公开(公告)号：US08119563B2

公开(公告)日：2012-02-21

申请号：US10595298

申请日：2004-10-04

申请人： George Theodoridis ,  David Rosen ,  Shunxiang Zhang ,  Walter H. Yeager ,  Robert N. Henrie, II ,  Syed Z. Ahmed ,  Hongbin Men ,  Stephen Donovan

发明人： George Theodoridis ,  David Rosen ,  Shunxiang Zhang ,  Walter H. Yeager ,  Robert N. Henrie, II ,  Syed Z. Ahmed ,  Hongbin Men ,  Stephen Donovan

IPC分类号： A01N43/22 ,  C07D211/06

CPC分类号： C07D211/48 ,  A01N43/40 ,  A01N43/54 ,  A01N43/58 ,  A01N43/713 ,  A01N43/90 ,  A01N47/06 ,  A01N47/20 ,  A01N47/22 ,  C07D211/94 ,  C07D401/10 ,  C07D401/12 ,  C07D451/02 ,  C07D471/10

摘要： N-substituted azacycle derivative compounds represented by formula (I): wherein m, q, r, t and u are independently selected from 0 or 1; and p is 0, 1, 2, or 3; and A, B, D, X, Y, R, R1, R2, R3, R4, R5, R6, R7, R8, R9, R10 and R11 are fully described herein. The compounds being particularly useful in compositions comprising an insecticidally effective amount of at least one compound of formula I, and an insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 由式（I）表示的N-取代的azacycle衍生物化合物：其中m，q，r，t和u独立地选自0或1; 且p为0,1,2或3; 并且A，B，D，X，Y，R，R 1，R 2，R 3，R 4，R 5，R 6，R 7，R 8，R 9，R 10和R 11在本文中被完整描述。 还公开了特别可用于包含杀虫有效量的至少一种式I化合物和杀虫相容载体的化合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US20090215821A1

公开(公告)日：2009-08-27

申请号：US10595298

申请日：2004-10-04

申请人： George Theodoridis ,  David Rosen ,  Shunxiang Zhang ,  Walter H. Yeager ,  Robert N. Henrie, II ,  Syed Z. Ahmed ,  Hongbin Men ,  Stephen Donovan

发明人： George Theodoridis ,  David Rosen ,  Shunxiang Zhang ,  Walter H. Yeager ,  Robert N. Henrie, II ,  Syed Z. Ahmed ,  Hongbin Men ,  Stephen Donovan

IPC分类号： A01N43/40 ,  C07D211/48 ,  C07D401/12

CPC分类号： C07D211/48 ,  A01N43/40 ,  A01N43/54 ,  A01N43/58 ,  A01N43/713 ,  A01N43/90 ,  A01N47/06 ,  A01N47/20 ,  A01N47/22 ,  C07D211/94 ,  C07D401/10 ,  C07D401/12 ,  C07D451/02 ,  C07D471/10

摘要： N-substituted azacycle derivative compounds represented by formula (I): wherein m, q, r, t and u are independently selected from 0 or 1; and p is 0, 1, 2, or 3; and A, B, D, X, Y, R, R1, R2, R3, R4, R5, R6, R7, R8, R9, R10 and R11 are fully described herein. The compounds being particularly useful in compositions comprising an insecticidally effective amount of at least one compound of formula I, and an insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 由式（I）表示的N-取代的azacycle衍生物化合物：其中m，q，r，t和u独立地选自0或1; 且p为0,1,2或3; 并且A，B，D，X，Y，R，R 1，R 2，R 3，R 4，R 5，R 6，R 7，R 8，R 9，R 10和R 11在本文中被完整描述。 还公开了特别可用于包含杀虫有效量的至少一种式I化合物和杀虫相容载体的化合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US07365082B2

公开(公告)日：2008-04-29

申请号：US10538997

申请日：2003-12-08

申请人： Ping Ding ,  Robert N. Henrie, II ,  Daniel H. Cohen ,  John W. Lyga ,  David S. Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter H. Yeager ,  Stephen F. Donovan ,  Steven Shunxiang Zhang ,  Inna Shulman ,  Seong Jae Yu ,  Guozhi Wang ,  Y. Larry Zhang ,  Ariamala Gopalsamy ,  Dennis L. Warkentin ,  Paul E. Rensner ,  Ian R. Silverman ,  Thomas G. Cullen

发明人： Ping Ding ,  Robert N. Henrie, II ,  Daniel H. Cohen ,  John W. Lyga ,  David S. Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter H. Yeager ,  Stephen F. Donovan ,  Steven Shunxiang Zhang ,  Inna Shulman ,  Seong Jae Yu ,  Guozhi Wang ,  Y. Larry Zhang ,  Ariamala Gopalsamy ,  Dennis L. Warkentin ,  Paul E. Rensner ,  Ian R. Silverman ,  Thomas G. Cullen

