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公开(公告)号:US5321000A
公开(公告)日:1994-06-14
申请号:US906107
申请日:1992-06-29
IPC分类号: A01N25/32 , C07C69/708 , A01N37/10 , C07C69/76
CPC分类号: C07C69/708 , A01N25/32
摘要: Acids, esters, amides and salts of benzhydryl compounds are antidotes for thiocarbamate and acetamide herbicides. These antidote compounds are especially effective to safen acetamide herbicides used to control grassy weeds and broadleaf weeds in rice, sorghum, corn and wheat.
摘要翻译: 二苯甲基化合物的酸,酯,酰胺和盐是硫代氨基甲酸盐和乙酰胺除草剂的解毒剂。 这些解毒剂化合物特别有效地安全用于控制水稻,高粱,玉米和小麦中的草地杂草和阔叶杂草的乙酰胺除草剂。
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公开(公告)号:US5162537A
公开(公告)日:1992-11-10
申请号:US550002
申请日:1990-07-09
IPC分类号: A01N25/32 , C07C69/708
CPC分类号: C07C69/708 , A01N25/32
摘要: Acids, esters, amides and salts of benzhydryl compounds are antidotes for thiocarbamate and acetamide herbicides. These antidote compounds are especially effective to safen acetamide herbicides used to control grassy weeds and broadleaf weeds in rice, sorghum, corn and wheat.
摘要翻译: 二苯甲基化合物的酸,酯,酰胺和盐是硫代氨基甲酸盐和乙酰胺除草剂的解毒剂。 这些解毒剂化合物特别有效地安全用于控制水稻,高粱,玉米和小麦中的草地杂草和阔叶杂草的乙酰胺除草剂。
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公开(公告)号:US4964893A
公开(公告)日:1990-10-23
申请号:US853301
申请日:1986-04-17
IPC分类号: A01N25/32 , C07C69/708
CPC分类号: C07C69/708 , A01N25/32
摘要: Acids, esters, amides and salts of benzhydryl compounds are antidotes for thiocarbamate and acetamide herbicides. These antidote compounds are especially effective to safen acetamide herbicides used to control grassy weeds and broadleaf weeds in rice, sorghum, corn and wheat.
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4.
公开(公告)号:US07138411B2
公开(公告)日:2006-11-21
申请号:US10303150
申请日:2002-11-22
申请人: Jeffery S Carter , Mark G Obukowicz , Balekudru Devadas , John J Talley , David L Brown , Matthew J Graneto , Stephen R Bertenshaw , Donald J Rogier, Jr. , Srinivasan Raj Nagarajan , Cathleen E Hanau , Susan J Hartmann , Cindy L Ludwig , Suzanne Metz , Donald E Korte
发明人: Jeffery S Carter , Mark G Obukowicz , Balekudru Devadas , John J Talley , David L Brown , Matthew J Graneto , Stephen R Bertenshaw , Donald J Rogier, Jr. , Srinivasan Raj Nagarajan , Cathleen E Hanau , Susan J Hartmann , Cindy L Ludwig , Suzanne Metz , Donald E Korte
IPC分类号: A61K31/47 , A61K31/38 , A61K31/35 , C07D307/77 , C07D335/04
CPC分类号: C07D215/54 , C07D311/22 , C07D311/58 , C07D311/92 , C07D335/06 , C07D401/12 , C07D405/04 , C07D407/04 , C07D407/12 , C07D409/04 , C07D471/04 , C07D491/04 , C07D493/04
摘要: A class of benzopyrans, benzothiopyrans, dihydroquinolines, dihydronaphthalenes, and analogs thereof, is described for use in treating cyclooxygenase-2 mediated disorders. Compounds of particular interest are defined by Formula I′ wherein X, A1, A2, A3, A4, R, R″, R1 and R2 are as described in the specification.
