公开(公告)号：US4891217A

公开(公告)日：1990-01-02

申请号：US186990

申请日：1988-04-27

Applicant: Terrence P. McGovern ,  Roy T. Cunningham

Inventor： Terrence P. McGovern ,  Roy T. Cunningham

IPC: A01N37/08 ,  C07C61/15

CPC classification number: C07C61/15 ,  A01N37/08

Abstract: Novel attractants for the Mediterrean Fruit Fly, "Medfly," are disclosed. The attractants comprise isomeric blends of esters of iodo-trans-2-methylcyclohexanecarboxylic acid. In use, the attractants are competitive in attraction with the "standard" Medfly attractant, Trimedlure, "TML," but are much more persistent than TML.

Abstract translation: Mediterrean Fruit Fly的新颖引诱剂“Medfly”被披露。 引诱剂包括碘 - 反-2-甲基环己烷羧酸的酯的异构共混物。 在使用中，引诱剂与“标准”Medfly引诱剂Trimedlure“TML”的吸引力具有竞争力，但比TML更加持久。

公开(公告)号：US4739112A

公开(公告)日：1988-04-19

申请号：US697508

申请日：1985-02-01

Applicant: Patricia M. Savu

Inventor： Patricia M. Savu

IPC: C07C17/12 ,  C07C17/00 ,  C07C17/26 ,  C07C23/18 ,  C07C23/20 ,  C07C23/36 ,  C07C27/00 ,  C07C31/44 ,  C07C51/00 ,  C07C61/15 ,  C07C67/00 ,  C07C69/54 ,  C07C69/753 ,  C07C69/52 ,  C07C19/08 ,  C07C51/58 ,  C09K5/00

CPC classification number: C07C23/36 ,  C07C23/18 ,  C07C61/15

Abstract: Perfluoropolycycloalkanes are provided. These perfluoropolycycloalkanes are ring assemblies having (a) at least two perfluorinated cyclohexane rings, (b) at least two perfluorinated fused ring systems, or (c) combinations of at least one perfluorinated cyclohexane ring with at least one perfluorinated fused ring system, each perfluorinated ring or fused ring system being directly joined to another perfluorinated ring or ring system by a single bond and the ring assemblies having a total of at least 13 carbon atoms.

Abstract translation: 提供全氟聚环烷烃。 这些全氟聚环烷烃是具有（a）至少两个全氟化环己烷环，（b）至少两个全氟化稠环体系，或（c）至少一个全氟化环己烷环与至少一个全氟化稠环系统的组合的环组件，每个全氟化 环或稠环系统通过单键直接连接到另一个全氟化环或环系统，并且环组件具有总共至少13个碳原子。

公开(公告)号：US4485116A

公开(公告)日：1984-11-27

申请号：US433866

申请日：1982-10-13

Applicant: Alan T. Hudson ,  Anthony W. Randall

Inventor： Alan T. Hudson ,  Anthony W. Randall

IPC: C07C50/12 ,  C07C50/32 ,  C07C51/08 ,  C07C51/36 ,  C07C51/487 ,  C07C53/134 ,  C07C61/08 ,  C07C61/15 ,  C07C61/22 ,  A01N9/24

CPC classification number: C07C61/22 ,  C07C50/32 ,  C07C51/08 ,  C07C51/36 ,  C07C51/487 ,  C07C53/134 ,  C07C61/08 ,  C07C61/15

Abstract: 1,4-Naphthoquinones of formula (I), methods for their preparation, veterinary formulations thereof, and the use thereof in animal therapy are disclosed. ##STR1## Particularly preferred compounds of formula (I) are, 2-[trans-(4-t-butylcyclohexyl)methyl]-3-hydroxy-1,4-naphthoquinone, and 2-[trans-(4-t-pentyl cyclohexyl)methyl]3-hydroxy-1,4-naphthoquinone. The compounds are of value as anti-protozoal agents, in particular as anti-theilerial agents.

