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21.发明申请公开(公告)号：US20080269298A1
公开(公告)日：2008-10-30
申请号：US12113224
申请日：2008-05-01
Applicant: Clarence W. Andrews , Mui Cheung , Ronda G. Davis-Ward , David Harold Drewry , Kyle Allen Emmitte , Robert Dale Hubbard , Kevin W. Kuntz , James Andrew Linn , Robert Anthony Mook , Gary Keith Smith , James Marvin Veal
Inventor： Clarence W. Andrews , Mui Cheung , Ronda G. Davis-Ward , David Harold Drewry , Kyle Allen Emmitte , Robert Dale Hubbard , Kevin W. Kuntz , James Andrew Linn , Robert Anthony Mook , Gary Keith Smith , James Marvin Veal
IPC: A61K31/4184 , A61P35/00 , A61K31/4439 , C07D409/14 , C07D409/04
CPC classification number: C07D491/04 , C07D409/04 , C07D409/14
Abstract: The present invention provides compounds of formula (I): pharmaceutical compositions containing the same, processes for preparing the same and their use as pharmaceutical agents.
Abstract translation: 本发明提供式（I）化合物：含有该化合物的药物组合物，其制备方法及其作为药剂的用途。
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公开(公告)号：US20070270437A1
公开(公告)日：2007-11-22
申请号：US11467577
申请日：2006-08-28
Applicant: Mui Cheung , Kyle Emmitte , James Salovich
Inventor： Mui Cheung , Kyle Emmitte , James Salovich
IPC: A61K31/4184 , A61K31/435 , A61K31/496 , A61P35/00 , C07D221/00 , C07D235/04 , C07D295/00
CPC classification number: C07D409/04 , C07D409/14
Abstract: The present invention provides benzimidazole thiophene compounds pharmaceutical compositions containing the same, processes for preparing the same and their use as pharmaceutical agents.
Abstract translation: 本发明提供苯并咪唑噻吩化合物，其含有它们的药物组合物，其制备方法及其作为药剂的用途。
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公开(公告)号：US07238813B2
公开(公告)日：2007-07-03
申请号：US10433128
申请日：2001-11-28
Applicant: Mui Cheung , Philip Anthony Harris , Masaichi Hasegawa , Satoru Ida , Kazuya Kano , Naohiko Nishigaki , Hideyuki Sato , James Marvin Veal , Yoshiaki Washio , Rob I. West
Inventor： Mui Cheung , Philip Anthony Harris , Masaichi Hasegawa , Satoru Ida , Kazuya Kano , Naohiko Nishigaki , Hideyuki Sato , James Marvin Veal , Yoshiaki Washio , Rob I. West
IPC: A61K31/4184 , C07D235/30
CPC classification number: C07D249/08 , C07D231/12 , C07D233/56 , C07D235/30 , C07D235/32 , C07D263/58 , C07D277/82 , C07D401/12 , C07D403/12 , C07D405/12 , C07D405/14 , C07D409/12 , C07D413/12 , C07D413/14 , C07D417/12 , C07D417/14 , C07D471/04 , C07D471/14 , C07D487/04
Abstract: Benzimidazole derivatives, which are useful as TIE-2 and/or VEGFR2 inhibitors are described herein. The described invention also includes methods of making such benzimidazole derivatives as well as methods of using the same in the treatment of hyperproliferative diseases.
Abstract translation: 本文描述了可用作TIE-2和/或VEGFR2抑制剂的苯并咪唑衍生物。 所述的发明还包括制备这种苯并咪唑衍生物的方法以及使用它们在治疗过度增殖性疾病中的方法。
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公开(公告)号：US20070142437A1
公开(公告)日：2007-06-21
申请号：US11670498
申请日：2007-02-02
Applicant: Matthew Brown , Mui Cheung , Scott Dickerson , Cassandra Gauthier , Philip Harris , Robert Hunter , Gregory Pacofsky , Michael Peel , Jeffrey Stafford
Inventor： Matthew Brown , Mui Cheung , Scott Dickerson , Cassandra Gauthier , Philip Harris , Robert Hunter , Gregory Pacofsky , Michael Peel , Jeffrey Stafford
IPC: A61K31/4439 , A61K31/427 , A61K31/423 , C07D413/02 , C07D417/02
CPC classification number: C07D263/48 , C07D413/04 , C07D413/10 , C07D413/12 , C07D413/14 , C07D417/10 , C07D417/12 , C07D417/14
Abstract: Oxazole derivatives, which are useful as VEGFR2, CDK2, and CDK4 inhibitors are described herein. The described invention also includes methods of making such oxazole derivatives as well as methods of using the same in the treatment of hyperproliferative diseases.
Abstract translation: 本文描述了可用作VEGFR2，CDK2和CDK4抑制剂的恶唑衍生物。 所述的发明还包括制备这种恶唑衍生物的方法以及使用它们在治疗过度增殖性疾病中的方法。
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公开(公告)号：US20070015756A1
公开(公告)日：2007-01-18
申请号：US11383229
申请日：2006-05-15
Applicant: Amogh Boloor , Mui Cheung , Ronda Davis , Philip Harris , Kevin Hinkle , Robert Mook , Jeffery Stafford , James Veal
Inventor： Amogh Boloor , Mui Cheung , Ronda Davis , Philip Harris , Kevin Hinkle , Robert Mook , Jeffery Stafford , James Veal
IPC: A61K31/53 , A61K31/506 , C07D403/02
CPC classification number: C07D239/30 , C07D231/56 , C07D235/08 , C07D403/12 , C07D413/14
Abstract: Pyrimidine derivatives, which are useful as VEGFR2 inhibitors are described herein. The described invention also includes methods of making such pyrimidine derivatives as well as methods of using the same in the treatment of hyperproliferative diseases.
