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    Pharmaceutically useful compounds
    4.
    发明申请
    Pharmaceutically useful compounds 有权
    药用有用化合物

    公开(公告)号：US20060040869A1

    公开(公告)日：2006-02-23

    申请号：US11059086

    申请日：2005-02-07

    Applicant: Stanley Roberts ,  Maria Gabriella Santoro ,  Vasudev Jadhav ,  Alan Happe ,  Jerome Dauvergne

    Inventor： Stanley Roberts ,  Maria Gabriella Santoro ,  Vasudev Jadhav ,  Alan Happe ,  Jerome Dauvergne

    IPC: A61K38/05 ,  A61K38/04 ,  A61K31/198 ,  C07C323/39 ,  C07K5/04 ,  C07K5/06

    CPC classification number: C07C323/59 ,  C07C45/673 ,  C07C49/647 ,  C07C49/653 ,  C07C49/657 ,  C07C49/753 ,  C07C205/45 ,  C07C225/20 ,  C07C233/32 ,  C07C233/76 ,  C07C271/24 ,  C07C271/36 ,  C07C271/56 ,  C07C271/66 ,  C07C311/20 ,  C07C311/53 ,  C07C323/43 ,  C07C2601/08 ,  C07C2601/10

    Abstract: A compound of formula (I) or (II): wherein A is hydrogen or CR1R2; Y and Z are each, independently, hydrogen or a halogen; X is —NR4R5, or R7; R1 is hydrogen, or a substituted or unsubstituted alkyl or alkenyl group containing 1-4 carbon atoms; when X is —NR4R5, R2 is a substituted or unsubstituted alkyl, alkenyl, alkynyl, aryl, aralkyl aralkenyl, or aralkynyl group, that optionally includes at least one heteroatom in its carbon skeleton and contains 1-12 carbon atoms; when X is R7, R2 is an unsubstituted alkyl, alkenyl or alkynyl group, or a substituted or unsubstituted aryl, aralkyl aralkenyl, or aralkynyl group, that optionally includes at least one heteroatom in its carbon skeleton and contains 1-12 carbon atoms; R3 is a substituted or unsubstituted alkyl, alkenyl, alkynyl, aryl, aralkyl aralkenyl, or aralkynyl group, that optionally includes at least one heteroatom in its carbon skeleton and contains 1-12 carbon atoms; R4 is hydrogen, a substituted or unsubstituted alkyl, alkenyl, alkynyl, aryl, aralkyl aralkenyl, or aralkynyl group, that optionally includes at least one heteroatom in its carbon skeleton and contains 1-12 carbon atoms, —COOR8, or —COR8; R5 is hydrogen, or a substituted or unsubstituted alkyl or alkenyl group containing 1-5 carbon atoms; R7 is an unsubstituted alkyl, alkenyl, or alkynyl group, that contains 1-4 carbon atoms; and, R8 is an unsubstituted or halo-substituted alkyl, aryl, or aralkyl group, that contains 1-12 carbon atoms.

    Abstract translation: 式（I）或（II）的化合物：其中A是氢或CR 1 R 2; Y和Z各自独立地为氢或卤素; X是-NR 4 R 5或R 7; R 1是氢或含有1-4个碳原子的取代或未取代的烷基或链烯基; 当X是-NR 4 R 5时，R 2是取代或未取代的烷基，烯基，炔基，芳基，芳烷基芳烯基或芳炔基 基团，其任选地在其碳骨架中包含至少一个杂原子并且含有1-12个碳原子; 当X是R 7时，R 2是未取代的烷基，烯基或炔基，或取代或未取代的芳基，芳烷基芳烯基或芳炔基，其任选地包括在 其碳骨架中至少有一个杂原子，含有1-12个碳原子; R 3是取代或未取代的烷基，烯基，炔基，芳基，芳烷基芳烯基或芳炔基，其任选地在其碳骨架中包含至少一个杂原子并含有1-12个碳原子; R 4是氢，取代或未取代的烷基，烯基，炔基，芳基，芳烷基芳烯基或芳炔基，其任选地在其碳骨架中包含至少一个杂原子并含有1-12个碳原子， -COOR 8或-COR 8; R 5是氢或含有1-5个碳原子的取代或未取代的烷基或链烯基; R 7是含有1-4个碳原子的未取代的烷基，烯基或炔基; R 8是含有1-12个碳原子的未取代或卤素取代的烷基，芳基或芳烷基。

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