Abstract translation: 公开了式（I）的1,4-萘醌，其制备方法，其兽用制剂及其在动物治疗中的用途。 （I）特别优选的式（I）化合物是2- [反式 - （4-叔丁基环己基）甲基] -3-羟基-1,4-萘醌和2- [反 - （4- 叔戊基环己基）甲基] -3-羟基-1,4-萘醌。 这些化合物作为抗原虫剂具有价值，特别是作为抗iler药。

公开(公告)号：US4391731A

公开(公告)日：1983-07-05

申请号：US289676

申请日：1981-08-03

Applicant: Arthur Boller ,  Martin Schadt ,  Alois Villiger

Inventor： Arthur Boller ,  Martin Schadt ,  Alois Villiger

IPC: C07C1/22 ,  C07C13/48 ,  C07C13/50 ,  C07C43/18 ,  C07C43/20 ,  C07C43/235 ,  C07C45/46 ,  C07C45/62 ,  C07C45/68 ,  C07C47/47 ,  C07C49/323 ,  C07C49/792 ,  C07C51/36 ,  C07C61/13 ,  C07C61/15 ,  C07C61/29 ,  C07C63/49 ,  C07C63/72 ,  C07C69/753 ,  C07C69/773 ,  C07C233/00 ,  C07C255/50 ,  C07C255/51 ,  C07C255/53 ,  C07D295/02 ,  C07D295/033 ,  C09K19/00 ,  C09K19/32 ,  C09K3/34 ,  C07C121/46

CPC classification number: C09K19/322 ,  C07C1/22 ,  C07C13/48 ,  C07C13/50 ,  C07C327/00 ,  C07C43/18 ,  C07C43/20 ,  C07C43/235 ,  C07C45/46 ,  C07C45/62 ,  C07C45/68 ,  C07C47/47 ,  C07C49/323 ,  C07C49/792 ,  C07C51/36 ,  C07C61/13 ,  C07C61/15 ,  C07C61/29 ,  C07C63/49 ,  C07C63/72 ,  C07D295/033 ,  C07C2102/28 ,  C09K2019/326

Abstract: Compounds of the formula ##STR1## wherein ring A is saturated or aromatic and a saturated ring A which may be present is trans-linked with the second ring; R.sup.1 is a straight-chain alkyl or alkoxy group containing 1 to 11 carbon atoms; R.sup.2 is cyano, a straight-chain alkyl group containing 1 to 11 carbon atoms, an ester group of the formula ##STR2## or, when ring A is saturated, additionally a straight-chain alkoxy group containing 1 to 11 carbon atoms; in the ester group of formula II ring B is either aromatic and X is oxygen or sulfur and R.sup.3 is cyano or a straight-chain alkyl or alkoxy group containing 1 to 10 carbon atoms, or ring B is a trans-1,4-disubstituted cyclohexane ring and X is oxygen and R.sup.3 is cyano or a straight-chain alkyl group containing 1 to 10 carbon atoms; and the total number of carbon atoms in the alkyl and/or alkoxy groups amounts to at most 12, are described. The compounds of formula I are useful in liquid crystal mixtures.

Abstract translation: 其中环A是饱和的或芳族的，其可以存在的饱和环A与第二个环反应的式I的化合物; R1是含有1至11个碳原子的直链烷基或烷氧基; R2是氰基，含有1至11个碳原子的直链烷基，式II的酯基或当A环饱和时，另外是含有1至11个碳原子的直链烷氧基; 在式II的酯基中，环B为芳族的，X为氧或硫，R 3为氰基或含有1至10个碳原子的直链烷基或烷氧基，或环B为反式-1,4-二取代 环己烷环，X为氧，R3为氰基或含有1〜10个碳原子的直链烷基; 并且烷基和/或烷氧基中的碳原子总数达到至多12。 式I化合物可用于液晶混合物。

公开(公告)号：US4339458A

公开(公告)日：1982-07-13

申请号：US147728

申请日：1980-05-08

Applicant: George Holan ,  David F. O'Keefe

Inventor： George Holan ,  David F. O'Keefe

IPC: C07C69/74 ,  A01N33/20 ,  A01N37/08 ,  A01N37/10 ,  A01N37/34 ,  A01N37/38 ,  A01N37/48 ,  A01N43/08 ,  A01N43/30 ,  C07C51/00 ,  C07C61/15 ,  C07C61/39 ,  C07C61/40 ,  C07C62/12 ,  C07C62/34 ,  C07C67/00 ,  C07C69/753 ,  C07C69/757 ,  C07C201/00 ,  C07C205/55 ,  C07C253/00 ,  C07C255/38 ,  C07C313/00 ,  C07C323/62 ,  C07D307/42 ,  C07D317/60 ,  C07D317/68 ,  A01N43/16

