-
公开(公告)号:US07279582B2
公开(公告)日:2007-10-09
申请号:US10280652
申请日:2002-10-25
申请人: Eric J. Stoner , Arthur J. Cooper , Lawrence Kolaczkowski , Ketan M. Patel , Hing Leung Sham , Daniel W. Norbeck , Xiaoqi Chen , David A. Betebenner , Thomas R. Herrin , Gondi N. Kumar , Stephen L. Condon , Daniel A. Dickman , Patricia A. Oliver , Jien-Heh J. Tien
发明人: Eric J. Stoner , Arthur J. Cooper , Lawrence Kolaczkowski , Ketan M. Patel , Hing Leung Sham , Daniel W. Norbeck , Xiaoqi Chen , David A. Betebenner , Thomas R. Herrin , Gondi N. Kumar , Stephen L. Condon , Daniel A. Dickman , Patricia A. Oliver , Jien-Heh J. Tien
IPC分类号: C07D233/32 , C07D239/10 , C07D239/12
CPC分类号: C07D207/27 , C07D207/404 , C07D207/408 , C07D223/10 , C07D233/32 , C07D233/42 , C07D239/10 , C07D239/22 , C07D241/08 , C07D241/18 , C07D253/06 , C07D263/22 , C07D307/20 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/12 , C07D405/14 , C07D407/12 , C07D409/12 , C07D409/14 , C07D417/12
摘要: A compound of the formula: is disclosed as an HIV protease inhibitor. Methods and compositions for inhibiting an HIV infection are also disclosed.
摘要翻译: 公开了下式的化合物作为HIV蛋白酶抑制剂。 还公开了用于抑制HIV感染的方法和组合物。
-
公开(公告)号:US06472529B2
公开(公告)日:2002-10-29
申请号:US09837280
申请日:2001-04-18
申请人: Hing Leung Sham , Daniel W. Norbeck , Xiaoqi Chen , David A. Betebenner , Dale J. Kempf , Thomas R. Herrin , Gondi N. Kumar , Stephen L. Condon , Arthur J. Cooper , Daniel A. Dickman , Steven M. Hannick , Lawrence Kolaczkowski , Patricia A. Oliver , Daniel J. Plata , Peter J. Stengel , Eric J. Stoner , Jieh-Heh J. Tien , Jih-Hua Liu , Ketan M. Patel
发明人: Hing Leung Sham , Daniel W. Norbeck , Xiaoqi Chen , David A. Betebenner , Dale J. Kempf , Thomas R. Herrin , Gondi N. Kumar , Stephen L. Condon , Arthur J. Cooper , Daniel A. Dickman , Steven M. Hannick , Lawrence Kolaczkowski , Patricia A. Oliver , Daniel J. Plata , Peter J. Stengel , Eric J. Stoner , Jieh-Heh J. Tien , Jih-Hua Liu , Ketan M. Patel
IPC分类号: C07D23332
CPC分类号: C07D207/27 , C07D207/404 , C07D207/408 , C07D223/10 , C07D233/32 , C07D233/42 , C07D239/10 , C07D239/22 , C07D241/08 , C07D241/18 , C07D253/06 , C07D263/22 , C07D307/20 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/12 , C07D405/14 , C07D407/12 , C07D409/12 , C07D409/14 , C07D417/12
摘要: A compound of the formula: is disclosed as an HIV protease inhibitor. Methods and compositions for inhibiting an HIV infection are also disclosed.
