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    2-[4-(4-Chlorophenoxymethyl)-phenoxy]-propionic acid compounds as herbicides
    1.
    发明授权
    2-[4-(4-Chlorophenoxymethyl)-phenoxy]-propionic acid compounds as herbicides 失效
    2- {8 4-（4-氯苯氧基甲基） - 苯氧基{9-丙酸化合物作为除草剂

    公开(公告)号：US4169720A

    公开(公告)日：1979-10-02

    申请号：US819823

    申请日：1977-07-28

    申请人： Erich Schacht ,  Gunter Lauterbach ,  Werner Mehrhof ,  Jurgen Curtze ,  Gerbert Linden ,  Siegmund Lust ,  Klaus Thomas

    发明人： Erich Schacht ,  Gunter Lauterbach ,  Werner Mehrhof ,  Jurgen Curtze ,  Gerbert Linden ,  Siegmund Lust ,  Klaus Thomas

    IPC分类号： A01N31/08 ,  A01N31/14 ,  A01N37/38 ,  A01N39/00 ,  A01N39/02 ,  A01N43/78 ,  A01N47/12 ,  A01N47/20 ,  C07C59/68 ,  C07C59/70 ,  C07C69/712 ,  C07C243/28 ,  C07D277/46 ,  A01N9/12 ,  A01N9/20 ,  A01N9/24

    CPC分类号： C07C243/00 ,  A01N39/02 ,  A01N43/78 ,  A01N47/12 ,  A01N47/20 ,  C07C243/28 ,  C07C251/72 ,  C07C59/68 ,  C07D277/46

    摘要： Compounds of the formula ##STR1## wherein R.sub.1 and R.sub.2 are each hydrogen, chlorine or fluorine; andR.sub.3 is --CH.sub.2 OH, --CH.sub.2 --O--COR.sub.4, --CH.sub.2 --O--CONHR.sub.5, --COOH, --COOCat, --COOR.sub.6, --CONR.sub.7 R.sub.8 or --CO--SR.sub.9 ;where Cat is one equivalent of an inorganic or organic cation;R.sub.4 is hydrogen or alkyl of 1 to 10 carbon atoms;R.sub.5 is alkyl of 1 to 4 carbon atoms, phenyl or halo-substituted phenyl;R.sub.6 is alkyl of 1 to 10 carbon atoms which may optionally have a chloro, hydroxyl, lower alkoxy, lower alkoxy-lower alkoxy, lower alkylthio, amino, mono-lower alkyl-amino, di-lower alkyl-amino, allyloxy or phenoxy substituent attached thereto; phenyl; benzyl; monochloro-benzyl; dichloro-benzyl; cyclohexyl; 1-ethynyl-cyclohexyl; lower alkenyl; lower alkynyl; --N.dbd.C(CH.sub.3).sub.2 ; 2--(2',4',5'-trichloro-phenoxy)-ethyl, 2-(2', 5'-dichloro-4'-bromo-phenoxy)-ethyl; or ##STR2## R.sub.7 is hydrogen, lower alkyl, hydroxy-lower alkyl, lower alkenyl, lower alkynyl, phenyl, chloro-substituted phenyl, hydroxyl, amino, phenyl-amino or thiazolyl;R.sub.8 is hydrogen, lower alkyl, lower alkenyl or hydroxy-lower alkyl;R.sub.9 is hydrogen or alkyl of 1 to 10 carbon atoms; andN is an integer from 2 to 6, inclusive.The compounds are useful as herbicides.

    摘要翻译： 其中R 1和R 2各自为氢，氯或氟的式“IMAGE”的化合物; 且R 3为-CH 2 OH，-CH 2 -O-COR 4，-CH 2 -O-CONHR 5，-COOH，-COOCat，-COOR 6，-CONR 7 R 8或-CO-SR 9; 其中Cat是1当量的无机或有机阳离子; R4是氢或1-10个碳原子的烷基; R5是1-4个碳原子的烷基，苯基或卤素取代的苯基; R6是具有1-10个碳原子的烷基，其可任选地具有氯，羟基，低级烷氧基，低级烷氧基 - 低级烷氧基，低级烷硫基，氨基，单低级烷基 - 氨基，二低级烷基 - 氨基，烯丙氧基或苯氧基取代基 附于其上 苯基; 苄基; 一氯 - 苄基; 二氯苄基; 环己基 1-乙炔基 - 环己基; 低级链烯基 低级炔基 -N = C（CH 3）2; 2-（2'，4'，5'-三氯 - 苯氧基） - 乙基，2-（2'，5'-二氯-4'-溴 - 苯氧基） - 乙基; 或者R 7是氢，低级烷基，羟基 - 低级烷基，低级烯基，低级炔基，苯基，氯取代的苯基，羟基，氨基，苯基 - 氨基或噻唑基。 R8是氢，低级烷基，低级烯基或羟基 - 低级烷基; R9是氢或1-10个碳原子的烷基; 并且N是从2到6的整数，包含。