IPC分类号： A61K31/44 ,  A61K31/445 ,  A61K31/4422 ,  C07D211/06 ,  C07D211/08 ,  C07D211/70 ,  C07D211/82

CPC分类号： C07D405/14 ,  A01N43/40 ,  A01N43/54 ,  A01N43/713 ,  C07D211/14 ,  C07D211/18 ,  C07D211/22 ,  C07D211/24 ,  C07D211/26 ,  C07D211/28 ,  C07D211/32 ,  C07D211/94 ,  C07D401/06 ,  C07D401/10 ,  C07D401/12 ,  C07D401/14 ,  C07D413/12 ,  C07D417/12 ,  C07D451/14 ,  C07D513/04

摘要： It has now been found that certain novel N-(substituted aryl)-4-(disubstituted methyl)piperidine and pyridine derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): wherein m, n, q, r, and s are independently selected from 0 or 1; and p is 0, 1, 2, or 3; A is CH or N; and B, D, E, R, R1, R2, R3, R4, R5, R6, R7 and R8 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 现在已经发现某些新的N-（取代的芳基）-4-（二取代的甲基）哌啶和吡啶衍生物提供了意想不到的杀虫活性。 这些化合物由式（I）表示：其中m，n，q，r和s独立地选自0或1; 且p为0,1,2或3; A是CH或N; 和B，D，E，R，R 1，R 2，R 3，R 4，R 本文完全描述了本发明的第5，第6，第七和第八和第八。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US07683070B2

公开(公告)日：2010-03-23

申请号：US11874015

申请日：2007-10-17

申请人： Ping Ding ,  Robert N. Henrie, II ,  Daniel H. Cohen ,  John W. Lyga ,  David S. Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter H. Yeager ,  Stephen F. Donovan ,  Stephen Shunxiang Zhang ,  Inna Shulman ,  Seong Jae Yu ,  Guozhi Wang ,  Y. Larry Zhang ,  Ariamala Gopalsamy ,  Dennis L. Warkentin ,  Paul E. Rensner ,  Ian R. Silverman ,  Thomas G. Cullen

发明人： Ping Ding ,  Robert N. Henrie, II ,  Daniel H. Cohen ,  John W. Lyga ,  David S. Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter H. Yeager ,  Stephen F. Donovan ,  Stephen Shunxiang Zhang ,  Inna Shulman ,  Seong Jae Yu ,  Guozhi Wang ,  Y. Larry Zhang ,  Ariamala Gopalsamy ,  Dennis L. Warkentin ,  Paul E. Rensner ,  Ian R. Silverman ,  Thomas G. Cullen

IPC分类号： A61K31/4523 ,  A61K31/4545 ,  C07D211/06 ,  C07D239/02

CPC分类号： C07D405/14 ,  A01N43/40 ,  A01N43/54 ,  A01N43/713 ,  C07D211/14 ,  C07D211/18 ,  C07D211/22 ,  C07D211/24 ,  C07D211/26 ,  C07D211/28 ,  C07D211/32 ,  C07D211/94 ,  C07D401/06 ,  C07D401/10 ,  C07D401/12 ,  C07D401/14 ,  C07D413/12 ,  C07D417/12 ,  C07D451/14 ,  C07D513/04

摘要： It has now been found that certain novel N-(substituted aryl)-4-(disubstituted methyl)piperidine and pyridine derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): wherein m, n, q, r, and s are independently selected from 0 or 1; and p is 0, 1, 2, or 3; A is C or CH; and B, D, E, R, R1, R2, R3, R4, R5, R6, R7 and R8 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 现在已经发现某些新的N-（取代的芳基）-4-（二取代的甲基）哌啶和吡啶衍生物提供了意想不到的杀虫活性。 这些化合物由式（I）表示：其中m，n，q，r和s独立地选自0或1; 且p为0,1,2或3; A是C或CH; 本文完整地描述了B，D，E，R，R 1，R 2，R 3，R 4，R 5，R 6，R 7和R 8。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US07300946B2

公开(公告)日：2007-11-27

申请号：US10538998

申请日：2003-12-08

申请人： Ping Ding ,  Robert N. Henrie, II ,  Daniel H. Cohen ,  John W. Lyga ,  David S. Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter H. Yeager ,  Stephen F. Donovan ,  Steven Shunxiang Zhang ,  Inna Shulman ,  Seong Jae Yu ,  Guozhi Wang ,  Y. Larry Zhang ,  Ariamala Gopalsamy ,  Dennis L. Warkentin ,  Paul E. Rensner ,  Ian R. Silverman ,  Thomas G. Cullen

