Acid amide derivatives, process for producing these, and pest control agent containing these
    2.
    发明授权
    Acid amide derivatives, process for producing these, and pest control agent containing these 有权
    酸酰胺衍生物,其制备方法,以及含有它们的害虫防治剂

    公开(公告)号:US07683096B2

    公开(公告)日:2010-03-23

    申请号:US10489778

    申请日:2002-09-18

    IPC分类号: A61K31/35

    摘要: The present invention relates to an acid amid derivative of the formula (I) or a salt thereof: wherein A is phenyl which may be substituted by X, benzyl which may be substituted by X, naphthyl which may be substituted by X, a heterocyclic group which may be substituted by X, a fused heterocyclic group which may be substituted by X, indanyl (the indanyl may be substituted by halogen, alkyl or alkoxy) or tetrahydronaphthyl (the tetrahydronaphthyl may be substituted by halogen, alkyl or alkoxy), B is alkyl, cycloalkyl, phenyl which may be substituted by Y, a heterocyclic group which may be substituted by Y, or a condensed heterocyclic group which may be substituted by Y, each of R1 and R2 is alkyl, cyano or —CO2R14, or R1 and R2 may together form a 3- to 6-membered saturated carbocyclic ring, R3 is hydrogen, alkyl, alkoxyalkyl, alkylthioalkyl, —COR15, —S(O)mR16 or —S(O)nNR17R18, which is useful as an active ingredient of pesticides.

    摘要翻译: 本发明涉及式(I)的酸酰胺衍生物或其盐:其中A为可被X取代的苯基,可被X取代的苄基,可被X取代的萘基,杂环基 其可以被X取代,可以被X取代的稠合杂环基,茚满基(茚满基可以被卤素,烷基或烷氧基取代)或四氢萘基(四氢萘基可以被卤素,烷基或烷氧基取代),B是 烷基,环烷基,可被Y取代的苯基,可被Y取代的杂环基或可被Y取代的稠合杂环基,R 1和R 2各自为烷基,氰基或-CO 2 R 14,或R 1和 R2可以一起形成3至6元饱和碳环,R 3是氢,烷基,烷氧基烷基,烷硫基烷基,-COR 15,-S(O)m R 16或-S(O)n NR 17 R 18,其可用作 农药。

    Phenacylamine derivatives, process for their production and pesticides containing them
    3.
    发明授权
    Phenacylamine derivatives, process for their production and pesticides containing them 有权
    苯甲酰胺衍生物,其生产工艺和含有它们的农药

    公开(公告)号:US07439366B2

    公开(公告)日:2008-10-21

    申请号:US10181963

    申请日:2001-02-09

    摘要: The present invention relates to a phenacylamine derivative of the formula (I) or a salt thereof: wherein A is alkyl, cycloalkyl, phenyl which may be substituted by Y, pyridyl which may be substituted by Y, or pyrazolyl which may be substituted by Y, R1 and R2 are each alkyl, or R1 and R2 may together form a 3- to 6-membered saturated carbocycle, R3 is hydrogen, alkyl, alkoxyalkyl, alkylthioalkyl or COR4, X is halogen, alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, alkoxy, haloalkoxy, alkenyloxy, haloalkenyloxy, alkynyloxy, haloalkynyloxy, alkylthio, haloalkylthio, alkenylthio, haloalkenylthio, alkynylthio, haloalkynylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, dialkylaminosulfonyl, nitro, cyano, phenyl which may be substituted by Y, phenoxy which may be substituted by Y, benzyloxy which may be substituted by Y, or pyridyloxy which may be substituted by Y, and n is an integer of from 0 to 5.

    摘要翻译: 本发明涉及式(I)的苯甲酰胺衍生物或其盐:其中A为烷基,环烷基,可被Y取代的苯基,可被Y取代的吡啶基或可被Y取代的吡唑基 R 1和R 2各自为烷基,或者R 1和R 2可以一起形成3- 至6元饱和碳环,R 3是氢,烷基,烷氧基烷基,烷硫基烷基或COR 4,X是卤素,烷基,卤代烷基,烯基,卤代烯基,炔基,卤代炔基 烷氧基,卤代烷氧基,烯氧基,卤代烯氧基,炔氧基,卤代炔氧基,烷硫基,卤代烷硫基,烯硫基,卤代链烯硫基,炔硫基,卤代炔硫基,烷基亚磺酰基,卤代烷基亚磺酰基,烷基磺酰基,卤代烷基磺酰基,二烷基氨基磺酰基,硝基,氰基,可被Y取代的苯基, 被Y取代的苄氧基,可被Y取代的苄氧基,或可被Y取代的吡啶氧基,n是整数 从0到5。

    Fungicidal composition containing acid amide derivative
    4.
    发明授权
    Fungicidal composition containing acid amide derivative 有权
    含有酰胺衍生物的杀真菌剂组合物

    公开(公告)号:US08039420B2

    公开(公告)日:2011-10-18

    申请号:US12822204

    申请日:2010-06-24

    IPC分类号: A01N43/56 A01N43/10 A01N43/08

    摘要: Conventional many fungicidal compositions have had practical problems such that either a preventive effect or a curing effect is inadequate, the residual effect tends to be inadequate, or the controlling effect against plant diseases tends to be inadequate depending upon the application site, and a fungicidal composition to overcome such problems has been desired. The present invention provides a fungicidal composition containing an acid amide derivative of the formula (I) or a salt thereof, as an active ingredient: wherein A is phenyl which may be substituted, benzyl which may be substituted, naphthyl which may be substituted, heterocyclic ring which may be substituted, fused heterocyclic ring which may be substituted, or the like; B is heterocyclic ring which may be substituted, fused heterocyclic ring which may be substituted, or naphthyl which may be substituted; each of R1 and R2 which are independent of each other, is alkyl, or the like; R3 is hydrogen, or the like; each of W1 and W2 which are independent of each other, is oxygen or sulfur.

