公开(公告)号：US2811554A

公开(公告)日：1957-10-29

申请号：US50583155

申请日：1955-05-03

Applicant: ROUSSEL UCLAF

Inventor： GEORGES MULLER ,  LEON VELLUZ

CPC classification number: C07C205/45

公开(公告)号：US5240960B1

公开(公告)日：1995-05-02

申请号：US78508791

申请日：1991-10-30

Applicant: ROUSSEL UCLAF

Inventor： HAMBLETON PHILIP T ,  HEDGECOCK CHARLES J R ,  KAY DAVID P ,  KUO ELIZABETH A ,  TULLY WILFRED R

IPC: A61K31/275 ,  A61K31/34 ,  A61K31/357 ,  A61P29/00 ,  A61P37/00 ,  C07C255/19 ,  C07C255/27 ,  C07C255/31 ,  C07C255/60 ,  C07C323/41 ,  C07D317/58 ,  C07D317/66

CPC classification number: C07D317/58 ,  C07C255/27 ,  C07C255/31 ,  C07C255/60 ,  C07C323/41 ,  C07C2601/02 ,  C07C2601/04 ,  C07C2601/06

公开(公告)号：US3925393A

公开(公告)日：1975-12-09

申请号：US37750373

申请日：1973-07-09

Applicant: ROUSSEL UCLAF

Inventor： HEURTAUX SIMONE ,  COSTEROUSSE GERMAIN

IPC: C07D461/00 ,  A61K20060101 ,  A61K31/395 ,  A61K31/435 ,  A61P9/08 ,  C07D471/22 ,  C07D487/22 ,  C07F20060101

CPC classification number: C07D461/00

Abstract: Novel racemic or optically active mixed alkali metal or ammonium phosphate salts with vincanol, methods for their preparation, and their pharmaceutical use.

Abstract translation: 新的外消旋或光学活性的与伐醇的混合碱金属或磷酸铵盐，其制备方法及其药物用途。

公开(公告)号：US3923800A

公开(公告)日：1975-12-02

申请号：US53963975

申请日：1975-01-09

Applicant: ROUSSEL UCLAF

Inventor： DERIBLE PIERRE HENRI ,  LAVAUX JEAN-PAUL ,  LAURENT JACQUES

IPC: A61K31/54 ,  C07D401/04 ,  C07D417/14 ,  C07D209/14

CPC classification number: C07D417/14 ,  A61K31/54

Abstract: Novel phenothiazines of the formula

WHEREIN X is selected from the group consisting of hydrogen, chlorine, trifluoromethyl, methylthio and methoxy, B is selected from the group consisting of hydrogen and alkyl of 1 to 3 carbon atoms, p is 0 or 1, R is selected from the group consisting of hydrogen and alkoxy of 1 to 3 carbon atoms and R1 and R2 are individually selected from the group consisting of hydrogen and alkyl of 1 to 3 carbon atoms and their non-toxic, pharmaceutically acceptable acid addition salts having neuroleptic activity and frequently antihistaminic activity and their preparation.

Abstract translation: 式WHEREIN X的新型吩噻嗪由氢，氯，三氟甲基，甲硫基和甲氧基组成的组中选择，B选自氢和1至3个碳原子的烷基，p为0或1，R为 选自氢和1至3个碳原子的烷氧基，R 1和R 2分别选自氢和1至3个碳原子的烷基及其无毒的药学上可接受的具有精神抑制活性的酸加成盐 并经常抗组胺活性及其制备。

公开(公告)号：US3910898A

公开(公告)日：1975-10-07

申请号：US45760474

申请日：1974-04-03

Applicant: ROUSSEL UCLAF

Inventor： ALLAIS ANDRE ,  MEIER JEAN

IPC: A61K31/47 ,  C07D215/44 ,  C07D401/12 ,  C07D405/12 ,  C07D413/12 ,  F24F3/04 ,  C07D295/04

CPC classification number: A61K31/47 ,  C07D215/44 ,  C07D401/12 ,  C07D405/12 ,  C07D413/12

Abstract: 7- OR 8-TRIFLUOROMETHYL-QUINOLINES OF THE FORMULA

WHEREIN N IS 1 OR 2 AND R is morpholino and their non-toxic, pharmaceutically acceptable acid addition salts having analgesic and anti-inflammatory activity and their preparation.

Abstract translation: 7-或8-三氟甲基喹啉，其中N为1或2，R为吗啉代及其无毒，药学上可接受的具有镇痛和抗炎活性的酸加成盐及其制备方法。

公开(公告)号：US3905996A

公开(公告)日：1975-09-16

申请号：US38419773

申请日：1973-07-31

Applicant: ROUSSEL UCLAF

Inventor： PERRONNET JACQUES ,  TECHE ANDRE

IPC: C07D243/04 ,  A01N43/48 ,  A01N43/50 ,  C07C275/64 ,  C07D233/32 ,  C07D233/38 ,  C07D239/10 ,  C07D243/08 ,  C07D245/02 ,  C07D247/02 ,  C07D233/02

CPC classification number: C07D239/10 ,  C07C265/12 ,  C07C275/64 ,  C07D233/38

Abstract: Novel compounds of the formula

wherein A is a straight or branched chain alkylene of 2 to 6 carbon atoms, X is selected from the group consisting of hydrogen, halogen, -CF3, -NO2, acyl of an organic carboxylic acid of 1 to 6 carbon atoms, alkyl and alkoxy of 1 to 6 carbon atoms and alkenyloxy of 2 to 6 carbon atoms optionally substituted with halogen, Y is selected from the group consisting of hydrogen, halogen and alkyl and alkoxy of 1 to 6 carbon atoms and R is selected from the group consisting of alkoxy of 1 to 4 carbon atoms, alkoxycarbonyl of 2 to 6 carbon atoms and chloroacetyl which have herbicidal properties.

