利索-全球专利检索

  1. 登录
  2. 注册

搜索结果

12 条记录 (耗时 0.022 秒)

    ANTIFUNGAL 4-SUBSTITUTED 5,6-DIHYDRO-4H-PYRROLO [1,2-a][1,4]BENZODIAZEPINES
    1.
    发明申请
    ANTIFUNGAL 4-SUBSTITUTED 5,6-DIHYDRO-4H-PYRROLO [1,2-a][1,4]BENZODIAZEPINES 有权
    反式4取代的5,6-二氢-4H-吡咯并[1,2-a] [1,4]苯并咪唑

    公开(公告)号：US20070232593A1

    公开(公告)日：2007-10-04

    申请号：US11680700

    申请日：2007-03-01

    申请人： Terence Gilkerson ,  Roger Nash ,  Jozef Van Gestel ,  Lieven Meerpoel

    发明人： Terence Gilkerson ,  Roger Nash ,  Jozef Van Gestel ,  Lieven Meerpoel

    IPC分类号： A61K31/55 ,  C07D487/12

    CPC分类号： C07D487/04 ,  A61K31/55 ,  A61K31/551

    摘要： The present invention concerns compounds for use as a medicine having the formula the N-oxide forms, the salts, the quaternary amines and stereochemically isomeric forms thereof, wherein R1 represents hydrogen, C1-6alkyl, C1-4alkylthio, C1-4alkyloxy, or halo; R2 represents hydrogen or C1-6alkyl; R3 represents phenyl substituted with halo, cyano, C1-4alkyloxy, C1-4alkylthio, C1-6alkyl, haloC1-6alkyl; 2-thienyl; or 3-thienyl, R4 represents hydrogen; or R2 and R4 form an extra bond, which are active against dermatophytes, and their preparation; it further relates to compositions comprising them, as well as their use as a medicine.

    摘要翻译： 本发明涉及用作具有N-氧化物形式的药物的化合物，其盐，季胺和立体化学异构形式，其中R 1表示氢，C 1〜 C 1 -C 6烷基，C 1-4烷基硫基，C 1-4烷基氧基或卤素; R 2表示氢或C 1-6烷基; R 3表示被卤素，氰基，C 1-4烷氧基，C 1-4烷基硫基，C 1-6烷基取代的苯基 烷基，卤代C 1-6烷基; 2-噻吩基; 或3-噻吩基，R 4表示氢; 或R 2和R 4形成对皮肤癣菌有活性的额外的结合，及其制备; 它还涉及包含它们的组合物以及它们作为药物的用途。

    Antifungal 4-substituted 5,6-dihydro-4h-pyrrolo[1,2-a][1,4] benzodiazepines
    2.
    发明授权
    Antifungal 4-substituted 5,6-dihydro-4h-pyrrolo[1,2-a][1,4] benzodiazepines 有权
    抗真菌剂4-取代的5,6-二氢-4H-吡咯并[1,2-a] [1,4]苯并二氮杂卓

    公开(公告)号：US07202240B2

    公开(公告)日：2007-04-10

    申请号：US10399596

    申请日：2001-10-17

    申请人： Terence Gilkerson ,  Roger John Nash ,  Jozel Frans Elisabetha Van Gestel ,  Lieven Meerpoel

    发明人： Terence Gilkerson ,  Roger John Nash ,  Jozel Frans Elisabetha Van Gestel ,  Lieven Meerpoel

    IPC分类号： A61K31/55 ,  A61P31/10 ,  C07D487/04

    CPC分类号： C07D487/04 ,  A61K31/55 ,  A61K31/551

    摘要： The present invention concerns compounds for use as a medicine having the formula (I), the N-oxide forms, the salts, the quaternary amines and stereochemically isomeric forms thereof, wherein R1 represents hydrogen, C1-6 alkyl, C1-4alkylthio, C1-4alkyloxy, or halo; R2 represents hydrogen or C1-6alkyl; R3 represents phenyl substituted with halo, cyano, C1-4alkyloxy, C1-4alkylthio, C1-6alkyl, haloC1-6alkyl; 2-thienyl; or 3-thienyl, R4 represents hydrogen; or R2 and R4 form an extra bond, which are active against dermatophytes, and their preparation; it further relates to compositions comprising them, as well as their use as a medicine.

