Cis-substituted fluoromethylpyrrolidine derivative
    1.
    发明授权
    Cis-substituted fluoromethylpyrrolidine derivative 失效
    顺式取代的氟甲基吡咯烷衍生物

    公开(公告)号:US06656952B2

    公开(公告)日:2003-12-02

    申请号:US09446696

    申请日:1999-12-23

    CPC classification number: C07D401/04

    Abstract: An antibacterial drug having potent antibacterial activities upon various bacteria including resistant strains and high safety is disclosed, which comprises as an active ingredient, quinolone derivatives represented by the following formula (I), its salts or hydrates thereof: wherein R1 represents a hydrogen atom or an alkyl group having 1 to 6 carbon atoms, R2 represents a halogenomethoxyl group or an alkoxyl group, R3 represents an alkyl group, an alkenyl group, a halogenoalkyl group, a cyclic alkyl group, a heteroaryl group, an alkoxyl group or an alkylamino group, and R4 represents a hydrogen atom, a phenyl group, an acetoxymethyl group, a pivaloyloxymethyl group, an ethoxycarbonyl group, a choline group, a dimethylaminoethyl group, a 5-indanyl group, a phthalidinyl group, a 5-alkyl-2-oxo-1,3-dioxol-4-ylmethyl group, 3-acetoxy-2-oxobutyl group, an alkyl group, an alkoxylmethyl group or a phenylalkyl group. These substituents may further have additional substituents.

    Abstract translation: 本发明公开了一种对各种细菌(包括耐药菌株)和高度安全性具有有效抗菌活性的抗菌药物,其包含作为活性成分的由下式(I)表示的喹诺酮衍生物,其盐或水合物:其中R 1表示 氢原子或碳原子数1〜6的烷基,R 2表示卤代甲氧基或烷氧基,R 3表示烷基,链烯基,卤代烷基,环状烷基,杂芳基 基团,烷氧基或烷基氨基,R 4表示氢原子,苯基,乙酰氧基甲基,新戊酰氧基甲基,乙氧基羰基,胆碱基,二甲基氨基乙基,5-二氢化茚基, 5-烷基-2-氧代-1,3-二氧杂环戊烯-4-基甲基,3-乙酰氧基-2-氧代丁基,烷基,烷氧基甲基或苯基烷基。 这些取代基还可以具有另外的取代基。

    Foldable and simplified water tank
    2.
    发明授权
    Foldable and simplified water tank 失效
    可折叠和简化的水箱

    公开(公告)号:US6021915A

    公开(公告)日:2000-02-08

    申请号:US714980

    申请日:1996-09-17

    CPC classification number: E04H4/0025

    Abstract: A foldable and simplified water tank characterized by a cylindrical shape and a side wall formed by a sheet made from synthetic resin, and the stiffness of said sheet, measured in accordance with the measuring method prescribed in Japan Industrial Standard L-1096 is from 100 to 1000. The water tank can be made to stand up by itself by only pouring water into it.

    Abstract translation: 一种折叠简化的水箱,其特征在于圆筒形状和由合成树脂制成的片形成的侧壁,并且根据日本工业标准L-1096中规定的测量方法测量的所述片材的刚度为100至 水罐可以自己立起来,只能把水倒入水中。

    Apparatus for testing optical fiber by using detector having virtually
broadened dynamic range
    3.
    发明授权
    Apparatus for testing optical fiber by using detector having virtually broadened dynamic range 失效
    用于通过使用具有虚拟宽带动态范围的探测器测试光纤的装置

    公开(公告)号:US5159400A

    公开(公告)日:1992-10-27

    申请号:US766238

    申请日:1991-09-24

    CPC classification number: G01M11/3172

    Abstract: An optical fiber testing apparatus for testing an optical fiber as to presence and location of a fault such as breakage by inputting a pulsed coherent light beam to the optical fiber and synthesizing a return light beam reflected back from the optical fiber with a reference light beam having a frequency deviated from the pulsed light beam by a predetermined amount, wherein the synthesized waveform is detected through optical heterodyning. The electric signal obtained from the heterodyning detection is detected by an envelope detector, of which dynamic range is effectively virtually broadened by using correcting data prepared previously. The optical fiber test can be accomplished through a single measurement without involving expensiveness of hardware.

