Psychotropic polycyclic imides
    3.
    发明授权
    Psychotropic polycyclic imides 失效
    精神药物多环酰胺

    公开(公告)号:US4824999A

    公开(公告)日:1989-04-25

    申请号:US248769

    申请日:1988-09-23

    申请人: Gary P. Stack

    发明人: Gary P. Stack

    摘要: The compound which is 2,3,3a,3b,4,5,6,6a,7,7a-decahydro-4,6,7-metheno-1H-cyclopenta[a]pentalene-1,3-dicarboxylic acid is useful as an intermediate for production of the corresponding anhydride from which several of the disclosed antipsychotic/anxiolytic agents are prepared.

    摘要翻译: 2,3,3a,3b,4,5,6,6a,7,7a-十氢-4,6,7-元苯-1H-环戊二烯并[a]精油烯-1,3-二羧酸的化合物是 可用作生产相应的酸酐的中间体,其中制备了几种所公开的抗精神病药/抗焦虑药物。

    Herbicidal n-octahydro-1,2,4-methenopentalenyl-(5)-ureas
    5.
    发明授权
    Herbicidal n-octahydro-1,2,4-methenopentalenyl-(5)-ureas 失效
    除草剂N-甲基吗啉-1,2,4-甲苯戊酸 - (5) -

    公开(公告)号:US3723415A

    公开(公告)日:1973-03-27

    申请号:US3723415D

    申请日:1970-09-04

    申请人: CIBA GEIGY CORP

    发明人: WEISS C RUMPF J

    摘要: New herbicidal compounds of the formula IN WHICH R1 and R2 represent hydrogen or certain substituents are described as particularly suitable for controlling weeds and undesirable grasses. Compositions containing these compounds as active ingredients in mixture with agriculturally acceptable carriers and a method of controlling weeds and undesirable grasses with the aid of such compounds or compositions containing them are also described, as well as novel intermediates which are methenopentalene derivatives from which the compounds of the above formula can be produced.

    Herbicidal n-octahydro-1,2,4-methenopentalenyl-(5)-ureas
    6.
    发明授权
    Herbicidal n-octahydro-1,2,4-methenopentalenyl-(5)-ureas 失效
    除草剂N-甲基吗啉-1,2,4-甲苯戊酸 - (5) -

    公开(公告)号:US3555086A

    公开(公告)日:1971-01-12

    申请号:US3555086D

    申请日:1967-12-18

    申请人: GEIGY CHEM CORP

    摘要: HERBICIDAL COMPOUNDS OF THE FORMULA

    5-(R1-N(-R2)-CO-NH-)OCTAHYDRO-1,2,4-METHENOPENTALENE

    IN WHICH

    R1 REPRESENTS HYDROGEN, LOWER ALIPHATIC HYDROCARBONS CYCLOALKYL, LOWER ALKOXY, OR PHENYL, R2 REPRESENTS HYDROGEN, LOWER ALKYL, OR LOWER ALKENYL, OR R1 AND R2 TOGETHER REPRESENT ETHYLENEOXYETHYLENE OR A POLYMETHYLENE BRIDGING MEMBER. ARE DESCRIBED AS PARTICULARLY SUITABLE FOR CONTROLLING WEEDS AND UNDESIRABLE GRASSES. COMPOSITIONS CONTAINING THESE COMPOUNDS AS ACTIVE INGREDIENTS IN MIXTURE WITH AGRICULTURALLY ACCEPTABLE CARRIRS AND A METHOD OF CONTROLLING WEEDS AND UNDESIRABLE GRASSES WITH THE AID OF SUCH COMPOUNDS OR COMPOSITIONS CONTAINING THEM ARE ALSO DESCRIBED, AS WELL AS INTERMEDIATES WHICH ARE METHENOPENTALENE DERIVATIVES FROM WHICH THE COMPOUNDS OF THE ABOVE FORMULA CAN BE PRODUCED.

    摘要翻译: 描述了R1和R2代表氢或某些取代基的新的除草化合物,特别适用于防治杂草和不希望的草。 还描述了含有这些化合物作为与农业上可接受的载体的混合物中的活性成分的组合物,以及借助于这些化合物或含有它们的组合物来控制杂草和不期望的草的方法,以及新颖的中间体,其是化合物 可以生产上述配方。

    NEUROACTIVE SUBSTITUTED CYCLOPENT[a]ANTHRACENES AS MODULATORS FOR GABA TYPE-A RECEPTORS
    8.
    发明申请
    NEUROACTIVE SUBSTITUTED CYCLOPENT[a]ANTHRACENES AS MODULATORS FOR GABA TYPE-A RECEPTORS 有权
    神经取代的循环[a]作为GABA型A受体的调节剂的蒽醌

    公开(公告)号:US20140275241A1

    公开(公告)日:2014-09-18

    申请号:US14203678

    申请日:2014-03-11

    发明人: Douglas Covey

    摘要: The present disclosure is generally directed to neuroactive substituted cyclopent[a]anthracenes as referenced herein, and pharmaceutically acceptable salts thereof, for use as, for example, an anesthetic, and/or in the treatment of disorders relating to GABA function and activity. The present disclosure is further directed to pharmaceutical compositions comprising such compounds.

    摘要翻译: 本公开一般涉及本文所述的神经活性取代的环戊烯[a]蒽及其药学上可接受的盐,用作例如麻醉剂和/或用于治疗与GABA功能和活性相关的疾病。 本公开进一步涉及包含这些化合物的药物组合物。