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    Pyrimidin-4-yl-3, 4-Dihydro-2H-Pyrrolo[1,2A] Pyrazin-1-one Compounds
    1.
    发明申请
    Pyrimidin-4-yl-3, 4-Dihydro-2H-Pyrrolo[1,2A] Pyrazin-1-one Compounds 有权
    嘧啶-4-基-3,4-二氢-2H-吡咯并[1,2A]吡嗪-1-酮化合物

    公开(公告)号：US20100035870A1

    公开(公告)日：2010-02-11

    申请号：US12083534

    申请日：2006-10-09

    申请人： Stuart Jones ,  Robert Westwood ,  Mark Thomas ,  Janice McLachlan ,  Kenneth Duncan ,  Fred Scaerou ,  Daniella I. Zheleva

    发明人： Stuart Jones ,  Robert Westwood ,  Mark Thomas ,  Janice McLachlan ,  Kenneth Duncan ,  Fred Scaerou ,  Daniella I. Zheleva

    IPC分类号： A61K31/506 ,  C07D487/04 ,  A61K31/538 ,  A61K31/5377 ,  A61K31/541 ,  A61P35/00 ,  A61P35/02 ,  A61P19/02 ,  A61P11/00 ,  A61P31/12 ,  C12Q1/48 ,  G01N33/53 ,  A61P25/00 ,  A61P25/28 ,  A61P17/14 ,  A61P3/10 ,  A61P27/02

    CPC分类号： C07D487/04

    摘要： The present invention relates to compounds of formula (I), or pharmaceutically acceptable salts thereof, wherein Z is NR11, NHCO, NHSO2, NHCH2, CH2, CH2CH2, or CH═CH; X is a hydrocarbyl group optionally substituted by one or more R12 groups; R10 and R11 are each independently II or alkyl; R1-R4 are each independently II or (CII2)mR12, where m is O, 1, 2, or 3; each R12 is independently (CH2)aR16, where each R16 is independently selected from O(CH2)bR13, R13, COR13, COOR13, CN, CONR13R14, NR13R14, NR13COR14, SR13, SOR13, SO2R13, NR13SO2R14, SO2OR13, SO2NR13R14, halogen, CF3, and NO2, and wherein each a is 0, 1, 2, or 3 and b is 0, 1, 2, or 3; R13 and R14 are each independently H or (CH2)nR15, where n is 0, 1, 2, or 3; and each R15 is independently selected from alkyl, cycloalkyl, heteroaryl, aralkyl, aryl and heterocycloalkyl, each of which may be optionally substituted by one or more substituents selected from halogen, OH, CN, COO-alkyl, aralkyl, SO2-alkyl, SO2-aryl, COOH, CO— alkyl, CO-aryl, NH2, NH-alkyl, N(alkyl)2, CF3, alkyl and alkoxy, wherein said alkyl and alkoxy groups may be further substituted by one or more OH groups. Further aspects of the invention relate to pharmaceutical compositions comprising compounds of formula I, and the use of compounds of formula (I) in the preparation of a medicament for treating a variety of disorders, including proliferative disorders, viral disorders, stroke, etc.

    摘要翻译： 本发明涉及式（I）化合物或其药学上可接受的盐，其中Z为NR11，NHCO，NHSO2，NHCH2，CH2，CH2CH2或CH-CH; X是任选被一个或多个R 12基团取代的烃基; R 10和R 11各自独立地为II或烷基; R1-R4各自独立地为II或（CII2）mR12，其中m为0,1,2或3; 每个R 12独立地为（CH 2）a R 16，其中每个R 16独立地选自O（CH 2）b R 13，R 13，COR 13，COOR 13，CN，CONR 13 R 14，NR 13 R 14，NR 13 COR 14，SR 13，SOR 13，SO 2 R 13，NR 13 SO 2 R 14，SO 2 R 13，SO 2 NR 13 R 14， CF 3和NO 2，并且其中每个a是0,1,2或3，b是0,1,2或3; R 13和R 14各自独立地为H或（CH 2）n R 15，其中n为0,1,2或3; 并且每个R 15独立地选自烷基，环烷基，杂芳基，芳烷基，芳基和杂环烷基，其各自可以任选被一个或多个选自卤素，OH，CN，COO-烷基，芳烷基，SO 2 - 烷基，SO 2 - 芳基，COOH，CO-烷基，CO-芳基，NH 2，NH-烷基，N（烷基）2，CF 3，烷基和烷氧基，其中所述烷基和烷氧基可进一步被一个或多个OH基取代。 本发明的其它方面涉及包含式I化合物的药物组合物，以及式（I）化合物在制备用于治疗多种病症（包括增殖性病症，病毒性疾病，中风等）的药物中的用途。

    Power Supply Systems For Electrical Devices
    2.
    发明申请
    Power Supply Systems For Electrical Devices 审中-公开
    电气设备电源系统

    公开(公告)号：US20070279011A1

    公开(公告)日：2007-12-06

    申请号：US10589105

    申请日：2005-02-11

    申请人： Stuart Jones ,  David Cross

    发明人： Stuart Jones ,  David Cross

    IPC分类号： H02J7/00

    CPC分类号： H02J7/345 ,  H01G9/14

    摘要： An electrically powered portable device, the device being other than a toothbrush, the device including means for providing a function to be performed by the device, an electrical power supply which incorporates at least one capacitor for storing electrical charge to power the device, electronic control circuitry to control electrical power drawn from the electrical power supply for driving the function providing means, and a recharge interface for recharging the electrical power supply, the recharge interface being arranged to be electrically connectable to a charging device.

