Aryl substituted pyrazoles, imidazoles, oxazoles, thiazoles and pyrroles, and the use thereof
    1.
    发明授权
    Aryl substituted pyrazoles, imidazoles, oxazoles, thiazoles and pyrroles, and the use thereof 有权
    芳基取代的吡唑,咪唑,恶唑,噻唑和吡咯,及其用途

    公开(公告)号:US06737418B2

    公开(公告)日:2004-05-18

    申请号:US10134697

    申请日:2002-04-30

    IPC分类号: A61K3142

    摘要: This invention relates to compounds having the Formula I: or a pharmaceutically acceptable salt, prodrug or solvate thereof, wherein Het and R5-R13 are set in the specification. The invention also is directed to the use of compounds of Formula I for the treatment of neuronal damage following global and focal ischemia, for the treatment or prevention of neurodegenerative conditions such as amyotrophic lateral sclerosis (ALS), and for the treatment, prevention or amelioration of both acute or chronic pain, as antitinnitus agents, as anticonvulsants, and as antimanic depressants, as local anesthetics, as antiarrhythmics and for the treatment or prevention of diabetic neuropathy.

    摘要翻译: 本发明涉及具有式I化合物或其药学上可接受的盐,前药或溶剂合物,其中Het和R5-R13在本说明书中设定。 本发明还涉及式I化合物用于治疗全身和局部缺血后的神经元损伤,用于治疗或预防神经变性疾病如肌萎缩性侧索硬化(ALS)以及治疗,预防或改善的用途 作为抗惊厥剂,作为抗惊厥剂,作为抗躁狂抑制剂,作为局部麻醉剂,作为抗心律失常药物和用于治疗或预防糖尿病性神经病变。

    Aryl substituted pyrazoles, and pyrroles, and the use thereof
    2.
    发明授权
    Aryl substituted pyrazoles, and pyrroles, and the use thereof 有权
    芳基取代的吡唑和吡咯及其用途

    公开(公告)号:US06414011B1

    公开(公告)日:2002-07-02

    申请号:US09533864

    申请日:2000-03-24

    IPC分类号: A61K31415

    摘要: This invention relates to compounds having the Formula I: or a pharmaceutically acceptable salt, prodrug or solvate thereof, wherein Het and R5-R13 are set in the specification. The invention also is directed to the use of compounds of Formula I for the treatment of neuronal damage following global and focal ischemia, for the treatment or prevention of neurodegenerative conditions such as amyotrophic lateral sclerosis (ALS), and for the treatment, prevention or amelioration of both acute or chronic pain, as antitinnitus agents, as anticonvulsants, and as antimanic depressants, as local anesthetics, as antiarrhythmics and for the treatment or prevention of diabetic neuropathy.

    摘要翻译: 本发明涉及具有式I化合物或其药学上可接受的盐,前药或溶剂合物,其中Het和R5-R13在本说明书中设定。 本发明还涉及式I化合物用于治疗全身和局部缺血后的神经元损伤,用于治疗或预防神经变性疾病如肌萎缩性侧索硬化(ALS)以及治疗,预防或改善的用途 作为抗惊厥剂,作为抗惊厥剂,作为抗躁狂抑制剂,作为局部麻醉剂,作为抗心律失常药物和用于治疗或预防糖尿病性神经病变。

    Adaptive pilot structure to assist channel estimation in spread spectrum systems
    5.
    发明授权
    Adaptive pilot structure to assist channel estimation in spread spectrum systems 有权
    自适应导频结构,用于在扩频系统中辅助信道估计

    公开(公告)号:US08094737B2

    公开(公告)日:2012-01-10

    申请号:US12064727

    申请日:2006-08-25

    申请人: Phong Nguyen

    发明人: Phong Nguyen

    IPC分类号: H04K1/10

    摘要: The present invention relates generally to methods for generating a dynamic pilot symbol structure in spread spectrum communication systems, and in particular to the use of pilot symbols by user equipment in channel estimation. In one form, the method includes, allocating basic pilot symbols (402) at the beginning of each data chunk (404, 406) and spread over the plurality of sub-carrier frequencies; and selectively replacing data symbols (408) in each data chunk (400) with adaptive pilot symbols (410) according to the speed of the user equipment.

