利索-全球专利检索

  1. 登录
  2. 注册

搜索结果

25 条记录 (耗时 0.016 秒)

    Process for preparation of iodopropargyl carbamates
    4.
    发明授权
    Process for preparation of iodopropargyl carbamates 失效
    碘代炔丙基氨基甲酸酯的制备方法

    公开(公告)号：US5326899A

    公开(公告)日：1994-07-05

    申请号：US76561

    申请日：1993-06-14

    申请人： Barry C. Lange

    发明人： Barry C. Lange

    IPC分类号： B01J21/04 ,  B01J27/08 ,  B01J27/26 ,  B01J31/02 ,  B01J31/04 ,  B01J31/12 ,  C07B61/00 ,  C07C269/04 ,  C07C271/12 ,  C07C261/00

    CPC分类号： C07C269/04 ,  C07C271/12

    摘要： A Process for producing N-alkyl iodopropargyl carbamate comprising:A. reacting a dialkyl(C.sub.1 -C.sub.3) carbonate with propargyl alcohol in the presence of a first catalyst under conditions to produce dipropargyl carbonate;B. reacting said dipropargyl carbonate with an alkyl(C.sub.1 -C.sub.6)amine, optionally in the presence of a second catalyst, to produce N-alkyl(C.sub.1 -C.sub.6) propargyl carbamate;C. reacting said N-alkyl(C.sub.1 -C.sub.6) propargyl carbamate with an iodinating agent to produce N-alkyl(C.sub.1 -C.sub.6) iodopropargyl carbamate is disclosed.

    摘要翻译： 一种N-烷基碘炔丙基氨基甲酸酯的制备方法，其包括：A.在第一催化剂存在下，在产生碳酸二丙酯的条件下，使碳酸二烷基酯（C 1 -C 3）与炔丙醇反应; B.任选在第二催化剂存在下，使所述碳酸二丙酯与烷基（C 1 -C 6）反应，生成N-烷基（C 1 -C 6）炔丙基氨基甲酸酯; C.公开了使所述N-烷基（C 1 -C 6）炔丙基氨基甲酸酯与碘化剂反应以制备N-烷基（C1-C6）碘炔丙基氨基甲酸酯。

    Substituted 3-thioacryloyl compounds and their use as antimicrobial agents
    7.
    发明授权
    Substituted 3-thioacryloyl compounds and their use as antimicrobial agents 失效
    取代的3-硫代丙烯酰化合物及其作为抗微生物剂的用途

    公开(公告)号：US5464832A

    公开(公告)日：1995-11-07

    申请号：US166498

    申请日：1993-12-13

    申请人： Peter Osei-Gyimah ,  Samuel E. Sherba ,  Barry C. Lange ,  Rai J. Mehta ,  Rhoda W. Joseph

    发明人： Peter Osei-Gyimah ,  Samuel E. Sherba ,  Barry C. Lange ,  Rai J. Mehta ,  Rhoda W. Joseph

    IPC分类号： A01N37/36 ,  A01N41/12 ,  A01N43/10 ,  A01N43/40 ,  A01N43/50 ,  A01N43/713 ,  A01N43/78 ,  A01N47/42 ,  A01N47/48 ,  C07C323/54 ,  C07C323/60 ,  C07C331/14 ,  C07C335/32 ,  C07D213/70 ,  C07D213/89 ,  C07D233/42 ,  C07D257/04 ,  C07D277/36 ,  C07D277/74 ,  C07D333/28 ,  C07D211/06 ,  A61K31/535 ,  C07D263/04 ,  C07D265/30

    CPC分类号： C07D213/70 ,  A01N37/36 ,  A01N41/12 ,  A01N43/10 ,  A01N43/40 ,  A01N43/50 ,  A01N43/713 ,  A01N43/78 ,  A01N47/42 ,  A01N47/48 ,  C07C323/54 ,  C07C323/60 ,  C07C331/14 ,  C07C335/32 ,  C07D213/89 ,  C07D233/42 ,  C07D257/04 ,  C07D277/36 ,  C07D277/74 ,  C07D333/28

