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154 条记录 (耗时 0.047 秒)

    Process for the preparation of thiazole derivatives
    31.
    发明授权
    Process for the preparation of thiazole derivatives 失效
    噻唑衍生物的制备方法

    公开(公告)号：US06677457B2

    公开(公告)日：2004-01-13

    申请号：US10047807

    申请日：2002-01-15

    申请人： Thomas Pitterna ,  Henry Szczepanski ,  Peter Maienfisch ,  Ottmar Franz Hüter ,  Thomas Rapold ,  Marcel Senn ,  Thomas Göbel ,  Anthony Cornelius O'Sullivan ,  Gottfried Seifert

    发明人： Thomas Pitterna ,  Henry Szczepanski ,  Peter Maienfisch ,  Ottmar Franz Hüter ,  Thomas Rapold ,  Marcel Senn ,  Thomas Göbel ,  Anthony Cornelius O'Sullivan ,  Gottfried Seifert

    IPC分类号： C07D27716

    CPC分类号： C07D277/32 ,  C07D277/16 ,  C07D277/36 ,  C07D417/06

    摘要： The invention relates to a process for the preparation of a compound of the formula wherein Q, Y, Z, R1, R2, R3, R4 and R5 are as defined in the specification, which comprises a) reacting a compound of the formula  with a halogenating agent to form a compound of the formula or b) converting a compound of formula (II) by means of a halogenating agent into a compound of the formula optionally c) converting the compound of formula (IV) into a compound of formula (III); d) converting a compound of formula (III) by means of a compound of the formula into a compound of the formula or e) converting a compound (IV) by means of a compound (V) into a compound (VI); and f) converting a compound (VI) by means of a chlorinating agent into a compound (I); a compound (IV); to a process for the preparation of a compound (III) and to a process for the preparation of a compound (IV).

    摘要翻译： 本发明涉及制备糠醛的化合物的方法，其中Q，Y，Z，R 1，R 2，R 3，R 4和R 5如本说明书中所定义，其包括：a）将卤化剂的化合物与 将式（II）化合物通过卤化剂转化成式（Ⅲ）的化合物，将式（Ⅳ）化合物转化为式（Ⅳ）化合物; d）将化合物 通过化学式（Ⅳ）将化合物（Ⅳ）转化为化合物（Ⅵ）;将式（Ⅳ）化合物与式 和（f）通过氯化剂将化合物（VI）转化为化合物（I）;化合物（IV）; 涉及制备化合物（III）的方法和制备化合物（IV）的方法。

    Thiazole compounds
    32.
    发明授权
    Thiazole compounds 失效
    噻唑化合物

    公开(公告)号：US06211381B1

    公开(公告)日：2001-04-03

    申请号：US09077569

    申请日：1998-06-01

    申请人： Henry Szczepanski ,  Thomas Göbel ,  Ottmar Franz Hüter ,  Anthony Cornelius O'Sullivan ,  Marcel Senn ,  Thomas Rapold ,  Peter Maienfisch ,  Thomas Pitterna

    发明人： Henry Szczepanski ,  Thomas Göbel ,  Ottmar Franz Hüter ,  Anthony Cornelius O'Sullivan ,  Marcel Senn ,  Thomas Rapold ,  Peter Maienfisch ,  Thomas Pitterna

    IPC分类号： C07D27732

    CPC分类号： C07D277/32 ,  C07D277/36 ,  C07D417/06

    摘要： The invention relates to a process for preparing a compound of formula (I), in which X is CH or N, Y is NO2 or CN, Z is CHR3, O, NR3 or S, R1 and R2 are either each, independently of the other, hydrogen or unsubstituted or R4-substituted alkyl or together a two- or three-membered alkylene bridge or a two- or three-membered alkylene bridge in which one member is replaced by a hetero member selected from the group, consisting of NR5, O and S, R3 is H or unsubstituted or R4-substituted alkyl, R4 is an unsubstituted or substituted aryl or heteroaryl group, and R5 is H or alkyl, which comprises a) reacting a compound of formula (II) with a chlorinating agent or b1) initially reacting a compound of formula (IV) with a compound of formula (V) and b2) further reacting the compound of formula (II) obtainable thereby, with or without intermediate isolation, with a chlorinating agent, to intermediates used in this process, to the use of these intermediates and to a process for the preparation of these intermediates.