摘要翻译: 描述了一类苯并吡喃,苯并噻喃,二氢喹啉,二氢萘及其类似物,用于治疗环氧合酶-2介导的病症。 特别感兴趣的化合物由式I'定义,其中X,A 1,A 2,A 3,A 4, SUP>,R,R“,R”1“和”R“2如说明书中所述。
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公开(公告)号:US06617324B1
公开(公告)日:2003-09-09
申请号:US10114297
申请日:2002-04-02
申请人: Ashok S. Naraian , Michael Clare , Paul W. Collins , Joyce Zuowu Crich , Rajesh Devraj , Daniel L. Flynn , Lifeng Geng , Matthew J. Graneto , Cathleen E. Hanau , Gunnar J. Hanson , Susan J. Hartmann , Michael Hepperle , He Huang , Francis J. Koszyk , Shuyuan Liao , Suzanne Metz , Richard A. Partis , Thao D. Perry , Shashidhar N. Rao , Shaun Raj Selness , Michael S. South , Michael A. Stealey , John Jeffrey Talley , Michael L. Vazquez , Richard M. Weier , Xiangdong Xi , Ish K. Khanna , Yi Yu
发明人: Ashok S. Naraian , Michael Clare , Paul W. Collins , Joyce Zuowu Crich , Rajesh Devraj , Daniel L. Flynn , Lifeng Geng , Matthew J. Graneto , Cathleen E. Hanau , Gunnar J. Hanson , Susan J. Hartmann , Michael Hepperle , He Huang , Francis J. Koszyk , Shuyuan Liao , Suzanne Metz , Richard A. Partis , Thao D. Perry , Shashidhar N. Rao , Shaun Raj Selness , Michael S. South , Michael A. Stealey , John Jeffrey Talley , Michael L. Vazquez , Richard M. Weier , Xiangdong Xi , Ish K. Khanna , Yi Yu
IPC分类号: A61K31496
CPC分类号: C07D409/14 , C07D401/04 , C07D401/14 , C07D403/04 , C07D405/14 , C07D413/14 , C07D417/14 , C07D453/02 , C07D471/04 , C07D473/00 , C07D487/04
摘要: A class of pyrazole derivatives described for use in treating p38 kinase mediated disorders. Compounds of particular interest are defined by Formula IA wherein R1, R2, R3 and R4 are as described in the specification.
摘要翻译: 一类描述用于治疗p38激酶介导的病症的吡唑衍生物。 特别感兴趣的化合物由式IA定义,其中R1,R2,R3和R4如说明书中所述。
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公开(公告)号:US6046211A
公开(公告)日:2000-04-04
申请号:US73929
申请日:1998-05-06
申请人: Donald W. Hansen, Jr. , Mark G. Currie , E. Ann Hallinan , Kam F. Fok , Timothy J. Hagen , Arija A. Bergmanis , Steven W. Kramer , Len F. Lee , Suzanne Metz , William M. Moore , Karen B. Peterson , Barnett S. Pitzele , Dale P. Spangler , R. Keith Webber , Mihaly V. Toth , Mahima Trivedi , Foe S. Tjoeng
发明人: Donald W. Hansen, Jr. , Mark G. Currie , E. Ann Hallinan , Kam F. Fok , Timothy J. Hagen , Arija A. Bergmanis , Steven W. Kramer , Len F. Lee , Suzanne Metz , William M. Moore , Karen B. Peterson , Barnett S. Pitzele , Dale P. Spangler , R. Keith Webber , Mihaly V. Toth , Mahima Trivedi , Foe S. Tjoeng
IPC分类号: C07D207/32 , A61K31/12 , A61K31/15 , A61K31/16 , A61K31/215 , A61K31/395 , A61K31/40 , A61K31/4015 , A61K31/4025 , A61K31/403 , A61K31/4035 , A61K31/415 , A61K31/42 , A61K31/425 , A61K31/435 , A61K31/44 , A61K31/443 , A61K31/445 , A61K31/4458 , A61K31/4468 , A61K31/451 , A61K31/47 , A61K31/505 , A61K31/535 , A61K31/54 , A61K31/55 , A61P3/08 , A61P9/00 , A61P9/08 , A61P9/10 , A61P29/00 , A61P31/04 , A61P35/00 , A61P37/00 , A61P43/00 , C07C251/44 , C07D207/22 , C07D207/263 , C07D207/273 , C07D207/28 , C07D209/44 , C07D209/46 , C07D211/72 , C07D211/74 , C07D211/76 , C07D213/16 , C07D215/38 , C07D217/22 , C07D221/22 , C07D221/24 , C07D223/12 , C07D223/16 , C07D225/02 , C07D233/46 , C07D239/12 , C07D239/14 , C07D263/28 , C07D265/08 , C07D277/18 , C07D279/06 , C07D405/06 , C07D471/08 , C07D498/04 , C07D513/04