    摘要： A thioacryloyl compound of the formula ##STR1## wherein Z is selected from the group consisting of OR, R and NR.sup.1 R.sup.2 ;R is selected from the group consisting of hydrogen; (C.sub.1 -C.sub.18)alkyl; (C.sub.1 -C.sub.8)alkenyl; (C.sub.1 -C.sub.8)haloalkynyl; 2-(5-chlorothienyl)methyl; phenyl optionally substituted with one or more substituents selected from the group consisting of halo-, (C.sub.1 -C.sub.3)alkoxy-, nitro-, and (C.sub.1 -C.sub.3)alkyl; phenacyl optionally substituted with one or more substituents selected from the group consisting of ring halo-, (C.sub.1 -C.sub.3)alkoxy-, nitro-, and (C.sub.1 -C.sub.3)alkyl; arylalkyl optionally substituted with one or more substituents selected from the group consisting of ring halo-, (C.sub.1 -C.sub.3)alkoxy-, nitro-, and (C.sub.1 -C.sub.3)alkyl;R.sup.1 and R.sup.2 are independently selected from (C.sub.1 -C.sub.8)alkyl and phenyl, or R.sup.1 and R.sup.2 may be joined together with the nitrogen atom to which they are attached to form a ring containing 4 to 5 carbon atoms with or without an oxygen heteroatom;X is selected from the group consisting of hydrogen, halogen, phenyl, CO.sub.2 CH.sub.3, and (C.sub.1 -C.sub.3)alkyl; andY is selected from the group consisting of CN, CH(COCH.sub.3).sub.2, CH.sub.2 COCH.sub.3, CH.sub.2 CN, CH.sub.2 CO.sub.2 C.sub.2 H.sub.5 -propargyl, SCH.dbd.CHCO.sub.2 CH.sub.3, C(.dbd.NH)NH.sub.2 hydrochloride, and 2-(5-chlorothienyl)methyl;provided that when Z is NR.sup.1 R.sup.2, Y is CN; andprovided that when Z is R, X is hydrogen, and Y is CN, R is not phenyl.

    摘要翻译： 式Ⅰ的硫代丙烯酰化合物，其中Z选自OR，R和NR1R2; R选自氢; （C 1 -C 18）烷基; （C1-C8）烯基; （C1-C8）卤代炔基; 2-（5-氯噻吩基）甲基; 任选被一个或多个选自卤代，（C 1 -C 3）烷氧基 - ，硝基 - 和（C 1 -C 3）烷基的取代基取代的苯基; 任选被一个或多个选自环卤，（C1-C3）烷氧基 - ，硝基 - 和（C1-C3）烷基的取代基取代的苯乙烯酰基; 任选被一个或多个选自环卤，（C 1 -C 3）烷氧基 - ，硝基 - 和（C 1 -C 3）烷基的取代基取代的芳基烷基; R 1和R 2独立地选自（C 1 -C 8）烷基和苯基，或者R 1和R 2可以与它们所连接的氮原子一起形成含有或不含有氧杂原子的含有4至5个碳原子的环; X选自氢，卤素，苯基，CO 2 CH 3和（C 1 -C 3）烷基; 并且Y选自CN，CH（COCH 3）2，CH 2 COCH 3，CH 2 CN，CH 2 CO 2 C 2 H 5 - 炔丙基，SCH = CHCO 2 CH 3，C（= NH）NH 2盐酸盐和2-（5-氯噻吩基）甲基; 条件是当Z为NR1R2时，Y为CN; 并且条件是当Z是R时，X是氢，Y是CN，R不是苯基。

    2-(3-oxoalk(en)yl)-3-isothiazolones and derivatives as antimicrobial agents
    9.
    发明授权
    2-(3-oxoalk(en)yl)-3-isothiazolones and derivatives as antimicrobial agents 失效
    2-（3-氧代烯（烯）基）-3-异噻唑酮及其衍生物作为抗微生物剂

    公开(公告)号：US5288693A

    公开(公告)日：1994-02-22

    申请号：US83958

    申请日：1993-06-25

    申请人： Peter Osei-Gyimah ,  Barry C. Lange

    发明人： Peter Osei-Gyimah ,  Barry C. Lange

    IPC分类号： A23L3/3544 ,  A01N43/80 ,  A61K8/49 ,  A61K31/425 ,  A61P31/04 ,  C07D275/02 ,  C07D275/03 ,  C07D275/04

    CPC分类号： C07D275/03 ,  A01N43/80

    摘要： Antimicrobial compounds of the formula ##STR1## wherein R is hydrogen, halogen or (C.sub.1 -C.sub.4)alkyl group;R.sub.1 is hydrogen or halogen; alternatively, R and R1 may be taken together with the carbons to which they are attached to form a 5- to 7-membered carbocyclic ring, said ring optionally being aromatic;R.sub.2 is hydrogen or (C.sub.1 -C.sub.3)alkyl group; andR3 is hydrogen, substituted or unsubstituted (C.sub.1 -C.sub.18)alkyl, substituted or unsubstituted (C.sub.2 -C.sub.18)alkenyl, substituted or unsubstituted (C.sub.2 -C.sub.18)alkynyl, substituted or unsubstituted (C.sub.4 -C.sub.8)cycloalkyl or cycloalkenyl, substituted or unsubstituted (C.sub.6 -C.sub.10)aryl or arylalkyl group are disclosed.