摘要翻译: 公开了下式的化合物作为HIV蛋白酶抑制剂。 还公开了用于抑制HIV感染的方法和组合物。
-
公开(公告)号:US06313296B1
公开(公告)日:2001-11-06
申请号:US09511390
申请日:2000-02-23
申请人: Hing Leung Sham , Daniel W. Norbeck , Xiaoqi Chen , David A. Betebenner , Dale J. Kempf , Thomas R. Herrin , Gondi N. Kumar , Stephen L. Condon , Arthur J. Cooper , Daniel A. Dickman , Steven M. Hannick , Lawrence Kolaczkowski , Patricia A. Oliver , Daniel J. Plata , Peter J. Stengel , Eric J. Stoner , Jieh-Heh J. Tien , Jih-Hua Liu , Ketan M. Patel
发明人: Hing Leung Sham , Daniel W. Norbeck , Xiaoqi Chen , David A. Betebenner , Dale J. Kempf , Thomas R. Herrin , Gondi N. Kumar , Stephen L. Condon , Arthur J. Cooper , Daniel A. Dickman , Steven M. Hannick , Lawrence Kolaczkowski , Patricia A. Oliver , Daniel J. Plata , Peter J. Stengel , Eric J. Stoner , Jieh-Heh J. Tien , Jih-Hua Liu , Ketan M. Patel
IPC分类号: C07D23902
CPC分类号: C07D207/27 , C07D207/404 , C07D207/408 , C07D223/10 , C07D233/32 , C07D233/42 , C07D239/10 , C07D239/22 , C07D241/08 , C07D241/18 , C07D253/06 , C07D263/22 , C07D307/20 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/12 , C07D405/14 , C07D407/12 , C07D409/12 , C07D409/14 , C07D417/12
摘要: A compound of the formula: is disclosed as an HIV protease inhibitor. Methods and compositions for inhibiting an HIV infection are also disclosed.
摘要翻译: 公开了下式的化合物作为HIV蛋白酶抑制剂。 还公开了用于抑制HIV感染的方法和组合物。
-
公开(公告)号:US07968707B2
公开(公告)日:2011-06-28
申请号:US11679227
申请日:2007-02-27
申请人: Hing Leung Sham , Daniel W. Norbeck , Xiaoqi Chen , David A. Betebenner , Dale J. Kempf , Thomas R. Herrin , Gondi N. Kumar , Stephen L. Condon , Arthur J. Cooper , Daniel A. Dickman , Steven M. Hannick , Lawrence Kolaczkowski , Patricia A. Oliver , Daniel J. Plata , Peter J. Stengel , Eric J. Stoner , Jieh-Heh J. Tien , Jih-Hua Liu , Ketan M. Patel
发明人: Hing Leung Sham , Daniel W. Norbeck , Xiaoqi Chen , David A. Betebenner , Dale J. Kempf , Thomas R. Herrin , Gondi N. Kumar , Stephen L. Condon , Arthur J. Cooper , Daniel A. Dickman , Steven M. Hannick , Lawrence Kolaczkowski , Patricia A. Oliver , Daniel J. Plata , Peter J. Stengel , Eric J. Stoner , Jieh-Heh J. Tien , Jih-Hua Liu , Ketan M. Patel
IPC分类号: C07D219/04 , C07D291/06 , C07D243/04 , C07D265/12 , C07D413/12 , C07D239/02
CPC分类号: C07D207/27 , C07D207/404 , C07D207/408 , C07D223/10 , C07D233/32 , C07D233/42 , C07D239/10 , C07D239/22 , C07D241/08 , C07D241/18 , C07D253/06 , C07D263/22 , C07D307/20 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/12 , C07D405/14 , C07D407/12 , C07D409/12 , C07D409/14 , C07D417/12
摘要: A compound of the formula: is disclosed as an HIV protease inhibitor. Methods and compositions for inhibiting an HIV infection are also disclosed.
