摘要:
2'-Methylidenepyrimidine nucleoside compounds of the general formula: ##STR1## wherein R.sup.1 stands for amino or hydroxy group; R.sup.2 stands for a halogen or a lower alkyl when R.sup.1 is amino or R.sup.2 stands for an alkyl having 2 to 4 carbon atoms, an alkynyl having 2 to 4 carbon atoms or a haloalkyl when R.sup.1 is hydroxy group; and R.sup.3 stands for hydrogen or a phosphoric acid residue, or salts thereof, compositions containing one or more of these compounds and methods for production of these compounds are disclosed.Said compounds and salts thereof exhibit noticeable antitumor activities.
摘要:
In a polycarbonate resin/silicone rubber integrally molded article, a polycarbonate resin having an aliphatic unsaturated group, typically an isopropenyl group is integrally joined to an addition type silicone rubber containing a tackifier component at high bond strength. It is prepared by injection molding a modified polycarbonate resin into a preform, injection molding a silicone rubber composition over the preform, and curing the composition at a temperature below the softening point of the polycarbonate resin.
摘要:
An optical fiber cable free from a generation of a microbent during manufacturing, and in which an impregnation of hydrogen and/or water to a cladding is prevented, and having high electrical conduction, tolerance to heat and mechanical strength, and a process for making same. The optical fiber cable includes a silica based glass optical fiber including a core and a cladding, a thin carbon coating formed on an outer surface of the optical fiber, and an electrically conductive coating formed on an outer surface of the carbon coating. The carbon coating functions as a layer for preventing the impregnation of hydrogen and/or water to the optical fiber, and the conductive coating functions as a heat tolerance member, a conductive member, and a mechanical support member. The carbon coating is preferably formed as an amorphous carbon layer. Preferably, the conductive coating can be made of materials having a good contact with the carbon coating, a high conductivity, a high heat tolerance, and a high strength, and can be formed as thin as possible. The conductive coating can be formed by a plurality of different metal layers having different thickness.
摘要:
Disclosed are imidazole derivatives represented by formula [I]: ##STR1## wherein R is a hydrogen atom or ##STR2## wherein R.sup.2 is a hydrogen atom or a hydroxy protecting group, R.sup.2 protecting either a single hydroxy or two hydroxies together when R.sup.2 is a hydroxy protecting group, and R.sup.3 is a hydrogen atom or OR.sup.2 ; A is CONH.sub.2 or CN; and R.sup.1 is a hydrogen atom, lower alkyl, hydroxy lower alkyl, or phenyl.Also disclosed are six processes for producing these novel compounds among which a typical process comprises reacting a starting imidazole compound having a halogen at the 5-position thereof with an acetylene derivative to alkynylate the 5-position.Furthermore, the compounds having remarkable antitumor activities and therefore can provide novel antitumor agents.
摘要:
This invention relates to a method for selectively enhancing absorption of 5-fluorouracil, bleomycins or bleomycin derivatives into the gastrointestinal tumor site by orally administering such substance together with an alkali metal salt of polyacrylic acid, and an orally administable antitumor composition used for such method.
摘要:
An inspection machine for detecting flaws in the surface of cylindrical fuel pellets, which comprises a pellet infeed section for successively transporting pellets to be inspected, a conveyer section for successively conveying delivered pellets to a plurality of inspection points, a plurality of inspection stations for detecting, at each inspection point, flaws at the corners, peripheral surface and end faces of the pellets by utilizing variations in back pressure prevailing in a sensor caused by the contact of an air stream with said flaws, an unacceptable pellet rejection station for rejecting pellets assessed to be unacceptable at any inspection station, and an acceptable pellet outfeed section for successively collecting pellets assessed as being acceptable.
摘要:
A disclosed vehicle navigation apparatus enables the issuance of an accurate and quick guidance. Voice uttered by an occupant of a vehicle is collected by a voice collecting unit and transmitted to an external facility by a voice transmitting unit. The external facility generates destination information based on the received voice, and transmits the destination information back to a destination information receiving unit of the apparatus. Based on the received destination information, the apparatus issues a guidance. The apparatus further includes a destination extracting unit by which the voice collected by the voice collecting unit is subjected to voice recognition in order to extract a destination from the collected voice. A tentative guidance is then issued based on the extracted destination until the destination information is received by the destination information receiving unit from the external facility.
摘要:
A copper foil reducing transmission loss at a high frequency and excellent in bond strength with a resin substrate, including at least a granular layer and a columnar layer in its thickness direction, the columnar layer being formed on at least one surface of the granular layer forming the copper foil or the granular layer being formed on at least one surface of the columnar layer forming the copper foil, the relation of the thickness A of the granular layer and the thickness B of the columnar layer in the copper foil being preferably A/(A+B)=40 to 99%, a method of production and apparatus for production for the same, and a high frequency circuit using the same.
摘要翻译:铜箔在高频下降低传输损耗,并且与树脂基板的粘合强度优异,其厚度方向至少包括粒状层和柱状层,所述柱状层形成在所述粒状层的至少一个表面上 铜箔或颗粒层形成在形成铜箔的柱状层的至少一个表面上,粒状层的厚度A与铜箔中柱状层的厚度B的关系优选为A /( A + B)= 40〜99%,制造方法及其制造装置以及使用该方法的高频电路。
摘要:
A convention appliance monitoring apparatus handles only the amount of gas used and security information for the case of a gas cutoff and can not address social needs for a desire to obtain information about influence (e.g., an amount of CO2 emission) of use of the gas combustion appliance on a terrestrial environment.Based on a gas appliance used by a client and a gas flow signal pertaining the gas appliance which are output from an appliance determination unit 2, CO2 emission data on the gas appliance stored in a CO2 emission data storage unit 3, and CO2 emission data which are to be compared with the gas appliance and stored in a comparative CO2 emission data storage unit 4, a CO2 emission calculation unit 5 calculates an amount of CO2 emission, an comparative amount of CO2 emission and a difference between the amount of CO2 emission and the comparative amount of CO2 emission. Accordingly, it is possible to determine the amount of CO2 emission produced by using the gas appliance and the difference between the amount of CO2 emission and the comparative amount of CO2 emission.
摘要:
The present invention provides a self-adhesive film which is a drawn polypropylene-based resin film comprising a laminated body containing an adhesive layer and a release layer which are provided on the surface of a base layer formed of a polypropylene-based resin, wherein an average surface roughness SRa of a surface of the above-described release layer is 0.200 μm or less, an average surface layer roughness SRa of a surface of the self-adhesive layer of the film is 0.030 μm or less, the contact area with the adherent, which is defined in the description, is 90% or more and 100% or less, and the film haze ranges from 1 to 40%. The self-adhesive film of the present invention is less likely to cause a blocking after the film is stored in a rolled state, and the processing suitability is excellent, and forming is less likely occur even when the film having been adhered to an adherend is processed at a high temperature, and further transparency is excellent.