    摘要翻译： 一种电动便携式设备，该设备不同于牙刷，该设备包括用于提供由该设备执行的功能的装置，包含至少一个用于存储电荷以为设备供电的电容器的电源，电子控制 用于控制从电源引出的用于驱动功能提供装置的电力的电路，以及用于对电源进行再充电的再充电接口，所述充电接口被布置成可电连接到充电装置。

    Automatic media switching apparatus and method
    7.
    发明授权
    Automatic media switching apparatus and method 失效
    自动介质切换装置及方法

    公开(公告)号：US06137802A

    公开(公告)日：2000-10-24

    申请号：US827014

    申请日：1997-03-25

    申请人： Wesley Stuart Jones ,  Louis P. Dellaverson

    发明人： Wesley Stuart Jones ,  Louis P. Dellaverson

    IPC分类号： H04L12/56 ,  H04Q11/04 ,  H04W36/14 ,  H04W36/18 ,  H04W88/02 ,  H04W88/06 ,  H04M11/00

    CPC分类号： H04W88/06 ,  H04Q11/0478 ,  H04L2012/5607 ,  H04L2012/5615 ,  H04L2012/5616 ,  H04W36/14 ,  H04W36/18

    摘要： A media switching apparatus automatically switches a user device between wired and wireless service mediums of communications networks. The switching apparatus includes a protocol stack having a network layer, a logical link control, a first set of lower layers specific to a wired service medium and a second set of lower layers specific to a wireless service medium. A selector is responsive to the availability of a wired service medium for selecting the first set of lower layers and is further responsive to the non-availability of a wired service medium and the availability of a wireless service medium for selecting the second set of lower layers.

    摘要翻译： 媒体交换设备在通信网络的有线和无线服务介质之间自动切换用户设备。 交换装置包括具有网络层，逻辑链路控制，特定于有线服务介质的第一组较低层的协议栈和对于无线服务介质特有的第二组较低层。 选择器响应于有线服务介质的可用性来选择第一组较低层，并且还响应于有线服务介质的不可用性以及用于选择第二组较低层的无线服务介质的可用性 。

    Network license server
    8.
    发明授权
    Network license server 失效
    网络许可证服务器

    公开(公告)号：US5023907A

    公开(公告)日：1991-06-11

    申请号：US252556

    申请日：1988-09-30

    申请人： Herrick J. Johnson ,  Margaret Olson ,  Stuart Jones ,  Stephanie Bodoff ,  Stephen C. Bertrand ,  Paul H. Levine

    发明人： Herrick J. Johnson ,  Margaret Olson ,  Stuart Jones ,  Stephanie Bodoff ,  Stephen C. Bertrand ,  Paul H. Levine

    IPC分类号： G06F1/00 ,  G06F21/00

    CPC分类号： G06F21/105 ,  G06F2221/2101 ,  G06F2221/2135

    摘要： A system for the management of computer programs in a computer network environment is presented. A network license server comprises a license server daemon which provides access to a computer program based on information stored in user and license databases. To track software usage, the daemon also maintains a log file which can be accessed by and interfaced with a network administration station. The network license server protects software vendors from unauthorized use of their software while permitting software programs and users to reside anywhere on the network.

    摘要翻译： 介绍了一种在计算机网络环境下管理计算机程序的系统。 网络许可证服务器包括许可证服务器守护程序，其基于存储在用户和许可证数据库中的信息来提供对计算机程序的访问。 为了跟踪软件使用情况，守护进程还维护一个日志文件，该日志文件可以由一个网络管理站访问并与其进行连接。 网络许可证服务器可以保护软件供应商免于未经授权使用其软件，同时允许软件程序和用户驻留在网络上的任何位置。

    Field replaceable management module
    10.
    发明授权
    Field replaceable management module 有权
    现场可更换管理模块

    公开(公告)号：US08427007B2

    公开(公告)日：2013-04-23

    申请号：US12711738

    申请日：2010-02-24

    申请人： Michael Jansma ,  Jeffrey Stuart Jones ,  Joseph Thomas Kramer

    发明人： Michael Jansma ,  Jeffrey Stuart Jones ,  Joseph Thomas Kramer

    IPC分类号： H02J3/38

    CPC分类号： H01R25/003 ,  G06F1/266 ,  H01R13/514 ,  H01R13/6683 ,  Y10T307/313

    摘要： Aspects of the invention are directed to a power distribution unit including a removable management module and methods for providing power using the power distribution units. According to one embodiment the power distribution unit comprises a housing having a length, a width and a depth with a front face of the housing extending across the width and along the length with the length being substantially greater than the width and the depth, and wherein the front face of the housing defines an opening to a docking space in an interior portion of the housing, a plurality of power outlets disposed on the front face of the housing, a management module configured to detect current through at least one of the plurality of power outlets, the management module being further configured and arranged to fit within the docking space, a memory component contained within the housing and configured to store operational data for the power distribution unit, and wherein the management module and the housing are configured and arranged such that the management module is removable from the docking space through the opening in the front face.

    摘要翻译： 本发明的方面涉及一种配电单元，其包括可拆卸管理模块和使用配电单元提供电力的方法。 根据一个实施例，功率分配单元包括具有长度，宽度和深度的壳体，其中壳体的前表面延伸穿过宽度并且沿长度方向延伸，其长度基本上大于宽度和深度，并且其中 壳体的前表面限定了在壳体的内部部分中的对接空间的开口，设置在壳体的前表面上的多个电源插座，管理模块，被配置为检测电流通过至少一个 电源插座，管理模块被进一步配置和布置成装配在对接空间内，容纳在外壳内并被配置为存储配电单元的操作数据的存储器组件，并且其中管理模块和壳体被配置和布置成 管理模块可以通过前面的开口从对接空间移除。