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    DIAZA-SPIRO [4.5] DECANES USEFUL AS PESTICIDES
    101.
    发明申请
    DIAZA-SPIRO [4.5] DECANES USEFUL AS PESTICIDES 有权
    DIAZA-SPIRO [4.5]代表有用的农药

    公开(公告)号：US20100227862A1

    公开(公告)日：2010-09-09

    申请号：US12161823

    申请日：2007-01-19

    申请人： Thomas Pitterna ,  Jerome Cassayre ,  Louis-Pierre Molleyres ,  Peter Maienfisch

    发明人： Thomas Pitterna ,  Jerome Cassayre ,  Louis-Pierre Molleyres ,  Peter Maienfisch

    IPC分类号： A01N43/90 ,  C07D221/20 ,  A01N43/54 ,  C07D239/00 ,  C07D265/30 ,  A01P5/00 ,  A01P7/00 ,  A01P9/00

    CPC分类号： C07D471/10 ,  A01N43/90

    摘要： A method of combating and controlling insects, acarines, nematodes or molluscs which comprises applying to a pest, to a locus of a pest, or to a plant susceptible to attack by a pest an insecticidally, acaricidally, nematicidally or molluscicidally effective amount of a compound of formula (I) wherein Y is a single bond, C═O, C═S or S(O)m where m is 0, 1 or 2; and R1, R3, R2 and R8 are defined organic, groups, p is 0, 1, 2, 3 or 4 or salts or N-oxides thereof; novel compounds and composition's containing them are also provided.

    摘要翻译： 一种防治昆虫，螨虫，线虫或软体动物的方法，其包括将有害生物施用于有害生物的场所或易受害虫攻击的植物，杀虫剂，杀螨剂，杀线虫剂或杀软体动物学上有效量的化合物 其中Y是单键的式（I），C = O，C = S或S（O）m，其中m是0,1或2; R1，R3，R2和R8定义为有机基团，p为0,1,2,3或4或其盐或N-氧化物; 还提供了含有它们的新化合物和组合物。

    "> AVERMECTIN B1 AND AVERMECTIN B1 MONOSACCHARIDE DERIVATIVES HAVING AN ALKOXYMETHYL SUBSTITUENT IN THE 4
    102.
    发明申请
    AVERMECTIN B1 AND AVERMECTIN B1 MONOSACCHARIDE DERIVATIVES HAVING AN ALKOXYMETHYL SUBSTITUENT IN THE 4"-OR 4'-POSITION 有权
    在4“-OR 4'-位置具有烷氧基取代基的AVERMECTIN B1和AVERMECTIN B1单糖衍生物

    公开(公告)号：US20100210574A1

    公开(公告)日：2010-08-19

    申请号：US12768280

    申请日：2010-04-27

    申请人： Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Thomas Pitterna ,  Ottmar Franz Hueter ,  Pierre Jung

    发明人： Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Thomas Pitterna ,  Ottmar Franz Hueter ,  Pierre Jung

    IPC分类号： A01N43/16 ,  C07H17/08 ,  A01P17/00

    CPC分类号： C07H17/08 ,  A61K31/7042

    摘要： What is described are a compound of the formula wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —NO2, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8-Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12-alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12-haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)—Z—R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.

    摘要翻译： 描述的是下式的化合物，其中n是0或1; A-B是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12-烷基，C3-C8-环烷基或C2-C12-烯基; R2是例如C1-C12-烷基，C2-C12-烯基或C2-C12-炔基; 其任选被一至五个选自OH，卤素，CN，-N 3，-NO 2，C 3 -C 8 - 环烷基，降冰片基 - ，C 3 -C 8 - 环烯基的取代基取代; C 3 -C 8卤代环烷基，C 1 -C 12烷氧基，C 1 -C 6烷氧基-C 1 -C 6 - 烷氧基，C 3 -C 8环烷氧基，C 1 -C 12卤代烷氧基，C 1 -C 12烷硫基，C 3 -C 8环烷硫基， C 1 -C 12烷基亚磺酰基，C 3 -C 8环烷基亚磺酰基，C 1 -C 12卤代烷基亚磺酰基，C 3 -C 8卤代环烷基亚磺酰基，C 1 -C 12烷基磺酰基，C 3 -C 8环烷基磺酰基，C 1 -C 12卤代烷基磺酰基， 卤代环烷基磺酰基，-NR4R6，-X-C（= Y）-R4，-X-C（= Y）-Z-R4，-P（= O）（OC1-C6-烷基）2，芳基，杂环基，芳氧基， 芳硫基和杂环氧基; R3是例如任选取代的H，C 1 -C 12 - 烷基或C 1 -C 12 - 烷基，并且在适用的情况下，E / Z异构体，E / Z异构体和/或互变异构体的混合物，在每种情况下为游离形式或 盐形式; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