    Phenylbutanol derivatives, processes for their preparation and compositions containing them
    4.
    发明授权
    Phenylbutanol derivatives, processes for their preparation and compositions containing them 失效
    苯乙醇衍生物及其制备方法及其组合物

    公开(公告)号：US4136200A

    公开(公告)日：1979-01-23

    申请号：US810712

    申请日：1977-06-28

    申请人： Erich Schacht ,  Werner Mehrhof ,  Albrecht Wild ,  Joachim Gante ,  Hans-Adolf Kurmeier

    发明人： Erich Schacht ,  Werner Mehrhof ,  Albrecht Wild ,  Joachim Gante ,  Hans-Adolf Kurmeier

    IPC分类号： C07C43/295 ,  C07C59/48 ,  C07C59/68 ,  C07C43/20

    CPC分类号： C07C59/68 ,  C07C43/295 ,  C07C59/48

    摘要： Phenylbutanol derivatives of the formula Z-C(CH.sub.3) (OH)-CH.sub.2 -Y wherein Z is 4-biphenyl or 4-phenoxyphenyl wherein the phenoxy group is unsubstituted or substituted by F, Cl or Br and Y is COOR.sup.2 or CH.sub.2 OR.sup.3 wherein R.sup.2 is H or alkyl of 1 to 6 carbon atoms and R.sup.3 is H or alkanoyl of 1 to 6 carbon atoms, and their physiologically acceptable salts, possess anti-inflammatory activity and are produced by (a) treating with a solvolyzing agent a compound of the formula Z-C(CH.sub.3) (OH)-CH.sub.2 -W or Z-CX(CH.sub.3)-CH.sub.2 -Y wherein W is a functionally modified carboxy or methylol group different from Y and X is Cl, Br or I or a functionally modified hydroxyl group; or (b) reducing a compound otherwise corresponding to a desired final product but having instead of one of the hydrogen atoms a group which can be reduced or replaced by a hydrogen atom; or (c) oxidizing a compound otherwise corresponding to a desired final product but lacking the tertiary hydroxyl group; or (d) converting a compound otherwise corresponding to a desired final product wherein Z is a 4-phenoxyphenyl group but having instead a 4-OH-, Cl-, Br- or 1-substituted phenyl group into a desired final product; or (e) diazotizing a compound otherwise corresponding to a desired final product wherein Z is a halogen-substituted 4-phenoxyphenyl group but having an --NH.sub.2 -substituted phenoxy group and reacting the resulting diazonium salt with a halogenating agent.

    Diphenoxyacetic acid derivatives
    5.
    发明授权
    Diphenoxyacetic acid derivatives 失效
    二苯氧基乙酸衍生物

    公开(公告)号：US4051170A

    公开(公告)日：1977-09-27

    申请号：US531475

    申请日：1974-12-11

    申请人： Erich Schacht ,  Werner Mehrhof ,  Zdenek Simane ,  Detlev Kayser ,  Herbert Nowak

    发明人： Erich Schacht ,  Werner Mehrhof ,  Zdenek Simane ,  Detlev Kayser ,  Herbert Nowak

    IPC分类号： C07D295/08 ,  C07C51/00 ,  C07C51/08 ,  C07C59/125 ,  C07C59/68 ,  C07C59/70 ,  C07C67/00 ,  C07C69/712 ,  C07D215/06 ,  C07D215/14 ,  C07D215/22 ,  C07D215/233 ,  C07D295/096 ,  C07D311/58 ,  C07D335/06

    CPC分类号： C07D215/233 ,  C07C51/08 ,  C07C59/68 ,  C07C59/70 ,  C07D215/06 ,  C07D215/14 ,  C07D295/096 ,  C07D311/58 ,  C07D335/06

