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126 条记录 (耗时 0.03 秒)

    Xanthine derivatives
    92.
    发明授权
    Xanthine derivatives 失效
    黄嘌呤衍生物

    公开(公告)号：US5756735A

    公开(公告)日：1998-05-26

    申请号：US483159

    申请日：1995-06-07

    申请人： Fumio Suzuki ,  Akio Ishii ,  Hiromi Nonaka ,  Nobuo Kosaka ,  Shunji Ichikawa ,  Junichi Shimada

    发明人： Fumio Suzuki ,  Akio Ishii ,  Hiromi Nonaka ,  Nobuo Kosaka ,  Shunji Ichikawa ,  Junichi Shimada

    IPC分类号： C07D473/06

    CPC分类号： C07D473/06

    摘要： The present invention relates to novel xanthine derivatives of the formula (I) which are selectively antagonistic to an adenosine A.sub.2 receptor, and pharmaceutically acceptable salts thereof. Formula (I): ##STR1## In the formula, R.sup.1 and R.sup.2 are the same or different and each represents a hydrogen atom, a propyl group, a butyl group or an allyl group; R.sup.3 represents a hydrogen atom or a lower alkyl group; Y.sup.1 and Y.sup.2 are the same or different and each represents a hydrogen atom or a methyl group; and Z represents a substituted or unsubstituted phenyl group, a pyridyl group, an imidazolyl group, a furyl group or a thienyl group.

    摘要翻译： 本发明涉及对腺苷A2受体选择性拮抗的式（I）的新颖黄嘌呤衍生物及其药学上可接受的盐。 式（I）：（I）式中，R 1和R 2相同或不同，表示氢原子，丙基，丁基或烯丙基; R3表示氢原子或低级烷基; Y1和Y2相同或不同，各自表示氢原子或甲基; Z表示取代或未取代的苯基，吡啶基，咪唑基，呋喃基或噻吩基。

    Semiconductor light emitting system
    94.
    发明授权
    Semiconductor light emitting system 失效
    半导体发光系统

    公开(公告)号：US5084895A

    公开(公告)日：1992-01-28

    申请号：US483853

    申请日：1990-02-23

    申请人： Junichi Shimada ,  Renshi Sawada

    发明人： Junichi Shimada ,  Renshi Sawada

    IPC分类号： H01S5/00 ,  G02B6/42 ,  H01S3/00 ,  H01S5/026 ,  H01S5/40

    CPC分类号： H01S5/026 ,  G02B6/42 ,  G02B6/4204 ,  H01L33/58 ,  H01S3/005 ,  H01S5/005 ,  H01S5/4025 ,  H01S5/4031

    摘要： A semiconductor light emitting element, a laser or a light emitting diode which is deposited on a first area of a semiconductor substrate, which also carries a microlens for focusing or diverging an output beam of the light emitting element on a second area of the substrate. Both the light emitting element and the microlens are deposited on a substrate through a photolithoetching process, and an alignment of an optical axis of the light emitting element and an optical axis of the microlens is accomplished in the steps of producing a light emitting semiconductor system. Thus, a semiconductor light emitting system which functions not only to generate light but also to focus or diverge the light, and is small in size and light in weight, can be obtained.

    Distributor for internal combustion engine
    96.
    发明授权
    Distributor for internal combustion engine 失效
    内燃机经销商

    公开(公告)号：US4960099A

    公开(公告)日：1990-10-02

    申请号：US404640

    申请日：1989-09-08

    申请人： Junichi Shimada ,  Kazutoshi Kobayashi ,  Norio Moriyama ,  Kazuhiko Kawakami

    发明人： Junichi Shimada ,  Kazutoshi Kobayashi ,  Norio Moriyama ,  Kazuhiko Kawakami

