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    Substituted guanidine derivatives
    24.
    发明授权
    Substituted guanidine derivatives 失效
    取代的胍衍生物

    公开(公告)号：US06503912B1

    公开(公告)日：2003-01-07

    申请号：US09582679

    申请日：2000-06-28

    Applicant: Klaus Wagner ,  Christoph Erdelen ,  Wolfram Andersch ,  Ulrike Wachendorff-Neumann ,  Andreas Turberg ,  Norbert Mencke

    Inventor： Klaus Wagner ,  Christoph Erdelen ,  Wolfram Andersch ,  Ulrike Wachendorff-Neumann ,  Andreas Turberg ,  Norbert Mencke

    IPC: C07D40106

    CPC classification number: C07D401/06 ,  A01N47/40 ,  A01N51/00 ,  C07D417/06

    Abstract: The present application relates to novel guanidine derivatives of the formula (I) in which R1 represents a five- or six-membered heterocyclic group; R2 represents hydrogen or alkyl, R3 represents the groupings —OR4, —OCOR5, —OCOOR6, —OCONR7R8 and —OSO2R9, where R4, R5 and R6 independently of one another represent alkyl, alkoxyalkyl, halogenoalkyl, alkenyl, alkinyl, alkylaminoalkyl, dialkylaminoalkyl, optionally substituted cycloalkyl and in each case optionally substituted phenyl or benzyl, R7 and R8 independently of one another represent hydrogen, alkyl, alkenyl and in each case optionally substituted phenyl or benzyl and R9 represents alkyl or optionally substituted phenyl, A represents the groupings —CH2CH2—, (CH2)3 and —CH═CH— and z represents cyano or nitro, with the proviso that, if Z represents NO2 and A represents —CH2CH2—, the radical R2 represents hydrogen; and the compound of the formula (I) in which R1 R2 H, R3 OCH3, A —CH2CH2— and Z NO2 is excluded. The compounds serve for controlling insects, arachnids and nematodes.

    Abstract translation: 本申请涉及式（I）的新型胍衍生物，其中R 1表示五元或六元杂环基; R 2表示氢或烷基，R 3表示基团-OR 4，-OCOR 5，-OCOOR 6，-OCONR 7 R 8和 - OSO 2 R 9，其中R 4，R 5和R 6彼此独立地表示烷基，烷氧基烷基，卤代烷基，烯基，炔基，烷基氨基烷基，二烷基氨基烷基，任选取代的环烷基，并且在每种情况下任选取代的苯基或苄基，R 7和R 8彼此独立地表示氢，烷基 ，烯基，并且在每种情况下为任选取代的苯基或苄基，R 9表示烷基或任选取代的苯基，A表示-CH 2 CH 2 - ，（CH 2）3和-CH = CH-并且Z表示氰基或硝基，条件是如果Z 表示NO 2，A表示-CH 2 CH 2 - ，基团R 2表示氢; 和其中R 1 R 2 H，R 3 OCH 3，A -CH 2 CH 2 - 和Z NO 2的式（I）化合物被排除。该化合物用于防治昆虫，蜘蛛和线虫。

    Octacyclodepsipeptides having an endoparasiticidal action
    25.
    发明授权
    Octacyclodepsipeptides having an endoparasiticidal action 失效
    具有内寄生性杀伤作用的Octacyclodepsipeptide

    公开(公告)号：US06369028B1

    公开(公告)日：2002-04-09

    申请号：US08246029

    申请日：1994-05-19

    Applicant: Jürgen Scherkenbeck ,  Peter Jeschke ,  Hans-Georg Lerchen ,  Hermann Hagemann ,  Achim Harder ,  Norbert Mencke ,  Andrew Plant

    Inventor： Jürgen Scherkenbeck ,  Peter Jeschke ,  Hans-Georg Lerchen ,  Hermann Hagemann ,  Achim Harder ,  Norbert Mencke ,  Andrew Plant

    IPC: A61K3800

    CPC classification number: C07D273/00 ,  C07C235/12 ,  C07C235/34

    Abstract: The present invention relates to compounds of the general formula (I) in which R1, R2, R11 and R12 represent the same or different radicals selected from the group of C1-8-alkyl, C1-8-halogenoalkyl, C3-6-cycloalkyl, aralkyl or aryl, R3, R5, R7, R9, represent the same or different radicals selected from the group of hydrogen or straight-chain C1-5-alkyl or branched C4-7-alkyl which may optionally be substituted by hydroxyl, C1-4-alkoxy, carboxyl  carboxamide,  imidazolyl, indolyl, guanidino, —SH or C1-4-alkylthio, and furthermore represents aryl, aralkyl or heteroarylmethyl which may be substituted by halogen, hydroxyl, C1-4-alkyl, C1-4-alkoxy, nitro or a —NR13R14 group in which R13 and R14 independently from each other represent hydrogen or alkyl or together with the adjoining nitrogen atom forms a 5, 6 or 7-membered ring which is optionally interrupted by O, S or N and which is optionally C1-4-alkyl substituted, R4, R6, R8, R10 represent the same or different radicals selected from the group of hydrogen, straight-chain C1-5-alkyl and represents isopropyl, sec.-butyl, t-butyl, C2-6-alkenyl, C3-7-cycloalkyl, which may optionally be substituted by hydroxyl, C1-4-alkoxy, carboxyl, carboxamide, imidazolyl, indolyl, guanidino, SH or C1-4-alkylthio and represent aryl, aralkyl or heteroarylmethyl which may be substituted by halogen, hydroxyl, C1-4-alkyl, C1-4-alkoxy, and stereoisomers thereof, to processes for their preparation and to their use as endoparasiticides.

    Abstract translation: 本发明涉及通式（I）的化合物，其中R 1，R 2，R 11和R 12表示相同或不同的选自C 1-8 - 烷基，C 1-8 - 卤代烷基，C 3-6 - 环烷基， 芳烷基或芳基，R 3，R 5，R 7，R 9表示相同或不同的选自氢或直链C 1-5烷基或支链C 4-7 - 烷基的基团，其可任选被羟基，C 1-4 烷氧基，羧基羧酰胺，咪唑基，吲哚基，胍基，-SH或C 1-4 - 烷硫基，此外表示可被卤素，羟基，C 1-4 - 烷基，C 1-4 - 烷氧基，硝基取代的芳基，芳烷基或杂芳基甲基 或-NR 13 R 14基团，其中R 13和R 14彼此独立地表示氢或烷基或与相邻的氮原子一起形成可选地被O，S或N中断的5,6或7-元环，并且其任选地为C1 R 4，R 6，R 8，R 10表示选自该基团的相同或不同的基团 的氢，直链C1-5 - 烷基，代表异丙基，仲丁基，叔丁基，C 2-6 - 烯基，C 3-7 - 环烷基，其可任选被羟基，C 1-4 - 烷氧基， 羧基，羧酰胺，咪唑基，吲哚基，胍基，SH或C 1-4 - 烷硫基，代表可被卤素，羟基，C 1-4 - 烷基，C 1-4 - 烷氧基及其立体异构体取代的芳基，芳烷基或杂芳基甲基， 其制备方法及其作为内寄生物杀虫剂的用途。

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