摘要翻译: 公开了下式的化合物作为HIV蛋白酶抑制剂。 还公开了用于抑制HIV感染的方法和组合物。
-
公开(公告)号:US06284767B1
公开(公告)日:2001-09-04
申请号:US09207873
申请日:1998-12-08
申请人: Hing Leung Sham , Daniel W. Norbeck , Dale J. Kempf , Xiaoqi Chen , David A. Betebenner , Thomas R. Herrin , Gondi N. Kumar , John M. Lipari , Laman Alani , Soumojeet Ghosh , Rong R. Gao , Dilip Kaul
发明人: Hing Leung Sham , Daniel W. Norbeck , Dale J. Kempf , Xiaoqi Chen , David A. Betebenner , Thomas R. Herrin , Gondi N. Kumar , John M. Lipari , Laman Alani , Soumojeet Ghosh , Rong R. Gao , Dilip Kaul
IPC分类号: A61K314166
CPC分类号: C07D207/27 , C07D207/404 , C07D207/408 , C07D223/10 , C07D233/32 , C07D233/42 , C07D239/10 , C07D239/22 , C07D241/08 , C07D241/18 , C07D253/06 , C07D263/22 , C07D307/20 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/12 , C07D405/14 , C07D407/12 , C07D409/12 , C07D409/14 , C07D417/12
摘要: A compound of the formula: is disclosed as an HIV protease inhibitor. Methods and compositions for inhibiting an HIV infection are also disclosed.
-
公开(公告)号:US5914332A
公开(公告)日:1999-06-22
申请号:US753201
申请日:1996-11-21
IPC分类号: C07D253/00 , A61K31/00 , A61K31/40 , A61K31/4015 , A61K31/41 , A61K31/415 , A61K31/4164 , A61K31/4166 , A61K31/4184 , A61K31/42 , A61K31/421 , A61K31/425 , A61K31/427 , A61K31/4427 , A61K31/443 , A61K31/4433 , A61K31/4439 , A61K31/47 , A61K31/495 , A61K31/496 , A61K31/4965 , A61K31/505 , A61K31/513 , A61K31/53 , A61K31/55 , A61K38/05 , A61K45/00 , A61P31/18 , A61P43/00 , C07C231/12 , C07C235/20 , C07C273/18 , C07C275/16 , C07D20060101 , C07D207/22 , C07D207/26 , C07D207/27 , C07D207/273 , C07D207/34 , C07D207/40 , C07D207/404 , C07D207/408 , C07D207/416 , C07D211/72 , C07D211/84 , C07D223/06 , C07D233/28 , C07D233/30 , C07D233/32 , C07D233/36 , C07D233/40 , C07D233/42 , C07D233/66 , C07D239/06 , C07D239/10 , C07D239/20 , C07D239/22 , C07D241/06 , C07D241/08 , C07D241/18 , C07D243/04 , C07D253/06 , C07D263/16 , C07D263/20 , C07D263/22 , C07D263/34 , C07D265/04 , C07D267/04 , C07D277/12 , C07D277/32 , C07D277/34 , C07D279/06 , C07D281/02 , C07D401/12 , C07D403/12 , C07D405/12 , C07D405/14 , C07D409/12 , C07D409/14 , C07D413/12 , C07D417/12 , A61K31/535
CPC分类号: C07D207/27 , C07D207/404 , C07D207/408 , C07D223/10 , C07D233/32 , C07D233/42 , C07D239/10 , C07D239/22 , C07D241/08 , C07D241/18 , C07D253/06 , C07D263/22 , C07D307/20 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/12 , C07D405/14 , C07D407/12 , C07D409/12 , C07D409/14 , C07D417/12
摘要: A compound of the formula: ##STR1## is disclosed as an HIV protease inhibitor. Methods and compositions for inhibiting an HIV infection are also disclosed.
