摘要:
Oxy-phenyl-(phenyl)gycinolamides with heterocyclic substituents are prepared by reaction of the corresponding oxyphenylcarboxylic acids with heterocyclic substituents with phenylglycinol. The new substances are suitable as active compounds in medicaments, in particular in agents having an antiatherosclerotic action.
摘要:
Novel substituted 2,4-imidazolidinediones are prepared either by reaction of .alpha.-aminocarboxylic acid derivatives with appropriately substituted biphenylmethyl halides and subsequent cyclization with isocyanates or by reaction of N-benzyl-substituted .alpha.-aminocarboxylic acid derivatives with tetrazolylphenylboronic acids or by reaction of sulphonyl-substituted benzyl halides with .alpha.-aminocarboxylic acid derivatives and subsequent cyclization with isocyanates. The compounds according to the invention can be employed as active compounds in medicaments, preferably for the treatment of arterial hypertension and arteriosclerosis.
摘要:
The invention relates to phenylacetic acid derivatives of the formula ##STR1## which are substituted by a five-membered nitrogen heterocycle bonded via an N atom. They are prepared by reaction of phenylacetic acid derivatives substituted with leaving groups with the appropriate nitrogen heterocycles and can be used as active substances in medicaments for the treatment of high blood pressure and atherosclerosis.
摘要:
Pyridinylmethyl-substituted pyridines and pyridones are prepared by reacting pyridine- or pyridone-substituted halogenopyridines with tetrazolylphenylboronic acids. The substances according to the invention can be used as active compounds in medicaments, in particular for the treatment of arterial hypertension and atherosclerosis.
摘要:
Propenoyl-imidazole derivatives are prepared by reaction of appropriate imidazoylaldehydes with CH-acidic compounds and subsequent dehydration of the intermediates. The propenoyl-imidazole derivatives can be employed as active compounds in medicaments for the treatment of arterial hypertension and atherosclerosis.
摘要:
This invention relates to the use of phosphorus-containing compounds, specifically cyclic organophosphorus compounds, as carbodiimidization catalysts in the preparation of open-celled flexible polyurethane foam for the purpose of controlling foam density and providing softer foams. foams that are softer and of lower density can be prepared with significantly reduced quantities of blowing agents in comparison to foams prepared in the absence of such phosphorus-containing compounds. Additionally, use of such catalysts provides for a reduced reaction exotherm during the preparation of the foam thereby minimizing foam discoloration or scorching. Preferred phosphorus-containing compounds are the 1-alkyl-1-oxophospholenes, especially 1-methyl-1-oxophospholene.
摘要:
The present invention relates to an arrangement for the discrete-time adaptive on-off switching control of a continuous-time process with a binary switching actuator, which uses for the determination of the on-off actuating signal a prediction of a process output sequence over several future sampling intervals as reaction to a possible process input sequence that is applied to a discrete-time linear process model and which estimates and updates in every sampling interval the parameters of the process model by means of a parameter estimation device in order to adapt them to the process to be controlled, even when the process behavior changes, and which has a device for the input and change of the setpoint, the limits of the process output and the sampling time as well as a measuring device for the periodical measurement of the process input. The arrangement further comprises two alternatively working control devices one of which is active in the stationary phase and the other of which is active in the start-up phase of the process or after setpoint changes, and a switching device which activates one or the other said control device in dependence of the result of the measurement of the process output and of input current setpoint, wherein the actuator is served by the active control device.
摘要:
An electronic key for wireless operation of a lock with a housing shell for g circuit electronics, wherein the housing shell—has a battery compartment, a battery compartment cover, an emergency key which has a key stem insertable into the housing shell for mechanical operation of the lock, wherein the key stem is movable between an insertion position, in which the key stem is fitted on a key shaft of the housing shell, and an end position in which the key stem is securely accommodated in the key shaft, and a seal arranged between the housing shell and the battery compartment cover for protecting the battery against environmental influences, wherein the battery compartment cover has a bearing surface for direct contact on the key stem, and, in the end position, the key stem exerts a contact pressure force against the seal via the bearing surface of the battery compartment cover.
摘要:
The invention relates to a switching device (1) for the keyless activation or deactivation of a consumer, especially an engine or the like in a vehicle, and/or for unlocking or locking a functionally essential component of a vehicle. Said device comprises at least one switching element (3), arranged inside a housing (2), which can be actuated by an actuation element (4), thereby generating at least one switching signal for the control unit (10). The aim of the invention is to provide a switching device which consists of only few components and which is incorporated into a keyless security system in a simple manner. For this purpose, an electrode (5) is provided on the housing (2) and is connected to the control unit (10). Said electrode (5) transmits data to a mobile ID transmitter (13) and the electrode (5) allows data being transmitted to a mobile ID transmitter (13) via a capacitative coupling (32, 34). The control unit (10) transmits a first encoded and/or modulated signal to the electrode (5) when the latter receives a first switching signal from the switching element (3). The invention also relates to a security system (25) for the keyless activation or deactivation of an installation or a device, especially of a steering wheel lock or of an engine in a vehicle. Said system comprises a switching device (1) according to the invention, and a mobile ID transmitter (13), capacitative data transmission between the switching device (1) and the ID transmitter (13) being possible, and a control unit (10) which controls data transmission between the switching device (1) and the mobile ID transmitter (13).
摘要:
Methods for ad-hoc trust establishment using visual verification are described. In a first embodiment, a visual representation of a shared data is generated on two or more devices and the visual representations generated can be visually compared by a user. This method can be used to verify that the correct devices are involved in a negotiation, when pre-existing trust relationships do not exist between the devices. The visual representation may, for example, comprise a picture with a number of different elements, each representing a part of the shared data. In another embodiment, a method of secure key exchange is described in which, before sharing the keys, the parties exchange information which encapsulates the key. This information can be used subsequently to check that a party has not changed the key that they are using and prevents a man in the middle attack.