    摘要翻译: 本发明一般涉及用于在扩展频谱通信系统中生成动态导频符号结构的方法,特别涉及用户设备在信道估计中使用导频符号的方法。 在一种形式中,该方法包括:在每个数据块(404,406)的开始处分配基本导频符号(402)并在多个子载波频率上分布; 以及根据所述用户设备的速度,用自适应导频符号(410)选择性地替换每个数据块(400)中的数据符号(408)。

    METHOD AND APPARATUS FOR ENCODING AND DECODING
    6.
    发明申请
    METHOD AND APPARATUS FOR ENCODING AND DECODING 有权
    编码和解码的方法和装置

    公开(公告)号:US20110283171A1

    公开(公告)日:2011-11-17

    申请号:US13125463

    申请日:2009-12-25

    IPC分类号: H03M13/09 G06F11/10

    CPC分类号: H04L1/0079 H04L1/0072

    摘要: A method of encoding a bit sequence over a Physical Downlink Control Channel (PDCCH) having Downlink Control Information (DCI) including: determining DCI bits to provide a DCI bit sequence; performing a CRC calculation on the DCI bit sequence to provide a CRC parity bit sequence; scrambling the CRC parity bit sequence to provide a scrambled CRC bit sequence; if the DCI format is LTE-A, further scrambling the DCI together with the attached scrambled CRC bit sequence to provide a LTE-A scrambled bit sequence; channel coding either the DCI attached scrambled CRC bit sequence or LTE-A scrambled bit sequence to provide a channel coded bit sequence; modulating the channel coded bit sequence to provide a modulated symbol sequence; layer mapping the modulated symbol sequence to one or more antennas associated with a transmitter to provide one or more layers having a symbol sequence; and precoding the layered symbol sequences.

    摘要翻译: 一种通过具有下行链路控制信息(DCI)的物理下行链路控制信道(PDCCH)编码比特序列的方法,包括:确定DCI比特以提供DCI比特序列; 对DCI比特序列执行CRC计算以提供CRC奇偶校验位序列; 对CRC校验位序列进行加扰以提供加扰CRC比特序列; 如果DCI格式是LTE-A,则进一步将DCI与附加的加扰CRC比特序列进行加扰,以提供LTE-A加扰比特序列; 信道编码DCI附加加扰CRC比特序列或LTE-A加扰比特序列以提供信道编码比特序列; 调制所述信道编码比特序列以提供调制符号序列; 将调制符号序列映射到与发射机相关联的一个或多个天线以提供具有符号序列的一个或多个层; 并对分层符号序列进行预编码。

    Method and System for Certifying Operators of X-ray Inspection Systems
    7.
    发明申请
    Method and System for Certifying Operators of X-ray Inspection Systems 有权
    X射线检测系统运行人员认证方法与系统

    公开(公告)号:US20080044801A1

    公开(公告)日:2008-02-21

    申请号:US11773735

    申请日:2007-07-05

    IPC分类号: G09B5/00

    摘要: A method and system for using Threat Imaging Projection (TIP) technology, and the operator testing data that it generates, in order to certify x-ray inspection system operators and thereby assure an acceptable and uniform level of operator performance. In a preferred configuration, the operator views x-ray images of objects on a screening system equipped with TIP technology. When the operator believes that a threat item image appears on the screening system, the operator indicates such via an indicating means. The system is capable of recording, storing and transmitting individual operator performance data relating to proper detections, missed detections, and false alarms, i.e., when an operator indicates that a threat item image appears when no such image actually appears on the screening system. The system preferably contains a library of various threat item images, e.g., guns, bombs, knives, etc., which are classified according to type of threat and difficulty of detection.

    摘要翻译: 一种使用威胁成像投影(TIP)技术的方法和系统,以及操作员对其生成的数据进行测试,以便对x射线检测系统操作人员进行认证,从而确保操作员性能可接受和统一的水平。 在优选的配置中,操作者在配有TIP技术的筛选系统上观察物体的X射线图像。 当操作者认为威胁物品图像出现在筛选系统上时,操作者通过指示装置来表示。 该系统能够记录,存储和发送与正确的检测,错过的检测和假警报有关的各个操作人员的性能数据,即当操作者在没有这样的图像实际上出现在筛选系统上时,显示出威胁物品图像。 系统优选地包含根据威胁类型和检测难度分类的各种威胁物品图像的文库,例如枪,炸弹,刀等。

    Method and system for certifying operators of x-ray inspection systems
    8.
    发明授权
    Method and system for certifying operators of x-ray inspection systems 有权
    X射线检测系统操作者认证方法及系统