    Avermectin and avemectin monosaccharide derivatives substituted in the 4″- or 4′-position having pesticidal properties
    103.
    发明授权
    Avermectin and avemectin monosaccharide derivatives substituted in the 4″- or 4′-position having pesticidal properties 有权
    在4“或4”位取代的具有杀虫性的阿维菌素和阿维菌素单糖衍生物

    公开(公告)号：US07632820B2

    公开(公告)日：2009-12-15

    申请号：US10543638

    申请日：2004-01-30

    申请人： Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung

    发明人： Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung

    IPC分类号： A01N43/04 ,  A61K31/40 ,  A61K31/335 ,  A61K31/70 ,  A61K31/397 ,  A61K31/445 ,  A61K31/44 ,  A01N43/38

    CPC分类号： A01N43/90 ,  C07H17/08

    摘要： Disclosed are compounds of the formulain which n is 0 or 1; X—Y is —CH═CH— or —CH2—CH2—; Z is —C(═O)—, —C(═S)— or —SO2—; R1 is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and R2 is R3-Z-, R3—O-Z-, R4 or -Z-N(R6)(R7); Q is O or —N—R5; R3 and R4 are for example H, C1C12alkyl, C2-C12alkenyl, C2-C12alkynyl, C3-C12zcycloalkyl, C5-C12cycloalkenyl, aryl or heterocyclyl; R5 is for example H, C1-C8alkyl, hydroxy-C1-C8alkyl, C3-C8cycloalkyl, C2-C8alkenyl, C2-C8alkynyl, phenyl or benzyl; R6 and R7 are for example, H, unsubstituted or mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C2-C12alkenyl or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form, are useful as pesticides.

    摘要翻译： 公开了n为0或1的甲醛化合物; X-Y是-CH-CH-或-CH 2 -CH 2 - ; Z是-C（-O） - ， - C（-S） - 或-SO 2 - ; R1是C1-C12烷基，C3-C8环烷基或C2-C12链烯基; R2为R3-Z-，R3-O-Z-，R4或-Z-N（R6）（R7）; Q是O或-N-R5; R 3和R 4例如是H，C 1 -C 12烷基，C 2 -C 12烯基，C 2 -C 12炔基，C 3 -C 12环烷基，C 5 -C 12环烯基，芳基或杂环基; R5是例如H，C1-C8烷基，羟基-C1-C8烷基，C3-C8环烷基，C2-C8链烯基，C2-C8炔基，苯基或苄基; R 6和R 7为例如未取代的或未被取代的一价或五价取代的C 1 -C 12烷基，未被取代的或一至五取代的C 2 -C 12链烯基或（如果合适的话）E / Z异构体，E / Z异构体混合物和/或其互变异构体， 在每种情况下以游离形式或盐形式，都可用作农药。

    PREPARATION OF THIAZOLES
    106.
    发明申请
    PREPARATION OF THIAZOLES 失效
    制备THIAZOLES

    公开(公告)号：US20080076920A1

    公开(公告)日：2008-03-27

    申请号：US11947891

    申请日：2007-11-30

    申请人： Thomas Pitterna ,  Henry Szczepanski ,  Peter Maienfisch ,  Ottmar Huter ,  Thomas Rapold ,  Marcel Senn ,  Thomas Gobel ,  Anthony O'Sullivan

    发明人： Thomas Pitterna ,  Henry Szczepanski ,  Peter Maienfisch ,  Ottmar Huter ,  Thomas Rapold ,  Marcel Senn ,  Thomas Gobel ,  Anthony O'Sullivan

    IPC分类号： C07D417/02 ,  C07D277/36 ,  C07D417/14

    CPC分类号： C07D277/32 ,  C07D277/16 ,  C07D277/36 ,  C07D277/70 ,  C07D277/74

    摘要： The present disclosure is directed to a process for the preparation of a compound having the formula: wherein R is unsubstituted or substituted C1-C12alkyl, unsubstituted or substituted C2-C4alkenyl, unsubstituted or substituted C2-C4alkynyl, unsubstituted or substituted C3-C6cycloalkyl, unsubstituted or substituted aryl, unsubstituted or substituted heteroaryl, or —SR1; R1 is unsubstituted or substituted C1-C12alkyl, unsubstituted or substituted C2-C4alkenyl, unsubstituted or substituted C2-C4alkynyl, unsubstituted or substituted cycloalkyl, unsubstituted or substituted aryl or unsubstituted or substituted heteroaryl; and X is a selected leaving group that is not halogen, and may specifically be methylsulfonate, trifluoromethylsulfonate, and p-toluenesulfonate. These compounds are valuable intermediates useful in the synthesis of compounds having pesticidal activity. Generally, the process includes reacting a water-removing reagent, with a compound having the formula Water-removing agents that may be used include thionyl chloride (SOCl2), thionyl bromide (SOBr2), phosphorus oxychloride (POCl3), phosphorus oxybromide (POBr3), phosphorus pentachloride or a sulfonic acid chloride or bromide.

