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公开(公告)号:US06936633B2
公开(公告)日:2005-08-30
申请号:US10750247
申请日:2003-12-31
申请人: Dong Zou , Olivier Dasse , Janelle Evans , Paul Higgins , Jeremy Kintigh , Rama Kondru , Eric Schwartz , Laurent Knerr , Hai-Xiao Zhai
发明人: Dong Zou , Olivier Dasse , Janelle Evans , Paul Higgins , Jeremy Kintigh , Rama Kondru , Eric Schwartz , Laurent Knerr , Hai-Xiao Zhai
IPC分类号: A61K31/40 , A61K31/4015 , A61K31/402 , A61K31/4025 , A61K31/422 , A61K31/4439 , A61P1/04 , A61P1/16 , A61P7/02 , A61P9/10 , A61P9/14 , A61P11/00 , A61P11/02 , A61P11/06 , A61P13/12 , A61P15/00 , A61P17/00 , A61P17/04 , A61P17/06 , A61P19/02 , A61P21/02 , A61P25/00 , A61P25/28 , A61P27/02 , A61P27/16 , A61P29/00 , A61P31/04 , A61P31/18 , A61P35/00 , A61P37/02 , A61P37/08 , A61P39/02 , C07D207/24 , C07D207/26 , C07D207/273 , C07D207/36 , C07D207/38 , C07D401/04 , C07D405/04 , C07D405/08 , C07D409/04 , C07D409/06 , C07D413/06 , C07D207/04
CPC分类号: C07D207/273 , A61K31/4015 , A61K31/4439 , C07D207/24 , C07D207/36 , C07D401/04 , C07D405/04 , C07D409/04 , C07D409/06 , C07D413/06
摘要: The present invention provides pharmaceutical compositions and novel compounds useful in the treatment of conditions mediated by CCR2, MCP-1 or the interaction thereof. The compounds of the present invention are pyrrolidinones and pyrrolidine-thiones.
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公开(公告)号:US20050004180A1
公开(公告)日:2005-01-06
申请号:US10489661
申请日:2002-09-26
申请人: Dong Zou , Olivier Dasse , Janelle Evans , Paul Higgins , Jeremy Kintigh , Laurent Knerr , Rama Kondru , Eric Schwartz , Hai-Xiao Zhai
发明人: Dong Zou , Olivier Dasse , Janelle Evans , Paul Higgins , Jeremy Kintigh , Laurent Knerr , Rama Kondru , Eric Schwartz , Hai-Xiao Zhai
IPC分类号: A61K31/40 , A61K31/4015 , A61K31/402 , A61K31/4025 , A61K31/422 , A61K31/4439 , A61P1/04 , A61P1/16 , A61P7/02 , A61P9/10 , A61P9/14 , A61P11/00 , A61P11/02 , A61P11/06 , A61P13/12 , A61P15/00 , A61P17/00 , A61P17/04 , A61P17/06 , A61P19/02 , A61P21/02 , A61P25/00 , A61P25/28 , A61P27/02 , A61P27/16 , A61P29/00 , A61P31/04 , A61P31/18 , A61P35/00 , A61P37/02 , A61P37/08 , A61P39/02 , C07D207/24 , C07D207/26 , C07D207/273 , C07D207/36 , C07D207/38 , C07D401/04 , C07D405/04 , C07D405/08 , C07D409/04 , C07D409/06 , C07D413/06
CPC分类号: C07D207/273 , A61K31/4015 , A61K31/4439 , C07D207/24 , C07D207/36 , C07D401/04 , C07D405/04 , C07D409/04 , C07D409/06 , C07D413/06
摘要: The present invention provides pharmaceutical compositions and novel compounds useful in the treatment of conditions mediated by CCR2, MCP-1 or the interaction thereof. The compounds of the present invention are pyrrolidinones and pyrrolidine-thiones.
摘要翻译: 本发明提供了用于治疗由CCR2,MCP-1介导的病症或其相互作用的药物组合物和新化合物。 本发明的化合物是吡咯烷酮和吡咯烷 - 硫堇。
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公开(公告)号:US06727275B2
公开(公告)日:2004-04-27
申请号:US10255494
申请日:2002-09-26
申请人: Dong Zou , Olivier Dasse , Janelle Evans , Paul Higgins , Jeremy Kintigh , Rama Kondru , Eric Schwartz , Laurent Knerr , Hai-Xiao Zhai
发明人: Dong Zou , Olivier Dasse , Janelle Evans , Paul Higgins , Jeremy Kintigh , Rama Kondru , Eric Schwartz , Laurent Knerr , Hai-Xiao Zhai
IPC分类号: C07D20726
CPC分类号: C07D207/273 , A61K31/4015 , A61K31/4439 , C07D207/24 , C07D207/36 , C07D401/04 , C07D405/04 , C07D409/04 , C07D409/06 , C07D413/06
摘要: The present invention provides pharmaceutical compositions and novel compounds useful in the treatment of conditions mediated by CCR2, MCP-1 or the interaction thereof. The compounds of the present invention are pyrrolidinones and pyrrolidine-thiones.