    摘要翻译： 本发明涉及用作具有式（I）的药物，N-氧化物形式，其盐，季胺及其立体化学异构形式的化合物，其中R 1表示氢， C 1-4烷基，C 1-4烷基硫基，C 1-4烷基氧基或卤素; R 2表示氢或C 1-6烷基; R 3表示被卤素，氰基，C 1-4烷氧基，C 1-4烷基硫基，C 1-6烷基取代的苯基 烷基，卤代C 1-6烷基; 2-噻吩基; 或3-噻吩基，R 4表示氢; 或R 2和R 4形成对皮肤癣菌有活性的额外的结合，及其制备; 它还涉及包含它们的组合物以及它们作为药物的用途。

    Antifungal 4-substituted 5,6-dihydro-4H-pyrrolo [1,2-a][1,4]benzodiazepines
    3.
    发明授权
    Antifungal 4-substituted 5,6-dihydro-4H-pyrrolo [1,2-a][1,4]benzodiazepines 有权
    抗真菌4-取代的5,6-二氢-4H-吡咯并[1,2-a] [1,4]苯并二氮杂卓

    公开(公告)号：US07820650B2

    公开(公告)日：2010-10-26

    申请号：US11680700

    申请日：2007-03-01

    申请人： Terence Gilkerson ,  Roger John Nash ,  Jozef Frans Elisabetha Van Gestel ,  Lieven Meerpoel

    发明人： Terence Gilkerson ,  Roger John Nash ,  Jozef Frans Elisabetha Van Gestel ,  Lieven Meerpoel

    IPC分类号： A61P31/10 ,  A61K31/55 ,  C07D487/04

    CPC分类号： C07D487/04 ,  A61K31/55 ,  A61K31/551

    摘要： The present invention concerns compounds for use as a medicine having the formula the N-oxide forms, the salts, the quaternary amines and stereochemically isomeric forms thereof, wherein R1 represents hydrogen, C1-6alkyl, C1-4alkylthio, C1-4alkyloxy, or halo; R2 represents hydrogen or C1-6alkyl; R3 represents phenyl substituted with halo, cyano, C1-4alkyloxy, C1-4alkylthio, C1-6alkyl, haloC1-6alkyl; 2-thienyl; or 3-thienyl, R4 represents hydrogen; or R2 and R4 form an extra bond, which are active against dermatophytes, and their preparation; it further relates to compositions comprising them, as well as their use as a medicine.

    摘要翻译： 本发明涉及用作具有N-氧化物形式的药物的化合物，其盐，季胺和立体化学异构形式，其中R 1表示氢，C 1-6烷基，C 1-4烷硫基，C 1-4烷氧基或卤素 ; R 2表示氢或C 1-6烷基; R 3表示被卤素，氰基，C 1-4烷氧基，C 1-4烷硫基，C 1-6烷基，卤代C 1-6烷基取代的苯基; 2-噻吩基; 或3-噻吩基，R 4表示氢; 或R2和R4形成额外的键，其对皮肤癣菌有活性，并且它们的制备; 它还涉及包含它们的组合物以及它们作为药物的用途。

    Herbicidal acrylonitrile derivatives
    5.
    发明授权
    Herbicidal acrylonitrile derivatives 失效
    除草丙烯腈衍生物