CPC classification number: A01N37/48 ,  A01N37/08 ,  A01N37/10 ,  A01N37/34 ,  A01N37/38 ,  A01N43/08 ,  A01N43/30 ,  C07C61/15 ,  C07C61/40 ,  C07C62/12 ,  C07C62/34 ,  C07C69/753 ,  C07C69/757 ,  C07D317/60

Abstract: Compounds of the general formula I ##STR1## wherein R.sup.1 is hydrogen or a methoxy, ethoxy, propoxy, butoxy, tetrafluoroethoxy, methylthio, ethylthio, propylthio, fluoro, chloro, bromo, methyl, ethyl, or nitro group, and R.sup.2 is hydrogen or a methyl group, or R.sup.1 and R.sup.2 together form a methylenedioxy group;R.sup.3 is hydrogen, or a lower alkyl group, or one of the following groups (a) to (f):(a) 3-phenoxybenzyl(b) 2-benzyl-4-furylmethyl(c) .alpha.-cyano-3-phenoxybenzyl(d) 3,4-methylenedioxybenzyl(e) .alpha.-ethynyl-3-phenoxybenzyl(f) .alpha.-cyano-3-(4'-chlorophenoxy)-benzyland Y.sup.1, Y.sup.2, Y.sup.3, Y.sup.4, Y.sup.5 and Y.sup.6 are the same or different groups and each is hydrogen or a fluoro, bromo or chloro group, with the proviso that when R.sup.1 is hydrogen, fluoro, chloro, bromo or methyl and R.sup.2 is hydrogen, then one of Y.sup.1 to Y.sup.6 is other than hydrogen.The compounds in which R.sup.3 is one of groups (a) to (f) are insecticides.

公开(公告)号：US4322374A

公开(公告)日：1982-03-30

申请号：US181015

申请日：1980-08-25

Applicant: Pierre Martin ,  Hans Greuter ,  Eginhard Steiner ,  Daniel Bellus

Inventor： Pierre Martin ,  Hans Greuter ,  Eginhard Steiner ,  Daniel Bellus

IPC: C07C51/60 ,  C07C51/62 ,  C07C53/50 ,  C07C61/15 ,  C07C61/40

CPC classification number: C07C45/45 ,  C07C45/67 ,  C07C51/60 ,  C07C51/62 ,  C07C53/50 ,  C07C61/15 ,  C07C61/40

Abstract: The preparation and use as an intermediate for making insecticides has been disclosed for a compound of the formula: ##STR1## in which X and Y are each chlorine or bromine.

Abstract translation: 已经公开了制备和用作制备杀虫剂的中间体的下式化合物：其中X和Y各自为氯或溴。

公开(公告)号：US4306077A

公开(公告)日：1981-12-15

申请号：US86033

申请日：1979-10-18

Applicant: Thomas Leigh

Inventor： Thomas Leigh

IPC: C07C61/04 ,  C07C51/00 ,  C07C51/487 ,  C07C61/15 ,  C07C61/37 ,  C07C61/40 ,  C07C67/00 ,  C07C255/48 ,  C07B19/00

CPC classification number: C07C51/487

Abstract: A process of separating cis and trans isomers of cyclopropane carboxylic acids comprising the step of treating an aqueous solution of a soluble salt of the cis and trans isomers with just sufficient of an acid, for example acetic acid or carbonic acid, to cause precipitation of one isomeric form of the cyclopropane carboxylic acid while substantially all or a major proportion of the other isomeric form remains in solution as the soluble salt. The process may be used, for example, to separate (+)-cis-3-(2,2-dichlorovinyl)-2,2-dimethylcyclopropane carboxylic acid (an intermediate for insecticides) from a mixture of the (+)-cis and (+)-trans acids.

