利索-全球专利检索

  1. 登录
  2. 注册

搜索结果

40 条记录 (耗时 0.034 秒)

    Substituted benzimidazoles
    22.
    发明授权
    Substituted benzimidazoles 失效
    取代的苯并咪唑

    公开(公告)号：US5863933A

    公开(公告)日：1999-01-26

    申请号：US822565

    申请日：1997-03-19

    申请人： Winfried Lunkenheimer ,  Bernd Baasner ,  Folker Lieb ,  Stefan Bohm ,  Albrecht Marhold ,  Ulrich Gorgens ,  Wilhelm Stendel ,  Heinz-Wilhelm Dehne ,  Hans-Joachim Santel

    发明人： Winfried Lunkenheimer ,  Bernd Baasner ,  Folker Lieb ,  Stefan Bohm ,  Albrecht Marhold ,  Ulrich Gorgens ,  Wilhelm Stendel ,  Heinz-Wilhelm Dehne ,  Hans-Joachim Santel

    IPC分类号： A01N43/52 ,  A01N43/90 ,  A01N47/12 ,  A01N47/18 ,  A01N47/20 ,  A01N47/30 ,  A01N47/34 ,  A01N57/24 ,  C07D235/10 ,  C07D405/12 ,  C07D491/04 ,  C07D491/056 ,  C07F9/6506

    CPC分类号： C07D405/12 ,  A01N43/52 ,  A01N43/90 ,  A01N47/12 ,  A01N47/18 ,  A01N47/20 ,  A01N47/30 ,  A01N47/34 ,  C07D235/10 ,  C07D491/04 ,  C07F9/65068

    摘要： The invention relates to new substituted benzimidazole of the general formula (I) ##STR1## in which R.sup.1 represents hydrogen, alkyl, alkoxy or optionally substituted aryl,R.sup.2 represents hydroxyl, cyano or in each case optionally substituted alkyl, alkenyl, alkinyl, alkoxy, alkenyloxy, alkinyloxy, alkylthio, amino, aminocarbonyl, alkylcarbonyl, alkoxycarbonyl, alkoxycarbonyloxy, dialkoxyphosphonyl, (hetero)aryl, (hetero)arylcarbonyl, (hetero)aryloxycarbonyl, (hetero)arylcarbonyloxy or (hetero)arylaminocarbonylaminocarbonyloxy, andR.sup.3 represents fluoroalkyl,X.sup.1, X.sup.2, X.sup.3 and X.sup.4 independently of one another in each case represent hydrogen, halogen, cyano, nitro, in each case optionally substituted alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl or cycloalkyl, optionally substituted, fused dioxyalkylene, or represent hydroxycarbonyl, alkylcarbonyl, alkoxycarbonyl or cycloalkyloxycarbonyl, in each case optionally substituted amino or aminocarbonyl or in each case optionally substituted aryl, aryloxy, arylthio, arylsulphinyl, arylsulphonyl, arylsulphonyloxy, arylcarbonyl, aryloxycarbonyl, arylazo or arylthiomethylsulphonyl, but where at least one of the substituents X.sup.1, X.sup.2, X.sup.3 or X.sup.4 represents halogenoalkyl, with the exception of the chloromethyl radical, halogenoalkoxy, halogenoalkylthio, halogenoalkylsulphinyl, halogenoalkylsulphonyl or alkylsulphonyl, optionally substituted, fused dioxyalkylene, or represent hydroxycarbonyl, alkylcarbonyl, alkoxycarbonyl or cycloalkyloxycarbonyl, in each case optionally substituted amino or aminocarbonyl, or in each case optionally substituted aryl, arylthio, arylsulphinyl, arylsulphonyl, arylsulphonyloxy, arylcarbonyl, aryloxycarbonyl, arylazo or arylthiomethylsulphonyl,their preparation and use as pesticides, and intermediates for their preparation.

    摘要翻译： 本发明涉及通式（I）的新取代的苯并咪唑，其中R 1表示氢，烷基，烷氧基或任选取代的芳基，R 2表示羟基，氰基或在各种情况下任选取代的烷基，烯基，炔基 （杂）芳基羰基，（杂）芳基羰基氧基或（杂）芳基氨基羰基氨基羰基氧基，R3代表氟代烷基，芳基羰氧基， 在各种情况下，X1，X2，X3和X4彼此独立地表示氢，卤素，氰基，硝基，在各种情况下均为任选取代的烷基，烷氧基，烷硫基，烷基亚磺酰基，烷基磺酰基或环烷基，任选取代的稠合二氧亚烷基，或代表羟基羰基 ，烷基羰基，烷氧基羰基或环烷氧基羰基，在每种情况下均为任选取代的氨基或氨基羰基，或在每种情况下任选取代 芳基，芳氧基，芳硫基，芳基亚磺酰基，芳基磺酰基，芳基磺酰氧基，芳基羰基，芳氧基羰基，芳基偶氮或芳基硫代甲基磺酰基，但其中至少一个取代基X1，X2，X3或X4表示卤代烷基，除了氯甲基，卤代烷氧基，卤代烷硫基 ，卤代烷基亚磺酰基，卤代烷基磺酰基或烷基磺酰基，任选取代的稠合的二氧亚烷基，或代表羟基羰基，烷基羰基，烷氧基羰基或环烷氧基羰基，在各种情况下均为任选取代的氨基或氨基羰基，或在每种情况下均为任选取代的芳基，芳硫基，芳基亚磺酰基，芳基磺酰基，芳基磺酰氧基，芳基羰基， 芳氧基羰基，芳基偶氮或芳基硫代甲基磺酰基，它们的制备和用作农药，以及其制备中间体。

