chiarello ,  George Theodoridis ,  Hongyan Qi

IPC分类号： A01N43/40 ,  A01N43/46 ,  C07D401/12

CPC分类号： C07D401/12 ,  A01N43/36 ,  A01N43/40 ,  A01N43/50 ,  A01N43/56 ,  A01N43/78 ,  C07D405/12 ,  C07D417/12

摘要： Certain novel N,N-di(heteroarylalkyl)amine derivatives have provided unexpected insecticidal and acaricidal activity. These compounds are represented by formula (I): wherein Ar Ar1, a, b, c, R, Rd, Re, Rf, Rg, Rh, R′, R3 and Rk are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 某些新的N，N-二（杂芳基烷基）胺衍生物已经提供了意想不到的杀虫和杀螨活性。 这些化合物由式（I）表示：其中Ar Ar1，a，b，c，R，Rd，Re，Rf，Rg，Rh，R'，R 3和R k在本文中被完整描述。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US20080287506A1

公开(公告)日：2008-11-20

申请号：US11577664

申请日：2005-10-27

申请人： David M. Roush ,  John F. Chiarello ,  George Theodoridis ,  Hongyan Qi

发明人： David M. Roush ,  John F. Chiarello ,  George Theodoridis ,  Hongyan Qi

IPC分类号： A01N43/40 ,  C07D401/12 ,  C07D207/02 ,  C07D231/12 ,  C07D233/61 ,  A01N43/36 ,  A01N43/56 ,  A01N43/50 ,  A01P7/04

CPC分类号： C07D401/12 ,  A01N43/36 ,  A01N43/40 ,  A01N43/50 ,  A01N43/56 ,  A01N43/78 ,  C07D405/12 ,  C07D417/12

摘要： Certain novel N,N-di(heteroarylalkyl)amine derivatives have provided unexpected insecticidal and acaricidal activity. These compounds are represented by formula (I): wherein Ar Ar1, a, b, c, R, Rd, Re, Rf, Rg, Rh, R′, R3 and Rk are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 某些新的N，N-二（杂芳基烷基）胺衍生物已经提供了意想不到的杀虫和杀螨活性。 这些化合物由式（I）表示：其中Ar Ar 1，a，b，c，R，R d，R e， 本文中完整地描述了R f，R g，R h，R'，R 3和R k。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US20110065710A1

公开(公告)日：2011-03-17

申请号：US10580481

申请日：2004-12-02

申请人： David M. Roush ,  John F. Chiarello ,  Jianming Yu ,  Benjamin J. Dugan ,  George Theodoridis ,  Manorama M. Patel ,  Walter H. Yeager ,  Steven W. Szczepanski

发明人： David M. Roush ,  John F. Chiarello ,  Jianming Yu ,  Benjamin J. Dugan ,  George Theodoridis ,  Manorama M. Patel ,  Walter H. Yeager ,  Steven W. Szczepanski

IPC分类号： A61K31/4965 ,  A61K31/50 ,  A61K31/426 ,  A61K31/44

CPC分类号： C07D213/26 ,  A01N43/40 ,  A01N43/50 ,  A01N43/78 ,  A01N43/82 ,  A01N43/88 ,  A01N47/40 ,  A01N51/00 ,  A01N57/26 ,  C07D213/38 ,  C07D213/64 ,  C07D213/70 ,  C07D213/73 ,  C07D233/64 ,  C07D237/08 ,  C07D237/12 ,  C07D239/30 ,  C07D241/16 ,  C07D261/08 ,  C07D263/34 ,  C07D273/00 ,  C07D277/32 ,  C07D285/06 ,  C07D307/14 ,  C07D401/12 ,  C07D401/14 ,  C07D405/12 ,  C07D413/12 ,  C07D413/14 ,  C07D417/12 ,  C07D417/14 ,  C07F9/58

摘要： Certain noel N-(heteroarylalkyl)alkanediamine derivatives have provided unexpected insecticidal and acaricidal activity. These compounds are represented by formula I: wherein Ar, a, r, R, Ra, Rb, Rc, Rd, b, c, Re, Rf, Rg, Rh, R5, d, e, U, V, X, WR6 and R7 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 某些Noel N-（杂芳基烷基）烷二胺衍生物提供了意想不到的杀虫和杀螨活性。 这些化合物由式I表示：其中Ar，a，r，R，Ra，Rb，Rc，Rd，b，c，Re，Rf，Rg，Rh，R5，d，e，U，V，X， 和R7完全描述于此。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US07977332B2

公开(公告)日：2011-07-12

申请号：US10580481

申请日：2004-12-02

申请人： David M. Roush ,  John F. Chiarello ,  Jianming Yu ,  Benjamin J. Dugan ,  George Theodoridis ,  Manorama M. Patel ,  Walter H. Yeager ,  Steven W. Szczepanski