Abstract translation: 分离环丙烷羧酸的顺式和反式异构体的方法，其包括用刚好足够的酸例如乙酸或碳酸处理顺式和反式异构体的可溶性盐的水溶液的步骤，以使一种 异构体形式的环丙烷羧酸，而基本上全部或大部分的其它异构形式作为可溶性盐保留在溶液中。 该方法可用于例如（+） - 顺式-3-（2,2-二氯乙烯基）-2,2-二甲基环丙烷羧酸（杀虫剂的中间体）从（+） - 顺式 和（+） - 反式酸。

公开(公告)号：US4283420A

公开(公告)日：1981-08-11

申请号：US31165

申请日：1979-04-18

Applicant: Charles Pigerol ,  Jean-Claude Vernieres ,  Pierre Eymard ,  Jacques Simiand ,  Madeleine Broll ,  Jean-Yves Lacolle

Inventor： Charles Pigerol ,  Jean-Claude Vernieres ,  Pierre Eymard ,  Jacques Simiand ,  Madeleine Broll ,  Jean-Yves Lacolle

IPC: A61K31/16 ,  A61K31/165 ,  A61K31/19 ,  A61P25/00 ,  A61P25/08 ,  A61P25/18 ,  A61P25/28 ,  C07C51/00 ,  C07C51/08 ,  C07C51/09 ,  C07C51/27 ,  C07C51/353 ,  C07C51/367 ,  C07C51/377 ,  C07C51/41 ,  C07C51/60 ,  C07C61/08 ,  C07C61/10 ,  C07C61/15 ,  C07C61/16 ,  C07C61/20 ,  C07C61/22 ,  C07C61/35 ,  C07C61/39 ,  C07C61/40 ,  C07C62/04 ,  C07C62/10 ,  C07C62/20 ,  C07C62/34 ,  C07C67/00 ,  C07C231/00 ,  C07C233/00 ,  C07C233/58 ,  C07C235/40 ,  C07C235/82

CPC classification number: C07C62/34 ,  C07C51/08 ,  C07C51/09 ,  C07C51/27 ,  C07C51/353 ,  C07C51/367 ,  C07C51/377 ,  C07C51/412 ,  C07C51/60 ,  C07C61/08 ,  C07C61/15 ,  C07C61/35 ,  C07C61/39 ,  C07C61/40 ,  C07C62/04 ,  C07C62/10 ,  C07C62/20

Abstract: The chemical compounds of the invention are useful as the active compound in drugs because of their anticonvulsant and/or antianoxic activity. They have the general formula ##STR1## wherein Z is a hydroxyl group; a group--OM wherein M is an alkali metal atom or an equivalent atom fraction of an alkaline-earth metal or an amino group such as --NH.sub.2, and R is a linear or branched alkyl group containing from 1 to 9 carbon atoms, and optionally substituted by one or more halogen atoms; a linear or branched alkenyl or alkynyl, alkoxyalkyl, or acylalkyl group containing from 2 to 9 carbon atoms and optionally substituted by one or more halogen atoms; an aryl or arylalkyl or aryloxyalkyl group comprising at least one aromatic radical and an alkyl chain having from 1 to 4 carbon atoms.

Abstract translation: 本发明的化合物由于其抗惊厥和/或抗氧化活性而可用作药物中的活性化合物。 它们具有通式，其中Z是羟基; 基团-M OM，其中M是碱金属原子或碱土金属或氨基的等价原子级分，例如-NH 2，R是含有1至9个碳原子的直链或支链烷基，并且任选地 被一个或多个卤素原子取代; 含有2至9个碳原子并且任选被一个或多个卤素原子取代的直链或支链烯基或炔基，烷氧基烷基或酰基烷基; 包含至少一个芳族基团和具有1至4个碳原子的烷基链的芳基或芳基烷基或芳氧基烷基。

公开(公告)号：US4224227A

公开(公告)日：1980-09-23

申请号：US18166

申请日：1979-03-07

Applicant: Jacques Martel ,  Jean Tessier ,  Jean-Pierre Demoute

Inventor： Jacques Martel ,  Jean Tessier ,  Jean-Pierre Demoute

IPC: C07C69/74 ,  A01N33/00 ,  A01N53/00 ,  A01N53/02 ,  A01N53/04 ,  A01N53/08 ,  A01P3/00 ,  A23K1/16 ,  A61K31/215 ,  A61K31/34 ,  A61K31/40 ,  A61K35/14 ,  A61P31/04 ,  C07C20060101 ,  C07C51/00 ,  C07C51/363 ,  C07C53/50 ,  C07C61/04 ,  C07C61/15 ,  C07C67/00 ,  C07C69/743 ,  C07C253/00 ,  C07C255/39 ,  C07D209/48 ,  C07D209/49 ,  C07D307/42 ,  C07D307/45 ,  C07D307/54 ,  C07D317/54 ,  G01G13/295 ,  A01N9/28

