Substituted guanidine derivatives
    7.
    发明授权
    Substituted guanidine derivatives 失效
    取代的胍衍生物

    公开(公告)号:US06503912B1

    公开(公告)日:2003-01-07

    申请号:US09582679

    申请日:2000-06-28

    IPC分类号: C07D40106

    摘要: The present application relates to novel guanidine derivatives of the formula (I) in which R1 represents a five- or six-membered heterocyclic group; R2 represents hydrogen or alkyl, R3 represents the groupings —OR4, —OCOR5, —OCOOR6, —OCONR7R8 and —OSO2R9, where R4, R5 and R6 independently of one another represent alkyl, alkoxyalkyl, halogenoalkyl, alkenyl, alkinyl, alkylaminoalkyl, dialkylaminoalkyl, optionally substituted cycloalkyl and in each case optionally substituted phenyl or benzyl, R7 and R8 independently of one another represent hydrogen, alkyl, alkenyl and in each case optionally substituted phenyl or benzyl and R9 represents alkyl or optionally substituted phenyl, A represents the groupings —CH2CH2—, (CH2)3 and —CH═CH— and z represents cyano or nitro, with the proviso that, if Z represents NO2 and A represents —CH2CH2—, the radical R2 represents hydrogen; and the compound of the formula (I) in which R1 R2 H, R3 OCH3, A —CH2CH2— and Z NO2 is excluded. The compounds serve for controlling insects, arachnids and nematodes.

    摘要翻译: 本申请涉及式(I)的新型胍衍生物,其中R 1表示五元或六元杂环基; R 2表示氢或烷基,R 3表示基团-OR 4,-OCOR 5,-OCOOR 6,-OCONR 7 R 8和 - OSO 2 R 9,其中R 4,R 5和R 6彼此独立地表示烷基,烷氧基烷基,卤代烷基,烯基,炔基,烷基氨基烷基,二烷基氨基烷基,任选取代的环烷基,并且在每种情况下任选取代的苯基或苄基,R 7和R 8彼此独立地表示氢,烷基 ,烯基,并且在每种情况下为任选取代的苯基或苄基,R 9表示烷基或任选取代的苯基,A表示-CH 2 CH 2 - ,(CH 2)3和-CH = CH-并且Z表示氰基或硝基,条件是如果Z 表示NO 2,A表示-CH 2 CH 2 - ,基团R 2表示氢; 和其中R 1 R 2 H,R 3 OCH 3,A -CH 2 CH 2 - 和Z NO 2的式(I)化合物被排除。该化合物用于防治昆虫,蜘蛛和线虫。