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    PREPARATION OF THIAZOLES
    61.
    发明申请
    PREPARATION OF THIAZOLES 失效
    制备THIAZOLES

    公开(公告)号：US20070055063A1

    公开(公告)日：2007-03-08

    申请号：US11552255

    申请日：2006-10-24

    申请人： Thomas Pitterna ,  Henry Szczepanski ,  Peter Maienfisch ,  Ottmar Huter ,  Thomas Rapold ,  Marcel Senn ,  Thomas Gobel ,  Anthony O'Sullivan

    发明人： Thomas Pitterna ,  Henry Szczepanski ,  Peter Maienfisch ,  Ottmar Huter ,  Thomas Rapold ,  Marcel Senn ,  Thomas Gobel ,  Anthony O'Sullivan

    IPC分类号： C07D417/02

    CPC分类号： C07D277/32 ,  C07D277/16 ,  C07D277/36 ,  C07D277/70 ,  C07D277/74

    摘要： A process for the preparation of a compound of the formula and, where applicable, its E/Z-isomers, mixtures of E/Z-isomers and/or tautomers and acid addition products thereof, in each case in free form or in salt form, wherein: R is unsubstituted or substituted C1-C12alkyl, unsubstituted or substituted C2-C4alkenyl, unsubstituted or substituted C2-C4alkynyl, unsubstituted or substituted C3-C6cycloalkyl, unsubstituted or substituted aryl, unsubstituted or substituted heteroaryl, or —SR1; R1 is unsubstituted or substituted C1-C12alkyl, unsubstituted or substituted C2-C4alkenyl, unsubstituted or substituted C2-C4alkynyl, unsubstituted or substituted cycloalkyl, unsubstituted or substituted aryl or unsubstituted or substituted heteroaryl; and X is a leaving group; The process comprises reacting a compound of the formula: with a halogenating agent or a sulfonylating agent. Alternatively, when X is a selected halogen, the process can comprise reacting a compound of the formula with a compound having a formula selected from the group consisting of halogen-C(═O)—O—C1-C8alkyl; halogen-C(═O)—O-aryl; and halogen-C(═O)—O-benzyl.

    摘要翻译： 制备下式化合物及其E / Z-异构体的方法，E / Z-异构体和/或互变异构体的混合物及其酸加成产物，各自为游离形式或盐形式 ，其中：R是未取代或取代的C 1 -C 12烷基，未取代或取代的C 2 -C 4 烯基，未取代或取代的C 2 -C 4炔基，未取代或取代的C 3 -C 6环烷基 ，未取代或取代的芳基，未取代或取代的杂芳基或-SR 1 N; R 1是未取代或取代的C 1 -C 12烷基，未取代或取代的C 2 -C 3 未取代或取代的C 2 -C 4炔基，未取代或取代的环烷基，未取代或取代的芳基或未取代或取代的杂芳基; X为离去群; 该方法包括使下式化合物与卤化剂或磺酰化剂反应。 或者，当X是选择的卤素时，该方法可以包括使下式的化合物与具有选自以下的式的化合物反应：卤素-C（ - ） - O-C 1 -C 烷基; 卤素-C（ - ） - O-芳基; 和卤素-C（ - ） - O-苄基。

    "> Avermectins and avermectin monosaccharides substituted in the 4'-and 4
    62.
    发明申请
    Avermectins and avermectin monosaccharides substituted in the 4'-and 4"-position having pesticidal properties 审中-公开
    在4'和4“位具有杀虫性质的阿维菌素和阿维菌素单糖被取代

    公开(公告)号：US20060094600A1

    公开(公告)日：2006-05-04

    申请号：US10544281

    申请日：2004-02-03

    申请人： Laura Quaranta ,  Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre

    发明人： Laura Quaranta ,  Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre

    IPC分类号： A01N43/04 ,  A01N25/26 ,  C07H17/08

    CPC分类号： C07H17/08 ,  A01N43/90

    摘要： What is described are a compound of the formula (I) wherein the bond of atoms C22 and C23 is a single or double bond; m is 0 or 1; n is 0, 1 or 2; p is 0 or 1; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12alkenyl; R2 is for example H, C1-C12-alkyl, C1-C12-haloalkyl or C1-C12-hydroxyalkyl; or together with R4 form with the carbon to which they are bound for example a three- to seven-membered ring; R3 is for example H, C1-C12-alkyl, halogen, halo-C1-C2alkyl, CN, NO2 or C3-C8-cycloalkyl; R4 has the same meanings as R2; R5 and R6 independently of each other are for example H, C1-C12-alkyl, CN, NO2, OH, SH, halogen, halo-C1-C2alkyl or C3-C8cycloalkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.