    公开(公告)号：US5366956A

    公开(公告)日：1994-11-22

    申请号：US026184

    申请日：1993-03-01

    申请人： Christopher J. Foster ,  Terence Gilkerson ,  Richard Stocker

    发明人： Christopher J. Foster ,  Terence Gilkerson ,  Richard Stocker

    IPC分类号： C07D213/64 ,  A01N43/40 ,  C07D213/643 ,  C07D413/06 ,  C07D213/84

    CPC分类号： C07D213/643 ,  A01N43/40

    摘要： Herbicidal compounds ##STR1## in which Q represents a group --C(O)--C(CN).dbd.CH--NR.sup.1 R.sup.2, R.sup.1 and R.sup.2 each independently represents alkyl, or together represent alkylene optionally interrupted by oxygen, m is O or m is an integer from 1 to 3 and the or each Y independently represents halogen or alkyl and n is O or n is an integer from 1 to 5 and the or each X independently represents halogen, alkyl, haloalkyl, cyanoalkyl, alkenyl, alkynyl, alkoxy, haloalkoxy, haloalkylthio, alkenyloxy, alkynyloxy, alkylthio, alkenylthio, alkynylthio, cyano, nitro, alkylsulphonyl, alkysulphinyl, sulphonamido, or phenyl optionally substituted by alkyl, haloalkyl, alkoxy or halogen.

    摘要翻译： 除草剂化合物（I）其中Q代表基团-C（O）-C（CN）= CH-NR1R2，R1和R2各自独立地表示烷基，或一起表示任选被氧中断的亚烷基，m是O或 m是1至3的整数，并且每个Y独立地表示卤素或烷基，n是0或n是1至5的整数，并且每个X独立地表示卤素，烷基，卤代烷基，氰基烷基，烯基，炔基， 烷氧基，卤代烷氧基，卤代烷硫基，烯氧基，炔氧基，烷硫基，烯硫基，炔硫基，氰基，硝基，烷基磺酰基，烷基亚磺酰基，磺酰氨基或任选被烷基，卤代烷基，烷氧基或卤素取代的苯基。

    Benzothiazinone derivatives
    8.
    发明授权
    Benzothiazinone derivatives 失效
    苯并噻嗪酮衍生物

    公开(公告)号：US4833137A

    公开(公告)日：1989-05-23

    申请号：US49245

    申请日：1987-05-13

    申请人： Terence Gilkerson ,  David C. Jennens ,  Mandy E. Coombs

    发明人： Terence Gilkerson ,  David C. Jennens ,  Mandy E. Coombs

    IPC分类号： A01N43/86 ,  A01P3/00 ,  C07D279/08 ,  C07D417/12 ,  C07D521/00

    CPC分类号： C07D417/12 ,  A01N43/86 ,  C07D279/08

    摘要： The invention provides benzothiazinone derivatives of formula ##STR1## wherein R.sub.1 represents a nitrogen-containing heteroaromatic group or a phenyl group substituted by 1 or 2 substituents selected from halogen atoms, alkyl, haloalkyl and alkoxy groups; a process for the preparation of such compounds; compositions containing them and a method of combating plant pathogenic fungi using such compositions or compounds.

    摘要翻译： 本发明提供了式I的苯并噻嗪酮衍生物，其中R 1表示含氮杂芳基或被1或2个选自卤原子，烷基，卤代烷基和烷氧基的取代基取代的苯基; 一种制备这种化合物的方法; 含有它们的组合物和使用这种组合物或化合物对抗植物致病真菌的方法。

    Herbicidal acrylonitrile derivatives
    9.
    发明授权
    Herbicidal acrylonitrile derivatives 失效
    除草丙烯腈衍生物

    公开(公告)号：US5426089A

    公开(公告)日：1995-06-20

    申请号：US293600

    申请日：1994-08-22

    申请人： Christopher J. Foster ,  Terence Gilkerson ,  Richard Stocker

    发明人： Christopher J. Foster ,  Terence Gilkerson ,  Richard Stocker

    IPC分类号： A01N43/40 ,  C07D213/64 ,  C07D213/643

    CPC分类号： C07D213/643 ,  A01N43/40

    摘要： Herbicidal compounds ##STR1## in which Q represents a group --C(O)--C(CN).dbd.CH--NR.sup.1 R.sup.2, R.sup.1 and R.sup.2 each independently represents alkyl, or together represent alkylene optionally interrupted by oxygen, m is O or m is an integer from 1 to 3 and the or each Y independently represents halogen or alkyl and n is O or n is an integer from 1 to 5 and the or each X independently represents halogen, alkyl, haloalkyl, cyanoalkyl, alkenyl, alkynyl, alkoxy, haloalkoxy, haloalkylthio, alkenyloxy, alkynyloxy, alkylthio, alkenylthio, alkynylthio, cyano, nitro, alkylsulphonyl, alkysulphinyl, sulphonamido, or phenyl optionally substituted by alkyl, haloalkyl, alkoxy or halogen.