    IPC分类号： F02P7/00 ,  F02P7/02 ,  F02P7/04 ,  F02P7/06 ,  F02P7/08 ,  H01F38/12

    CPC分类号： H01F38/12 ,  F02P7/021 ,  F02P7/026 ,  F02P7/028 ,  F02P7/061 ,  F02P7/08

    摘要： A distributor for an internal combustion engine has a housing, a shaft inserted in the housing, a head mounted on the shaft, a cap attached to the housing so as to cover the rotor head, a signal detector accommodated in the housing, a connector projecting outside the housing, and an ignition coil accommodated in the housing. The housing has a cut-out portion formed in a side wall thereof from an abutment between the cap and the housing and extending toward the bottom of the housing for receiving the connector, and the cap and the connector are tightly engaged with the housing through a gasket. Silicon rubber is charged in the gap between the housing and the ignition coil. A heat release plate may be provided between the housing and the signal detector so that a path formed by the plate and the housing and surrounding a section of the core is electrically cut off, whereby no current flows in the path.

    摘要翻译： 用于内燃机的分配器具有壳体，插入壳体中的轴，安装在轴上的头部，附接到壳体以覆盖转子头部的盖，容纳在壳体中的信号检测器，突出的连接器 外壳外部和容纳在壳体中的点火线圈。 壳体具有形成在其侧壁中的切口部分，该切口部分从盖和壳体之间的邻接部分延伸并且朝向壳体的底部延伸以接收连接器，并且帽和连接器通过一个与壳体紧密接合 垫片 硅橡胶在壳体和点火线圈之间的间隙中充电。 可以在壳体和信号检测器之间设置放热板，使得由板和壳体形成并且围绕芯的一部分的路径被电切断，由此在路径中不流过电流。

    3-heteroaralkylthio carbacephem compounds and antibacterial pharmaceutical composition
    97.
    发明授权
    3-heteroaralkylthio carbacephem compounds and antibacterial pharmaceutical composition 失效
    3-杂芳烷硫基碳化合物和抗菌药物组成

    公开(公告)号：US4760060A

    公开(公告)日：1988-07-26

    申请号：US798320

    申请日：1985-11-15

    申请人： Kenichi Mochida ,  Takehiro Ogasa ,  Junichi Shimada ,  Tadahi Hirata ,  Kiyoshi Sato ,  Ryo Okachi

    发明人： Kenichi Mochida ,  Takehiro Ogasa ,  Junichi Shimada ,  Tadahi Hirata ,  Kiyoshi Sato ,  Ryo Okachi

    IPC分类号： A61K31/435 ,  A61K31/545 ,  A61K31/546 ,  A61P31/04 ,  C07D463/00 ,  C07D501/59 ,  C07D487/06 ,  C07D501/14

    CPC分类号： C07D463/22 ,  Y02P20/55

    摘要： Carbacephem and cephem compounds represented by the formula: ##STR1## [Wherein X is S or CH.sub.2 ; n is an integer of 1 to 5; R.sub.1 is an unsubstituted or substituted heterocyclic group (where the heterocyclic group is a 5- or 6-membered heterocyclic group having 1 to 4 of O, S and N); R.sub.2 is a group represented by the formula: ##STR2## (where R.sub.4 is an unsubstituted or substituted phenyl or 2-aminothiazolyl) or a group represented by the formula: ##STR3## (where R.sub.5 is an unsubstituted or substituted lower alkyl); R.sub.3 is hydrogen, an alkali metal, an alkaline earth metal, an organic ammonium group or an ester residue, and R.sub.1 may be a quaternary ammonium group, where --CO.sub.2 R.sub.3 represents --CO.sub.2.sup.- ] have strong antibacterial activity against Gram-positive and Gram-negative bacteria, and are useful for treating various infections.