    摘要翻译： 描述的是式（I）的化合物，其中原子C 22和C 23的键是单键或双键; m为0或1; n为0,1或2; p为0或1; R 1是C 1 -C 12 - 烷基，C 3 -C 8亚烷基，C 3 -C 12 - 烷基，C 3 -C 12 - 环烷基或C 2 -C 12链烯基; R 2是例如H，C 1 -C 12 - 烷基，C 1 -C 3 - 12个 - 卤代烷基或C 1 -C 12 - 羟基烷基; 或与R 4 S形成的碳与它们所键合的碳例如为三至七元环; R 3是例如H，C 1 -C 12 - 烷基，卤素，卤素-C 1 - C 2 -C 12烷基，CN，NO 2或C 3 -C 8 - 环烷基; R 4具有与R 2'相同的含义; R 5和R 6彼此独立地是例如H，C 1 -C 12 - 烷基， CN，NO 2，OH，SH，卤素，卤代-C 1 -C 2烷基或C 3 - -C 8环烷基; 或者如果适用，E / Z异构体，E / Z异构体混合物和/或其互变异构体在每种情况下以游离形式或盐形成用于制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

    Process for the preparation of thiazole derivatives
    64.
    发明授权
    Process for the preparation of thiazole derivatives 失效
    噻唑衍生物的制备方法

    公开(公告)号：US06677457B2

    公开(公告)日：2004-01-13

    申请号：US10047807

    申请日：2002-01-15

    申请人： Thomas Pitterna ,  Henry Szczepanski ,  Peter Maienfisch ,  Ottmar Franz Hüter ,  Thomas Rapold ,  Marcel Senn ,  Thomas Göbel ,  Anthony Cornelius O'Sullivan ,  Gottfried Seifert

    发明人： Thomas Pitterna ,  Henry Szczepanski ,  Peter Maienfisch ,  Ottmar Franz Hüter ,  Thomas Rapold ,  Marcel Senn ,  Thomas Göbel ,  Anthony Cornelius O'Sullivan ,  Gottfried Seifert

    IPC分类号： C07D27716

    CPC分类号： C07D277/32 ,  C07D277/16 ,  C07D277/36 ,  C07D417/06

    摘要： The invention relates to a process for the preparation of a compound of the formula wherein Q, Y, Z, R1, R2, R3, R4 and R5 are as defined in the specification, which comprises a) reacting a compound of the formula  with a halogenating agent to form a compound of the formula or b) converting a compound of formula (II) by means of a halogenating agent into a compound of the formula optionally c) converting the compound of formula (IV) into a compound of formula (III); d) converting a compound of formula (III) by means of a compound of the formula into a compound of the formula or e) converting a compound (IV) by means of a compound (V) into a compound (VI); and f) converting a compound (VI) by means of a chlorinating agent into a compound (I); a compound (IV); to a process for the preparation of a compound (III) and to a process for the preparation of a compound (IV).

    摘要翻译： 本发明涉及制备糠醛的化合物的方法，其中Q，Y，Z，R 1，R 2，R 3，R 4和R 5如本说明书中所定义，其包括：a）将卤化剂的化合物与 将式（II）化合物通过卤化剂转化成式（Ⅲ）的化合物，将式（Ⅳ）化合物转化为式（Ⅳ）化合物; d）将化合物 通过化学式（Ⅳ）将化合物（Ⅳ）转化为化合物（Ⅵ）;将式（Ⅳ）化合物与式 和（f）通过氯化剂将化合物（VI）转化为化合物（I）;化合物（IV）; 涉及制备化合物（III）的方法和制备化合物（IV）的方法。

    Thiazole compounds
    65.
    发明授权
    Thiazole compounds 失效
    噻唑化合物

    公开(公告)号：US06211381B1

    公开(公告)日：2001-04-03

    申请号：US09077569

    申请日：1998-06-01

    申请人： Henry Szczepanski ,  Thomas Göbel ,  Ottmar Franz Hüter ,  Anthony Cornelius O'Sullivan ,  Marcel Senn ,  Thomas Rapold ,  Peter Maienfisch ,  Thomas Pitterna

    发明人： Henry Szczepanski ,  Thomas Göbel ,  Ottmar Franz Hüter ,  Anthony Cornelius O'Sullivan ,  Marcel Senn ,  Thomas Rapold ,  Peter Maienfisch ,  Thomas Pitterna

    IPC分类号： C07D27732

    CPC分类号： C07D277/32 ,  C07D277/36 ,  C07D417/06

    摘要： The invention relates to a process for preparing a compound of formula (I), in which X is CH or N, Y is NO2 or CN, Z is CHR3, O, NR3 or S, R1 and R2 are either each, independently of the other, hydrogen or unsubstituted or R4-substituted alkyl or together a two- or three-membered alkylene bridge or a two- or three-membered alkylene bridge in which one member is replaced by a hetero member selected from the group, consisting of NR5, O and S, R3 is H or unsubstituted or R4-substituted alkyl, R4 is an unsubstituted or substituted aryl or heteroaryl group, and R5 is H or alkyl, which comprises a) reacting a compound of formula (II) with a chlorinating agent or b1) initially reacting a compound of formula (IV) with a compound of formula (V) and b2) further reacting the compound of formula (II) obtainable thereby, with or without intermediate isolation, with a chlorinating agent, to intermediates used in this process, to the use of these intermediates and to a process for the preparation of these intermediates.