CPC classification number: C07D209/49 ,  A01N53/00 ,  C07C255/00 ,  C07C61/15 ,  C07D307/42 ,  Y10S514/949

Abstract: Novel cyclopropane carboxylic acid esters of the formula ##STR1## wherein X.sub.1 is selected from the group consisting of hydrogen, fluorine, chlorine and bromine, X.sub.2 is selected from the group consisting of fluorine, chlorine and bromine, X.sub.3 is selected from the group consisting of chlorine, bromine and iodine and R is selected from the group consisting of ##STR2## and benzyl optionally substituted with at least one member of the group consisting of alkyl of 1 to 4 carbon atoms, alkenyl of 2 to 6 carbon atoms, alkenyloxy of 2 to 6 carbon atoms, alkadienyl of 4 to 8 carbon atoms, methylenedioxy, benzyl and halogens, R.sub.1 is selected from the group consisting of hydrogen and methyl, R.sub.2 is selected from the group consisting of monocyclic aryl and --CH.sub.2 --C.tbd.CH,R.sub.3 is an aliphatic of 2 to 6 carbon atoms having at least one double bond, R.sub.4 is selected from the group consisting of hydrogen, --CN and --C.tbd.CH, R.sub.5 is selected from the group consisting of chlorine and methyl, n is 0, 1 or 2, R.sub.6, R.sub.7, R.sub.8 and R.sub.9 are individually selected from the group consisting of hydrogen, chlorine and methyl and S/I indicates that the ring may be aromatic, dihydro or tetrahydro having pesticidal properties, and a process for their preparation.

Abstract translation: 新的式（I）的环丙烷羧酸酯，其中X 1选自氢，氟，氯和溴，X 2选自氟，氯和溴，X 3选自 的氯，溴和碘，R选自 和任选被至少一个由1至4个碳原子的烷基取代的苄基， 2至6个碳原子的烯氧基，2至6个碳原子的链烯氧基，4至8个碳原子的链二烯基，亚甲二氧基，苄基和卤素，R1选自氢和甲基，R2选自单环 芳基和-CH 2 -C 3 CH 3，R 3是具有至少一个双键的2至6个碳原子的脂族基，R 4选自氢，-CN和-C 3位CH，R 5选自 由氯和甲基组成 n为0,1或2，R6，R7，R8和R9分别选自氢，氯和甲基，S / I表示该环可为具有杀虫性质的芳香族二氢或四氢，以及 一个他们准备的过程。

公开(公告)号：US3641148A

公开(公告)日：1972-02-08

申请号：US3641148D

申请日：1969-03-05

Applicant: SMITH KLINE FRENCH LAB

Inventor： STEDMAN ROBERT JOHN

IPC: C07C49/423 ,  C07C49/473 ,  C07C61/125 ,  C07C61/15 ,  C07D317/72 ,  C07C87/40

CPC classification number: C07C61/15 ,  C07C49/423 ,  C07C49/473 ,  C07C61/125 ,  C07D317/72

Abstract: 1-AMINO AND AMINIMETHYLPENTACYCLO

(6.2.4.02,7.04.10.05,9)

DECANES, 3-AMINO AND AMINOMETHYLTETRACYCLO

(5.3.0.02,6.04,9)

DECANES, AND 1-AMINO AND AMINOMETHYLTETRACYCLO(5.2.0.02,6.04,9)-NONANES ARE PREPARED STARTING FROM TETRACHLOROCYCLOPENTADIENONE CYCLIC ETHYLENE KETAL AND 1,4-CYCLOHEXADIENE AND PROCEEDING WITH RING-CLOSURE, HYDROLYSIS AND FAVORSKII REACTIONS. THE PRODUCTS ARE ANTIVIRALS.