发明人： Ping Ding ,  Robert N. Henrie, II ,  Daniel H. Cohen ,  John W. Lyga ,  David S. Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter H. Yeager ,  Stephen F. Donovan ,  Steven Shunxiang Zhang ,  Inna Shulman ,  Seong Jae Yu ,  Guozhi Wang ,  Y. Larry Zhang ,  Ariamala Gopalsamy ,  Dennis L. Warkentin ,  Paul E. Rensner ,  Ian R. Silverman ,  Thomas G. Cullen

IPC分类号： A61K31/44 ,  A61K31/445 ,  A61K31/4422 ,  C07D211/06 ,  C07D211/08 ,  C07D211/70 ,  C07D211/82

CPC分类号： C07D405/14 ,  A01N43/40 ,  A01N43/54 ,  A01N43/713 ,  C07D211/14 ,  C07D211/18 ,  C07D211/22 ,  C07D211/24 ,  C07D211/26 ,  C07D211/28 ,  C07D211/32 ,  C07D211/94 ,  C07D401/06 ,  C07D401/10 ,  C07D401/12 ,  C07D401/14 ,  C07D413/12 ,  C07D417/12 ,  C07D451/14 ,  C07D513/04

摘要： It has now been found that certain novel N-(substituted aryl)-4(disubstituted methyl)piperidine and pyridine derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): wherein m, n, q, r, and s are independently selected from 0 or 1; and p is 0, 1, 2, or 3; A is C or CH; and B, D, E, R, R1, R2, R3, R4, R5, R6, R7 and R8 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present

摘要翻译： 现在已经发现，某些新的N-（取代的芳基）-4（二取代的甲基）哌啶和吡啶衍生物已经提供了意想不到的杀虫活性。 这些化合物由式（I）表示：其中m，n，q，r和s独立地选自0或1; 且p为0,1,2或3; A是C或CH; 和B，D，E，R，R 1，R 2，R 3，R 4，R 本文中充分描述了本发明的第5，第6，第七和第八和第八。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所

公开(公告)号：US20060135504A1

公开(公告)日：2006-06-22

申请号：US10538998

申请日：2003-12-08

申请人： Ping Ding ,  Robert Henrie II ,  Daniel Cohen ,  John Lyga ,  David Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter Yeager ,  Stephen Donovan ,  Steven Zhang ,  Inna Shulman ,  Seong Yu ,  Guozhi Wang ,  Y. Larry Zhang ,  Araimala Gopalsamy ,  Dennis Warkentin ,  Paul Rensner ,  Ian Silverman ,  Thomas Cullen

发明人： Ping Ding ,  Robert Henrie II ,  Daniel Cohen ,  John Lyga ,  David Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter Yeager ,  Stephen Donovan ,  Steven Zhang ,  Inna Shulman ,  Seong Yu ,  Guozhi Wang ,  Y. Larry Zhang ,  Araimala Gopalsamy ,  Dennis Warkentin ,  Paul Rensner ,  Ian Silverman ,  Thomas Cullen

IPC分类号： A61K31/397 ,  C07D213/63 ,  C07D205/10

CPC分类号： C07D405/14 ,  A01N43/40 ,  A01N43/54 ,  A01N43/713 ,  C07D211/14 ,  C07D211/18 ,  C07D211/22 ,  C07D211/24 ,  C07D211/26 ,  C07D211/28 ,  C07D211/32 ,  C07D211/94 ,  C07D401/06 ,  C07D401/10 ,  C07D401/12 ,  C07D401/14 ,  C07D413/12 ,  C07D417/12 ,  C07D451/14 ,  C07D513/04

摘要： It has now been found that certain novel N-(substituted aryl)-4(disubstituted methyl)piperidine and pyridine derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): wherein m, n, q, r, and s are independently selected from 0 or 1; and p is 0, 1, 2, or 3; A is C or CH; and B, D, E, R, R1, R2, R3, R4, R5, R6, R7 and R8 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 现在已经发现，某些新的N-（取代的芳基）-4（二取代的甲基）哌啶和吡啶衍生物已经提供了意想不到的杀虫活性。 这些化合物由式（I）表示：其中m，n，q，r和s独立地选自0或1; 且p为0,1,2或3; A是C或CH; 和B，D，E，R，R 1，R 2，R 3，R 4，R 本文中充分描述了本发明的第5，第6，第七和第八和第八。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US20080090828A1

