Sulfonamide derivatives, insecticides for agricultural and horticultural use, and usage thereof
    2.
    发明授权
    Sulfonamide derivatives, insecticides for agricultural and horticultural use, and usage thereof 失效
    磺酰胺衍生物,农业和园艺用杀虫剂及其用途

    公开(公告)号:US07161032B2

    公开(公告)日:2007-01-09

    申请号:US10525504

    申请日:2003-08-26

    摘要: Sulfonamide derivatives represented by general formula (I) or salts thereof; insecticides for agricultural and horticultural use containing the same as the active ingredient; and usage thereof: [wherein A is optionally substituted (C1–C6)alkylene, (C3–C6)alkenylene or the like; R1 is H, optionally substituted (C1–C6)alkyl, (C3–C6)alkenyl, (C3–C6)cycloalkyl or the like; R2, R3 and R4 are each H, (C1–C6)alkyl, (C3–C6)alkenyl or the like, or R2 and A or R2 and R1 may form a 3- to 8-membered ring which may be interrupted by one to three atoms selected from among O, S and N; Q is C or N; X and Y are each halogen, CN, NO2, (C1–C6)alkyl, (C2–C6)alkenyl or the like; m is 0 to 2; n is 0 to 3; and two adjacent Xs or Ys on the aromatic ring may be united to form a fused ring]. The compounds exhibit excellent insecticidal activity against insect pests resistant to existing pesticides even when applied in dosages lower than those of similar pesticides.

    摘要翻译: 由通式(I)表示的磺酰胺衍生物或其盐; 含有与活性成分相同的农业和园艺用杀虫剂; 及其用途:[其中A是任选取代的(C 1 -C 6 -C 6)亚烷基,(C 3 -C 6 - 亚烷基等; R 1是H,任选取代的(C 1 -C 6 -C 6)烷基,(C 3 -C 6 - (C 3 -C 6 -C 6)环烷基等;(C 3 -C 6)烷基,(C 3 -C 6 -C 6)环烷基等; R 2,R 3和R 4各自为H,(C 1 -C 6)烷基, (C 1 -C 6)烷基,(C 3 -C 6 -C 6)链烯基等,或R 2和A或R 2 R 1和R 2可以形成3至8元环,其可以被选自O,S和N中的一至三个原子间隔; Q是C或N; X和Y各自为卤素,CN,NO 2,(C 1 -C 6)烷基,(C 1 -C 6)烷基, 链烯基或类似物; m为0〜2; n为0〜3; 并且芳环上的两个相邻的X或Y可以结合形成稠环]。 该化合物对于现有农药抗性的昆虫害虫具有优异的杀虫活性,即使施用量低于类似农药的剂量。

    Sulfonamide derivatives, insecticides for agricultural and horticultural use, and usage thereof
    3.
    发明申请
    Sulfonamide derivatives, insecticides for agricultural and horticultural use, and usage thereof 失效
    磺酰胺衍生物,农业和园艺用杀虫剂及其用途

    公开(公告)号:US20060167315A1

    公开(公告)日:2006-07-27

    申请号:US10525504

    申请日:2003-08-26

    IPC分类号: C07D213/72 C07C311/30

    摘要: Sulfonamide derivatives represented by general formula (I) or salts thereof; insecticides for agricultural and horticultural use containing the same as the active ingredient; and usage thereof: [wherein A is optionally substituted (C1-C6)alkylene, (C3-C6)alkenylene or the like; R1 is H, optionally substituted (C1-C6)alkyl, (C3-C6)alkenyl, (C3-C6)cycloalkyl or the like; R2, R3 and R4 are each H, (C1-C6)alkyl, (C3-C6)alkenyl or the like, or R2 and A or R2 and R1 may form a 3- to 8-membered ring which may be interrupted by one to three atoms selected from among Of S and N; Q is C or N; X and Y are each halogen, CN, NO2, (C1-C6)alkyl, (C2-C6)alkenyl or the like; m is 0 to 2; n is 0 to 3; and two adjacent Xs or Ys on the aromatic ring may be united to form a fused ring]. The compounds exhibit excellent insecticidal activity against insect pests resistant to existing pesticides even when applied in dosages lower than those of similar pesticides.