Abstract translation: 新型式O的化合物其中A是2至6个碳原子的直链或支链亚烷基，X选自氢，卤素，-CF 3，-NO 2， 1至6个碳原子的有机羧酸的酰基，1至6个碳原子的烷基和烷氧基以及2至6个碳原子的任选被卤素取代的烯氧基，Y选自氢，卤素和烷基和烷氧基 1至6个碳原子，R选自1至4个碳原子的烷氧基，2至6个碳原子的烷氧基羰基和具有除草性质的氯乙酰基。

公开(公告)号：US3904624A

公开(公告)日：1975-09-09

申请号：US39407873

申请日：1973-09-04

Applicant: ROUSSEL UCLAF

Inventor： PERRONNET JACQUES ,  TALIANI LAURENT

IPC: A01N57/08 ,  A01N57/16 ,  C07D471/04 ,  C07F9/08 ,  C07F9/24 ,  C07F9/40 ,  C07F9/6561 ,  C07D239/70 ,  A01N9/36

CPC classification number: C07D471/04 ,  C07F9/6561

Abstract: Novel organo-phosphorus compounds of the formula

WHEREIN R is selected from the group consisting of methine and nitrogen, R1 is selected from the group consisting of hydrogen, alkyl of 1 to 3 carbon atoms and NO2, R2 is selected from the group consisting of hydrogen, straight or branched alkyl of 1 to 3 carbon atoms, chlorine, bromine, alkoxycarbonyl of 2 to 4 carbon atoms, phenyl and thioalkyl of 1 to 4 carbon atoms, R3 is branched or straight chain alkyl of 1 to 3 carbon atoms and R4 is selected from the group consisting of straight and branched chain alkyl of 1 to 3 carbon atoms, alkoxy of 1 to 3 carbon atoms and

wherein R5 and R6 are individually selected from the group consisting of hydrogen and branched and straight chain alkyl of 1 to 3 carbon atoms having pesticidal properties and their preparation.

公开(公告)号：US3904586A

公开(公告)日：1975-09-09

申请号：US48703674

申请日：1974-07-10

Applicant: ROUSSEL UCLAF

Inventor： DERIBLE PIERRE HENRI ,  HUMBERT DANIEL ,  DUMONT CLAUDE

IPC: C07C307/02 ,  C07C67/00 ,  C07C301/00 ,  C07C303/34 ,  C07D209/48 ,  C07C143/80

CPC classification number: C07D209/48

Abstract: Novel benzyloxysulfamides of the formula

WHEREIN X is a halogen and m is 0, 1, 2 or 3 and their nontoxic, pharmaceutically acceptable alkaline salts having tranquillizing, anticonvulsant and anxiolytic properties and their preparation.

公开(公告)号：US3903270A

公开(公告)日：1975-09-02

申请号：US34567273

申请日：1973-03-28

Applicant: ROUSSEL UCLAF

Inventor： QUEUILLE ANDRE

IPC: A61K20060101 ,  A61K36/02 ,  A61K36/04 ,  C08B20060101 ,  C08L5/00 ,  A61K27/00

CPC classification number: A61K36/04 ,  Y10S514/926 ,  Y10S514/927

Abstract: Novel pharmaceutical compositions having as the active ingredient at least one alkali metal salt of the sulfuric acid ester of a high molecular weight polysaccharide extracted from Furcellaria fastigiata algae (Rhodophyces - gigantinals) and a method of treating pepsic hyperactivity in warm-blooded animals by oral administration of said alkali metal salts.

Abstract translation: 作为活性成分的新型药物组合物，其是从毛细丝藻（Rhodophyces-gigantinals）中提取的高分子量多糖的硫酸酯的至少一种碱金属盐和通过口服给药在温血动物中治疗多囊卵巢综合征的方法 的所述碱金属盐。

公开(公告)号：US3903114A

公开(公告)日：1975-09-02

申请号：US40203073

申请日：1973-10-01

Applicant: ROUSSEL UCLAF

Inventor： LE MARTRET ODILE ,  CLEMENCE FRANCOIS

IPC: A61K31/38 ,  A61K31/381 ,  A61P25/04 ,  A61P25/06 ,  A61P29/00 ,  C07D333/22 ,  C07D333/38

CPC classification number: C07D333/22

Abstract: Novel thiophene derivatives of the formula

WHEREIN R and R2 are individually selected from the group consisting of hydrogen and methyl with R2 being in the 3- or 4position of the thienyl ring, R1 is selected from the group consisting of hydrogen and acyl of an organic carboxylic acid of 1 to 18 carbon atoms and X is selected from the group consisting of hydrogen, halogen, methyl, methoxy, CF3- and CF3O- in any position on the benzene ring, the compounds being in racemic or optically active form when R is methyl having anti-inflammatory and analgesic activity.

Abstract translation: 式WHEREIN R和R2的新型噻吩衍生物分别选自氢和甲基，R2在噻吩环的3-或4-位，R1选自氢和酰基， 1至18个碳原子的有机羧酸，X选自氢，卤素，甲基，甲氧基，CF3-和CF3O-在苯环上的任何位置，该化合物当R 是具有抗炎和止痛活性的甲基。