Fused 1-(2,6-dichloro-4-trifluoromethylphenyl)-pyrazoles, the synthesis thereof and the use thereof as pesticides
    5.
    发明授权
    Fused 1-(2,6-dichloro-4-trifluoromethylphenyl)-pyrazoles, the synthesis thereof and the use thereof as pesticides 有权
    熔融的1-(2,6-二氯-4-三氟甲基苯基) - 吡唑,其合成及其作为农药的用途

    公开(公告)号:US06545033B1

    公开(公告)日:2003-04-08

    申请号:US09680275

    申请日:2000-10-06

    IPC分类号: A61K31416

    摘要: The present invention is directed to novel pyrazole derivatives and their use as pesticidal agents. The pyrazole derivatives have Formula I: or a salt thereof, where R1 is amino, hydrogen, alkyl, hydroxy, halo, alkoxy, alkylamino, dialkylamino, alkylthio, alkylsulfinyl, alkylsulfonyl, trifluoroalkylsulfinyl, trifluoroalkylsulfonyl, hydroxy, amino, trifluoromethyl, acetylamino, —OSO2R2, —OS(O)R2, —OC(O)R2, —OC(O)NHR2, or —NHC(O)NHR2 where R2 is C1-4 alkyl or optionally substituted aryl; X, Y and Z are each independently (CH)n, (CR3R4)n, S, S(O), or SO2, wherein n is 1-2, R3 and R4 are defined herein; Q is N or C—R6, wherein R6 is fluoro, chloro, bromo, or iodo; R5 is halo, C1-C6 alkyl, C1-C4 alkenyl, C1-C4 alkoxy, C1-C4 alkylamino, C1-C4 dialkylamino, C1-C4 alkylthio, C1-C4 alkylsulfinyl, C1-C4 alkylsulfonyl, C1-C4 trifluoroalkylsulfinyl, C1-C4 trifluoroalkylsulfonyl, hydroxy, amino, or trifluoromethyl; and with the proviso that only one of X, Y and Z can be S, S(O) or SO2.

    摘要翻译: 本发明涉及新颖的吡唑衍生物及其作为杀虫剂的用途。 吡唑衍生物具有式I或其盐,其中R 1是氨基,氢,烷基,羟基,卤素,烷氧基,烷基氨基,二烷基氨基,烷硫基,烷基亚磺酰基,烷基磺酰基,三氟烷基亚磺酰基,三氟烷基磺酰基,羟基,氨基,三氟甲基,乙酰氨基, ,-OS(O)R 2,-OC(O)R 2,-OC(O)NHR 2或-NHC(O)NHR 2,其中R 2为C 1-4烷基或任选取代的芳基; X,Y和Z各自独立地为 CH)n,(CR 3 R 4)n,S,S(O)或SO 2,其中n为1-2,R 3和R 4如本文所定义; Q为N或C-R6,其中R6为氟,氯,溴, 或碘; R5是卤素,C1-C6烷基,C1-C4链烯基,C1-C4烷氧基,C1-C4烷基氨基,C1-C4二烷基氨基,C1-C4烷硫基,C1-C4烷基亚磺酰基,C1-C4烷基磺酰基,C1-C4 三氟烷基亚磺酰基,C 1 -C 4三氟烷基磺酰基,羟基,氨基或三氟甲基; 并且条件是X,Y和Z中只有一个可以是S,S(O)或SO 2。