    摘要翻译: 常规的许多杀真菌组合物具有实际的问题,即预防效果或固化效果不足,残留效果趋于不足,或根据施用部位对植物病害的防治效果往往不足,杀真菌组合物 克服这些问题一直是希望的。 本发明提供含有式(I)的酰胺衍生物或其盐作为活性成分的杀真菌组合物,其中A为可被取代的苯基,可被取代的苄基,可被取代的萘基,杂环基 可被取代的环,可被取代的稠合杂环等; B是可被取代的杂环,可被取代的稠合杂环,或可被取代的萘基; R 1和R 2各自独立地为烷基等; R3是氢等; W1和W2彼此独立的是氧或硫。

    Fungicidal composition containing acid amide derivative
    6.
    发明授权
    Fungicidal composition containing acid amide derivative 有权
    含有酰胺衍生物的杀真菌剂组合物

    公开(公告)号:US07829501B2

    公开(公告)日:2010-11-09

    申请号:US11659423

    申请日:2005-08-10

    IPC分类号: A01N43/10 C07D333/16

    摘要: Conventional many fungicidal compositions have had practical problems such that either a preventive effect or a curing effect is inadequate, the residual effect tends to be inadequate, or the controlling effect against plant diseases tends to be inadequate depending upon the application site, and a fungicidal composition to overcome such problems has been desired. The present invention provides a fungicidal composition containing an acid amide derivative of the formula (I) or a salt thereof, as an active ingredient: wherein A is phenyl which may be substituted, benzyl which may be substituted, naphthyl which may be substituted, heterocyclic ring which may be substituted, fused heterocyclic ring which may be substituted, or the like; B is heterocyclic ring which may be substituted, fused heterocyclic ring which may be substituted, or naphthyl which may be substituted; each of R1 and R2 which are independent of each other, is alkyl, or the like; R3 is hydrogen, or the like; each of W1 and W2 which are independent of each other, is oxygen or sulfur.

    摘要翻译: 常规的许多杀真菌组合物具有实际的问题,即预防效果或固化效果不足,残留效果趋于不足,或根据施用部位对植物病害的防治效果往往不足,杀真菌组合物 克服这些问题一直是希望的。 本发明提供含有式(I)的酰胺衍生物或其盐作为活性成分的杀真菌组合物,其中A为可被取代的苯基,可被取代的苄基,可被取代的萘基,杂环基 可被取代的环,可被取代的稠合杂环等; B是可被取代的杂环,可被取代的稠合杂环,或可被取代的萘基; R 1和R 2各自独立地为烷基等; R3是氢等; W1和W2彼此独立的是氧或硫。

    Geometrical isomers of acrylonitrile compounds, mixture thereof, and process for producing these
    9.
    发明授权
    Geometrical isomers of acrylonitrile compounds, mixture thereof, and process for producing these 有权
    丙烯腈化合物的几何异构体,其混合物,及其制备方法

    公开(公告)号:US06624179B1

    公开(公告)日:2003-09-23

    申请号:US10030122

    申请日:2002-01-24

    IPC分类号: A61K3144

    摘要: A geometrical isomer of an acrylonitrile compound represented by the formula (I) or of its salt, or a mixture thereof: [wherein T is phenyl or pyridyl, which is substituted by R2, Q is phenyl, thienyl, pyridyl or benzyl, which may be substituted by R3, R1 is —C(═O)R4 or —C(═S)R4, R4 is alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy, alkylthio, alkenylthio, alkynylthio, cycloalkyl, cycloalkyloxy, cycloalkylthio, —N(R5)R6, phenyl, phenoxy, phenylthio, benzyl, benzyloxy, benzylthio, —J, —O—J or —S—J], wherein the geometrical isomer has a longer retention time when analyzed by reversed phase liquid chromatography in which a packing comprising silica having chemically bonded thereto an alkyl group selected from trimethyl, octyl and octadecyl, is used as the stationary phase, and a polar solvent selected from water, methanol and acetonitrile, is used as the mobile phase, and the geometrical isomer mixture contains such geometrical isomer in a larger proportion.

    摘要翻译: 由式(I)表示的丙烯腈化合物或其盐的几何异构体或其混合物:[其中T是被R 2取代的苯基或吡啶基,Q是苯基,噻吩基,吡啶基或苄基,其可以 被R 3取代,R 1是-C(= O)R 4或-C(= S)R 4,R 4是烷基,烯基,炔基,烷氧基,烯氧基,炔氧基,烷硫基,链烯硫基,炔硫基,环烷基,环烷氧基, N(R 5)R 6,苯基,苯氧基,苯硫基,苄基,苄氧基,苄硫基,-J,-OJ或-SJ],其中几何异构体在通过反相液相色谱分析时具有更长的保留时间, 化学键合有选自三甲基,辛基和十八烷基的烷基作为固定相,使用选自水,甲醇和乙腈的极性溶剂作为流动相,几何异构体混合物含有这种几何异构体 比例较大。