-
公开(公告)号:US08748443B2
公开(公告)日:2014-06-10
申请号:US13260199
申请日:2010-03-25
申请人: David A. Betebenner , John K. Pratt , David A. DeGoey , Pamela L. Donner , Charles A. Flentge , Douglas K. Hutchinson , Warren M. Kati , Allan C. Krueger , Kenton L. Longenecker , Clarence J. Maring , John T. Randolph , Todd W. Rockway , Michael D. Tufano , Rolf Wagner , Dachun Liu
发明人: David A. Betebenner , John K. Pratt , David A. DeGoey , Pamela L. Donner , Charles A. Flentge , Douglas K. Hutchinson , Warren M. Kati , Allan C. Krueger , Kenton L. Longenecker , Clarence J. Maring , John T. Randolph , Todd W. Rockway , Michael D. Tufano , Rolf Wagner , Dachun Liu
IPC分类号: A01N43/54 , A61K31/505 , A61K31/503 , C07D239/54
CPC分类号: C07D409/10 , A61K31/18 , A61K31/27 , A61K31/402 , A61K31/4166 , A61K31/421 , A61K31/425 , A61K31/4418 , A61K31/503 , A61K31/513 , A61K45/06 , C07C311/08 , C07D207/27 , C07D213/64 , C07D233/32 , C07D233/72 , C07D239/10 , C07D239/54 , C07D263/22 , C07D263/24 , C07D275/02 , C07D403/10 , C07D405/10 , Y02P20/55
摘要: This invention relates to: (a) compounds and salts thereof that, inter alia, inhibit HCV; (b) intermediates useful for the preparation of such compounds and salts; (c) compositions comprising such compounds and salts; (d) methods for preparing such intermediates, compounds, salts, and compositions; (e) methods of use of such compounds, salts, and compositions; and (f) kits comprising such compounds, salts, and compositions.
-
公开(公告)号:US08691938B2
公开(公告)日:2014-04-08
申请号:US12813301
申请日:2010-06-10
申请人: David A. DeGoey , Warren M. Kati , Charles W. Hutchins , Pamela L. Donner , Allan C. Krueger , John T. Randolph , Christopher E. Motter , Lissa T. Nelson , Sachin V. Patel , Mark A. Matulenko , Ryan G. Keddy , Tammie K. Jinkerson , Yi Gao , Dachun Liu , John K. Pratt , Todd W. Rockway , Clarence J. Maring , Douglas K. Hutchinson , Charles A. Flentge , Rolf Wagner , Michael D. Tufano , David A. Betebenner , Kathy Sarris , Kevin R. Woller , Seble H. Wagaw , Jean C. Califano , Wenke Li , Daniel D. Caspi , Mary E. Bellizzi
发明人: David A. DeGoey , Warren M. Kati , Charles W. Hutchins , Pamela L. Donner , Allan C. Krueger , John T. Randolph , Christopher E. Motter , Lissa T. Nelson , Sachin V. Patel , Mark A. Matulenko , Ryan G. Keddy , Tammie K. Jinkerson , Yi Gao , Dachun Liu , John K. Pratt , Todd W. Rockway , Clarence J. Maring , Douglas K. Hutchinson , Charles A. Flentge , Rolf Wagner , Michael D. Tufano , David A. Betebenner , Kathy Sarris , Kevin R. Woller , Seble H. Wagaw , Jean C. Califano , Wenke Li , Daniel D. Caspi , Mary E. Bellizzi
CPC分类号: C07F9/65583 , C07C33/26 , C07C201/06 , C07C205/19 , C07D207/08 , C07D207/09 , C07D207/16 , C07D401/14 , C07D403/14 , C07D405/14 , C07D413/14 , C07D417/14 , C07D453/00 , C07D471/04 , C07D491/113 , C07K5/06
摘要: Compounds effective in inhibiting replication of Hepatitis C virus (“HCV”) are described. This invention also relates to processes of making such compounds, compositions comprising such compounds, and methods of using such compounds to treat HCV infection.
摘要翻译: 描述了有效抑制丙型肝炎病毒(“HCV”)复制的化合物。 本发明还涉及制备这种化合物的方法,包含这些化合物的组合物,以及使用这些化合物治疗HCV感染的方法。
-
公开(公告)号:US08236950B2
公开(公告)日:2012-08-07
申请号:US11960298
申请日:2007-12-19
申请人: David A. Betebenner , Clarence J. Maring , Todd W. Rockway , Curt S. Cooper , David D. Anderson , Rolf Wagner , Rong Zhang , Akhteruzzaman Molla , Hongmei Mo , Tami J. Pilot-Matias , Sherie V L. Masse , Robert J. Carrick , Wenping He , Liangjun Lu
发明人: David A. Betebenner , Clarence J. Maring , Todd W. Rockway , Curt S. Cooper , David D. Anderson , Rolf Wagner , Rong Zhang , Akhteruzzaman Molla , Hongmei Mo , Tami J. Pilot-Matias , Sherie V L. Masse , Robert J. Carrick , Wenping He , Liangjun Lu
IPC分类号: C07D491/02
CPC分类号: C07D471/04 , C07D239/94 , C07D487/04 , C07D487/14 , C07D519/00
摘要: Compounds effective in inhibiting replication of Hepatitis C virus (“HCV”) or other viruses are disclosed. This invention is also directed to compositions comprising such compounds, co-formulation or co-administration of such compounds with other anti-viral or therapeutic agents, processes and intermediates for the syntheses of such compounds, and methods of using such compounds for the treatment of HCV or other viral infections.
