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    1-oxa-a-nor steroids
    112.
    发明授权
    1-oxa-a-nor steroids 失效
    1-OXA-A-NOR STEROIDS

    公开(公告)号：US3714203A

    公开(公告)日：1973-01-30

    申请号：US3714203D

    申请日：1969-07-07

    Applicant: ROUSSEL UCLAF

    Inventor： NEDELEC L ,  TORELLI V

    IPC: B05B1/14 ,  B05B17/04 ,  C07D303/32 ,  C07D303/40 ,  C07J73/00 ,  C07D5/10

    CPC classification number: C07D303/32 ,  C07D303/40 ,  C07J73/003

    Abstract: 1-OXA-A-Nor steroids of the formula

    WHEREIN R is selected from the group consisting of hydrogen, acyl of an organic carboxylic acid of one to 18 carbon atoms and alkyl of one to five carbon atoms which may be further substituted with an aryl, alkoxy and alkylthio which have antiandrogenic activity and their preparation and use.

    Abstract translation: 1-OXA-A-型甾体，式WHEREIN R选自氢，1至18个碳原子的有机羧酸的酰基和1至5个碳原子的烷基，可以进一步被芳基取代 ，烷氧基和烷硫基，其具有抗雄激素活性及其制备和用途。

    Novel 2,2-dimethyl steroids
    113.
    发明授权
    Novel 2,2-dimethyl steroids 失效
    新二氢二异丙基苯甲酸酯

    公开(公告)号：US3708474A

    公开(公告)日：1973-01-02

    申请号：US3708474D

    申请日：1971-02-03

    Applicant: ROUSSEL UCLAF

    Inventor： NEDELEC L ,  GASC J

    IPC: C07J1/00 ,  C07J75/00 ,  C07C169/22 ,  C07C173/00

    CPC classification number: C07J1/00 ,  C07J75/00

    Abstract: 2A,2B,17A A-TRIMETHYL - 13B - ALKYL-$4,9,11-GONATRIENE-17BOL-3-ONES OF THE FORMULA

    2,2,17-TRI(H3C-),4-R1,7-R2,17-(Z-O-),18-R-GONA-4,9,11-

    TRIEN-3-ONE

    WHEREIN Z IS HYDROGEN, ALKYL OF 1 TO 6 CARBON ATOMS OR TETRAHYDROPYRANYL, R IS ALKYL OF 1 TO 4 CARBON ATOMS, R1 IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, HYDROXY, LOWER ALKANOYLOXY OF 1 TO 7 CARBON ATOMS AND HALOGEN, AND R2 IS HYDROGEN ALKYL OF 1 TO 4 CARBON ATOMS HAVING ANTI-ANDROGENIC ACTIVITY AND THEIR PREPARATION.

    1,3-thiazines and their preparation
    114.
    发明授权
    1,3-thiazines and their preparation 失效
    1,3-THIAZINES及其制备

    公开(公告)号：US3707540A

    公开(公告)日：1972-12-26

    申请号：US3707540D

    申请日：1966-12-07

    Applicant: ROUSSEL UCLAF

    Inventor： AMIARD GASTON ,  HEYMES RENE

    IPC: C07D307/60 ,  C07D501/08 ,  C07D513/04 ,  G03C5/39 ,  C07D93/08 ,  C07D99/24

    CPC classification number: C07D513/04 ,  C07D307/60 ,  G03C5/39

    Abstract: LACTONES OF 2-(CARBONYL-AMINO-METHYL)-5-HYDROXYMETHYL-3,6-DIHYDRO-2H-1,3-THIAZINE-4 -CARBOXYLIC ACIDS USEFUL AS INTERMEDIATES FOR ANTIBIOTICS OF THE C-CEPHALOSPORINE FAMILY AND THEIR PREPARATION. THE INVENTION RELATES TO NOVEL DIHYDRO-1,3-THIAZINE COMPOUNDS OF THE FORMULA

    2-(R-OOC-CH(-Y)-),7-(O=)-1,2,5,7-TETRAHYDRO-4H-FURO(3,4-D)

    (3,1)THIAZINE

    WHEREIN R IS SELECTED FROM THE GROUP CONSISTING OF ALKYL AND ARALKYL, Y IS SELECTED FROM THE GROUP CONSISTING OF -HN-AC, PHTHALIMIDO AND-NH-R'',R'' IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, ALKYL AND ARALKYL AND AC IS THE ACYL RADICAL OF AN ORGANIC CARBOXYLIC ACID OF 1 TO 18 CARBON ATOMS AND TO A NOVEL PROCESS FOR THE PREPARATION OF THE SAID COMPOUNDS.

    Preparation of 7{60 -methyl steroids
    115.
    发明授权
    Preparation of 7{60 -methyl steroids 失效
    制备7种{6-甲基异烟肼

    公开(公告)号：US3697556A

    公开(公告)日：1972-10-10

    申请号：US3697556D

    申请日：1970-07-27

    Applicant: ROUSSEL UCLAF

    Inventor： BOUCOURT ROBERT ,  NEDELEC LUCIEN ,  GASC JEAN-CLAUDE

    IPC: A61K31/565 ,  B65H31/10 ,  C07J1/00 ,  C07J75/00 ,  C07C169/22

    CPC classification number: A61K31/565 ,  B65H31/10 ,  C07J1/00 ,  C07J75/00

    Abstract: WHEREIN R is alkyl of one to four carbon atoms and R'' is selected from the group consisting of hydrogen, acyl of an organic carboxylic acid of one to 18 carbon atoms and an organic ether radical, a novel process for preparing the corresponding Delta 4,9,11-gonatrienes and novel intermediates produced by the said processes.