    摘要翻译： 式（I）其中R为氢，卤素或（C 1 -C 4）烷基的式I的化合物; R1是氢或卤素; 或者，R和R 1可以与它们所连接的碳一起形成5-至7-元碳环，所述环任选是芳族的; R2是氢或（C1-C3）烷基; 取代或未取代的（C 2 -C 18）烯基，取代或未取代的（C 2 -C 18）炔基，取代或未取代的（C 1 -C 8）环烷基或环烯基，取代或未取代的 （C6-C10）芳基或芳基烷基。

    Microbicidal and plant growth regulating compounds
    10.
    发明授权
    Microbicidal and plant growth regulating compounds 失效
    杀菌剂和植物生长调节化合物

    公开(公告)号：US4975459A

    公开(公告)日：1990-12-04

    申请号：US450127

    申请日：1989-12-13

    申请人： Raj J. Mehta ,  Colin Swithenbank ,  Zev Lidert ,  Margaret M. Bowers-Daines ,  David H. Young ,  Barry C. Lange

    发明人： Raj J. Mehta ,  Colin Swithenbank ,  Zev Lidert ,  Margaret M. Bowers-Daines ,  David H. Young ,  Barry C. Lange

    IPC分类号： C07D331/02 ,  A01N35/06 ,  A01N43/20 ,  A01N43/44 ,  C07C50/24 ,  C07C50/34 ,  C07C50/38 ,  C07C225/30 ,  C07C225/34 ,  C07C233/61 ,  C07D203/08 ,  C07D303/04 ,  C07D303/08 ,  C07D303/12 ,  C07D303/34 ,  C07D303/36 ,  C07D303/48

    CPC分类号： C07C50/34 ,  A01N35/06 ,  A01N43/20 ,  C07C225/30 ,  C07C225/34 ,  C07C233/61 ,  C07C50/24 ,  C07C50/38 ,  C07D303/36 ,  C07C2101/02 ,  C07C2103/24

    摘要： Process comprising the use as a microbicide or plant growth regulator of a compound of the formula ##STR1## wherein A, B, C and D is each independently selected from the group consisting of O,NR.sup.1, CR.sup.1 R.sup.1, CO, S,SO, and SO.sub.2, except for the A-C, C-A, B-D,D-B combinations: O--O, SO--SO, SO.sub.2 --SO.sub.2, S--O, S--NR.sup.2, SONR.sup.2, SO--CO, SO.sub.2 --CO, SO.sub.2 --SO;each group of the groups R.sup.1 is independently selected from the group consisting of H and (C.sub.1 -C.sub.4)alkyl;Y.sup.1 and Y.sup.2 may each be independently selected from the group consisting of H, (C.sub.1 -C.sub.4)alkyl, halogen, OR,SOR,SO.sub.2 R, SO.sub.3 R, CN, CO.sub.2 R, COR, CF.sub.3, NO.sub.2, NHCOR, and OCOR; or alternatively Y.sup.1 and Y.sup.2 and the carbons to which they are attached may comprise a cyclic structure selected from the group consisting of ##STR2## where R.sup.11 is aryl or (C.sub.1 -C.sub.4)alkylX.sup.1 to X.sup.8 is each independently selected from the group consisting of H, (C.sub.1 -C.sub.4)alkyl, halogen, OR, SOR, SO.sub.2 R, SO.sub.3 R, CN,CO.sub.2 R, COR, CF.sub.3, NO.sub.2, NHCOR, and OCOR: and furthermore optionally any pair or pairs of adjacent X's may be in the form of a divalent group attached across the adjacent X position;Z.sup.1 and Z.sup.2 is each independently selected from the group consisting of NR.sup.2, O, S, CR.sup.2 R.sup.2 where each of the groups R.sup.2 is independently selected from the group consisting of H and (C.sub.1 -C.sub.4)alkyl;each of the groups R.sup.3 is independently selected from the group consisting of CO.sub.2 R, COR, CN CF.sub.3, SOR, SO.sub.2 R, (C.sub.1 -C.sub.4)alkyl and H.

    摘要翻译： 其中A，B，C和D分别独立地选自O，NR 1，CR 1 R 1，CO，S，SO，以及其中A，B，C和D的化合物的杀微生物剂或植物生长调节剂 SO2，除了AC，CA，BD，DB组合：OO，SO-SO，SO2-SO2，SO，S-NR2，SONR2，SO-CO，SO2-CO，SO2-SO; 每个基团R 1独立地选自H和（C 1 -C 4）烷基; Y 1和Y 2可各自独立地选自H，（C 1 -C 4）烷基，卤素，OR，SOR，SO 2 R，SO 3 R，CN，CO 2 R，COR，CF 3，NO 2，NHCOR和OCOR; 或者Y1和Y2以及它们所连接的碳可以包含选自下列的环状结构：其中R11为芳基或（C1-C4）烷基X1至X8各自独立地选自 由H，（C 1 -C 4）烷基，卤素，OR，SOR，SO 2 R，SO 3 R，CN，CO 2 R，COR，CF 3，NO 2，NHCOR和OCOR组成的组： 为相邻X位置附近的二价基团的形式; Z 1和Z 2各自独立地选自NR 2，O，S，CR 2 R 2，其中每个基团R 2独立地选自H和（C 1 -C 4）烷基; 基团R3各自独立地选自CO 2 R，COR，CN CF 3，SOR，SO 2 R，（C 1 -C 4）烷基和H.