    摘要翻译： 本发明涉及制备式（I）化合物的方法，其中X是CH或N，Y是NO 2或CN，Z是CHR 3，O，NR 3或S，R 1和R 2各自独立地是 另一个，氢或未取代的或R4取代的烷基或二元或三元亚烷基桥或二元或三元亚烷基桥，其中一个成员被选自NR5， O和S，R 3是H或未取代的或R 4取代的烷基，R 4是未取代或取代的芳基或杂芳基，R 5是H或烷基，其包括a）使式（II）化合物与氯化剂或 b1）最初使式（Ⅳ）化合物与式（Ⅴ）化合物反应，和b2）使可得到的式（Ⅱ）化合物进一步与中间体分离与氯化剂反应，得到本发明的中间体 过程，使用这些中间体和制备过程 这些中间体。

    Oxadiazine derivatives
    66.
    发明授权
    Oxadiazine derivatives 失效
    恶二嗪衍生物

    公开(公告)号：US5852012A

    公开(公告)日：1998-12-22

    申请号：US464931

    申请日：1995-06-05

    申请人： Peter Maienfisch ,  Laurenz Gsell

    发明人： Peter Maienfisch ,  Laurenz Gsell

    IPC分类号： A01N43/88 ,  A01N43/72 ,  A01N43/84 ,  A01N47/40 ,  A01N47/44 ,  A01N51/00 ,  A01P7/04 ,  C07D20060101 ,  C07D273/04 ,  C07D413/06 ,  C07D417/06 ,  C07D471/04 ,  C07D487/04 ,  C07D498/04 ,  C07D513/04

    CPC分类号： C07D413/06 ,  A01N47/40 ,  A01N51/00 ,  C07D273/00 ,  C07D273/04 ,  C07D417/06

    摘要： Compounds of the formula ##STR1## in which A is an unsubstituted or mono- to tetrasubstituted, aromatic or non-aromatic, monocyclic or bicyclic heterocyclic radical, where one to two of the substituents of A can be selected from the group consisting of halo-C.sub.1 -C.sub.3 alkyl, cyclopropyl, halocyclopropyl, C.sub.2 -C.sub.3 alkenyl, C.sub.2 -C.sub.3 alkynyl, halo-C.sub.2 -C.sub.3 alkenyl, halo-C.sub.2 -C.sub.3 alkynyl, halo-C.sub.1 -C.sub.3 alkoxy, C.sub.1 -C.sub.3 alkylthio, halo-C.sub.1 -C.sub.3 alkylthio, allyloxy, propargyloxy, allylthio, propargylthio, haloallyloxy, haloallylthio, cyano and nitro, and one to four of the substituents of A can be selected from the group consisting of C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 alkoxy and halogen; R is hydrogen, C.sub.1 -C.sub.6 alkyl, phenyl-C.sub.1 -C.sub.4 alkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.2 -C.sub.6 alkenyl or C.sub.2 -C.sub.6 alkynyl; and X is N--NO.sub.2 or N--CN, and, if appropriate, tautomers thereof, in each case in free form or in salt form, can be used as insecticidal active ingredients and can be prepared in a manner known per se.

    摘要翻译： 式（I）的化合物，其中A是未取代或单取代或单取代的，芳香族或非芳族的单环或双环杂环基，其中A的一至两个取代基可以选自 卤代C 1 -C 3烷基，环丙基，卤代环丙基，C 2 -C 3烯基，C 2 -C 3炔基，卤代-C 2 -C 3烯基，卤代-C 2 -C 3炔基，卤代-C 1 -C 3烷氧基，C 1 -C 3烷硫基，卤代C 1 -C 3烷硫基，烯丙氧基，炔丙氧基 ，烯丙硫基，炔丙硫基，卤代烯丙氧基，卤代烯硫基，氰基和硝基，A至1-4个取代基可以选自C 1 -C 3烷基，C 1 -C 3烷氧基和卤素; R是氢，C 1 -C 6烷基，苯基-C 1 -C 4烷基，C 3 -C 6环烷基，C 2 -C 6烯基或C 2 -C 6炔基; 且X为N-NO 2或N-CN，并且如果合适，其互变异构体在各种情况下以游离形式或盐形式可用作杀虫活性成分，并且可以以本身已知的方式制备。