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公开(公告)号:US09012462B2
公开(公告)日:2015-04-21
申请号:US12736910
申请日:2009-05-21
申请人: Yihan Wang , Wei-Sheng Huang , Shuangying Liu , William C. Shakespeare , R. Mathew Thomas , Jiwei Qi , Feng Li , Xiaotian Zhu , Anna Kohlman , David C. Dalgarno , Jan Antoinette C. Romero , Dong Zou
发明人: Yihan Wang , Wei-Sheng Huang , Shuangying Liu , William C. Shakespeare , R. Mathew Thomas , Jiwei Qi , Feng Li , Xiaotian Zhu , Anna Kohlman , David C. Dalgarno , Jan Antoinette C. Romero , Dong Zou
IPC分类号: A61K31/506 , C07F9/30 , C07D239/48 , C07F9/6509 , C07F9/6512 , C07F9/6521 , C07F9/6558 , C07F9/6561 , C07F9/6568 , C07F9/6571
CPC分类号: C07F9/6533 , C07D239/48 , C07F9/58 , C07F9/650905 , C07F9/6512 , C07F9/6521 , C07F9/65218 , C07F9/65583 , C07F9/65586 , C07F9/6561 , C07F9/65616 , C07F9/65685 , C07F9/657172 , C07F9/65846
摘要: The invention features compounds of the general formula (I) in which the variable groups are as defined herein, and to their preparation and use.
摘要翻译: 本发明的特征在于其中可变基团如本文所定义的通式(I)的化合物及其制备和用途。
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5.Substituted acetylenic imidazo[1,2-A]pyridine compounds as kinase inhibitors 有权
标题翻译: 取代的炔属咪唑并[1,2-A]吡啶化合物作为激酶抑制剂公开(公告)号:US08470851B2
公开(公告)日:2013-06-25
申请号:US13357745
申请日:2012-01-25
申请人: Dong Zou , Wei-Sheng Huang , R. Mathew Thomas , Jan Antoinette C. Romero , Jiwei Qi , Yihan Wang , Xiaotian Zhu , William C. Shakespeare , Rajeswari Sundaramoorthi , Chester A. Metcalf, III , David C. Dalgarno , Tomi K. Sawyer
发明人: Dong Zou , Wei-Sheng Huang , R. Mathew Thomas , Jan Antoinette C. Romero , Jiwei Qi , Yihan Wang , Xiaotian Zhu , William C. Shakespeare , Rajeswari Sundaramoorthi , Chester A. Metcalf, III , David C. Dalgarno , Tomi K. Sawyer
IPC分类号: A61K31/44
CPC分类号: C07D471/04 , C07D473/34 , C07D487/04
摘要: This invention relates to compounds of the general formula: in which the variable groups are as defined herein, and to their preparation and use.
摘要翻译: 本发明涉及以下通式的化合物:其中可变基团如本文所定义,及其制备和用途。
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公开(公告)号:US20130274273A1
公开(公告)日:2013-10-17
申请号:US13832240
申请日:2013-03-15
申请人: Chester A. Metcalf, III , Yu Gui Gu , Spencer D. Kimball , Qingy Li , Blaise S. Lippa , Dominic Ryan , Xinyuan Wu , Dong Zou
发明人: Chester A. Metcalf, III , Yu Gui Gu , Spencer D. Kimball , Qingy Li , Blaise S. Lippa , Dominic Ryan , Xinyuan Wu , Dong Zou
IPC分类号: C07D473/08
CPC分类号: C07D473/08
摘要: This disclosure describes a novel compounds and pharmaceutical compositions for inhibiting the TRPA1 ion channel and/or medical conditions related to TRPA1, such as pain.
摘要翻译: 本公开描述了用于抑制TRPA1离子通道和/或与TRPA1相关的医学状况的新型化合物和药物组合物,例如疼痛。
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公开(公告)号:US20120135986A1
公开(公告)日:2012-05-31
申请号:US13357745
申请日:2012-01-25
申请人: Dong Zou , Wei-Sheng Huang , R. Mathew Thomas , Jan Antionette C. Romero , Jiwei Qi , Yihan Wang , Xiaotian Zhu , William C. Shakespeare , Rajeswari Sundaramoorthi , Chester A. Metcalf, III , David C. Dalgarno , Tomi K. Sawyer
发明人: Dong Zou , Wei-Sheng Huang , R. Mathew Thomas , Jan Antionette C. Romero , Jiwei Qi , Yihan Wang , Xiaotian Zhu , William C. Shakespeare , Rajeswari Sundaramoorthi , Chester A. Metcalf, III , David C. Dalgarno , Tomi K. Sawyer
IPC分类号: A61K31/5377 , A61K31/4985 , C07D471/04 , A61K31/437 , A61P35/00 , A61K31/5025 , A61K31/53 , A61K31/519 , C07D473/34 , A61K31/52 , C07D487/04 , A61K31/496
CPC分类号: C07D471/04 , C07D473/34 , C07D487/04
摘要: This invention relates to compounds of the general formula: in which the variable groups are as defined herein, and to their preparation and use.