    摘要： Diphenoxyacetic acid derivatives of the general formula ##STR1## wherein R.sub.1 is H or alkyl of 1-4 carbon atoms, R.sub.2 is H or Cl, R.sub.2 is H or Cl, R.sub.3 is piperidino, 4-piperidinophenyl, 1,2,3,4-tetrahydroquinolino, 1-R.sub.4 -1,2,3,4-tetrahydro-4-quinolyl, 4-oxo-1,2,3,4-tetrahydroquinolino, 4-chromanyl, 4-thiochromanyl or 4-chlorophenoxy, and R.sub.4 is H or alkyl of 1-4 carbon atoms, and the physiologically acceptable salts thereof, possess cholesterol level lowering activity and can be prepared by reacting a phenol of the formula ##STR2## with a compound of the formula ##STR3## wherein X is OH, esterified OH, Cl, Br or I, one R is R.sub.2 and the other is R.sub.3 ; or by cyclizing a compound of the formula ##STR4## wherein X.sub.1 is Cl, Br, I, NH.sub.2 OH or an esterified or etherified OH-group and n is 0 or 1; or by treating a compound of the formula ##STR5## wherein Z is a functionally modified carboxyl group different from COOR.sub.1, with a solvolyzing agent, R.sub.1, R.sub.2 and R.sub.3 in each instance having the values given above.

    摘要翻译： 其中R 1为H或1-4个碳原子的烷基，R 2为H或Cl，R 2为H或Cl，R 3为哌啶子基，4-哌啶子基苯基，1,2,3,4 1-四氢喹啉，1-R4-1,2,3,4-四氢-4-喹啉基，4-氧代-1,2,3,4-四氢喹啉，4-苯并二氢吡喃基，4-硫代苯并二氢吡喃基或4-氯苯氧基，R4是 H或1-4个碳原子的烷基及其生理上可接受的盐具有降低胆固醇水平的活性，并且可以通过使下式的苯酚与下式化合物（IMAGE）反应来制备，其中X是OH， 酯化的OH，Cl，Br或I，一个R是R 2，另一个是R 3; 或者通过环化式（VI）的化合物，其中X 1是Cl，Br，I，NH 2 + L，OH或酯化或醚化的OH-基团，n是0或1; 或者通过用溶剂分解剂，R 1，R 2和R 3在每种情况下处理具有上述给定值的式“IMAGE”的化合物，其中Z是不同于COOR1的官能改性羧基。

    2-Methyl-2-[4-(4-piperidinophenyl)-phenoxy]-propionic acid 1-methyl-4-piperidyl ester
    8.
    发明授权
    2-Methyl-2-[4-(4-piperidinophenyl)-phenoxy]-propionic acid 1-methyl-4-piperidyl ester 失效
    2-甲基-2- {8 4-（4-哌啶基苯基） - 苯氧基{9-丙酸1-甲基-4-哌啶基酯

    公开(公告)号：US3956334A

    公开(公告)日：1976-05-11

    申请号：US483408

    申请日：1974-06-26

    申请人： Erich Schacht ,  Werner Mehrhof ,  Herbert Nowak ,  Zdenek Simane

    发明人： Erich Schacht ,  Werner Mehrhof ,  Herbert Nowak ,  Zdenek Simane

    IPC分类号： C07D295/08 ,  C07D295/096 ,  C07D211/46

    CPC分类号： C07D295/096

    摘要： Piperidines of the formula ##SPC1##Wherein R is --CH.sub.2 OH, CO--NR,R.sub.2 in which R.sub.1 and R.sub.2 each are H or alkyl of 1-4 carbon atoms, --NHCH.sub.2 CH.sub.2 OH, --N(CH.sub.2 CH.sub.2 OH).sub.2, --NHCH.sub.2 CH.sub.2 SO.sub.3 H, --NHNH.sub.2 or --NHCH.sub.2 COOH, or --COOR.sub.3 in which R.sub.3 is 3-pyridylmethyl, 2-acetamidoethyl, 1-methyl-4-piperidyl or 2,3-dihydroxypropyl and the physiologically acceptable salts thereof, have cholesterol-level-lowering and triglyceride-level-lowering activity and can be prepared from 2-methyl-2-[4-(4-piperidinophenyl)-phenoxy]-propionic acid or a functional derivative thereof by reduction or by reaction with a compound of the formula HZ.

    摘要翻译： 式WHEREIN R是-CH 2 OH，CO-NR，R 2，其中R 1和R 2各自为H或1-4个碳原子的烷基，-NHCH 2 CH 2 OH，-N（CH 2 CH 2 OH）2，-NHCH 2 CH 2 SO 3 H，-NHNH 2或-NHCH 2 COOH 或其中R3为3-吡啶基甲基，2-乙酰氨基乙基，1-甲基-4-哌啶基或2,3-二羟基丙基的-COOR 3及其生理学上可接受的盐具有降低胆固醇含量和降低甘油三酯水平的活性， 可以由2-甲基-2- [4-（4-哌啶基苯基） - 苯氧基] - 丙酸或其官能衍生物通过还原或与式HZ的化合物反应来制备。