Abstract translation: 本文描述了可用作VEGFR2抑制剂的嘧啶衍生物。 所述的发明还包括制备此类嘧啶衍生物的方法以及使用该嘧啶衍生物的方法来治疗过度增殖性疾病。
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Patent Agency Ranking
公开(公告)号：US07163940B2
公开(公告)日：2007-01-16
申请号：US10433881
申请日：2001-11-26
Applicant: F. Leslie Boyd , Stanley D Chamberlain , Mui Cheung , Kristjan Gudmundsson , Philip Anthony Harris , Brian A Johns , David Kendall Jung , Michael Robert Peel , Jennifer G Badiang , Connie Jo Sexton
Inventor： F. Leslie Boyd , Stanley D Chamberlain , Mui Cheung , Kristjan Gudmundsson , Philip Anthony Harris , Brian A Johns , David Kendall Jung , Michael Robert Peel , Jennifer G Badiang , Connie Jo Sexton
IPC: C07D471/04 , A61K31/435 , C07D401/04
CPC classification number: C07D471/04
Abstract: The present invention provides compounds of formula (I): wherein all variables are as defined herein, pharmaceutical compositions containing the same, processes for preparing the same and their use as pharmaceutical agents.
Abstract translation: 本发明提供式（I）化合物：其中所有变量如本文所定义，含有该化合物的药物组合物，其制备方法及其作为药剂的用途。
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公开(公告)号：US08114885B2
公开(公告)日：2012-02-14
申请号：US11830608
申请日：2007-07-30
Applicant: Amogh Boloor , Mui Cheung , Philip Anthony Harris , Kevin Hinkle , Jeffery Alan Stafford , James Marvin Veal
Inventor： Amogh Boloor , Mui Cheung , Philip Anthony Harris , Kevin Hinkle , Jeffery Alan Stafford , James Marvin Veal
IPC: C07D239/48 , A61K31/506 , A61P35/00
CPC classification number: C07D239/30 , C07D231/56 , C07D235/08 , C07D403/12 , C07D413/14
Abstract: Pyrimidine derivatives, which are useful as VEGFR2 inhibitors are described herein. The described invention also includes methods of making such pyrimidine derivatives as well as methods of using the same in the treatment of hyperproliferative diseases.
Abstract translation: 本文描述了可用作VEGFR2抑制剂的嘧啶衍生物。 所述的发明还包括制备此类嘧啶衍生物的方法以及使用该嘧啶衍生物的方法来治疗过度增殖性疾病。
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公开(公告)号：US07858626B2
公开(公告)日：2010-12-28
申请号：US11830024
申请日：2007-07-30
Applicant: Amogh Boloor , Mui Cheung , Ronda Gayle Davis-Ward , Philip Anthony Harris , Kevin Hinkle , Christopher P. Lauderman , Robert Anthony Mook, Jr. , Jeffery Alan Stafford , James Marvin Veal
Inventor： Amogh Boloor , Mui Cheung , Ronda Gayle Davis-Ward , Philip Anthony Harris , Kevin Hinkle , Christopher P. Lauderman , Robert Anthony Mook, Jr. , Jeffery Alan Stafford , James Marvin Veal
IPC: C07D403/04 , A61K31/53 , A61P35/00
CPC classification number: C07D239/30 , C07D231/56 , C07D235/08 , C07D403/12 , C07D413/14
Abstract: Pyrimidine derivatives, which are useful as VEGFR2 inhibitors are described herein. The described invention also includes methods of making such pyrimidine derivatives as well as methods of using the same in the treatment of hyperproliferative diseases.
Abstract translation: 本文描述了可用作VEGFR2抑制剂的嘧啶衍生物。 所述的发明还包括制备此类嘧啶衍生物的方法以及使用该嘧啶衍生物的方法来治疗过度增殖性疾病。
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公开(公告)号：US20100105712A1
公开(公告)日：2010-04-29
申请号：US12609398
申请日：2009-10-30
Applicant: Amogh Boloor , Mui Cheung , Philip Anthony Harris , Kevin Hinkle , Jeffery Alan Stafford , James Marvin Veal
Inventor： Amogh Boloor , Mui Cheung , Philip Anthony Harris , Kevin Hinkle , Jeffery Alan Stafford , James Marvin Veal
IPC: A61K31/506 , A61P7/00 , A61P27/10 , C07D403/12
CPC classification number: C07D239/30 , C07D231/56 , C07D235/08 , C07D403/12 , C07D413/14
Abstract: Pyrimidine derivatives, which are useful as VEGFR2 inhibitors are described herein. The described invention also includes methods of making such pyrimidine derivatives as well as methods of using the same in the treatment of hyperproliferative diseases.
Abstract translation: 本文描述了可用作VEGFR2抑制剂的嘧啶衍生物。 所述的发明还包括制备此类嘧啶衍生物的方法以及使用该嘧啶衍生物的方法来治疗过度增殖性疾病。
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公开(公告)号：US20060217382A1
公开(公告)日：2006-09-28
申请号：US10550434
申请日：2004-03-29
Applicant: Mui Cheung , Nigel King , Kevin Kuntz , Robert Mook , Mark Pobanz , James Salovich , Brian Wilson
Inventor： Mui Cheung , Nigel King , Kevin Kuntz , Robert Mook , Mark Pobanz , James Salovich , Brian Wilson
IPC: A61K31/53 , C07D487/04
CPC classification number: C07D487/04
Abstract: The present invention provides compounds of formula (I): wherein all variables are as defined herein, pharmaceutical compositions containing the same, processes for preparing the same and their use as pharmaceutical agents.
Abstract translation: 本发明提供式（I）化合物：其中所有变量如本文所定义，含有该化合物的药物组合物，其制备方法及其作为药剂的用途。
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