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154 条记录 (耗时 0.046 秒)

    Pesticidal compositions
    111.
    发明授权
    Pesticidal compositions 有权
    杀虫剂组合物

    公开(公告)号：US06867169B1

    公开(公告)日：2005-03-15

    申请号：US09716656

    申请日：2000-11-20

    申请人： Robert Senn ,  Peter Maienfisch ,  Peter Wyss

    发明人： Robert Senn ,  Peter Maienfisch ,  Peter Wyss

    IPC分类号： A01N31/14 ,  A01N33/26 ,  A01N37/34 ,  A01N41/10 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/88 ,  A01N47/12 ,  A01N47/18 ,  A01N47/22 ,  A01N47/24 ,  A01N47/34 ,  A01N47/38 ,  A01N47/40 ,  A01N51/00 ,  A01N53/04 ,  A01N53/06 ,  A01N53/08 ,  A01N53/14 ,  A01N55/00 ,  A01N57/12 ,  A01N57/14 ,  A01N57/16 ,  A01N57/28 ,  A01N57/36 ,  A01N63/00 ,  A01N63/02 ,  A61N43/72 ,  A61K31/535

    CPC分类号： A01N53/00 ,  A01N43/88 ,  A01N47/40 ,  A01N51/00 ,  A01N43/56 ,  A01N43/40 ,  A01N43/30 ,  A01N2300/00 ,  A01N57/12

    摘要： Composition for controlling insects and representatives of the order Acarina, which comprises a combination of variable amounts of one or more compounds of the formula in which A is an unsubstituted or, depending on the possibility of substitution on the ring system, mono- to tetrasubstituted, aromatic or non-aromatic monocyclic or bicyclic heterocyclic radical, in which the substituents of A can be chosen from the group consisting of C1-C3alkyl, C1-C3alkoxy, halogen, halo-C1-C3alkyl, cyclopropyl, halocyclopropyl, C2-C3alkenyl, C2-C3alkynyl, halo-C2-C3alkenyl, halo-C2-C3alkynyl, halo-C1-C3alkoxy, C1-C3alkylthio, Halo-C1-C3alkylthio, allyloxy, propargyloxy, allylthio, propargylthio, haloallyloxy, haloallylthio, cyano and nitro, R is hydrogen, C1-C6alkyl, phenyl-C1-C4alkyl, C3-C6cycloalkyl, C2-C6alkenyl or C2-C6alkynyl, and X is N—NO2 or N—CN, in the free form or in salt form, if appropriate tautomers, in the free form or salt form, and one or more of the compounds (I) to (CLXXXIV) mentioned according to the invention and at least one auxiliary. A method of controlling pests, a process for the preparation of the composition, its use and plant propagation material treated with it, and the use of the compound of the formula (A) for the preparation of the composition, are described.

    摘要翻译： 用于控制昆虫的组合物和Acarina序列的代表，其包含可变量的一种或多种下列组分的一种或多种化学式的组合：A是未取代的，或取决于在环系上取代的可能性为单 - 四取代的，芳族的或芳族的 非芳族单环或双环杂环基，其中A的取代基可以选自C 1 -C 3烷基，C 1 -C 3烷氧基，卤素，卤代C 1 -C 3烷基，环丙基，卤代环丙基，C 2 -C 3烯基，C 2 -C 3炔基 卤代C 2 -C 3烯基，卤代C 2 -C 3炔基，卤代-C 1 -C 3烷氧基，C 1 -C 3烷硫基，卤代C 1 -C 3烷硫基，烯丙氧基，炔丙氧基，烯丙硫基，炔丙硫基，卤代烯氧基，卤代烯硫基，氰基和硝基， C 6烷基，苯基-C 1 -C 4烷基，C 3 -C 6环烷基，C 2 -C 6烯基或C 2 -C 6炔基，X为N-NO 2或N-CN，以游离形式或盐形式，如果合适的互变异构体以游离形式或盐形式 ，和一种或多种化合物（I）至（CLXXXIV） 本发明的方法和至少一种辅助剂。一种防治害虫的方法，用其制备组合物，其用途和植物繁殖材料的方法，以及式（A）化合物在制备中的用途 的描述。