    摘要翻译： 碳水化合物和头孢烯化合物，其由下式表示：其中X是S或CH 2; n为1〜5的整数， R1是未取代或取代的杂环基（其中杂环基是具有1至4个O，S和N的5或6元杂环基）; R2是由下式表示的基团：其中R 4是未取代或取代的苯基或2-氨基噻唑基）或由下式表示的基团：其中R5是未取代或取代的低级烷基; R3是氢，碱金属，碱土金属，有机铵基或酯残基，R1可以是季铵基，其中-CO 2 R 3表示-CO 2 - ]对革兰氏阳性和革兰氏阳性菌具有很强的抗菌活性， 阴性细菌，可用于治疗各种感染。

    3-substituted carbacepem compounds having antibacterial effect
    98.
    发明授权
    3-substituted carbacepem compounds having antibacterial effect 失效
    具有抗菌作用的3-取代的碳水化合物

    公开(公告)号：US4640919A

    公开(公告)日：1987-02-03

    申请号：US702623

    申请日：1985-02-19

    申请人： Kenichi Mochida ,  Takehiro Ogasa ,  Junichi Shimada ,  Tadashi Hirata ,  Kiyoshi Sato ,  Ryo Okachi

    发明人： Kenichi Mochida ,  Takehiro Ogasa ,  Junichi Shimada ,  Tadashi Hirata ,  Kiyoshi Sato ,  Ryo Okachi

    IPC分类号： A61K31/435 ,  A61P31/04 ,  C07D463/00 ,  C07D493/14 ,  A61K31/53 ,  C07D251/00 ,  C07D253/00

    CPC分类号： C07D493/14 ,  C07D463/22

    摘要： Carbacephem compounds represented by the formula: ##STR1## [wherein R.sub.1 is a lower alkylsulfonyloxy, unsubstituted or substituted arylsulfonyloxy, azido, cyano, carbamoyloxy, unsubstituted or substituted heterocyclic thio ("heterocyclic" means a 5- or 6-membered heterocyclic group having 1 to 4 O, S or N atoms), unsubstituted or substituted lower alkylthio, or unsubstituted or substituted arylthio group; R.sub.2 and R.sub.3 are groups frequently used in the cephalosporin chemistry] have strong antibacterial activity against Gram-positive and Gram-negative bacteria, and are useful for curing various infections.

    摘要翻译： 由下式表示的碳水化合物化合物[其中R1是低级烷基磺酰氧基，未取代或取代的芳基磺酰氧基，叠氮基，氰基，氨基甲酰氧基，未取代或取代的杂环硫基（“杂环”是指具有1 至4 O，S或N原子），未取代或取代的低级烷硫基，或未取代或取代的芳硫基; R2和R3是头孢菌素化学中经常使用的基团]对革兰氏阳性和革兰氏阴性菌具有很强的抗菌活性，可用于治疗各种感染。

    Mounting for a heat producing element of an automobile
    99.
    发明授权
    Mounting for a heat producing element of an automobile 失效
    安装汽车的发热元件

    公开(公告)号：US4349078A

    公开(公告)日：1982-09-14

    申请号：US168469

    申请日：1980-07-10

    申请人： Junichi Shimada ,  Kazutake Ogawa

    发明人： Junichi Shimada ,  Kazutake Ogawa

    IPC分类号： F01N13/08 ,  B60K13/04 ,  F01N3/28 ,  F01N13/18 ,  F16L59/06 ,  F16L59/12

    CPC分类号： F01N13/1822 ,  B60K13/04

    摘要： A mounting for a heat producing element of an automobile is described, in which elastic support members of rubber or an elastomeric material are positioned externally of a heat shield in a position in which they are exposed to unobstructed air flow beneath the automobile, and are isolated from radiant heat produced by the heat producing element in a manner minimizing the conduction of heat from said heat producing element.

    摘要翻译： 描述了一种用于汽车的发热元件的安装件，其中橡胶或弹性体材料的弹性支撑构件定位在隔热罩的外部，在它们暴露于汽车下方的无障碍空气流动的位置，并且被隔离 从由发热元件产生的辐射热以最小化来自所述发热元件的热​​传导的方式。