CPC分类号: C07D213/06 , A61K31/395 , A61K31/40 , A61K31/415 , A61K31/42 , A61K31/425 , A61K31/435 , A61K31/44 , A61K31/445 , A61K31/47 , A61K31/505 , A61K31/535 , A61K31/54 , A61K31/55 , C07D207/22 , C07D209/44 , C07D211/72 , C07D211/74 , C07D215/38 , C07D217/22 , C07D221/22 , C07D221/24 , C07D223/12 , C07D225/02 , C07D233/46 , C07D239/12 , C07D239/14 , C07D263/28 , C07D265/08 , C07D277/18 , C07D279/06 , C07D405/06
摘要: The current invention discloses useful pharmaceutical compositions containing amidino derivative useful as nitric oxide synthase inhibitors.
摘要翻译: 本发明公开了含有用作一氧化氮合酶抑制剂的脒基衍生物的有用的药物组合物。
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公开(公告)号:US5854234A
公开(公告)日:1998-12-29
申请号:US448473
申请日:1995-06-06
申请人: Donald W. Hansen, Jr. , Mark G. Currie , E. Ann Hallinan , Kam F. Fok , Timothy J. Hagen , Arija A. Bergmanis , Steven W. Kramer , Len F. Lee , Suzanne Metz , William M. Moore , Karen B. Peterson , Barnett S. Pitzele , Dale P. Spangler , R. Keith Webber , Mihaly V. Toth , Mahima Trivedi , Foe S. Tjoeng
发明人: Donald W. Hansen, Jr. , Mark G. Currie , E. Ann Hallinan , Kam F. Fok , Timothy J. Hagen , Arija A. Bergmanis , Steven W. Kramer , Len F. Lee , Suzanne Metz , William M. Moore , Karen B. Peterson , Barnett S. Pitzele , Dale P. Spangler , R. Keith Webber , Mihaly V. Toth , Mahima Trivedi , Foe S. Tjoeng
IPC分类号: C07D207/32 , A61K31/12 , A61K31/15 , A61K31/16 , A61K31/215 , A61K31/395 , A61K31/40 , A61K31/4015 , A61K31/4025 , A61K31/403 , A61K31/4035 , A61K31/415 , A61K31/42 , A61K31/425 , A61K31/435 , A61K31/44 , A61K31/443 , A61K31/445 , A61K31/4458 , A61K31/4468 , A61K31/451 , A61K31/47 , A61K31/505 , A61K31/535 , A61K31/54 , A61K31/55 , A61P3/08 , A61P9/00 , A61P9/08 , A61P9/10 , A61P29/00 , A61P31/04 , A61P35/00 , A61P37/00 , A61P43/00 , C07C251/44 , C07D207/22 , C07D207/263 , C07D207/273 , C07D207/28 , C07D209/44 , C07D209/46 , C07D211/72 , C07D211/74 , C07D211/76 , C07D213/16 , C07D215/38 , C07D217/22 , C07D221/22 , C07D221/24 , C07D223/12 , C07D223/16 , C07D225/02 , C07D233/46 , C07D239/12 , C07D239/14 , C07D263/28 , C07D265/08 , C07D277/18 , C07D279/06 , C07D405/06 , C07D471/08 , C07D498/04 , C07D513/04 , C07D267/06 , C07D281/02
CPC分类号: C07D213/06 , A61K31/395 , A61K31/40 , A61K31/415 , A61K31/42 , A61K31/425 , A61K31/435 , A61K31/44 , A61K31/445 , A61K31/47 , A61K31/505 , A61K31/535 , A61K31/54 , A61K31/55 , C07D207/22 , C07D209/44 , C07D211/72 , C07D211/74 , C07D215/38 , C07D217/22 , C07D221/22 , C07D221/24 , C07D223/12 , C07D225/02 , C07D233/46 , C07D239/12 , C07D239/14 , C07D263/28 , C07D265/08 , C07D277/18 , C07D279/06 , C07D405/06
摘要: The current invention discloses useful pharmaceutical compositions containing azepine derivatives useful as nitric oxide synthase inhibitors.