公开(公告)日：2008-04-17

申请号：US11874015

申请日：2007-10-17

申请人： Ping Ding ,  Robert Henrie ,  Daniel Cohen ,  John Lyga ,  David Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter Yeager ,  Stephen Donovan ,  Stephen Zhang ,  Inna Shulman ,  Seong Yu ,  Guozhi Wang ,  Y. Zhang ,  Ariamala Gopalsamy ,  Dennis Warkentin ,  Paul Rensner ,  Ian Silverman ,  Thomas Cullen

发明人： Ping Ding ,  Robert Henrie ,  Daniel Cohen ,  John Lyga ,  David Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter Yeager ,  Stephen Donovan ,  Stephen Zhang ,  Inna Shulman ,  Seong Yu ,  Guozhi Wang ,  Y. Zhang ,  Ariamala Gopalsamy ,  Dennis Warkentin ,  Paul Rensner ,  Ian Silverman ,  Thomas Cullen

IPC分类号： C07D453/02 ,  A61K31/4745 ,  A61K31/50

CPC分类号： C07D405/14 ,  A01N43/40 ,  A01N43/54 ,  A01N43/713 ,  C07D211/14 ,  C07D211/18 ,  C07D211/22 ,  C07D211/24 ,  C07D211/26 ,  C07D211/28 ,  C07D211/32 ,  C07D211/94 ,  C07D401/06 ,  C07D401/10 ,  C07D401/12 ,  C07D401/14 ,  C07D413/12 ,  C07D417/12 ,  C07D451/14 ,  C07D513/04

摘要： It has now been found that certain novel N-(substituted aryl)-4-(disubstituted methyl)piperidine and pyridine derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): wherein m, n, q, r, and s are independently selected from 0 or 1; and p is 0, 1, 2, or 3; A is C or CH; and B, D, E, R, R1, R2, R3, R4, R5, R6, R7 and R8 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 现在已经发现某些新的N-（取代的芳基）-4-（二取代的甲基）哌啶和吡啶衍生物提供了意想不到的杀虫活性。 这些化合物由式（I）表示：其中m，n，q，r和s独立地选自0或1; 且p为0,1,2或3; A是C或CH; 和B，D，E，R，R 1，R 2，R 3，R 4，R 本文中充分描述了本发明的第5，第6，第七和第八和第八。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US06987194B2

公开(公告)日：2006-01-17

申请号：US10832624

申请日：2004-04-27

申请人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  David M. Roush ,  Stephen F. Donovan ,  Frank J. Zawacki ,  Walter H. Yeager ,  John W. Lyga ,  Daniel H. Cohen

发明人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  David M. Roush ,  Stephen F. Donovan ,  Frank J. Zawacki ,  Walter H. Yeager ,  John W. Lyga ,  Daniel H. Cohen

IPC分类号： C07D307/83 ,  C07D311/04 ,  A61K31/343 ,  A61K31/353

CPC分类号： A01N43/30 ,  A01N43/32 ,  A01N43/40 ,  A01N43/60 ,  A01N47/16 ,  C07D211/22 ,  C07D307/79 ,  C07D307/83 ,  C07D311/04 ,  C07D401/04 ,  C07D495/10

摘要： Insecticidal (dihalopropenyl) phenylalkyl substituted dihydrobenzofuran and dihydrobenzopyran derivatives of Formula I are disclosed. These compounds provide unexpected insecticidal activity across a spectrum of insect pests combined with desirable physical properties including improved photostability. wherein x and y are integers independently selected from 0 or 1; and B is a bridging group *—(CR16R17)q—(CR18R19)r—(CR20R21)s—Lt—(CR22R23)u—(CR24R25)v—(CR26R27)w—, where the asterisk denotes attachment at A; and q, r, s, u, v and w are integers independently selected from 0, 1 and 2; and t is an integer selected from 0 and 1. A, D, E, G, M, R through R11, and R16 through R27, inclusively, are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I and methods of controlling insects by applying said compositions to a locus where insects are present or are expected to be present are also disclosed.

