FUSED BICYCLIC OXAZINONE AND THIAZINONE FUNGICIDES
    7.
    发明申请
    FUSED BICYCLIC OXAZINONE AND THIAZINONE FUNGICIDES 审中-公开
    熔化双相氧化亚锡酮和噻唑酮类杀真菌剂

    公开(公告)号:WO00051992A1

    公开(公告)日:2000-09-08

    申请号:PCT/US2000/004578

    申请日:2000-02-23

    摘要: Compounds of Formulae (I) and (II), and their N-oxides and agriculturally suitable salts, are disclosed which are useful as fungicides wherein Z is O, S(O)n or NR ; n is 0, 1, or 2; Q is O or S; G is, together with the two linking carbons, a substituted fused phenyl or a substituted fused 5- or 6-membered aromatic heterocyclic ring; and R , R and R are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formulae (I) and (II) and a method for controlling plant diseases caused by fungal plant pathogens which involves applying an effective amount of a compound of Formulae (I) or (II).

    摘要翻译: 公开了式(I)和(II)化合物及其N-氧化物和农业上合适的盐,其可用作杀真菌剂,其中Z为O,S(O)n或NR 5; n为0,1或2; Q是O或S; G与两个连接的碳一起为取代的稠合苯基或取代的稠合的5元或6元芳族杂环; 且R 1,R 2和R 5如本公开所定义。 还公开了含有式(I)和(II)化合物的组合物以及用于控制由真菌植物病原体引起的植物病害的方法,其涉及施用有效量的式(I)或(II)化合物。

    4H-3,1-BENZOXAZIN-4-ONE DERIVATIVES AND ANALOGS AS ANTIVIRAL AGENTS
    8.
    发明申请
    4H-3,1-BENZOXAZIN-4-ONE DERIVATIVES AND ANALOGS AS ANTIVIRAL AGENTS 审中-公开
    4H-3,1-BENZOXAZIN-4-ONE衍生物和类似物作为抗病毒剂

    公开(公告)号:WO1997048707A1

    公开(公告)日:1997-12-24

    申请号:PCT/EP1997003158

    申请日:1997-06-16

    IPC分类号: C07D498/04

    CPC分类号: C07D265/22

    摘要: Herpesvirus protease inhibitor 4H-3,1-benzoxazin-4-one, 4H-thieno[3,2-d][1,3]oxazin-4-one, or 4H-thieno[2,3-d][1,3]oxazin-4-one; derivatives which are 2-substituted by C(XY)-R1, C(XY)-CH2-R1, C(XY)-C2H4-R1, or CX=CY-R1 wherein one of X and Y is hydrogen or halo or an alkyl substituent and the other is hydrogen or an alkyl substituent, and R1 is aryl or heteroaryl substituted by ZR4 wherein Z is CO, NRxCO, NRxCOCO, NRxCOCH2, or NRxSO2 wherein Rx is hydrogen or alkyl and R4 is aryl or heteroaryl.

    摘要翻译: 疱疹病毒蛋白酶抑制剂4H-3,1-苯并恶嗪-4-酮,4H-噻吩并[3,2-d] [1,3]恶嗪-4-酮或4H-噻吩并[2,3-d] 3]恶嗪-4-酮; 由C(XY)-R1,C(XY)-CH2-R1,C(XY)-C2H4-R1或CX = CY-R1 2-取代的衍生物,其中X和Y中的一个是氢或卤素或 烷基取代基,另一个是氢或烷基取代基,并且R 1是被ZR 4取代的芳基或杂芳基,其中Z是CO,NR x CO,NR x COCO,NR x COCH 2或NR x SO 2,其中R x是氢或烷基,且R 4是芳基或杂芳基。

    BENZOXAZINONES AND BENZOTHIAZINONES ENDOWED WITH THERAPEUTIC ACTIVITY
    9.
    发明申请
    BENZOXAZINONES AND BENZOTHIAZINONES ENDOWED WITH THERAPEUTIC ACTIVITY 审中-公开
    含有治疗活性的苯并嗪和苯并噻嗪酮

    公开(公告)号:WO1995004048A1

    公开(公告)日:1995-02-09

    申请号:PCT/EP1994002354

    申请日:1994-07-18

    IPC分类号: C07D265/22

    CPC分类号: C07D265/22 C07D279/08

    摘要: Compounds of general formula (I) wherein X is an oxygen or sulfur atom; Y is alkylene or cycloalkylene; A is hydroxy, alkoxy, acyloxy, mercapto, alkyl-sulfonyloxy, phenyl-sulfonyloxy, (a) or (b) wherein R3 is an alkyl or alkylene group omega -substituted by 2,3-dihydro-4H-1,3-benzoxazin-4-one-N-yl; R is hydrogen, alkyl or phenyl; R1 and R2 are independently hydrogen, halogen, alkoxy, trifluoromethyl or alkyl; and the pharmaceutically acceptable acid and base salts thereof, are useful as therapeutically active substances.

    摘要翻译: 通式(I)的化合物,其中X是氧或硫原子; Y是亚烷基或亚环烷基; A是羟基,烷氧基,酰氧基,巯基,烷基磺酰氧基,苯基磺酰氧基,(a)或(b)其中R3是被2,3-二氢-4H-1,3-苯并恶嗪 -4-酮-N基; R是氢,烷基或苯基; R1和R2独立地是氢,卤素,烷氧基,三氟甲基或烷基; 及其药学上可接受的酸和碱盐可用作治疗活性物质。

    PROCESS FOR THE PRODUCTION OF 2-PHENYL-BENZOXAZIN-4-ONE
    10.
    发明申请
    PROCESS FOR THE PRODUCTION OF 2-PHENYL-BENZOXAZIN-4-ONE 审中-公开
    2-苯基苯并噻嗪-4-酮的制备方法

    公开(公告)号:WO1993022300A1

    公开(公告)日:1993-11-11

    申请号:PCT/GB1993000822

    申请日:1993-04-20

    IPC分类号: C07D265/22

    CPC分类号: C07D265/22

    摘要: This invention relates to a process for the production of compounds of the 2-phenyl-benzoxazin-4-one (2PB4) type by reacting the corresponding isatoic anhydride with benzoic anhydride at elevated temperature, optionally in the presence of a solvent. The process has the advantage that the reaction is carried out without resorting to the use of acid halides or nitrogeneous bases. The 2PB4 type products are useful as bleach activators.

    摘要翻译: 本发明涉及通过在升高的温度下,任选地在溶剂存在下,通过使相应的酸酐与苯甲酸酐反应来生产2-苯基 - 苯并恶嗪-4-酮(2PB4)型化合物的方法。 该方法具有的优点是反应在不使用酰卤或含氮碱的情况下进行。 2PB4型产品可用作漂白活化剂。