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公开(公告)号：US20160251372A1
公开(公告)日：2016-09-01
申请号：US15059142
申请日：2016-03-02
Applicant: SENOMYX, INC.
Inventor： Catherine Tachdjian , Xiao Qing Tang , Donald S. Karanewsky , Guy Servant , Xiaodong Li , Feng Zhang , Qing Chen , Hong Zhang , Timothy Davis , Vincent Darmohusodo , Melissa Wong , Victor Selchau
IPC: C07D495/04 , A61K47/22 , A23L2/56 , C07D401/12 , C07D405/12 , C07D215/54 , C07D471/04
CPC classification number: C07D495/04 , A23L2/56 , A23L27/2054 , A23L27/88 , A23V2002/00 , A61K47/22 , C07D215/54 , C07D215/60 , C07D401/12 , C07D405/12 , C07D471/04 , C07D491/048
Abstract: The present invention includes compounds having structural formula (I), or pharmaceutically acceptable salts, solvate, and/or ester thereof. These compounds are useful as sweet flavor modifiers. The present invention also includes compositions comprising the present compounds and methods of enhancing the sweet taste of ingestible compositions. Furthermore, the present invention provides methods for preparing the compounds.
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Patent Agency Ranking
公开(公告)号：US20150265711A1
公开(公告)日：2015-09-24
申请号：US14731224
申请日：2015-06-04
Applicant: SENOMYX, INC.
Inventor： Catherine Tachdjian , Xiao Qing Tang , Donald S. Karanewsky , Guy Servant , Xiaodong Li , Feng Zhang , Qing Chen , Hong Zhang , Timothy Davis , Vincent Darmohusodo , Melissa Wong , Victor Selchau
CPC classification number: C07D495/04 , A23L2/56 , A23L27/2054 , A23L27/88 , A23V2002/00 , A61K47/22 , C07D215/54 , C07D215/60 , C07D401/12 , C07D405/12 , C07D471/04 , C07D491/048
Abstract: The present invention includes compounds having structural formula (I), or pharmaceutically acceptable salts, solvate, and/or ester thereof. These compounds are useful as sweet flavor modifiers. The present invention also includes compositions comprising the present compounds and methods of enhancing the sweet taste of ingestible compositions. Furthermore, the present invention provides methods for preparing the compounds.
Abstract translation: 本发明包括具有结构式（I）的化合物或其药学上可接受的盐，溶剂化物和/或酯。 这些化合物可用作甜味调味剂。 本发明还包括包含本发明化合物的组合物和增强可摄入组合物的甜味的方法。 此外，本发明提供了制备化合物的方法。
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公开(公告)号：US09181276B2
公开(公告)日：2015-11-10
申请号：US14077749
申请日：2013-11-12
Applicant: SENOMYX, INC.
Inventor： Catherine Tachdjian , Donald S. Karanewsky , Xiao-Qing Tang , Xiaodong Li , Feng Zhang , Guy Servant , Qing Chen , Vincent Darmohusodo , Richard Fine , Joseph R. Fotsing , Jeffrey Robert Hammaker , Xinshan Kang , Rachel D. A. Kimmich , Boris Klebansky , Haitian Liu , Goran Petrovic , Marketa Rinnova , Sara Adamski-Werner , Jeffrey Yamamoto , Hong Zhang , Albert Zlotnik
IPC: C07D239/95 , C07D285/16 , A61K31/517 , A61K31/54 , C07D513/04 , C07D417/04 , C07D417/12 , A23L1/236 , A23L2/60 , A23L2/39 , A23L1/22
CPC classification number: C07D513/04 , A23L2/39 , A23L2/60 , A23L27/30 , A23L27/31 , A23L27/33 , A23L27/34 , A23L27/88 , C07D215/42 , C07D215/54 , C07D215/56 , C07D239/70 , C07D239/84 , C07D239/94 , C07D239/95 , C07D285/16 , C07D417/04 , C07D417/12 , C07D471/04 , C07D487/04 , C07D491/04 , C07D491/056 , C07D493/04 , C07D495/04 , C07D495/14 , C07D513/20 , G01N33/566
Abstract: The present invention includes methods for identifying modifiers of chemosensory receptors and their ligands, e.g., by determining whether a test entity is suitable to interact with one or more interacting sites within the Venus flytrap domains of the chemosensory receptors, and modifiers capable of modulating chemosensory receptors and their ligands. The present invention also includes modifiers of chemosensory receptors and their ligands having Formula (I), its subgenus, and specific compounds. Furthermore, the present invention includes ingestible compositions comprising the modifiers of chemosensory receptors and their ligands and methods of using the modifiers of chemosensory receptors and their ligands to enhance the sweet taste of an ingestible composition or treat a condition associated with a chemosensory receptor. In addition, the present invention include processes for preparing the modifiers of chemosensory receptors and their ligands.
