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公开(公告)号:US4960884A
公开(公告)日:1990-10-02
申请号:US399448
申请日:1989-08-28
申请人: David M. Roush , Donald A. Shaw , Michael L. Jones , Jun H. Chang
发明人: David M. Roush , Donald A. Shaw , Michael L. Jones , Jun H. Chang
IPC分类号: A01N31/04 , A01N31/14 , A01N31/16 , A01N33/10 , A01N33/20 , A01N33/22 , A01N35/02 , A01N35/04 , A01N35/10 , A01N37/00 , A01N37/38 , A01N37/40 , A01N37/48 , A01N41/10 , A01N43/10 , A01N43/12 , C07C43/174 , C07C43/225 , C07C43/23 , C07C45/62 , C07C45/71 , C07C45/72 , C07C47/575 , C07C49/255 , C07C49/84 , C07C59/64 , C07C65/21 , C07C69/92 , C07C205/34 , C07C205/37 , C07C205/59 , C07C217/76 , C07C217/84 , C07C235/46 , C07C235/60 , C07C251/24 , C07C255/54 , C07C323/03
CPC分类号: C07C323/03 , A01N31/04 , A01N31/14 , A01N31/16 , A01N33/10 , A01N33/20 , A01N33/22 , A01N35/02 , A01N35/04 , A01N35/10 , A01N37/00 , A01N37/38 , A01N37/40 , A01N37/48 , A01N41/10 , A01N43/10 , A01N43/12 , C07C205/34 , C07C205/37 , C07C205/59 , C07C217/76 , C07C217/84 , C07C235/46 , C07C235/60 , C07C251/24 , C07C255/54 , C07C43/174 , C07C43/1742 , C07C43/1745 , C07C43/225 , C07C43/23 , C07C45/62 , C07C45/71 , C07C45/72 , C07C47/575 , C07C49/255 , C07C49/84 , C07C59/64 , C07C65/21 , C07C69/92
摘要: Pesticidal mono-, di-, and tri-2-fluoroethyl ethers of the formula R.sup.1 R.sup.2.sub.m Ar(OCH.sub.2 CH.sub.2 F).sub.n, compositions thereof and their insecticidal, acaricidal and nematicidal uses are described and claimed.
摘要翻译: 描述和要求保护的式R1R2mAr(OCH2CH2F)n的杀虫单,二和三氟乙基醚及其杀虫,杀螨和杀线虫剂的组合物。
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公开(公告)号:US4486588A
公开(公告)日:1984-12-04
申请号:US435164
申请日:1982-10-19
IPC分类号: C07D295/155
CPC分类号: C07D295/155
摘要: Precursors to benzyl compounds, useful in the manufacture of pyrethroid insecticides, are prepared by regiospecific addition of an enamine to a heterocyclic diene accompanied by elimination of volatile by-products.
摘要翻译: 可用于制造拟除虫菊酯杀虫剂的苄基化合物的前体是通过将烯胺区域特异性加成到伴随着挥发性副产物消除的杂环二烯中制备的。
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公开(公告)号:US20090012070A1
公开(公告)日:2009-01-08
申请号:US12196893
申请日:2008-08-22
申请人: John A. Dixson , Zeinab M. Elshenawy , Harvey R. Wendt , Saroj Sehgel , Robert H. Henrie, II , David M. Roush , Ping Ding , John W. Lyga , Stephen F. Donovan
发明人: John A. Dixson , Zeinab M. Elshenawy , Harvey R. Wendt , Saroj Sehgel , Robert H. Henrie, II , David M. Roush , Ping Ding , John W. Lyga , Stephen F. Donovan
IPC分类号: A01N43/50 , A61P7/04 , C07D233/20 , C07D405/04 , C07D409/04 , C07D403/04 , C07D207/30 , C07D239/06 , A01N43/38 , A01N43/88 , A01N43/76 , A01N43/78 , A01N43/54 , A01N43/36 , C07D277/08 , C07D417/04 , C07D263/08 , C07D413/04 , C07D495/04 , C07D491/048 , C07D271/10
CPC分类号: A01N43/88 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/76 , A01N43/78 , C07D211/70 , C07D211/74 , C07D233/10 , C07D233/20 , C07D233/22 , C07D233/24 , C07D233/26 , C07D233/64 , C07D263/14 , C07D273/04 , C07D277/14 , C07D307/06 , C07D307/12 , C07D307/20 , C07D309/18 , C07D309/20 , C07D309/22 , C07D309/30 , C07D333/08 , C07D333/16 , C07D333/32 , C07D401/04 , C07D405/04 , C07D409/04 , C07D413/04 , C07F9/6506 , C07F9/6533 , C07F9/65586
摘要: It has now been found that certain novel heterocyclic derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): R Preferred are those compounds of formula (I) where R2 and R3 taken together is ═NCH(R6)CH(R7)N(R8)—, ═NC(R6)=C(R7)N(R8)-, or ═CHN═C(R7)N(R8)—, and tautomers thereof, and where R4 and R5 taken together is —C(R11)=C(R12)C(R13)=C(R14) 112, -, where R, R, R6, R7, R8, R11, R R13, R14, and X are described. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula (I), and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.