    2-cyanobenzimidazoles and their use
    25.
    发明授权
    2-cyanobenzimidazoles and their use 失效
    2-氰基苯并咪唑及其用途

    公开(公告)号：US5571830A

    公开(公告)日：1996-11-05

    申请号：US586119

    申请日：1996-01-16

    申请人： Winfried Lunkenheimer ,  Heinz-Wilheim Dehne ,  Ulrike Wachendorff-Neumann

    发明人： Winfried Lunkenheimer ,  Heinz-Wilheim Dehne ,  Ulrike Wachendorff-Neumann

    IPC分类号： A01N43/90 ,  C07D491/04 ,  C07D491/056 ,  C07D491/113 ,  C07D235/02

    CPC分类号： C07D491/04 ,  A01N43/90

    摘要： New 2-cyanobenzimidazoles of the formula (I) ##STR1## in which R.sup.1, R.sup.2 and A have the meaning given in the description, a preparation process, their use in agriculture, for example against fungi, insects etc., and new intermediates.Formula (I) provides a definition of the compounds; for example they are obtained from suitable 2-cyanobenzimidazoles which are unsubstituted in the 1-position with N,N-dimethylsulphamoyl halide. The 2-cyanobenzimidazoles which are unsubstituted in the 1-position are equally new and can be reacted from suitable phenylenediamines of the formula (IV) with methyl 2,2,2-trichloroacetimidate of the formula (V) to give the 2-trichloromethylbenzimidazoles of the formula (VI), which are equally new and from which the compounds of the formula (II) can subsequently be obtained with ammonia.

    摘要翻译： 式（I）的新的2-氰基苯并咪唑其中R1，R2和A具有说明书中给出的含义，制备方法，它们在农业中的用途，例如抗真菌，昆虫等，以及 新中间体 式（I）提供化合物的定义; 例如，它们可由合适的2-氰基苯并咪唑得到，其中N，N-二甲基氨磺酰卤在1位未被取代。 在1-位未被取代的2-氰基苯并咪唑是同等新的，并且可以由适当的式（Ⅳ）亚苯基二胺与式（Ⅴ）的2,2,2-三氯乙酰亚氨酸甲酯反应得到2-（三氟甲基）苯并咪唑 式（VI）同样新，随后可以用氨获得式（II）化合物。

    2-cyanobenzimidazoles and their use, and new precursors
    30.
    发明授权
    2-cyanobenzimidazoles and their use, and new precursors 失效
    2-氰基苯并咪唑及其用途和新前体

    公开(公告)号：US5510364A

    公开(公告)日：1996-04-23

    申请号：US981035

    申请日：1992-11-24

    申请人： Winfried Lunkenheimer ,  Heinz-Wilhelm Dehne ,  Ulrike Wachendorff-Neumann

    发明人： Winfried Lunkenheimer ,  Heinz-Wilhelm Dehne ,  Ulrike Wachendorff-Neumann

    IPC分类号： A01N43/90 ,  C07D491/04 ,  C07D491/056 ,  C07D491/113 ,  C07D235/02

    CPC分类号： C07D491/04 ,  A01N43/90

    摘要： New 2-cyanobenzimidazoles of the formula (I) ##STR1## in which R.sup.1, R.sup.2 and A have the meaning given in the description, a preparation process, their use in agriculture, for example against fungi, insects etc., and new intermediates.Formula (I) provides a definition of the compounds; for example they are obtained from suitable 2-cyanobenzimidazoles which are unsubstituted in the 1-position with N,N-dimethylsulphamoyl halide. The 2-cyanobenzimidazoles which are unsubstituted in the 1-position are equally new and can be reacted from suitable phenylenediamines of the formula (IV) with methyl 2,2,2-trichloroacetimidate of the formula (V) to give the 2-trichloromethylbenzimidazoles of the formula (VI), which are equally new and from which the compounds of the formula (II) can subsequently be obtained with ammonia.

    摘要翻译： 式（I）的新的2-氰基苯并咪唑其中R1，R2和A具有说明书中给出的含义，制备方法，它们在农业中的用途，例如抗真菌，昆虫等，以及 新中间体 式（I）提供化合物的定义; 例如，它们可由合适的2-氰基苯并咪唑得到，其中N，N-二甲基氨磺酰卤在1位未被取代。 在1-位未被取代的2-氰基苯并咪唑是同等新的，并且可以由适当的式（Ⅳ）亚苯基二胺与式（Ⅴ）的2,2,2-三氯乙酰亚氨酸甲酯反应得到2-（三氟甲基）苯并咪唑 式（VI）同样新，随后可以用氨获得式（II）化合物。