发明人： David M. Roush ,  John F. Chiarello ,  Jianming Yu ,  Benjamin J. Dugan ,  George Theodoridis ,  Manorama M. Patel ,  Walter H. Yeager ,  Steven W. Szczepanski

IPC分类号： C07D213/02 ,  A01N43/08

CPC分类号： C07D213/26 ,  A01N43/40 ,  A01N43/50 ,  A01N43/78 ,  A01N43/82 ,  A01N43/88 ,  A01N47/40 ,  A01N51/00 ,  A01N57/26 ,  C07D213/38 ,  C07D213/64 ,  C07D213/70 ,  C07D213/73 ,  C07D233/64 ,  C07D237/08 ,  C07D237/12 ,  C07D239/30 ,  C07D241/16 ,  C07D261/08 ,  C07D263/34 ,  C07D273/00 ,  C07D277/32 ,  C07D285/06 ,  C07D307/14 ,  C07D401/12 ,  C07D401/14 ,  C07D405/12 ,  C07D413/12 ,  C07D413/14 ,  C07D417/12 ,  C07D417/14 ,  C07F9/58

摘要： Certain noel N-(heteroarylalkyl)alkanediamine derivatives have provided unexpected insecticidal and acaricidal activity. These compounds are represented by formula I: wherein Ar, a, r, R, Ra, Rb, Rc, Rd, b, c, Re, Rf, Rg, Rh, R5, d, e, U, V, X, WR6 and R7 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 某些Noel N-（杂芳基烷基）烷二胺衍生物提供了意想不到的杀虫和杀螨活性。 这些化合物由式I表示：其中Ar，a，r，R，Ra，Rb，Rc，Rd，b，c，Re，Rf，Rg，Rh，R5，d，e，U，V，X， 和R7完全描述于此。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US20100261757A1

公开(公告)日：2010-10-14

申请号：US12223279

申请日：2007-01-15

申请人： John F. Chiarello ,  Harvey R. Wendt ,  Najing Zhang ,  George Theodoridis

发明人： John F. Chiarello ,  Harvey R. Wendt ,  Najing Zhang ,  George Theodoridis

IPC分类号： A01N43/40 ,  A01N43/78 ,  A01N47/40 ,  C07D401/12 ,  C07D417/12 ,  C07D213/59 ,  C07D277/30 ,  C07D407/12 ,  A01P7/04

CPC分类号： C07D401/12 ,  C07D213/61 ,  C07D277/32 ,  C07D401/14 ,  C07D407/12 ,  C07D417/12 ,  C07D417/14

摘要： Certain novel N-(heteroarylalkyl)alkanediamine derivatives have provided unexpected insecticidal and acaricidal activity. These compounds are represented by formula I: wherein Ar, a, b, c, T, W, Y R, Rf, Rg, Rh, Ri, Rj, Rk, Rm, Rn, and R are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 某些新的N-（杂芳基烷基）烷二胺衍生物提供了意想不到的杀虫和杀螨活性。 这些化合物由式I表示：其中Ar，a，b，c，T，W，Y R，R f，R g，Rh，R 1，R j，R k，R m，R n和R在本文中被完整描述。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US07932393B2

公开(公告)日：2011-04-26

申请号：US12223279

申请日：2007-01-15

申请人： John F. Chiarello ,  Harvey R. Wendt ,  Nanjing Zhang ,  George Theodoridis

发明人： John F. Chiarello ,  Harvey R. Wendt ,  Nanjing Zhang ,  George Theodoridis

IPC分类号： C07D213/04

CPC分类号： C07D401/12 ,  C07D213/61 ,  C07D277/32 ,  C07D401/14 ,  C07D407/12 ,  C07D417/12 ,  C07D417/14

摘要： Certain novel N-(heteroarylalkyl)alkanediamine derivatives have provided unexpected insecticidal and acaricidal activity. These compounds are represented by formula I: wherein Ar, a, b, c, T, W, Y, R, Rf, Rg, Rh, Ri, Rj, Rk, Rm, Rn, and R7 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 某些新的N-（杂芳基烷基）烷二胺衍生物提供了意想不到的杀虫和杀螨活性。 这些化合物由式I表示：其中Ar，a，b，c，T，W，Y，R，R f，R g，Rh，R 1，R j，R k，R m，R n和R 7在本文中被完整描述。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US06987194B2

公开(公告)日：2006-01-17

申请号：US10832624

申请日：2004-04-27

申请人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  David M. Roush ,  Stephen F. Donovan ,  Frank J. Zawacki ,  Walter H. Yeager ,  John W. Lyga ,  Daniel H. Cohen

发明人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  David M. Roush ,  Stephen F. Donovan ,  Frank J. Zawacki ,  Walter H. Yeager ,  John W. Lyga ,  Daniel H. Cohen