    摘要翻译: 由通式(I)表示的磺酰胺衍生物或其盐; 含有与活性成分相同的农业和园艺用杀虫剂; 及其用途:[其中A是任选取代的(C 1 -C 6 -C 6)亚烷基,(C 3 -C 6 - 亚烷基等; R 1是H,任选取代的(C 1 -C 6 -C 6)烷基,(C 3 -C 6 - (C 3 -C 6 -C 6)环烷基等;(C 3 -C 6)烷基,(C 3 -C 6 -C 6)环烷基等; R 2,R 3和R 4各自为H,(C 1 -C 6)烷基, (C 1 -C 6)烷基,(C 3 -C 6 -C 6)链烯基等,或R 2和A或R 2 R 1和R 2可以形成3至8元环,其可以被选自S和N中的一至三个原子间隔; Q是C或N; X和Y各自为卤素,CN,NO 2,(C 1 -C 6)烷基,(C 1 -C 6)烷基, 链烯基或类似物; m为0〜2; n为0〜3; 并且芳环上的两个相邻的X或Y可以结合形成稠环]。 该化合物对于现有农药抗性的昆虫害虫具有优异的杀虫活性,即使施用量低于类似农药的剂量。

    Benzamide derivatives, insecticides for agricultural and horticultural use and usage thereof
    10.
    发明授权
    Benzamide derivatives, insecticides for agricultural and horticultural use and usage thereof 失效
    苯甲酰胺衍生物,农业和园艺用杀虫剂及其用途

    公开(公告)号:US06642379B1

    公开(公告)日:2003-11-04

    申请号:US10018687

    申请日:2002-04-04

    IPC分类号: C07D26504

    摘要: Benzamide derivatives represented by the general formula (I): and insecticides for agricultural and horticultural use and usage thereof, wherein Z1 is O or S; R is H, (substituted) alkyl, or alkoxycarbonyl; X is halogeno, cyano, nitro, C3-C6(halo)cycloalkyl, (substituted) phenyl, a (substituted) heterocyclic group, or —A1—R1 [wherein A1 is —O—, —S—, —SO—, —SO2—, —C(═O)—, or —C(═NOR2)— (wherein R2 is H, C1-C6(halo)alkyl, (substituted) phenylated C1-C4 alkyl, or the like); and R1 is halogeno, C3-C6 cycloalkyl, C3-C6 halocycloalkenyl, (substituted) phenyl, or the like]; n is 0 to 4; Y is halogeno, cyano, nitro, C3-C6 halocycloalkyl, (substituted) phenyl, or the like; m is 1 to 5; Q is a heterocycle such as oxazoline; and B1 to B4 are each CH or N.

    摘要翻译: 由通式(I)表示的苯甲酰胺衍生物:和农业和园艺用途的杀虫剂及其用途,其中Z 1是O或S; R为H,(取代的)烷基或烷氧基羰基; X是卤代,氰基,硝基,C 3 -C 6(卤代)环烷基,(取代的)苯基,(取代的)杂环基或-A 1 -R 1 [其中A 1是-O-, -S-,-SO-,-SO 2 - , - C(= O) - 或-C(= NOR 2) - (其中R 2是H,C 1 -C 6(卤代)烷基,(取代的) -C4烷基等); 和R 1是卤代,C 3 -C 6环烷基,C 3 -C 6卤代环烯基,(取代的)苯基等]。 n为0〜4; Y是卤代,氰基,硝基,C 3 -C 6卤代环烷基,(取代的)苯基等; m为1〜5; Q是杂环,如恶唑啉; 和B 1至B 4各自为CH或N.