摘要翻译: 公开了有效抑制丙型肝炎病毒(“HCV”)或其他病毒复制的化合物。 本发明还涉及包含这些化合物的组合物,这些化合物与其它抗病毒剂或治疗剂的共同配制或共同给药,用于合成这些化合物的方法和中间体,以及使用这些化合物治疗 HCV或其他病毒感染。
-
公开(公告)号:US20120004196A1
公开(公告)日:2012-01-05
申请号:US13100827
申请日:2011-05-04
申请人: David A. DeGoey , Warren M. Kati , Charles W. Hutchins , Pamela L. Donner , Allan C. Krueger , John T. Randolph , Christopher E. Motter , Lissa T. Nelson , Sachin V. Patel , Mark A. Matulenko , Ryan G. Keddy , Tammie K. Jinkerson , Yi Gao , Dachun Liu , John K. Pratt , Todd W. Rockway , Clarence J. Maring , Douglas K. Hutchinson , Charles A. Flentge , Rolf Wagner , Michael D. Tufano , David A. Betebenner , Kathy Sarris , Kevin R. Woller , Seble H. Wagaw , Jean C. Califano , Wenke Li , Daniel D. Caspi , Mary E. Bellizzi , William A. Carroll
发明人: David A. DeGoey , Warren M. Kati , Charles W. Hutchins , Pamela L. Donner , Allan C. Krueger , John T. Randolph , Christopher E. Motter , Lissa T. Nelson , Sachin V. Patel , Mark A. Matulenko , Ryan G. Keddy , Tammie K. Jinkerson , Yi Gao , Dachun Liu , John K. Pratt , Todd W. Rockway , Clarence J. Maring , Douglas K. Hutchinson , Charles A. Flentge , Rolf Wagner , Michael D. Tufano , David A. Betebenner , Kathy Sarris , Kevin R. Woller , Seble H. Wagaw , Jean C. Califano , Wenke Li , Daniel D. Caspi , Mary E. Bellizzi , William A. Carroll
IPC分类号: A61K31/4184 , C07D401/14 , C07D405/14 , C07D413/14 , C07F7/10 , A61K31/454 , A61K31/4439 , A61K31/422 , A61K31/438 , A61K31/4545 , A61K31/695 , A61K31/496 , A61K31/506 , A61K31/5377 , A61P31/14 , C07D403/14
CPC分类号: A61K31/454 , A61K31/4178 , A61K31/4184 , A61K31/422 , A61K31/435 , A61K31/4355 , A61K31/438 , A61K31/4418 , A61K31/4439 , A61K31/4545 , A61K31/496 , A61K31/506 , A61K31/5377 , A61K31/695 , A61K45/06 , C07D401/14 , C07D403/14 , C07D405/14 , C07D413/14 , C07D417/14 , C07D453/00 , C07D491/113 , C07F7/02 , Y02P20/582
摘要: Compounds effective in inhibiting replication of Hepatitis C virus (“HCV”) are described. This invention also relates to processes of making such compounds, compositions comprising such compounds, and methods of using such compounds to treat HCV infection.
摘要翻译: 描述了有效抑制丙型肝炎病毒(“HCV”)复制的化合物。 本发明还涉及制备这种化合物的方法,包含这些化合物的组合物,以及使用这些化合物治疗HCV感染的方法。
-
-
-
-
-
-
-
-
-