    摘要翻译： 本公开涉及制备具有下式的化合物的方法：其中R是未取代或取代的C 1 -C 12烷基，未取代或取代的C 1 -C 12烷基， 未取代或取代的C 2 -C 4炔基，未取代或取代的C 1 -C 4烷基， 3个C 6环烷基，未取代或取代的芳基，未取代或取代的杂芳基或-SR 1 N; R 1是未取代或取代的C 1 -C 12烷基，未取代或取代的C 2 -C 3 未取代或取代的C 2 -C 4炔基，未取代或取代的环烷基，未取代或取代的芳基或未取代或取代的杂芳基; X是不是卤素的选择的离去基团，可以具体为甲基磺酸酯，三氟甲基磺酸酯和对甲苯磺酸酯。 这些化合物是有用的合成具有杀虫活性的化合物的中间体。 通常，该方法包括使除水试剂与具有式的化合物反应可以使用的除水剂包括亚硫酰氯（SOCl 2/2），亚硫酰溴（SO 2 R 2） （POCl 3 3），三溴氧化磷（POBr 3 N），五氯化磷或磺酰氯或溴化物。

    "> Avermectin and avemectin monosaccharide derivatives substituted in the 4
    108.
    发明申请
    Avermectin and avemectin monosaccharide derivatives substituted in the 4"-or 4'-position having pesticidal properties 有权
    在4“ - 或4”位取代的具有杀虫性的阿维菌素和阿维菌素单糖衍生物

    公开(公告)号：US20060166824A1

    公开(公告)日：2006-07-27

    申请号：US10543638

    申请日：2004-01-30

    申请人： Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung

    发明人： Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung

    IPC分类号： A01N43/04 ,  A61K31/7048

    CPC分类号： A01N43/90 ,  C07H17/08

    摘要： Disclosed are compounds of the formula in which n is 0 or 1; X—Y is —CH═CH— or —CH2—CH2—; Z is —C(═O)—, —C(═S)— or —S02—; R1 is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and R2 is R3-Z-, R3—O-Z-, R4 or -Z-N(R6)(R7); Q is O or —N—R5; R3 and R4 are for example H, C1C12alkyl, C2-C12alkenyl, C2-C12alkynyl, C3-C12zcycloalkyl, C5-C12cycloalkenyl, aryl or heterocyclyl; R5 is for example H, C1-C8alkyl, hydroxy-C1-C8alkyl, C3-C8cycloalkyl, C2-C8alkenyl, C2-C8alkynyl, phenyl or benzyl; R6 and R7 are for example, H, unsubstituted or mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C2-C12alkenyl or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form, are useful as pesticides.

    摘要翻译： 公开了下式的化合物，其中n为0或1; X-Y是-CH-CH-或-CH 2 -CH 2 - 。 Z是-C（-O） - ， - C（-S） - 或-SO 2 - 。 R 1是C 1 -C 12烷基，C 3 -C 8烷基，C 1 -C 12烷基，C 3 -C 12烷基， 环烷基或C 2 -C 12 - 烯基; 和R 2是R 3 -Z-，R 3 -OZ-，R 4或-ZN（ R 6）（R 7）; Q是O或-N-R 5; R 3和R 4是例如H，C 1 -C 12烷基，C 2， C 1 -C 12亚烷基，C 2 -C 12炔基，C 3 -C 12链烯基，C 2 -C 12亚炔基，C 3 -C 12亚烷基， 12个环烷基，C 5 -C 12环烯基，芳基或杂环基; R 5是例如H，C 1 -C 8烷基，羟基-C 1 -C 3 C 1 -C 8烷基，C 3 -C 8环烷基，C 2 -C 8链烯基，C 1 -C 8烷基， C 2 -C 8炔基，苯基或苄基; R 6和R 7是例如H，未取代的或一至五取代的C 1 -C 12 - 烷基，未取代的或一至五取代的C 2 -C 12链烯基，或者如果合适的话，E / Z异构体，E / Z异构体混合物和/或其互变异构体， 在每种情况下以游离形式或盐形式，都可用作农药。

    "> Avermectin b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substitutent in the 4
    109.
    发明申请
    Avermectin b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substitutent in the 4"-or 4'-position 有权

    公开(公告)号：US20060148729A1

    公开(公告)日：2006-07-06

    申请号：US10539274

    申请日：2003-12-19

    申请人： Peter Maienfisch ,  Fiona Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Thomas Pitterna ,  Ottmar Hueter ,  Pierre Jung

    发明人： Peter Maienfisch ,  Fiona Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Thomas Pitterna ,  Ottmar Hueter ,  Pierre Jung

    IPC分类号： A01N43/04 ,  C07H17/08

    CPC分类号： C07H17/08 ,  A61K31/7042

    摘要： What is described are a compound of the formula (I): wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —N02, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12 alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)-Z-R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.