    摘要翻译： 本发明涉及制备式（I）化合物的方法，其中X是CH或N，Y是NO 2或CN，Z是CHR 3，O，NR 3或S，R 1和R 2各自独立地是 另一个，氢或未取代的或R4取代的烷基或二元或三元亚烷基桥或二元或三元亚烷基桥，其中一个成员被选自NR5， O和S，R 3是H或未取代的或R 4取代的烷基，R 4是未取代或取代的芳基或杂芳基，R 5是H或烷基，其包括a）使式（II）化合物与氯化剂或 b1）最初使式（Ⅳ）化合物与式（Ⅴ）化合物反应，和b2）使可得到的式（Ⅱ）化合物进一步与中间体分离与氯化剂反应，得到本发明的中间体 过程，使用这些中间体和制备过程 这些中间体。

    Chemical compounds
    34.
    发明授权
    Chemical compounds 失效
    化合物

    公开(公告)号：US08524896B2

    公开(公告)日：2013-09-03

    申请号：US12921000

    申请日：2009-03-02

    申请人： Peter Maienfisch ,  Ottmar Hueter ,  Peter Renold ,  Werner Zambach ,  Thomas Pitterna

    发明人： Peter Maienfisch ,  Ottmar Hueter ,  Peter Renold ,  Werner Zambach ,  Thomas Pitterna

    IPC分类号： C07D293/10 ,  C07D251/00 ,  C07D253/00 ,  C07D237/02 ,  C07D211/78 ,  C07D213/63 ,  A01N25/26 ,  A01N43/54 ,  A01N41/12 ,  A61K31/53 ,  A61K31/501 ,  A61K31/435

    CPC分类号： C07D207/48 ,  A01N43/36 ,  A01N43/78 ,  C07D277/04 ,  C07D277/10 ,  C07D277/22

    摘要： A compound of the formula (I) where, for example, W, X and Y are each CH; R1 and R6 together with the adjacent nitrogen forms a 3 to 10-membered saturated ring, wherein the ring may contain, in addition to the nitrogen and carbon ring members, 1, 2 or 3 heteroatoms and/or heteroatom groups as ring members, independently of one another, selected from the group consisting of sulfur, CO, SO, SO2 and N—R7 and/or the ring may carry 1, 2 or 3 radicals, independently of one another, each selected, for example, from the group consisting of halogen, cyano, nitro, amino, and C1-C6-alkyl. R2 is, for example, halogen, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C1-C6-haloalkoxy or C1-C6-alkoxy-C1-C6-alkoxy, and R7 is for example, R10C(═O), C1-C6 alkyl or C1-C6-haloalkyl; and/or salts thereof; and their use as pesticidal agents.

    摘要翻译： 式（I）的化合物，其中例如W，X和Y各自为CH; R1和R6与相邻的氮一起形成3至10元饱和环，其中除了氮和碳环成员之外，环可以独立地包含1,2或3个杂原子和/或杂原子基团作为环成员 彼此相互选择，选自硫，CO，SO，SO 2和N-R 7和/或环可以彼此独立地携带1,2或3个基团，每个选自例如 的卤素，氰基，硝基，氨基和C 1 -C 6 - 烷基。 R 2是例如卤素，C 1 -C 6烷基，C 1 -C 6卤代烷基，C 1 -C 6 - 烷氧基，C 1 -C 6 - 卤代烷氧基或C 1 -C 6 - 烷氧基-C 1 -C 6 - 烷氧基， R 10 C（= O），C 1 -C 6烷基或C 1 -C 6 - 卤代烷基; 和/或其盐; 并将其用作杀虫剂。

    Avermectins and avermectin monosacharides substituted in the 4′-and 4″ position having pesticidal properties
    39.
    发明授权
    Avermectins and avermectin monosacharides substituted in the 4′-and 4″ position having pesticidal properties 有权
    在具有杀虫性的4'和4“位置取代的阿维菌素和阿维菌素单糖苷

    公开(公告)号：US07704961B2

    公开(公告)日：2010-04-27

    申请号：US10568715

    申请日：2004-08-27

    申请人： Fiona Murphy Kessabi ,  Thomas Pitterna ,  Peter Maienfisch ,  Jérôme Cassayre ,  Laura Quaranta ,  Pierre Jung ,  Ottmar Franz Hueter

    发明人： Fiona Murphy Kessabi ,  Thomas Pitterna ,  Peter Maienfisch ,  Jérôme Cassayre ,  Laura Quaranta ,  Pierre Jung ,  Ottmar Franz Hueter

    IPC分类号： A61K31/70 ,  A61K31/7028 ,  C07H17/08

    CPC分类号： A01N43/90 ,  C07H19/01

    摘要： Described is a compound of the formula (I) wherein the bond between carbon atoms 22 and 23 is a single or double bond; m is 0 or 1; R1, is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and either (A) R2 is —N(R3)R4, and (1) X is 0, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C3-C12cycloalkyl; or (2) X is S, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl; or (3) X is 0 or S, wherein R3 and R4 together are, for instance, a three- to seven membered alkylene or a four- to seven-membered alkenylene bridge; or (B) R2 is OR5, X is 0 or S, wherein R5 is, for instance, C1-C12alkyl, mono- to pentasubstituted C1-C12alkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form; such a compound demonstrates pesticidal activity.