Abstract translation: 本发明包括用于鉴定化学感受器及其配体的调节剂的方法，例如通过确定测试实体是否适合与化学感应受体的金星蝇捕获区域内的一个或多个相互作用位点相互作用，以及能够调节化学感应受体 及其配体。 本发明还包括具有式（I），其亚属和特定化合物的化学感应受体及其配体的改性剂。 此外，本发明包括含有化学感应受体调节剂及其配体的可摄入组合物，以及使用化学感应受体及其配体改性剂增强可摄入组合物的甜味或治疗与化学感觉受体相关的病症的方法。 此外，本发明包括制备化学感受器及其配体的改性剂的方法。
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公开(公告)号：US09049878B2
公开(公告)日：2015-06-09
申请号：US14061013
申请日：2013-10-23
Applicant: SENOMYX, INC.
Inventor： Catherine Tachdjian , Xiao Qing Tang , Donald S. Karanewsky , Guy Servant , Xiaodong Li , Feng Zhang , Qing Chen , Hong Zhang , Timothy Davis , Vincent Darmohusodo , Melissa Wong , Victor Selchau
IPC: A23L1/236 , A23L1/22 , A23L1/226 , C07D215/54 , C07D215/60 , C07D401/12 , C07D405/12 , C07D471/04 , C07D491/048 , C07D495/04 , A61K47/22
CPC classification number: C07D495/04 , A23L2/56 , A23L27/2054 , A23L27/88 , A23V2002/00 , A61K47/22 , C07D215/54 , C07D215/60 , C07D401/12 , C07D405/12 , C07D471/04 , C07D491/048
Abstract: The present invention includes compounds having structural formula (I), or pharmaceutically acceptable salts, solvate, and/or ester thereof. These compounds are useful as sweet flavor modifiers. The present invention also includes compositions comprising the present compounds and methods of enhancing the sweet taste of ingestible compositions. Furthermore, the present invention provides methods for preparing the compounds.
Abstract translation: 本发明包括具有结构式（I）的化合物或其药学上可接受的盐，溶剂化物和/或酯。 这些化合物可用作甜味调味剂。 本发明还包括包含本发明化合物的组合物和增强可摄入组合物的甜味的方法。 此外，本发明提供了制备化合物的方法。
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公开(公告)号：US09834544B2
公开(公告)日：2017-12-05
申请号：US14337764
申请日：2014-07-22
Applicant: SENOMYX, INC.
Inventor： Catherine Tachdjian , Xiao Qing Tang , Donald S. Karanewsky , Guy Servant , Xiaodong Li , Feng Zhang , Qing Chen , Hong Zhang , Timothy James Davis , Vincent Darmohusodo , Melissa S. Wong , Victor Selchau
IPC: C07D405/12 , A23L2/60 , C07D401/12 , C07D215/54 , C07D451/06 , A61K47/22 , C07D215/42 , A23L27/00
CPC classification number: C07D405/12 , A23L2/60 , A23L27/88 , A23V2002/00 , A61K47/22 , C07D215/42 , C07D215/54 , C07D401/12 , C07D451/06
Abstract: The present invention includes compounds having structural formula (I), or salts or solvates thereof. These compounds are useful as sweet flavor modifiers. The present invention also includes compositions comprising the present compounds and methods of enhancing the sweet taste of compositions.
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公开(公告)号：US09902737B2
公开(公告)日：2018-02-27
申请号：US15059142
申请日：2016-03-02
Applicant: SENOMYX, INC.
Inventor： Catherine Tachdjian , Xiao Qing Tang , Donald S. Karanewsky , Guy Servant , Xiaodong Li , Feng Zhang , Qing Chen , Hong Zhang , Timothy Davis , Vincent Darmohusodo , Melissa S. Wong , Victor Selchau
IPC: C07D495/04 , C07D215/54 , C07D215/60 , C07D401/12 , C07D405/12 , C07D471/04 , C07D491/048 , A61K47/22 , A23L2/56 , A23L27/00 , A23L27/20
CPC classification number: C07D495/04 , A23L2/56 , A23L27/2054 , A23L27/88 , A23V2002/00 , A61K47/22 , C07D215/54 , C07D215/60 , C07D401/12 , C07D405/12 , C07D471/04 , C07D491/048
Abstract: The present invention includes compounds having structural formula (I), or pharmaceutically acceptable salts, solvate, and/or ester thereof. These compounds are useful as sweet flavor modifiers. The present invention also includes compositions comprising the present compounds and methods of enhancing the sweet taste of ingestible compositions. Furthermore, the present invention provides methods for preparing the compounds.
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