    Pyridine compounds which are useful as pesticides
    68.
    发明授权
    Pyridine compounds which are useful as pesticides 失效
    可用作杀虫剂的吡啶化合物

    公开(公告)号：US5223520A

    公开(公告)日：1993-06-29

    申请号：US858910

    申请日：1992-03-27

    申请人： Odd Kristiansen ,  Laurenz Gsell ,  Peter Maienfisch

    发明人： Odd Kristiansen ,  Laurenz Gsell ,  Peter Maienfisch

    IPC分类号： A01N43/40 ,  A01N43/78 ,  A01N47/44 ,  A01N51/00 ,  C07D213/36 ,  C07D213/40 ,  C07D213/61 ,  C07D213/89 ,  C07D277/20 ,  C07D277/32

    CPC分类号： C07D213/40 ,  A01N43/40 ,  A01N43/78 ,  A01N47/44 ,  A01N51/00 ,  C07D213/61 ,  C07D213/89 ,  C07D277/32

    摘要： Compounds of formula ##STR1## wherein R.sub.1 is hydrogen, C.sub.1 -C.sub.4 alkyl or C.sub.3 -C.sub.6 cycloalkyl, R.sub.2 is hydrogen or C.sub.1 -C.sub.4 alkyl, R.sub.3 is hydrogen, C.sub.1 -C.sub.4 alkyl or C.sub.3 -C.sub.6 cycloalkyl and R.sub.4 is C.sub.1 -C.sub.4 alkyl, C.sub.3 -C.sub.6 cycloalkyl or --CH.sub.2 CH.sub.2 COOR.sub.7, or R.sub.3 and R.sub.4 together are --(CH.sub.2).sub.4 -- or --(CH.sub.2).sub.5 --, R.sub.5 is hydrogen, C.sub.1 -C.sub.4 alkyl, ##STR2## --CH.sub.2 OCH.sub.3, --CN, --COOR.sub.7 or ##STR3## R.sub.6 is hydrogen, chlorine, methyl or nitro, R.sub.7 and R.sub.8 are each methyl or ethyl, A is an unsubstituted or mono- to tetra-substituted, aromatic or non-aromatic, monocyclic or bicyclic, heterocyclic radical, one or two substituents being selected from the group consisting of C.sub.1 -C.sub.3 haloalkyl, cyclopropyl, halocyclopropy, C.sub.2 -C.sub.3 alkenyl, C.sub.2 -C.sub.3 alkynyl, C.sub.2 -C.sub.3 haloalkenyl, C.sub.2 -C.sub.3 haloalkynyl, C.sub.1 -C.sub.3 haloalkoxy, C.sub.1 -C.sub.3 alkylthio, C.sub.1 -C.sub.3 haloalkylthio, allyloxy, propargyloxy, allylthio, propargylthio, haloallyloxy, haloallylthio, cyano and nitro, and from one to four substituents being selected from the group consisting of C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 alkoxy and halogen, and .dbd.X is .dbd.N--NO.sub.2, .dbd.CH--NO.sub.2, .dbd.N--CN or .dbd.CH--CO--CF.sub.3, in free form or in the form of acid addition salts, can be used as agrochemical active ingredients and can be prepared in a manner known per se.

    摘要翻译： 式（I）的化合物其中R 1是氢，C 1 -C 4烷基或C 3 -C 6环烷基，R 2是氢或C 1 -C 4烷基，R 3是氢，C 1 -C 4烷基或C 3 -C 6环烷基，R 4是C 1 -C 4烷基， C 6环烷基或-CH 2 CH 2 COOR 7，或者R 3和R 4一起是 - （CH 2）4 - 或 - （CH 2）5 - ，R 5是氢，C 1 -C 4烷基，-CH 2 OCH 3，-CN，-COOR 7或者R 6是 氢，氯，甲基或硝基，R 7和R 8各自为甲基或乙基，A为未取代或单取代或四取代的芳族或非芳族单环或双环杂环基，一个或两个选自 由C 1 -C 3卤代烷基，环丙基，卤代环丙基，C 2 -C 3烯基，C 2 -C 3炔基，C 2 -C 3卤代烯基，C 2 -C 3卤代炔基，C 1 -C 3卤代烷氧基，C 1 -C 3烷硫基，C 1 -C 3卤代烷硫基，烯丙氧基，炔丙氧基，烯丙硫基，炔丙基硫代，卤代烯氧基，卤代烯硫基 氰基和硝基，以及一至四个选自C 1 -C 3烷基，C 1 -C 3烷氧基和卤素的取代基，X = N-NO 2 = 游离形式或以酸加成盐形式的CH-NO 2，= N-CN或= CH-CO-CF 3可用作农业化学活性成分，并且可以以本身已知的方式制备。