    公开(公告)号:US07257189B2

    公开(公告)日:2007-08-14

    申请号:US11343747

    申请日:2006-01-30

    IPC分类号: G01N23/04 G09B19/00

    CPC分类号: G09B19/00 G01V5/0008

    摘要: A method and system for using Threat Imaging Projection (TIP) technology, and the operator testing data that it generates, in order to certify x-ray inspection system operators and thereby assure an acceptable and uniform level of operator performance. In a preferred configuration, the operator views x-ray images of objects on a screening system equipped with TIP technology. When the operator believes that a threat item image appears on the screening system, the operator indicates such via an indicating means. The system is capable of recording, storing and transmitting individual operator performance data relating to proper detections, missed detections, and false alarms, i.e., when an operator indicates that a threat item image appears when no such image actually appears on the screening system. The system preferably contains a library of various threat item images, e.g., guns, bombs, knives, etc., which are classified according to type of threat and difficulty of detection.

    摘要翻译: 一种使用威胁成像投影(TIP)技术的方法和系统,以及操作员对其生成的数据进行测试,以便对x射线检测系统操作人员进行认证,从而确保操作员性能可接受和统一的水平。 在优选的配置中,操作者在配有TIP技术的筛选系统上观察物体的X射线图像。 当操作者认为威胁物品图像出现在筛选系统上时,操作者通过指示装置来表示。 该系统能够记录,存储和发送与正确的检测,错过的检测和假警报有关的各个操作人员的性能数据,即当操作者在没有这样的图像实际上出现在筛选系统上时,显示出威胁物品图像。 系统优选地包含根据威胁类型和检测难度分类的各种威胁物品图像的文库,例如枪,炸弹,刀等。

    Method for decoding channelisation code set information in a spread spectrum receiver

    公开(公告)号:US20070177496A1

    公开(公告)日:2007-08-02

    申请号:US11570104

    申请日:2005-06-07

    申请人: Phong Nguyen

    发明人: Phong Nguyen

    IPC分类号: H04J11/00

    CPC分类号: H04B1/707

    摘要: A method of decoding channelisation code set information to determine the number P of channelisation codes and the code offset O in a spread spectrum data transmission, wherein the channelisation code set information 32 includes a first group of bits encoding the number of channelisation codes and a second group of bits encoding the code offset, the method including the steps of: deriving (30-40) the number P of channelisation codes according to P = C + ⌊ m - A n ⌋ ; and deriving (42-48) the code offset O according to O = ⌊ P n ⌋ × ( m - 2 ⁢ B ) + ( B + 1 ) ; where m is the maximum number of multicodes allocated from the spread spectrum data transmission, n = ⌊ m 2 ⌋ + 1 , A is the value of the first group of bits of the channelisation code set information, B is the value of the second group of bits of the channelisation code set information, and C = A + ⌊ B m - A ⌋ × ( m - 2 ⁢ A ) .

    Aryl substituted pyrazoles, triazoles, and tetrazoles, and the use thereof
    10.
    发明授权
    Aryl substituted pyrazoles, triazoles, and tetrazoles, and the use thereof 有权
    芳基取代的吡唑,三唑和四唑,及其用途

    公开(公告)号:US07078426B2

    公开(公告)日:2006-07-18

    申请号:US09814123

    申请日:2001-03-22

    IPC分类号: A61K31/4155 C07D231/10

    摘要: This invention relates to compounds having the Formula I: or a pharmaceutically acceptable salt, prodrug or solvate thereof, wherein Het and R5-R8 are set in the specification. The invention also is directed to the use of compounds of Formula I for the treatment of neuronal damage following global and focal ischemia, for the treatment or prevention of neurodegenerative conditions such as amyotrophic lateral sclerosis (ALS), and for the treatment, prevention or amelioration of both acute or chronic pain, as antitinnitus agents, as anticonvulsants, and as antimanic depressants, as local anesthetics, as antiarrhythmics and for the treatment or prevention of diabetic neuropathy.

    摘要翻译: 本发明涉及具有式I化合物或其药学上可接受的盐,前药或溶剂化物,其中Het和R 5 -R 8被定义在说明书中。 本发明还涉及式I化合物用于治疗全身和局部缺血后的神经元损伤,用于治疗或预防神经变性疾病如肌萎缩性侧索硬化(ALS)以及治疗,预防或改善的用途 作为抗惊厥剂,作为抗惊厥剂,作为抗躁狂抑制剂,作为局部麻醉剂,作为抗心律失常药物和用于治疗或预防糖尿病性神经病变。