    Abstract translation: 一种光纤测试装置,用于通过向光纤输入脉冲相干光束并合成从光纤反射回来的返回光束,用参考光束来测试光纤是否存在和定位故障,例如断裂,所述参考光束具有 频率偏离脉冲光束预定量,其中通过光学外差检测合成波形。 由外部检测获得的电信号由包络检测器检测,其中动态范围通过使用之前准备的校正数据被有效地扩大。 光纤测试可以通过单个测量来实现,而不涉及硬件的昂贵性。

    Method and container for insecticidally storing grains
    5.
    发明授权
    Method and container for insecticidally storing grains 失效
    杀虫剂储存方法和容器

    公开(公告)号:US6063418A

    公开(公告)日:2000-05-16

    申请号:US77095

    申请日:1998-07-14

    CPC classification number: A23B9/22 A23B9/18 A23B9/20

    Abstract: A method and a container for long-term storage in a state in which harmful insects do not propagate, in a case in which grains such as unpolished rice or the like are filled and stored. An inner bag (10) made of a flexible material is accommodated in an outer bag (12) which has high-strength. After grains are filled in the inner bag, the inner bag (10) is filled with carbon dioxide gas and is closed. The grains are stored in a state in which harmful insects are exterminated. It is preferable from the standpoint of the insecticidal effect that the inner portion of the inner bag (10) is able to maintain a carbon dioxide gas concentration of 40% or more for 7 days or more. Because the inner bag has the property of a CO.sub.2 permeation amount of less than or equal to 6300 cc/m.sup.2 .multidot.24 hr 1 atm, an oxygen-deficient state can be maintained.

    Abstract translation: PCT No.PCT / JP96 / 03704 Sec。 371日期:1998年7月14日 102(e)日期1998年7月14日PCT 1996年12月19日PCT PCT。 出版物WO97 / 22258 日期1997年6月26日在填充并储存诸如未磨光米等的颗粒的情况下,在有害昆虫不传播的状态下长期储存的方法和容器。 由柔性材料制成的内袋(10)容纳在具有高强度的外袋(12)中。 在内袋中填充颗粒后,内袋(10)填充有二氧化碳气体并关闭。 谷物被储存在有害昆虫被灭绝的状态。 从杀虫效果的观点出发,优选内袋(10)的内部能够将二氧化碳气体浓度保持在40%以上,持续7天以上。 因为内袋具有小于或等于6300cc / m2×24小时1atm的CO 2渗透量的性质,因此可以保持缺氧状态。

    Electronic circuit capable of stably keeping a frequency during presence
of a burst
    7.
    发明授权
    Electronic circuit capable of stably keeping a frequency during presence of a burst 失效
    能够在存在突发时稳定地保持频率的电子电路

    公开(公告)号:US4633510A

    公开(公告)日:1986-12-30

    申请号:US687343

    申请日:1984-12-28

    CPC classification number: H04B1/40 H03L7/14

    Abstract: In a radio communication system, a transmitting section of a substation comprises a controlling circuit (21) for controlling a carrier frequency of a local oscillator (24) in response to a frequency deviation signal. A burst generating circuit (26) generates a burst in response to the input signal, a burst control signal, and a local oscillation signal of the carrier frequency. The transmitting section further comprises a holding circuit (34) responsive to a frequency control signal and the burst control signal. During presence of the burst control signal, the holding circuit holds the frequency control signal received before a beginning of the burst control signal to keep the carrier frequency of the local oscillation signal invariable until an end of the burst control signal. Otherwise, the frequency control signal passes through the holding circuit as it stands. Consequently, the carrier frequency of the local oscillation signal is controlled only during absence of the input signal and is kept invariable during presence of the input signal.

    Abstract translation: 在无线电通信系统中,变电站的发送部分包括用于响应于频率偏差信号来控制本地振荡器(24)的载波频率的控制电路(21)。 突发发生电路(26)响应于输入信号,脉冲串控制信号和载波频率的本地振荡信号产生脉冲串。 发送部分还包括响应于频率控制信号和突发控制信号的保持电路(34)。 在脉冲串控制信号的存在期间,保持电路保持在突发控制信号开始之前接收到的频率控制信号,以保持本地振荡信号的载波频率不变,直到脉冲串控制信号的结束。 否则,频率控制信号就一直通过保持电路。 因此,本地振荡信号的载波频率仅在没有输入信号的情况下被控制,并且在存在输入信号的过程中保持不变。

    Disc brake for motor vehicles
    8.
    发明授权
    Disc brake for motor vehicles 有权
    机动车盘式制动器

    公开(公告)号:US06851524B2

    公开(公告)日:2005-02-08

    申请号:US10606802

    申请日:2003-06-27

    Abstract: The disc brake for a motor vehicle contains a caliper bracket to be secured to a vehicle body on the outer side of a disc rotor with respect to the vehicle body, a caliper body supported by the caliper bracket to be slidable in the axial direction of the disc rotor and a pair of friction pads disposed to oppose each other through the disc rotor. The caliper bracket contains a bracket main body and a connecting arm which are disposed respectively on the outer side and on the inner side of the disc rotor with respect to the vehicle body, as well as, a pair of caliper supporting arms, which connect the bracket main body with the connecting arm at their disc turning-in side end portions and at their disc turning-out side end portions, respectively. The bracket main body and the connecting arm have torque receiving portions at least on the disc turning-out side respectively to receive braking torques from the respective friction pads; the bracket main body has a disc turning-out side fixing portion, where the caliper bracket is secured to the vehicle body, located outer than the disc turning-out side torque receiving portion toward the disc turning-out side and substantially on the peripheral edge of the disc rotor.