    摘要翻译： 描述了式（I）的化合物，其中碳原子22和23之间的键是单键或双键; m为0或1; R1是C1-C12烷基，C3-C8环烷基或C2-C12链烯基; （A）R 2是-N（R 3）R 4，和（1）X是0，其中R 3是例如氢，未被取代的或单取代到五取代的C 1 -C 12烷基，R 4是例如， 至五取代的C 1 -C 12烷基，未取代的或一至五取代的C 3 -C 12环烷基; 或（2）X为S，其中R 3为例如氢，未取代或单价至五价取代的C 1 -C 12烷基，R 4为例如氢，未取代或单价至五价取代的C 1 -C 12烷基; 或（3）X为0或S，其中R3和R4一起为例如三至七元亚烷基或四至七元亚烯基桥; 或（B）R 2是OR 5，X是0或S，其中R 5是例如C 1 -C 12烷基，一至五取代的C 1 -C 12烷基; 或者如果合适的话，E / Z异构体，E / Z异构体混合物和/或其互变异构体在每种情况下都是游离形式或盐形式; 这种化合物显示出杀虫活性。

    Avermectin and avermectin monosaccharide derivatives substituted in the 4″-or 4′-position having pesticidal properties
    40.
    发明授权
    Avermectin and avermectin monosaccharide derivatives substituted in the 4″-or 4′-position having pesticidal properties 有权
    在4“ - 或4”位取代的具有杀虫性的阿维菌素和阿维菌素单糖衍生物

    公开(公告)号：US07678740B2

    公开(公告)日：2010-03-16

    申请号：US10543637

    申请日：2004-01-30

    申请人： Thomas Pitterna ,  Fiona Murphy Kessabi ,  Peter Maienfisch ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung

    发明人： Thomas Pitterna ,  Fiona Murphy Kessabi ,  Peter Maienfisch ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung

    IPC分类号： A01N25/26 ,  A01N43/02 ,  A01N43/04 ,  C07H17/08

    CPC分类号： A01N43/90 ,  C07H17/08

    摘要： What is described are a compound of the formula (I) Wherein U is —N(R2)OR3 or —N+(O−)═C(RE)RZ); n is 0 or 1; X—Y is —CH═CH— or —CH2—CH2—; R1 is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; R2 and R3 are, for example; independently from each other, —Q, —C(═O)—Z—Q or —CN; RZ and RE are, independently from each other, —Q, —C(═O)—Z—Q or —CN; or RZ and RE together are a three- to seven membered alkylene or alkenylene bridge, which is unsubstituted or mono- to tri-substituted; Z is a bond, O or —NR4—; Q is H, C1-C12alkyl, C2-C12alkenyl, C2-C12alkynyl, C3-C12-Cycloalkyl, C5-C12-cycloalkenyl, aryl, or heterocyclyl, which are unsubstituted or mono- to pentasubstituted; R4 is for example H, C1-C8alkyl, hydroxy-C1-C8alkyl, C3-C8cycloalkyl or C2-C8alkenyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof; a process for preparing these compounds, their isomers and tautomers and the use of these compounds, their isomers and tautomers; pesticidal compositions whose active compound is selected from these compounds and their tautomers; intermediates for the preparation of the said compounds of the formula (I), methods for the preparation of the compounds of the formula (I), and a method for controlling pests using these compositions.

    摘要翻译： 描述的是式（I）的化合物，其中U是-N（R 2）OR 3或-N +（O-）= C（RE）R Z）; n为0或1; X-Y是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12烷基，C3-C8环烷基或C2-C12链烯基; R2和R3例如是： 独立地为-Q，-C（= O）-Z-Q或-CN; RZ和RE彼此独立地为-Q，-C（= O）-Z-Q或-CN; 或RZ和RE一起是三至七元的亚烷基或亚烯基桥，其是未取代的或一至三取代的; Z是O或-NR4-键; Q是未被取代或被一取代或五取代的H，C 1 -C 12烷基，C 2 -C 12烯基，C 2 -C 12炔基，C 3 -C 12环烷基，C 5 -C 12 - 环烯基，芳基或杂环基， R4是例如H，C1-C8烷基，羟基-C1-C8烷基，C3-C8环烷基或C2-C8链烯基; 或者，如果合适的话，E / Z异构体，E / Z异构体混合物和/或其互变异构体; 制备这些化合物，其异构体和互变异构体的方法以及这些化合物，其异构体和互变异构体的用途; 活性化合物选自这些化合物及其互变异构体的杀虫组合物; 用于制备所述式（I）化合物的中间体，式（I）化合物的制备方法和使用这些组合物来控制害虫的方法。