摘要翻译： 公开了杀虫（二卤代丙烯基）苯基烷基取代的二氢苯并呋喃和式I的二氢苯并吡喃衍生物。 这些化合物在一系列昆虫害虫中提供了意想不到的杀虫活性，并结合所需的物理性质，包括改善的光稳定性。 其中x和y是独立地选自0或1的整数; 并且B是桥接基团<？in-line-formula description =“In-line Formulas”end =“lead”？> * - （CR ^{16 17 ） - （CR 20） - （CR 20） - （CR 20） - （CR 20） - （CR 22）23 - - - （CR 22）23 （CR 26）25（ - ） - （CR 26）25 ） q，r，s，u，v和w是独立地选自0,1和2的整数; A，D，E，G，M，R至R 11和R 16至R 27中的一个整数。 / SUP>，包括这里完全描述。 此外，还公开了包含杀虫有效量的至少一种式I化合物的组合物和通过将所述组合物施用于存在昆虫或预期存在的场所来控制昆虫的方法。}

公开(公告)号：US07247756B2

公开(公告)日：2007-07-24

申请号：US10353471

申请日：2003-01-29

申请人： George Theodoridis ,  Edward Barron ,  Daniel H. Cohen ,  Ellen M. Crawford ,  Thomas G. Cullen ,  Hongyan Qi ,  Elizabeth Rowley ,  Syed F. Ali ,  Walter H. Yeager ,  Christina B. Duggan

发明人： George Theodoridis ,  Edward Barron ,  Daniel H. Cohen ,  Ellen M. Crawford ,  Thomas G. Cullen ,  Hongyan Qi ,  Elizabeth Rowley ,  Syed F. Ali ,  Walter H. Yeager ,  Christina B. Duggan

IPC分类号： C07C43/20

CPC分类号： C07D215/233 ,  C07C211/59 ,  C07C217/20 ,  C07C217/58 ,  C07C217/92 ,  C07C233/43 ,  C07C235/56 ,  C07C251/24 ,  C07C271/28 ,  C07C275/34 ,  C07C275/40 ,  C07C291/04 ,  C07C2602/08 ,  C07C2602/10 ,  C07D209/46 ,  C07D215/24 ,  C07D215/38 ,  C07D215/40 ,  C07D215/44 ,  C07D217/22 ,  C07D295/088 ,  C07D295/096 ,  C07D295/205 ,  C07D491/10

摘要： Compounds of formula I: wherein A, B, D, and R are as defined herein and their agriculturally acceptable salts are disclosed as effective insecticides. In addition, compositions comprising an insecticidally effective amount of a compound of Formula I in admixture with at least one agriculturally acceptable extender or adjuvant and methods of controlling insects comprising applying the compositions to locus on crops where control is desired are disclosed.

摘要翻译： 式I化合物：其中A，B，D和R如本文所定义，其农业上可接受的盐被公开为有效的杀虫剂。 此外，公开了包含杀虫有效量的式I化合物与至少一种农业上可接受的增量剂或佐剂混合的组合物和控制昆虫的方法，其包括将组合物施用于需要控制的作物上的位点。

公开(公告)号：US20110065710A1

公开(公告)日：2011-03-17

申请号：US10580481

申请日：2004-12-02

申请人： David M. Roush ,  John F. Chiarello ,  Jianming Yu ,  Benjamin J. Dugan ,  George Theodoridis ,  Manorama M. Patel ,  Walter H. Yeager ,  Steven W. Szczepanski

发明人： David M. Roush ,  John F. Chiarello ,  Jianming Yu ,  Benjamin J. Dugan ,  George Theodoridis ,  Manorama M. Patel ,  Walter H. Yeager ,  Steven W. Szczepanski

IPC分类号： A61K31/4965 ,  A61K31/50 ,  A61K31/426 ,  A61K31/44

CPC分类号： C07D213/26 ,  A01N43/40 ,  A01N43/50 ,  A01N43/78 ,  A01N43/82 ,  A01N43/88 ,  A01N47/40 ,  A01N51/00 ,  A01N57/26 ,  C07D213/38 ,  C07D213/64 ,  C07D213/70 ,  C07D213/73 ,  C07D233/64 ,  C07D237/08 ,  C07D237/12 ,  C07D239/30 ,  C07D241/16 ,  C07D261/08 ,  C07D263/34 ,  C07D273/00 ,  C07D277/32 ,  C07D285/06 ,  C07D307/14 ,  C07D401/12 ,  C07D401/14 ,  C07D405/12 ,  C07D413/12 ,  C07D413/14 ,  C07D417/12 ,  C07D417/14 ,  C07F9/58

摘要： Certain noel N-(heteroarylalkyl)alkanediamine derivatives have provided unexpected insecticidal and acaricidal activity. These compounds are represented by formula I: wherein Ar, a, r, R, Ra, Rb, Rc, Rd, b, c, Re, Rf, Rg, Rh, R5, d, e, U, V, X, WR6 and R7 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 某些Noel N-（杂芳基烷基）烷二胺衍生物提供了意想不到的杀虫和杀螨活性。 这些化合物由式I表示：其中Ar，a，r，R，Ra，Rb，Rc，Rd，b，c，Re，Rf，Rg，Rh，R5，d，e，U，V，X， 和R7完全描述于此。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。