    Oxadiazine derivatives
    112.
    发明授权
    Oxadiazine derivatives 失效
    恶二嗪衍生物

    公开(公告)号：US06627753B1

    公开(公告)日：2003-09-30

    申请号：US09669209

    申请日：2000-09-25

    申请人： Peter Maienfisch ,  Laurenz Gsell

    发明人： Peter Maienfisch ,  Laurenz Gsell

    IPC分类号： C07D27304

    CPC分类号： C07D413/06 ,  A01N47/40 ,  A01N51/00 ,  C07D273/00 ,  C07D273/04 ,  C07D417/06

    摘要： Compounds of the formula in which A is an unsubstituted or mono- to tetrasubstituted, aromatic or non-aromatic, monocyclic or bicyclic heterocyclic radical, where one to two of the substituents of A can be selected from the group consisting of halo-C1-C3alkyl, cyclopropyl, halocyclopropyl, C2-C3alkenyl, C2-C3alkynyl, halo-C2-C3alkenyl, halo-C2-C3alkynyl, halo-C1-C3alkoxy, C1-C3alkylthio, halo-C1-C3alkylthio, allyloxy, propargyloxy, allylthio, propargylthio, haloallyloxy, haloallylthio, cyano and nitro, and one to four of the substituents of A can be selected from the group consisting of C1-C3alkyl, C1-C3alkoxy and halogen; R is hydrogen, C1-C6alkyl, phenyl-C1-C4alkyl, C3-C6cycloalkyl, C2-C6alkenyl or C2-C6alkynyl; and X is N—NO2 or N—CN, and, if appropriate, tautomers thereof, in each case in free form or in salt form, can be used as agrochemical active ingredients and can be prepared in a manner known per se.

    摘要翻译： 其中A是未取代或单取代或单取代的芳香族或非芳香族单环或双环杂环基的化合物，其中A的一个至两个取代基可以选自卤代-C 1 -C 3烷基，环丙基 卤代环丙基，C 2 -C 3烯基，C 2 -C 3炔基，卤代-C 2 -C 3烯基，卤代-C 2 -C 3炔基，卤代-C 1 -C 3烷氧基，C 1 -C 3烷硫基，卤代C 1 -C 3烷硫基，烯丙氧基，炔丙氧基，烯丙硫基，炔丙硫基，卤代烯氧基，卤代烯硫基 氰基和硝基，A至1-4个取代基可以选自C 1 -C 3烷基，C 1 -C 3烷氧基和卤素; R 2是氢，C 1 -C 6烷基，苯基-C 1 -C 4烷基，C 3 -C 6环烷基， C 2 -C 6烯基或C 2 -C 6炔基; 且X是N-NO 2或N-CN，并且如果合适，其互变异构体在各种情况下以游离形式或盐形式可用作农业化学活性成分，并且可以以本身已知的方式制备。

    Preparation of thiazoles
    113.
    发明授权
    Preparation of thiazoles 失效
    噻唑的制备

    公开(公告)号：US06548676B1

    公开(公告)日：2003-04-15

    申请号：US09331433

    申请日：1999-06-18

    申请人： Thomas Pitterna ,  Henry Szczepanski ,  Peter Maienfisch ,  Ottmar Franz Hüter ,  Thomas Rapold ,  Marcel Senn ,  Thomas Göbel ,  Anthony Cornelius O'Sullivan

    发明人： Thomas Pitterna ,  Henry Szczepanski ,  Peter Maienfisch ,  Ottmar Franz Hüter ,  Thomas Rapold ,  Marcel Senn ,  Thomas Göbel ,  Anthony Cornelius O'Sullivan