IPC分类号： C07D307/83 ,  C07D311/04 ,  A61K31/343 ,  A61K31/353

CPC分类号： A01N43/30 ,  A01N43/32 ,  A01N43/40 ,  A01N43/60 ,  A01N47/16 ,  C07D211/22 ,  C07D307/79 ,  C07D307/83 ,  C07D311/04 ,  C07D401/04 ,  C07D495/10

摘要： Insecticidal (dihalopropenyl) phenylalkyl substituted dihydrobenzofuran and dihydrobenzopyran derivatives of Formula I are disclosed. These compounds provide unexpected insecticidal activity across a spectrum of insect pests combined with desirable physical properties including improved photostability. wherein x and y are integers independently selected from 0 or 1; and B is a bridging group *—(CR16R17)q—(CR18R19)r—(CR20R21)s—Lt—(CR22R23)u—(CR24R25)v—(CR26R27)w—, where the asterisk denotes attachment at A; and q, r, s, u, v and w are integers independently selected from 0, 1 and 2; and t is an integer selected from 0 and 1. A, D, E, G, M, R through R11, and R16 through R27, inclusively, are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I and methods of controlling insects by applying said compositions to a locus where insects are present or are expected to be present are also disclosed.

摘要翻译： 公开了杀虫（二卤代丙烯基）苯基烷基取代的二氢苯并呋喃和式I的二氢苯并吡喃衍生物。 这些化合物在一系列昆虫害虫中提供了意想不到的杀虫活性，并结合所需的物理性质，包括改善的光稳定性。 其中x和y是独立地选自0或1的整数; 并且B是桥接基团<？in-line-formula description =“In-line Formulas”end =“lead”？> * - （CR ^{16 17 ） - （CR 20） - （CR 20） - （CR 20） - （CR 20） - （CR 22）23 - - - （CR 22）23 （CR 26）25（ - ） - （CR 26）25 ） q，r，s，u，v和w是独立地选自0,1和2的整数; A，D，E，G，M，R至R 11和R 16至R 27中的一个整数。 / SUP>，包括这里完全描述。 此外，还公开了包含杀虫有效量的至少一种式I化合物的组合物和通过将所述组合物施用于存在昆虫或预期存在的场所来控制昆虫的方法。}

公开(公告)号：US06753429B2

公开(公告)日：2004-06-22

申请号：US09941812

申请日：2001-08-29

申请人： George Theodoridis ,  Edward Barron ,  Daniel H. Cohen ,  Ellen M. Crawford ,  Thomas G. Cullen ,  Hongyan Qi ,  Elizabeth Rowley ,  Syed F. Ali ,  Walter H. Yeager ,  Christina B. Duggan

发明人： George Theodoridis ,  Edward Barron ,  Daniel H. Cohen ,  Ellen M. Crawford ,  Thomas G. Cullen ,  Hongyan Qi ,  Elizabeth Rowley ,  Syed F. Ali ,  Walter H. Yeager ,  Christina B. Duggan

IPC分类号： C07D24104

CPC分类号： C07D215/233 ,  C07C211/59 ,  C07C217/20 ,  C07C217/58 ,  C07C217/92 ,  C07C233/43 ,  C07C235/56 ,  C07C251/24 ,  C07C271/28 ,  C07C275/34 ,  C07C275/40 ,  C07C291/04 ,  C07C2602/08 ,  C07C2602/10 ,  C07D209/46 ,  C07D215/24 ,  C07D215/38 ,  C07D215/40 ,  C07D215/44 ,  C07D217/22 ,  C07D295/088 ,  C07D295/096 ,  C07D295/205 ,  C07D491/10

摘要： Compounds of formula I: wherein A, B, D, and R are as defined herein and their agriculturally acceptable salts are disclosed as effective insecticides. In addition, compositions comprising an insecticidally effective amount of a compound of Formula I in admixture with at least one agriculturally acceptable extender or adjuvant and methods of controlling insects comprising applying said compositions to locus on crops where control is desired are disclosed. It is emphasized that this abstract is provided to comply with the rules requiring an abstract that will allow a searcher or other reader to quickly ascertain the subject matter of the technical disclosure. It is submitted with the understanding that it will not be used to interpret or limit the scope or meaning of the claims (see 37 C.F.R. 1.72(b)).