摘要翻译: 现在已经发现某些新的杂环衍生物已经提供了意想不到的杀虫活性。 这些化合物由式(I)表示:R优选的是其中R 2和R 3一起为-NCH(R 6)CH(R 7)N(R 8) - , - C(R 6)= C( R 7)N(R 8) - 或-CHN-C(R 7)N(R 8) - 及其互变异构体,其中R 4和R 5一起为-C(R 11)= C(R 12)C(R 13)= C (R14)112, - ,其中描述了R,R,R 6,R 7,R 8,R 11,R 13,R 14和X。 此外,还公开了包含杀虫有效量的至少一种式(I)化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法,包括将所述组合物施用于存在昆虫或预期存在的场所。
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公开(公告)号:US4814325A
公开(公告)日:1989-03-21
申请号:US908493
申请日:1986-09-17
IPC分类号: A01N57/16 , C07F9/6553 , A01N43/32 , A01N43/24 , C07D339/00 , C07D339/08
CPC分类号: A01N57/16 , C07F9/6553
摘要: Dithiacycloalkenyl phosphoric esters of the following formula are effective for the control of soil and foliar insects, acarids and nematodes: ##STR1## wherein R.sub.1 is lower alkyl;R.sub.2 is lower alkoxy or lower alkylthio;R.sub.3 is hydrogen, lower alkyl or phenyl;R.sub.4, R.sub.5 and R.sub.6 are independently hydrogen or lower alkyl;Z is oxygen or sulfur;x is 0 or 1;y is 0, 1 or 2; andn is 0, 1 or 2.
摘要翻译: 下式的二硫代环烯基磷酸酯对于控制土壤和叶面昆虫,螨虫和线虫是有效的:其中R1是低级烷基; R2是低级烷氧基或低级烷硫基; R3是氢,低级烷基或苯基; R4,R5和R6独立地是氢或低级烷基; Z是氧或硫; x为0或1; y为0,1或2; n为0,1或2。
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公开(公告)号:US4782079A
公开(公告)日:1988-11-01
申请号:US148194
申请日:1988-01-26
IPC分类号: A01N43/10 , A01N47/06 , C07D333/12 , A01N43/02 , C07D333/00 , C07D333/24
CPC分类号: C07D333/12 , A01N43/10 , A01N47/06
摘要: Thiophene derivatives of the following formula are effective as acaricides: ##STR1## wherein R.sub.A is selected from -hydrogen, -halogen, -lower alkyl, hydroxy, -lower alkoxy, -lower alkylthio, -lower alkoxyalkoxy, -lower alkoxycarbonyl, -aryloxycarbonyl, -lower alkoxycarbonyloxy, -lower alkylsulfonyl, -lower alkylsulfonyloxy, -arylsulfonyloxy, and -lower alkyl phosphonyloxy;R.sub.B is -hydrogen, or R.sub.A and R.sub.B together are --C.sub.4 H.sub.4 --bridging 2'-3' or 3'-4';R.sub.3 and R.sub.4 are selected from -hydrogen, -lower alkyl, and -aryl;X is -halogen; andY is selected from -hydrogen and -halogen.