    摘要翻译： 除草剂化合物（I）其中Q代表基团-C（O）-C（CN）= CH-NR1R2，R1和R2各自独立地表示烷基，或一起表示任选被氧中断的亚烷基，m是O或 m是1至3的整数，并且每个Y独立地表示卤素或烷基，n是0或n是1至5的整数，并且每个X独立地表示卤素，烷基，卤代烷基，氰基烷基，烯基，炔基， 烷氧基，卤代烷氧基，卤代烷硫基，烯氧基，炔氧基，烷硫基，烯硫基，炔硫基，氰基，硝基，烷基磺酰基，烷基亚磺酰基，磺酰氨基或任选被烷基，卤代烷基，烷氧基或卤素取代的苯基。

    Herbicidal carboxamide compounds
    10.
    发明授权
    Herbicidal carboxamide compounds 失效
    除草甲酰胺化合物

    公开(公告)号：US5384305A

    公开(公告)日：1995-01-24

    申请号：US787647

    申请日：1991-11-04

    申请人： Christopher J. Foster ,  Terence Gilkerson ,  Richard Stocker ,  Ian J. Gilmore

    发明人： Christopher J. Foster ,  Terence Gilkerson ,  Richard Stocker ,  Ian J. Gilmore

    IPC分类号： A01N43/40 ,  A01P13/00 ,  C07D213/79 ,  C07D213/81 ,  C07D213/83 ,  C07D213/86 ,  C07D213/56

    CPC分类号： C07D213/79 ,  C07D213/81 ,  C07D213/83 ,  C07D213/86

    摘要： Compounds of the formula ##STR1## wherein n is 1 to 5 and the/each X is hydrogen, halogen, cyano, nitro, optionally substituted alkyl or alkoxy alkenyloxy, alkynyloxy, haloalkylthio, alkenylthio or alkynylthio;m is 0 or 1 to 3 and the/each Y is halogen, alkyl or haloalkyl;Z is oxygen or sulphur;andR.sup.1 and R.sup.2 each, independently, is hydrogen, alkyl optionally substituted by halogen, hydroxy, cyano, alkoxy, alkylthio, alkoxycarbonyl, or mono- or di-alkylamino, alkenyl, alkynyl, hydroxy, alkoxy, alkenyloxy, alkynyloxy, alkoxycarbonyl, amino, mono- or di-alkylamino, alkoxycarbonylamino, arylamino, dialkylcarbamoyl, cycloalkyl, or optionally substituted cycloalkylalkyl;orR.sup.1 and R.sup.2 together form an alkylene chain optionally interrupted by oxygen, sulphur or --NR--, R being hydrogen or alkyl;are herbicides.

    摘要翻译： 式（I）的化合物，其中n为1至5，并且每个X为氢，卤素，氰基，硝基，任选取代的烷基或烷氧基烯氧基，炔氧基，卤代烷硫基，烯硫基或炔硫基; m为0或1至3，并且每个Y为卤素，烷基或卤代烷基; Z是氧或硫; 羟基，氰基，烷氧基，烷硫基，烷氧基羰基或单 - 或二 - 烷基氨基，烯基，炔基，羟基，烷氧基，烯氧基，炔氧基，烷氧基羰基，氨基 ，单 - 或二 - 烷基氨基，烷氧基羰基氨基，芳基氨基，二烷基氨基甲酰基，环烷基或任选取代的环烷基烷基; 或R 1和R 2一起形成任选被氧，硫或-NR-中断的亚烷基链，R是氢或烷基; 是除草剂。