    A novel process for the preparation of 7 Alpha -methyl- Delta 4,9-gonadienes of the formula

    Abstract translation: 用于制备式WHEREIN R的7个α-甲基-TATA 4,9-基那烯的新方法是1至4个碳原子的烷基，R'选自氢，有机羧酸的酰基， 1至18个碳原子和有机醚基团，一种制备相应的DELTA 4,9,11-三烯的新方法和由所述方法制备的新型中间体。

    Novel 7{60 -methyl-{66 {11 {11 {11 {11 -gonadienes
    116.
    发明授权
    Novel 7{60 -methyl-{66 {11 {11 {11 {11 -gonadienes 失效
    第7号{60 -METHYL- {66 {11 {11}

    公开(公告)号：US3679718A

    公开(公告)日：1972-07-25

    申请号：US3679718D

    申请日：1970-07-27

    Applicant: ROUSSEL UCLAF

    Inventor： BUCOURT ROBERT ,  NEDELEC LUCIEN ,  GASC JEAN-CLAUDE

    IPC: A61K31/565 ,  C07J1/00 ,  C07C169/22

    CPC classification number: A61K31/565 ,  C07J1/00 ,  Y10S514/925

    Abstract: Novel 7 Alpha -methyl- Delta 4,11-gonadiene of the formula

    WHEREIN R is alkyl of one to four carbon atoms and R'' is selected from the group consisting of hydrogen, acyl of an organic carboxylic acid of one to 18 carbon atoms and an organic ether radical which have anabolic and androgenic activities and their preparation.

    Abstract translation: 具有式IV的新型7α-甲基-TATA 4,11-二氢二环，其中R是具有1至4个碳原子的烷基，R'选自氢，1至18个碳原子的有机羧酸的酰基和 具有合成代谢和雄激素活性及其制备的有机醚基团。

    10,11-DIHYDRO-,9,10-DIHYDRO-10,10-DIMETHYL-5-OR 9-{8 3-AMINO-2-oxo -OR-HYDROXY-PROPYLIDENE{9 {11 -5H-DIBENZO{8 a,d{9 {11 CYCLOHEPTENES AND-ANTHRACENES
    117.
    发明授权
    10,11-DIHYDRO-,9,10-DIHYDRO-10,10-DIMETHYL-5-OR 9-{8 3-AMINO-2-oxo -OR-HYDROXY-PROPYLIDENE{9 {11 -5H-DIBENZO{8 a,d{9 {11 CYCLOHEPTENES AND-ANTHRACENES 失效
    10,11-二氢 - ，9,10-二氢-10,10-二甲基-5 - 或9- {8 3-氨基-2-氧代-OR-羟基 - 丙基} {9 {11-5H-二苯并[{a ，d {9 {11 CYCLOHEPTENES AND-ANTHRACENES

    公开(公告)号：US3674841A

    公开(公告)日：1972-07-04

    申请号：US3674841D

    申请日：1969-03-03

    Applicant: ROUSSEL UCLAF

    Inventor： BOISSIER JACQUES ROBERT ,  RATOUIS ROGER

    IPC: C07C91/02 ,  C07C97/10

    CPC classification number: C07C215/30

    Abstract: The products are new tricyclic amino compounds and acid addition salts thereof, said tricyclic amino compounds corresponding to the general formula : WHERE X represents one of the following divalent hydrocarbon radicals : A represents a carbonyl (CO) or a hydroxymethylene (CHOH) group and R represents a monoalkylamino or a dialkylamino radical. They are very useful substances for human therapeutics, namely as antidepressants and antianxiety agents. The process for preparing compounds of formula (1) and their salts is disclosed.

    Abstract translation: 产物是新的三环氨基化合物及其酸加成盐，所述三环氨基化合物对应于通式：

    2-oxa-steroid and the production thereof
    119.
    发明授权
    2-oxa-steroid and the production thereof 失效
    2-OXA-STEROID及其生产

    公开(公告)号：US3595877A

    公开(公告)日：1971-07-27

    申请号：US3595877D

    申请日：1968-08-14

    Applicant: ROUSSEL UCLAF

    Inventor： BUCOURT ROBERT ,  NEDELEC LUCIEN

    IPC: C07D295/096 ,  C07D295/116 ,  C07J73/00 ,  C07D7/20

    CPC classification number: C07D295/096 ,  C07C2603/16 ,  C07D295/116 ,  C07J73/003

    Abstract: 2-OXA-13B-R-17A-METHYL-$4,9,11-GONATRIENES OF THE FORMULA

    13-R,16-(R''-O-),16-(CH3-)-2-OXA-GONA-4,9,11-TRIENE

    WHEREIN R IS SELECTED FROM THE GROUP CONSISTING OF METHYL AND ETHYL AND R'' IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, SATRUATED ALKYL OF 1 TO 5 CARBON ATOMS WHICH MAY CONTAIN A HETERO OXYGEN ATOM, UNSATURATED ALKYL OF 2 TO 5 CARBON ATOMS, CYCLOALKYL OF 3 TO 5 CARBON ATOMS WHICH MAY CONTAIN A HETERO OXYGEN ATOM, WITH THE PROVISO THAT R IS ETHYL WHEN R'' IS HYDROGEN WHCIH COMPOUNDS POSSESS ANABLOIC AND ANDROGENIC ACTIVITY. THE INVENTION ALSO RELATES TO A NOVEL PROCESS AND NOVEL INTERMEDIATES FOR THE PREPARATION OF THE COMPOUNDS OF FORMULA I.

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