摘要翻译: PCT No.PCT / US94 / 11832 Sec。 371日期:1998年6月6日 102(e)1998年6月6日PCT 1994年10月20日PCT PCT。 出版物WO95 / 11231 日期1995年04月27日本发明公开了含有用作一氧化氮合酶抑制剂的吖庚因衍生物的有用的药物组合物。
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8.
公开(公告)号:US07109211B2
公开(公告)日:2006-09-19
申请号:US10922036
申请日:2004-08-19
申请人: Jeffery S Carter , Mark G Obukowicz , Balekudru Devadas , John J Talley , David L Brown , Matthew J Graneto , Stephen R Bertenshaw , Donald J. Rogier, Jr. , Srinivasan Raj Nagarajan , Cathleen E Hanau , Susan J Hartmann , Cindy L Ludwig , Suzanne Metz , Donald E Korte
发明人: Jeffery S Carter , Mark G Obukowicz , Balekudru Devadas , John J Talley , David L Brown , Matthew J Graneto , Stephen R Bertenshaw , Donald J. Rogier, Jr. , Srinivasan Raj Nagarajan , Cathleen E Hanau , Susan J Hartmann , Cindy L Ludwig , Suzanne Metz , Donald E Korte
IPC分类号: A61K31/47 , C07D211/30
CPC分类号: C07D335/06 , C07D215/54 , C07D311/22 , C07D311/58 , C07D311/92 , C07D401/12 , C07D405/04 , C07D407/04 , C07D407/12 , C07D409/04 , C07D471/04 , C07D491/04 , C07D493/04
摘要: A class of benzopyran, derivatives is described for use in treating cyclooxygenase-2 mediated disorders. Compounds of particular interest are defined by Formula I′ wherein X, A1, A2, A3, A4, R, R″, R1 and R2 are as described in the specification.
摘要翻译: 描述了一类苯并吡喃衍生物用于治疗环氧合酶-2介导的病症。 特别感兴趣的化合物由式I'定义,其中X,A 1,A 2,A 3,A 4, SUP>,R,R“,R”1“和”R“2如说明书中所述。
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公开(公告)号:US06956052B2
公开(公告)日:2005-10-18
申请号:US10247096
申请日:2002-09-19
申请人: Arija A. Bergmanis , Michael Clare , Joyce Z. Crich , Lifeng Geng , Timothy J. Hagen , Gunnar J. Hanson , Stephen C. Houdek , He Huang , Donna M. Iula , Francis J. Koszyk , Shuyuan Liao , Scott B. Mohler , Maria Nguyen , Richard A. Partis , Michael A. Stealey , Michael B. Tollefson , Richard M. Weier , Xiangdong Xu , Dominique Bonafoux , Theresa R. Fletcher , Bruce C. Hamper , Patrick J. Lennon , Subo Liao , Suzanne Metz , David S. Oburn , Thomas J. Owen , Angela M. Scates , Michael L. Vazquez , Serge G. Wolfson
发明人: Arija A. Bergmanis , Michael Clare , Joyce Z. Crich , Lifeng Geng , Timothy J. Hagen , Gunnar J. Hanson , Stephen C. Houdek , He Huang , Donna M. Iula , Francis J. Koszyk , Shuyuan Liao , Scott B. Mohler , Maria Nguyen , Richard A. Partis , Michael A. Stealey , Michael B. Tollefson , Richard M. Weier , Xiangdong Xu , Dominique Bonafoux , Theresa R. Fletcher , Bruce C. Hamper , Patrick J. Lennon , Subo Liao , Suzanne Metz , David S. Oburn , Thomas J. Owen , Angela M. Scates , Michael L. Vazquez , Serge G. Wolfson