摘要翻译： 式I化合物：其中A，B，D和R如本文所定义，其农业上可接受的盐被公开为有效的杀虫剂。 此外，公开了包含杀虫有效量的式I化合物与至少一种农业上可接受的增量剂或佐剂混合的组合物和控制昆虫的方法，其包括将所述组合物施用于需要控制的作物上的位点。 要强调的是，该摘要被提供以符合要求抽象的规则，允许搜索者或其他读者快速确定技术公开的主题。 提交它的理解是，它不会用于解释或限制权利要求的范围或含义（见C.C.R. 1.72（b））。

公开(公告)号：US07247756B2

公开(公告)日：2007-07-24

申请号：US10353471

申请日：2003-01-29

申请人： George Theodoridis ,  Edward Barron ,  Daniel H. Cohen ,  Ellen M. Crawford ,  Thomas G. Cullen ,  Hongyan Qi ,  Elizabeth Rowley ,  Syed F. Ali ,  Walter H. Yeager ,  Christina B. Duggan

发明人： George Theodoridis ,  Edward Barron ,  Daniel H. Cohen ,  Ellen M. Crawford ,  Thomas G. Cullen ,  Hongyan Qi ,  Elizabeth Rowley ,  Syed F. Ali ,  Walter H. Yeager ,  Christina B. Duggan

IPC分类号： C07C43/20

CPC分类号： C07D215/233 ,  C07C211/59 ,  C07C217/20 ,  C07C217/58 ,  C07C217/92 ,  C07C233/43 ,  C07C235/56 ,  C07C251/24 ,  C07C271/28 ,  C07C275/34 ,  C07C275/40 ,  C07C291/04 ,  C07C2602/08 ,  C07C2602/10 ,  C07D209/46 ,  C07D215/24 ,  C07D215/38 ,  C07D215/40 ,  C07D215/44 ,  C07D217/22 ,  C07D295/088 ,  C07D295/096 ,  C07D295/205 ,  C07D491/10

摘要： Compounds of formula I: wherein A, B, D, and R are as defined herein and their agriculturally acceptable salts are disclosed as effective insecticides. In addition, compositions comprising an insecticidally effective amount of a compound of Formula I in admixture with at least one agriculturally acceptable extender or adjuvant and methods of controlling insects comprising applying the compositions to locus on crops where control is desired are disclosed.

摘要翻译： 式I化合物：其中A，B，D和R如本文所定义，其农业上可接受的盐被公开为有效的杀虫剂。 此外，公开了包含杀虫有效量的式I化合物与至少一种农业上可接受的增量剂或佐剂混合的组合物和控制昆虫的方法，其包括将组合物施用于需要控制的作物上的位点。

公开(公告)号：US07576224B2

公开(公告)日：2009-08-18

申请号：US11292023

申请日：2005-12-01

申请人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  David M. Roush ,  Stephen F. Donovan ,  Frank J. Zawacki ,  Walter H. Yeager ,  John W. Lyga ,  Daniel H. Cohen

发明人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  David M. Roush ,  Stephen F. Donovan ,  Frank J. Zawacki ,  Walter H. Yeager ,  John W. Lyga ,  Daniel H. Cohen

IPC分类号： C07D307/80 ,  C07D495/10

CPC分类号： A01N43/30 ,  A01N43/32 ,  A01N43/40 ,  A01N43/60 ,  A01N47/16 ,  C07D211/22 ,  C07D307/79 ,  C07D307/83 ,  C07D311/04 ,  C07D401/04 ,  C07D495/10

摘要： Insecticidal (dihalopropenyl) phenylalkyl substituted dihydrobenzofuran and dihydrobenzopyran derivatives of Formula I are disclosed. These compounds provide unexpected insecticidal activity across a spectrum of insect pests combined with desirable physical properties including improved photostability. wherein x and y are integers independently selected from 0 or 1; and B is a bridging group *—(CR16R17)q—(CR18R19)r—(CR20R21)s-Lt-(CR22R23)u—(CR24R25)v—(CR26R27)w—, where the asterisk denotes attachment at A; and q, r, s, u, v and w are integers independently selected from 0, 1 and 2; and t is an integer selected from 0 and 1. A, D, E, G, M, R through R11, and R16 through R27, inclusively, are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I and methods of controlling insects by applying said compositions to a locus where insects are present or are expected to be present are also disclosed.

摘要翻译： 公开了杀虫（二卤代丙烯基）苯基烷基取代的二氢苯并呋喃和式I的二氢苯并吡喃衍生物。 这些化合物在一系列昆虫害虫中提供了意想不到的杀虫活性，并结合所需的物理性质，包括改善的光稳定性。 其中x和y是独立地选自0或1的整数; * - （CR16R17）q-（CR18R19）r-（CR20R21）s-Lt-（CR22R23），而B是桥接基团<？in-line-formula description =“In-line Formulas”end =“lead” u-（CR24R25）v-（CR26R27）w - ，<？在线公式描述=“在线公式”end =“tail”？>其中星号表示在A附近; q，r，s，u，v和w是独立地选自0,1和2的整数; 并且t是选自0和1的整数。本文充分描述了A，D，E，G，M，R至R 11和R 16至R 27。 此外，还公开了包含杀虫有效量的至少一种式I化合物的组合物和通过将所述组合物施用于存在昆虫或预期存在的场所来控制昆虫的方法。