2-phenyl-7-chloro-perhydroimidazo[1,5A]pyridines
    6.
    发明授权
    2-phenyl-7-chloro-perhydroimidazo[1,5A]pyridines 失效
    2-苯基-7-氯 - 全氢咪唑并[1,5A]吡啶

    公开(公告)号:US5665681A

    公开(公告)日:1997-09-09

    申请号:US492687

    申请日:1995-06-20

    CPC分类号: C07D471/04 A01N43/90

    摘要: The invention discloses compounds of formula I ##STR1## wherein X is oxygen or sulfur,R is hydrogen, chlorine or fluorine,R.sub.1 is fluorine, chlorine, bromine, cyano or methyl,R.sub.2 is halogen, C.sub.1-6 alkyl, C.sub.1-6 alkoxy, C.sub.1-6 alkylcarbonyloxy, C.sub.3-6 cycloalkoxy, C.sub.3-6 alkynyloxy, C.sub.3-6 alkenyloxy, --COOH, --CO--R.sub.3, --CO--NR.sub.4 R.sub.5, --NR.sub.6 R.sub.7, C.sub.2-6 alkenyl, N-pyrrolyl, 2-oxo-3-tetrahydrofuranyl or isC.sub.1-6 alkyl substituted with halogen, COOH, --CO--R.sub.3, --CO--NR.sub.8 R.sub.9, .dbd.N--OH, .dbd.N--C.sub.1-4 alkoxy, --O--CO--R.sub.3 or --O--C.sub.2-3 alkylene-O--; or isC.sub.2-6 alkenyl substituted with halogen, COOH, --CO--R.sub.3, --CO--NR.sub.8 R.sub.9 or C.sub.1-4 alkoxy; or isC.sub.1-6 alkoxy substituted with cyano, --CO--R.sub.3, C.sub.1-4 alkoxy, C.sub.3-6 cycloalkyl, oxiranyl, orC.sub.1-4 alkoxy or halogen; or isC.sub.3-6 alkenyloxy substituted by C.sub.2-5 alkynyl;R.sub.3 is C.sub.1-6 alkyl, C.sub.1-6 haloalkyl, C.sub.1-6 cyanoalkyl, C.sub.1-6 alkoxy, C.sub.3-6 cycloalkoxy, C.sub.3-6 alkenyloxy, C.sub.3-6 alkynyloxy or C.sub.1-6 alkoxy substituted with cyano, halogen, C.sub.1-6 alkoxy, C.sub.1-6 alkoxycarbonyl, C.sub.3-6 alkynyloxycarbonyl orC.sub.1-4 alkoxy-C.sub.1-4 alkoxycarbonyl;the use of such compounds for the control of phytopathogens, compositions for facilitating such use, and the preparation of the compounds of formula I.

    摘要翻译: 本发明公开了式I的化合物其中X是氧或硫,R是氢,氯或氟,R1是氟,氯,溴,氰基或甲基,R2是卤素,C1-6烷基,C1- 6-烷氧基,C 1-6烷基羰氧基,C 3-6环烷氧基,C 3-6炔基氧基,C 3-6烯氧基,-COOH,-CO-R 3,-CO-NR 4 R 5,-NR 6 R 7,C 2-6烯基,N-吡咯基,2-氧代-3-四氢呋喃基或 被卤素,COOH,-CO-R 3,-CO-NR 8 R 9,= N-OH,= N-C 1-4烷氧基,-O-CO-R 3或-O-C 2-3亚烷基-O-取代的C 1-6烷基; 或是被卤素,COOH,-CO-R 3,-CO-NR 8 R 9或C 1-4烷氧基取代的C 2-6烯基; 或被氰基,-CO-R 3,C 1-4烷氧基,C 3-6环烷基,环氧乙烷基或C 1-4烷氧基或卤素取代的C 1-6烷氧基; 或是被C 2-5炔基取代的C 3-6烯氧基; R 3是C 1-6烷基,C 1-6卤代烷基,C 1-6氰基烷基,C 1-6烷氧基,C 3-6环烷氧基,C 3-6烯氧基,C 3-6炔基氧基或被氰基,卤素,C 1-6烷氧基,C 1-6烷氧基羰基,C 3-6炔基氧基羰基取代的C 1-6烷氧基 或C 1-4烷氧基-C 1-4烷氧基羰基; 使用这些化合物来控制植物病原体,促进这种用途的组合物和式I化合物的制备。