    IPC分类号： C07D27732

    CPC分类号： C07D277/32 ,  C07D277/16 ,  C07D277/36 ,  C07D277/70 ,  C07D277/74

    摘要： Described is a process for the preparation of a compound of formula (I) wherein R is unsubstituted or substituted C1-C12alkyl, C2-C4alkenyl, C2-C4alkynyl, C3-C6cycloalkyl, aryl or heteroaryl, or —SR1; R1 is unsubstituted or substituted C1-C12alkyl, C2-C4alkenyl, C2-C4alkynyl, cycloalkyl, aryl or heteroaryl; and X is a leaving group; which comprises: a) reacting a compound of formula (II) wherein R is as defined for formula (I), with a water-removing reagent; or b) for the preparation of a compound of formula (I) wherein X is halogen or a sulfonate, reacting a compound of the formula (III) wherein R is as defined for formula (I), with a halogenating or a sulfonylating agent; or c) for the preparation of a compound of formula (I) wherein X is halogen, reacting a compound of formula (IV) wherein R is as defined for formula (I); and wherein R2 and R3 are for example H, C1-C6alkyl, C3-C6cycloalkyl, phenyl or benzyl; with a compound of the formula halogen-C(═O)—O—C1-C8alkyl, halogen-C(═O)—O-aryl or halogen-C(═O)—O-benzyl. Intermediates for the preparation of the synthesis of compounds (II) to (IV) and method of the preparation thereof.

    摘要翻译： 描述了制备式（I）化合物的方法，其中R是未取代的或取代的C 1 -C 12烷基，C 2 -C 4烯基，C 2 -C 4炔基，C 3 -C 6环烷基，芳基或杂芳基或-SR 1; R1是未取代的或取代的C1-C12烷基，C2-C4链烯基，C2-C4炔基，环烷基，芳基或杂芳基; X为离去群; 其包括：a）使其中R如式（I）所定义的式（II）化合物与除水试剂反应; 或者b）用于制备其中X为卤素或磺酸盐的式（I）化合物，其中R为式（I）所定义的式（III）化合物与卤化剂或磺酰化剂反应; 或c）用于制备其中X为卤素的式（I）化合物，其中R为式（I）所定义的式（IV）化合物; 并且其中R 2和R 3是例如H，C 1 -C 6烷基，C 3 -C 6环烷基，苯基或苄基; 与卤素-C（= O）-O-C 1 -C 8烷基，卤素-C（= O）-O-芳基或卤素-C（= O）-O-苄基的化合物反应。 用于制备化合物（II）至（IV）的合成的中间体及其制备方法。

    Method for producing nitroguanidine derivatives
    114.
    发明授权
    Method for producing nitroguanidine derivatives 失效
    制备硝基胍衍生物的方法

    公开(公告)号：US06252072B1

    公开(公告)日：2001-06-26

    申请号：US09445608

    申请日：1999-12-08

    申请人： Peter Maienfisch ,  Hansjürg Widmer

    发明人： Peter Maienfisch ,  Hansjürg Widmer

    IPC分类号： C07D23104

    CPC分类号： C07D213/89 ,  C07D213/61 ,  C07D277/28 ,  C07D307/14 ,  C07D403/06

    摘要： A process for the preparation of compounds of formula is described, wherein R1 is hydrogen or C1-C4-alkyl; R2 is hydrogen, C1-C6-alkyl, C3-C6-cycloalkyl or a radical —CH2B; A is an unsubstituted or mono- to penta-substituted, aromatic or non-aromatic, monocyclic to bicyclic heterocyclic radical; and B is phenyl, 3-pyridyl or thiazolyl, which are optionally substituted by one to rhee substituents; by means of the hydrolysis of a compound of formula wherein R1, R2 and A have the same significances as given for formula (I), and R3 signifies unsubstituted or substituted C1-C10-alkyl, C3-C6-cycloalkyl, phenyl or benzyl; whereby the reaction is carried out at a pH value of between 7 and 14, as well as starting materials for carrying out the process. The compounds of formula (I) are suitable as intermediates in the preparation of pesticidal compositions.