摘要翻译: 下式的噻吩衍生物作为杀螨剂是有效的:其中RA选自氢,卤素,低级烷基,羟基,低级烷氧基,低级烷硫基,低级烷氧基烷氧基,低级烷氧基羰基, 低级烷氧基羰基氧基,低级烷基磺酰基, - 低级烷基磺酰氧基, - 芳基磺酰氧基和 - 低级烷基膦酰氧基; RB是氢,或RA和RB一起是-C4H4-桥接2'-3'或3'-4'; R3和R4选自氢,低级烷基和 - 芳基; X是卤素; 并且Y选自氢和卤素。
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公开(公告)号:US4645777A
公开(公告)日:1987-02-24
申请号:US724224
申请日:1985-04-17
IPC分类号: A01N43/10 , A01N57/24 , C07D333/08 , C07D333/12 , C07D333/16 , C07D333/18 , C07D333/28 , C07D333/32 , C07D333/34 , C07D333/38 , C07F9/6553 , A01N43/02
CPC分类号: A01N43/10 , A01N57/24 , C07D333/08 , C07D333/12 , C07D333/16 , C07D333/18 , C07D333/28 , C07D333/32 , C07D333/34 , C07D333/38 , C07F9/655345
摘要: Bithienyl compounds of the following structural formula are phototoxic insecticides and acaricides: ##STR1## wherein R.sub.1 is selected from hydrogen, halogen, alkyl, haloalkyl, alkoxy, and haloalkoxy;R.sub.2 is selected from hydrogen and halogen;R.sub.3 is selected from hydrogen, alkyl, phenyl, and thienyl; andR.sub.4 is selected from hydrogen, halogen, alkyl, and haloalkyl.
摘要翻译: 具有下列结构式的双噻吩基化合物是光毒杀虫剂和杀螨剂:其中R 1选自氢,卤素,烷基,卤代烷基,烷氧基和卤代烷氧基; R2选自氢和卤素; R3选自氢,烷基,苯基和噻吩基; 并且R 4选自氢,卤素,烷基和卤代烷基。
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公开(公告)号:US4621078A
公开(公告)日:1986-11-04
申请号:US709483
申请日:1985-03-07
申请人: David M. Roush
发明人: David M. Roush
摘要: Vinyl phosphoric esters of the following formula are effective in the control of insects and acarids: ##STR1## wherein R.sub.1 is lower alkoxy;R.sub.2 is selected from lower alkoxy and lower thioalkyl;R.sub.3 is selected from lower alkyl, phenyl, and halophenyl;R.sub.4 is selected from hydrogen, lower alkyl, halogen, and lower thioalkyl;V is selected from hydrogen, halogen, lower alkyl, lower alkoxy, lower haloalkyl, amino, mono and dialkyl substituted amino, lower alkoxy carbonyl, lower thioalkyl, lower alkyl sulfonyl, nitro, and phenyl;W is oxygen or sulfur;Y is halogen;m is 0-2; andn is 0-2.
摘要翻译: 下式的乙烯基磷酸酯可有效控制昆虫和螨类:其中R1是低级烷氧基; R2选自低级烷氧基和低级硫代烷基; R3选自低级烷基,苯基和卤代苯基; R4选自氢,低级烷基,卤素和低级硫代烷基; V选自氢,卤素,低级烷基,低级烷氧基,低级卤代烷基,氨基,一烷基和二烷基取代的氨基,低级烷氧基羰基,低级硫代烷基,低级烷基磺酰基,硝基和苯基; W是氧或硫; Y为卤素; m为0-2; n为0-2。
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公开(公告)号:US07977332B2
公开(公告)日:2011-07-12
申请号:US10580481
申请日:2004-12-02
申请人: David M. Roush , John F. Chiarello , Jianming Yu , Benjamin J. Dugan , George Theodoridis , Manorama M. Patel , Walter H. Yeager , Steven W. Szczepanski
发明人: David M. Roush , John F. Chiarello , Jianming Yu , Benjamin J. Dugan , George Theodoridis , Manorama M. Patel , Walter H. Yeager , Steven W. Szczepanski
IPC分类号: C07D213/02 , A01N43/08
CPC分类号: C07D213/26 , A01N43/40 , A01N43/50 , A01N43/78 , A01N43/82 , A01N43/88 , A01N47/40 , A01N51/00 , A01N57/26 , C07D213/38 , C07D213/64 , C07D213/70 , C07D213/73 , C07D233/64 , C07D237/08 , C07D237/12 , C07D239/30 , C07D241/16 , C07D261/08 , C07D263/34 , C07D273/00 , C07D277/32 , C07D285/06 , C07D307/14 , C07D401/12 , C07D401/14 , C07D405/12 , C07D413/12 , C07D413/14 , C07D417/12 , C07D417/14 , C07F9/58
摘要: Certain noel N-(heteroarylalkyl)alkanediamine derivatives have provided unexpected insecticidal and acaricidal activity. These compounds are represented by formula I: wherein Ar, a, r, R, Ra, Rb, Rc, Rd, b, c, Re, Rf, Rg, Rh, R5, d, e, U, V, X, WR6 and R7 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.