IPC分类号: A61K31/416 , A61K31/4178 , A61K31/4245 , A61K31/427 , A61K31/433 , A61K31/437 , A61K31/4439 , A61K31/444 , A61K31/4709 , A61K31/4725 , A61K31/496 , A61K31/506 , A61K31/5377 , A61K31/551 , A61P19/02 , A61P25/04 , A61P29/00 , A61P35/00 , C07D231/54 , C07D333/62 , C07D401/04 , C07D401/10 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/04 , C07D405/10 , C07D405/12 , C07D405/14 , C07D409/12 , C07D409/14 , C07D413/12 , C07D417/12 , C07D417/14 , C07D471/04
CPC分类号: C07D403/12 , C07D231/54 , C07D333/62 , C07D401/12 , C07D401/14 , C07D405/10 , C07D405/12 , C07D405/14 , C07D409/12 , C07D409/14 , C07D413/12 , C07D417/12
摘要: The present invention relates to substituted pyrazolyl derivatives, compositions comprising such, intermediates, methods of making substituted pyrazolyl derivatives, and methods for treating cancer, inflammation, and inflammation-associated disorders, such as arthritis.
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10.Substituted pyrazolyl benzenesulfamide compounds for the treatment of inflammation 失效
标题翻译: 用于治疗炎症的取代的吡唑基苯磺酰胺化合物公开(公告)号:US06849653B2
公开(公告)日:2005-02-01
申请号:US10247021
申请日:2002-09-19
申请人: Michael Clare , Lifeng Geng , Gunnar J. Hanson , He Huang , Donna M. Iula , Shuyuan Liao , Michael A. Stealey , Richard M. Weier , Suzanne Metz , Michael L. Vazquez
发明人: Michael Clare , Lifeng Geng , Gunnar J. Hanson , He Huang , Donna M. Iula , Shuyuan Liao , Michael A. Stealey , Richard M. Weier , Suzanne Metz , Michael L. Vazquez
IPC分类号: A61K31/416 , A61K31/4439 , A61K31/444 , A61K31/63 , A61P1/02 , A61P1/04 , A61P3/10 , A61P5/14 , A61P7/06 , A61P7/10 , A61P9/00 , A61P9/10 , A61P9/14 , A61P11/00 , A61P11/06 , A61P13/08 , A61P13/12 , A61P15/00 , A61P17/00 , A61P17/02 , A61P17/06 , A61P19/00 , A61P19/02 , A61P19/06 , A61P19/10 , A61P21/00 , A61P21/04 , A61P25/00 , A61P25/06 , A61P27/02 , A61P29/00 , A61P31/12 , A61P35/00 , A61P35/02 , A61P35/04 , A61P37/08 , A61P43/00 , C07C311/29 , C07D231/54 , C07D231/56 , C07D401/12 , C07D401/14 , C07D405/04 , C07D405/12 , C07D405/14
CPC分类号: C07D231/56 , C07D231/54 , C07D405/04 , C07D405/12 , C07D405/14
摘要: The present invention relates to substituted pyrazolyl derivatives, compositions comprising such, intermediates, methods of making substituted pyrazolyl derivatives, and methods for treating cancer, inflammation, and inflammation-associated disorders, such as arthritis.
摘要翻译: 本发明涉及取代的吡唑基衍生物,包含这些的组合物,中间体,制备取代的吡唑基衍生物的方法,以及用于治疗癌症,炎症和炎症相关疾病如关节炎的方法。
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