    摘要翻译： 一种制备式中化合物的方法，其中R 1是氢或C 1 -C 4 - 烷基; R 2是氢，C 1 -C 6烷基，C 3 -C 6环烷基或基团-CH 2 B; A是未取代的或单 - 五取代的，芳族的或非芳香的单环到双环杂环基; 和B是苯基，3-吡啶基或噻唑基，它们任选地被一个取代基取代;通过水解式I的化合物，R 2和A具有与式（I）给出的相同的含义，并且R 3表示 未取代或取代的C 1 -C 10 - 烷基，C 3 -C 6 - 环烷基，苯基或苄基; 由此反应在7-14之间的pH值下进行，以及用于进行该方法的起始原料。式（I）化合物适合作为制备杀虫剂组合物的中间体。

    Oxadiazine derivatives
    116.
    发明授权
    Oxadiazine derivatives 有权

    公开(公告)号：US6022871A

    公开(公告)日：2000-02-08

    申请号：US252541

    申请日：1999-02-18

    申请人： Peter Maienfisch ,  Laurenz Gsell

    发明人： Peter Maienfisch ,  Laurenz Gsell

    IPC分类号： A01N43/88 ,  C07D273/04 ,  C07D417/06

    CPC分类号： A01N51/00 ,  A01N47/40 ,  C07D273/04 ,  C07D413/06 ,  C07D417/06

    摘要： Compounds of the formula ##STR1## in which A is an unsubstituted or mono- to tetrasubstituted, aromatic or non-aromatic, monocyclic or bicyclic heterocyclic radical, where one to two of the substituents of A can be selected from the group consisting of halo-C.sub.1 -C.sub.3 alkyl, cyclopropyl, halocyclopropyl, C.sub.2 -C.sub.3 alkenyl, C.sub.2 -C.sub.3 alkynyl, halo-C.sub.2 -C.sub.3 alkenyl, halo-C.sub.2 -C.sub.3 alkynyl, halo-C.sub.1 -C.sub.3 alkoxy, C.sub.1 -C.sub.3 alkylthio, halo-C.sub.1 -C.sub.3 alkylthio, allyloxy, propargyloxy, allylthio, propargylthio, haloallyloxy, haloallylthio, cyano and nitro, and one to four of the substituents of A can be selected from the group consisting of C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 alkoxy and halogen;R is hydrogen, C.sub.1 -C.sub.6 alkyl, phenyl-C.sub.1 -C.sub.4 alkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.2 -C.sub.6 alkenyl or C.sub.2 -C.sub.6 alkynyl; andX is N--NO.sub.2 or N--CN,and, if appropriate, tautomers thereof, in each case in free form or in salt form, can be used as agrochemical active ingredients and can be prepared in a manner known per se.

    Microbial process for the preparation of milbemycin derivatives
    119.
    发明授权
    Microbial process for the preparation of milbemycin derivatives 失效
    微生物制备米尔倍霉素衍生物的方法

    公开(公告)号：US5183749A

    公开(公告)日：1993-02-02

    申请号：US496183

    申请日：1990-03-20

    申请人： Gerado Ramos ,  Oreste Ghisalba ,  Hans-Peter Schar ,  Bruno Frei ,  Peter Maienfisch ,  Anthony C. O'Sullivan

    发明人： Gerado Ramos ,  Oreste Ghisalba ,  Hans-Peter Schar ,  Bruno Frei ,  Peter Maienfisch ,  Anthony C. O'Sullivan

    IPC分类号： A01N49/00 ,  C07H19/01 ,  C12P17/18

    CPC分类号： C07H19/01 ,  A01N49/00 ,  C12P17/181 ,  C12R1/525 ,  C12R1/685 ,  Y10S435/822 ,  Y10S435/886 ,  Y10S435/911 ,  Y10S435/917