摘要翻译: 某些Noel N-(杂芳基烷基)烷二胺衍生物提供了意想不到的杀虫和杀螨活性。 这些化合物由式I表示:其中Ar,a,r,R,Ra,Rb,Rc,Rd,b,c,Re,Rf,Rg,Rh,R5,d,e,U,V,X, 和R7完全描述于此。 此外,还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法,包括将所述组合物施用于存在昆虫或预期存在的场所。
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公开(公告)号:US20080287506A1
公开(公告)日:2008-11-20
申请号:US11577664
申请日:2005-10-27
IPC分类号: A01N43/40 , C07D401/12 , C07D207/02 , C07D231/12 , C07D233/61 , A01N43/36 , A01N43/56 , A01N43/50 , A01P7/04
CPC分类号: C07D401/12 , A01N43/36 , A01N43/40 , A01N43/50 , A01N43/56 , A01N43/78 , C07D405/12 , C07D417/12
摘要: Certain novel N,N-di(heteroarylalkyl)amine derivatives have provided unexpected insecticidal and acaricidal activity. These compounds are represented by formula (I): wherein Ar Ar1, a, b, c, R, Rd, Re, Rf, Rg, Rh, R′, R3 and Rk are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.
摘要翻译: 某些新的N,N-二(杂芳基烷基)胺衍生物已经提供了意想不到的杀虫和杀螨活性。 这些化合物由式(I)表示:其中Ar Ar 1,a,b,c,R,R d,R e, 本文中完整地描述了R f,R g,R h,R',R 3和R k。 此外,还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法,包括将所述组合物施用于存在昆虫或预期存在的场所。
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公开(公告)号:US07417057B2
公开(公告)日:2008-08-26
申请号:US10512377
申请日:2003-04-28
申请人: John A. Dixson , Zeinab M. Elshenawy , Harvey R. Wendt , Saroj Sehgel , Robert H. Henrie, II , David M. Roush , Ping Ding , John W. Lyga , Stephen F. Donovan
发明人: John A. Dixson , Zeinab M. Elshenawy , Harvey R. Wendt , Saroj Sehgel , Robert H. Henrie, II , David M. Roush , Ping Ding , John W. Lyga , Stephen F. Donovan
CPC分类号: A01N43/88 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/76 , A01N43/78 , C07D211/70 , C07D211/74 , C07D233/10 , C07D233/20 , C07D233/22 , C07D233/24 , C07D233/26 , C07D233/64 , C07D263/14 , C07D273/04 , C07D277/14 , C07D307/06 , C07D307/12 , C07D307/20 , C07D309/18 , C07D309/20 , C07D309/22 , C07D309/30 , C07D333/08 , C07D333/16 , C07D333/32 , C07D401/04 , C07D405/04 , C07D409/04 , C07D413/04 , C07F9/6506 , C07F9/6533 , C07F9/65586
摘要: It has now been found that certain novel heterocyclic derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): R Preferred are those compounds of formula (I) where R2 and R3 taken together is ═NCH(R6)CH(R7)N(R8)—, ═NC(R6)═C(R7)N(R8)—, or ═CHN═C(R7)N(R8)—, and tautomers thereof, and where R4 and R5 taken together is —C(R11)═C(R12)C(R13)═C(R14) 1 12, —, where R,R,R 6, R 7, R8, R I1, R R 13, R 14, and X are described. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula (I), and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present
摘要翻译: 现在已经发现某些新的杂环衍生物已经提供了意想不到的杀虫活性。 这些化合物由式(I)表示:R优选的是式(I)的那些化合物,其中R 2和R 3一起是-NCH(R 6)CH( N(R 8) - (R 8)N(R 8) - 或-CHN-C(R' 7)N(R 8) - 及其互变异构体,其中R 4和R 5一起是-C (R 11)-C(R 12)C(R 13)-C(R 14)12, - ,其中R,R,R 6,R 7,R 8,R 11,R R 13,R 14和X。 此外,还公开了包含杀虫有效量的至少一种式(I)化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法,包括将所述组合物施用于存在昆虫或预期存在的场所
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