摘要翻译: 本发明涉及以下通式的化合物:其中可变基团如本文所定义,以及其制备和用途。
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公开(公告)号:US20060264405A1
公开(公告)日:2006-11-23
申请号:US11429582
申请日:2006-05-05
申请人: Chester Metcalf , Leonard Rozamus , Yihan Wang , R. Thomas , Dong Zou , David Berstein
发明人: Chester Metcalf , Leonard Rozamus , Yihan Wang , R. Thomas , Dong Zou , David Berstein
IPC分类号: A61K31/675 , C07F9/6527
CPC分类号: C07F9/6561 , A61K31/407 , A61K31/4745 , A61K31/675 , C07F9/6527
摘要: This invention concerns a new family of phosphorus-containing macrocycles containing various phosphonate- and phosphonate-containing moieties.
摘要翻译: 本发明涉及含有各种含膦酸盐和膦酸盐的部分的含磷大环的新家族。
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公开(公告)号:US09090561B2
公开(公告)日:2015-07-28
申请号:US13614838
申请日:2012-09-13
申请人: Yihan Wang , Xiaotian Zhu , Rajeswari Sundaramoorthi , Wei-Sheng Huang , Dong Zou , R. Mathew Thomas , Jiwei Qi , Jan Antoinette C. Romero , David C. Dalgarno , William C. Shakespeare , Tomi K. Sawyer , Chester A. Metcalf, III
发明人: Yihan Wang , Xiaotian Zhu , Rajeswari Sundaramoorthi , Wei-Sheng Huang , Dong Zou , R. Mathew Thomas , Jiwei Qi , Jan Antoinette C. Romero , David C. Dalgarno , William C. Shakespeare , Tomi K. Sawyer , Chester A. Metcalf, III
IPC分类号: C07D471/04 , A61K31/4375 , C07D213/56 , C07D213/73 , C07D213/75 , C07D213/78 , C07D217/14 , C07D217/22 , C07D237/20 , C07D237/28 , C07D239/26 , C07D241/12 , C07D241/20 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/06 , C07D413/12 , C07D417/12
CPC分类号: C07D213/56 , C07D213/73 , C07D213/75 , C07D213/78 , C07D217/14 , C07D217/22 , C07D237/20 , C07D237/28 , C07D239/26 , C07D241/12 , C07D241/20 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/06 , C07D413/12 , C07D417/12 , C07D471/04
摘要: This invention relates to compounds of the general formula: in which the variable groups are as defined herein, and to their preparation and use.
摘要翻译: 本发明涉及以下通式的化合物:其中可变基团如本文所定义,及其制备和用途。
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公开(公告)号:US20130018046A1
公开(公告)日:2013-01-17
申请号:US13614838
申请日:2012-09-13
申请人: Yihan Wang , Xiaotian Zhu , Rajeswari Sundaramoorthi , Wei-Sheng Huang , Dong Zou , R. Mathew Thomas , Jiwei Qi , Jan Antoinette C. Romero , David C. Dalgarno , William C. Shakespeare , Tomi K. Sawyer , Chester A. Metcalf, III
发明人: Yihan Wang , Xiaotian Zhu , Rajeswari Sundaramoorthi , Wei-Sheng Huang , Dong Zou , R. Mathew Thomas , Jiwei Qi , Jan Antoinette C. Romero , David C. Dalgarno , William C. Shakespeare , Tomi K. Sawyer , Chester A. Metcalf, III
IPC分类号: A61K31/4439 , C07D403/12 , A61K31/506 , C07D401/12 , A61K31/496 , C07D471/04 , A61K31/4375 , C07D413/12 , A61K31/4725 , A61K31/502 , A61K31/497 , C07D498/04 , A61K31/5383 , A61K31/551 , A61K31/5377 , A61K31/53 , A61P35/00 , C07D401/14
CPC分类号: C07D213/56 , C07D213/73 , C07D213/75 , C07D213/78 , C07D217/14 , C07D217/22 , C07D237/20 , C07D237/28 , C07D239/26 , C07D241/12 , C07D241/20 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/06 , C07D413/12 , C07D417/12 , C07D471/04
摘要: This invention relates to compounds of the general formula: in which the variable groups are as defined herein, and to their preparation and use.
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