    摘要： The present invention relates to a one-step microbial process for the preparation of 13.beta.-hydroxy- or 14,15-epoxy-milbemycins of the following formulae I and II ##STR1## in which R.sub.1 and R.sub.1 ' represent methyl, ethyl, isopropyl or sec.-butyl or represent the group ##STR2## in which X represents methyl, ethyl or isopropyl, and A and A' represent the group ##STR3## in which R.sub.2 represents hydrogen, --C(O)-CH.sub.2 O-C(O)-CH.sub.2 CH.sub.2 -COOH or --C(O)-CH.sub.2 CH.sub.2 -COOH, or mixtures of compounds of the formulae I and II, which process comprises bringing a milbemycin of the formula III ##STR4## dissolved in a liquid phase, in which R.sub.3 represents R.sub.1 or R.sub.1 ' and R.sub.4 represents A or A', and R.sub.1, R.sub.1 ', A and A' have the meanings given for formulae I and II, into contact with a microorganism that is capable of 13.beta.-hydroxylation or 14,15-epoxidation or of both reactions, or into contact with active constituents thereof. The microorganism or its active constituents may be either in free form or immobilized form.

    摘要翻译： 本发明涉及一种用于制备下式I和II的13β-羟基或14,15-环氧 - 米尔倍霉素的一步微生物方法。其中R1 并且R 1'表示甲基，乙基，异丙基或仲丁基，或表示其中X表示甲基，乙基或异丙基的基团，A和A'表示其中R 2表示氢的基团，-C （O）-CH 2 O-C（O）-CH 2 CH 2 -COOH或-C（O）-CH 2 CH 2 -COOH，或式I和II化合物的混合物，该方法包括使式III的米尔倍霉素 III）溶解在液相中，其中R3表示R1或R1'，R4表示A或A'，R1，R1'，A和A'具有式I和II给出的含义，与微生物接触， 能够进行13β-羟基化或14,15-环氧化或两种反应，或与其活性成分接触。 微生物或其活性成分可以是游离形式或固定化形式。

    Pest control agents
    120.
    发明授权
    Pest control agents 失效
    害虫控制剂

    公开(公告)号：US5179094A

    公开(公告)日：1993-01-12

    申请号：US672763

    申请日：1991-03-19

    申请人： Odd Kristiansen ,  Manfred Boger ,  Haukur Kristinsson ,  Peter Maienfisch

    发明人： Odd Kristiansen ,  Manfred Boger ,  Haukur Kristinsson ,  Peter Maienfisch

    IPC分类号： A01N43/707 ,  C07D401/12

    CPC分类号： C07D401/12 ,  A01N43/707

    摘要： There are disclosed novel substituted N-amino-1,2,4-triazinones of formula I ##STR1## wherein R.sub.1 is C.sub.1 -C.sub.12 alkyl or C.sub.3 -C.sub.7 cycloalkyl,R.sub.2 and R.sub.3 are each independently of the other hydrogen or C.sub.1 -C.sub.6 alkyl,R.sub.4, R.sub.5, R.sub.6 and R.sub.7 are each independently of one another hydrogen, halogen, C.sub.1 -C.sub.3 alkyl, ##STR2## C.sub.1 -C.sub.3 alkoxy or C.sub.1 -C.sub.3 alkylthio, and n is 0 or 1, or a salt thereof, with the proviso that n is 1, if simultaneously the pyridine ring is attached via the 3-position to the methylidene group and R.sub.4, R.sub.5, R.sub.6 and R.sub.7 are each hydrogen; their use in pest control and pesticidal compositions which contain a compound of formula I as active component. The preferred utility is the control of pests of animals and plants.

    摘要翻译： 公开了式I（I）的新的取代的N-氨基-1,2,4-三嗪酮，其中R 1是C 1 -C 12烷基或C 3 -C 7环烷基，R 2和R 3各自独立地是另一个氢或C 1 -C 6烷基 ，R 4，R 5，R 6和R 7各自独立地为氢，卤素，C 1 -C 3烷基，C 1 -C 3烷氧基或C 1 -C 3烷硫基，n为0或1，或其盐，条件是n 是1，如果同时吡啶环通过3-位连接到亚甲基上，并且R4，R5，R6和R7各自为氢; 它们在害虫控制中的用途和含有式I化合物作为活性成分的杀虫组合物。 优选的效用是控制动物和植物的害虫。