    Abstract translation: 用于机动车辆的盘式制动器包括卡钳支架,其被固定到相对于车身的盘形转子的外侧上的车身,由卡钳托架支撑的卡钳体可沿着该车辆的轴向方向滑动 盘形转子和通过盘形转子彼此相对设置的一对摩擦垫。 卡钳支架包括分别设置在盘转子相对于车体的外侧和内侧的支架主体和连接臂,以及一对卡钳支撑臂,其连接 支架主体,其连接臂分别在盘的转动侧端部和盘的转出侧端部。 支架主体和连接臂分别至少在盘转出侧上具有转矩接收部分,以从各个摩擦垫接收制动力矩; 支架主体具有盘转出侧固定部,卡钳支架固定在车体上,位于盘转出侧转矩接收部的外侧,朝向盘转出侧且基本上位于周缘 的圆盘转子。

    Method for preparing water-soluble lacquer
    9.
    发明授权
    Method for preparing water-soluble lacquer 失效
    制备水溶性漆的方法

    公开(公告)号:US4312895A

    公开(公告)日:1982-01-26

    申请号:US230881

    申请日:1981-02-02

    CPC classification number: C09K11/02 C08G65/30 C09D171/02

    Abstract: This invention relates to a method for preparing a water soluble lacquer, which comprises dissolving polyethylene oxide having a molecular weight of at least 2,500,000 in water to form a polyethylene oxide aqueous solution, adding acid to said solution in such a manner as to adjust the pH of the solution in the range of from 3.0 to 5.0, heating the resultant solution at a temperature of not lower than 95.degree. C., cooling the solution and removing the remaining acid with an ion exchange resin.

    Abstract translation: 本发明涉及一种制备水溶性漆的方法,其包括将分子量至少为2,500,000的聚环氧乙烷溶于水中以形成聚环氧乙烷水溶液,向所述溶液中加入酸以调节pH 的溶液在3.0至5.0的范围内,在不低于95℃的温度下加热所得溶液,冷却溶液并用离子交换树脂除去剩余的酸。

    Cycloalkyl-substituted aminomethylpyrrolidine derivatives
    10.
    发明授权
    Cycloalkyl-substituted aminomethylpyrrolidine derivatives 失效
    环烷基取代的氨基甲基吡咯烷衍生物

    公开(公告)号:US06573260B1

    公开(公告)日:2003-06-03

    申请号:US09856631

    申请日:2001-05-24

    CPC classification number: C07D401/04

    Abstract: This invention provides a quinolone derivative which exerts strong antibacterial action upon various bacteria and has high safety, and it relates to a compound having a structure of formula (I), its salts and hydrates thereof: {R1 and R2: hydrogen, alkyl; n: 1 to 4; Q: following structure (Ia): [R3: alkyl, alkenyl, halogenoalkyl, cyclic alkyl, aryl, heteroaryl, alkoxyl, alkylamino; R4: hydrogen, alkylthio; R5: hydrogen, amino, hydroxyl, thiol, halogenomethyl, alkyl, alkenyl, alkynyl, alkoxyl; X1: halogen, hydrogen, A1: nitrogen, structure of formula (II): (X2: hydrogen, amino, halogen, cyano, halogenomethyl, halogenomethyl, alkyl, alkenyl, alkynyl, alkoxyl; R4 and R3 or X2 and R3 may together form a cyclic structure; Y: hydrogen, various ester forming groups]}.

    Abstract translation: 本发明提供了一种喹诺酮衍生物,其对各种细菌具有强烈的抗菌作用并具有高度的安全性,它涉及具有式(I)结构的化合物及其盐和水合物:{R1和R2:氢,烷基; n:1到4; Q:以下结构(Ia):[R3:烷基,烯基,卤代烷基,环烷基,芳基,杂芳基,烷氧基,烷基氨基; R4:氢,烷硫基; R5:氢,氨基,羟基,硫醇,卤代甲基,烷基,烯基,炔基,烷氧基; X1:卤素,氢,A1:氮,式(II)的结构:(X2:氢,氨基,卤素,氰基,卤代甲基,卤代甲基,烷基,烯基,炔基,烷氧基; R4和R3或X2和R3可以一起形成 环状结构; Y:氢,各种酯形成基团]}。

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