Quinazoline(di)ones for invertebrate pest control
    25.
    发明申请
    Quinazoline(di)ones for invertebrate pest control 失效
    喹唑啉(二)用于无脊椎害虫防治

    公开(公告)号:US20050124600A1

    公开(公告)日:2005-06-09

    申请号:US10496724

    申请日:2003-01-16

    摘要: Compounds of Formula I including all geometric and stereoisomers, N-oxides, and agriculturally suitable salts thereof, are disclosed which are useful as invertebrate pest control agents, (I) wherein A, B, J, K, L and R3 are as defined in the disclosure. Also disclosed are compositions for controlling an invertebrate pest comprising a biologically effective amount of a compound of Formula I an N-oxide thereof or a suitable salt thereof and at least one additional component selected from the group consisting of surfactants, solid diluents and liquid diluents. Also disclosed are methods for controlling an invertebrate pest comprising contacting the invertebrate pest or its environment with a biologically effective amount of a compound of Formula I, its N-oxide or a suitable salt of the compound (e.g., as a composition described herein).

    摘要翻译: 公开了包含所有几何和立体异构体,N-氧化物和农业上合适的盐的式I化合物,其可用作无脊椎害虫防治剂,(I)其中A,B,J,K,L和R 3 如本公开中所定义。 还公开了用于控制无脊椎害虫的组合物,其包含生物有效量的式I化合物及其N-氧化物或其合适的盐和至少一种选自表面活性剂,固体稀释剂和液体稀释剂的另外的组分。 还公开了用于控制无脊椎害虫的方法,包括使无脊椎害虫或其环境与生物有效量的式I化合物,其N-氧化物或该化合物的合适盐(例如本文所述的组合物)接触。

    System for routing and tracking deliverables
    26.
    发明申请
    System for routing and tracking deliverables 审中-公开
    用于路由和跟踪可交付成果的系统

    公开(公告)号:US20050108076A1

    公开(公告)日:2005-05-19

    申请号:US10712983

    申请日:2003-11-13

    IPC分类号: G06K17/00 G06F17/60

    摘要: A system for routing and tracking deliverables, the system including a flexible label having a flexible transponder associated therewith or formed therein for association with a respective deliverable, at least one transceiver configured to communicate with the transceivers to receive control signals; and a routing device coupled to the transceiver and configured to route and sort deliverables in response to control signals received at the transceiver from the transponder.

    摘要翻译: 一种用于路由和跟踪可交付物的系统,所述系统包括具有与其相关联或在其中形成的灵活的应答器的灵活标签,用于与相应的可递送的至少一个收发器相关联,所述收发器经配置以与收发器通信以接收控制信号; 以及路由设备,其耦合到所述收发器并且被配置为响应于在所述收发器处从所述应答器接收的控制信号来路由和分类可交付物。

    Bicyclic fused pyridinyl amides and advantagesous compositons thereof for use as fungicides
    29.
    发明申请
    Bicyclic fused pyridinyl amides and advantagesous compositons thereof for use as fungicides 审中-公开
    双环稠合吡啶基酰胺和其有用的组合物用作杀真菌剂

    公开(公告)号:US20050020644A1

    公开(公告)日:2005-01-27

    申请号:US10501258

    申请日:2003-02-20

    摘要: Compounds of Formula I, including all geometric and stereoisomers, N-oxides, and agriculturally suitable salts thereof: (Formula I); wherein X and either Y or Z are a linking chain 3 or 4 atoms in length attached to contiguous carbon atoms and are taken together with said carbon atoms to form a fused phenyl ring, a fused 5- or 6-membered nonaromatic carbocyclic or heterocyclic ring optionally including one or two ring members selected from the group consisting of C(═O), SO or S(O)2, or a fused 5- or 6-membered heteroaromatic ring, each fused ring optionally substituted with one to three substituents independently selected from R7; and R1, R2, R5, R6R7, m and p are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula I and a method for controlling plant diseases caused by fungal plant pathogens that involves applying an effective amount of a compound of Formula I.

    摘要翻译: 式I的化合物,包括所有几何和立体异构体,N-氧化物及其农业上合适的盐:(式I); 其中X和Y或Z是连接在连接碳原子上的长度为3或4个原子的连接链,并与所述碳原子一起形成稠合苯环,稠合的5或6元非芳族碳环或杂环 任选地包括一个或两个选自C(= O),SO或S(O)2的环成员或稠合的5或6元杂芳环,每个稠环任选被一至三个取代基独立地取代 选自R 7; 和R 1,R 2,R 5,R 6 R 7,m和p如本公开所定义。 还公开了含有式I化合物的组合物和用于控制由真菌植物病原体引起的植物病害的方法,其涉及施用有效量的式I化合物。

    Certain polycyclic compounds useful as tubulin-binding agents
    30.
    发明授权
    Certain polycyclic compounds useful as tubulin-binding agents 失效
    某些多环化合物可用作微管蛋白结合剂

    公开(公告)号:US06433187B1

    公开(公告)日:2002-08-13

    申请号:US09464217

    申请日:1999-12-15

    IPC分类号: C07D33708

    摘要: Derivatives of known tubulin-binding compounds are provided in which a (poly)fluorobenzene, a fluoropyridine, or a fluoronitrobenzene moiety is incorporated or added to the structure. These derivatives can be used as antimitotic agents and can be considered covalent modifiers of tubulin. The strategy developed for each of the compounds is to i) append a fluorinated electrophile (e.g., pentafluorophenylsulfonamido, 2-fluoropyridyl, or 3,5-dinitro-4-fluorophenyl) to an existing functional group in a natural product, ii) replace an aromatic ring in a natural product with a fluorinated electrophile, or iii) attach a fluorinated electrophile to an open valence in a portion of the molecule that will not interfere with recognition and binding to the tubulin site. Derivatives are provided based on colchicine, steganacin, podophyllotoxin, nocodazole, combretastatin, curacin A, vinblastine, vincristine, dolastatin, 2-methoxyestradiol, dihydroxy-pentamethoxyflavanone and others.

    摘要翻译: 提供了已知的微管蛋白结合化合物的衍生物,其中(聚)氟苯,氟代吡啶或氟硝基苯部分被结合或添加到该结构中。 这些衍生物可用作抗有丝分裂剂并且可以被认为是微管蛋白的共价修饰剂。 为每种化合物制定的策略是i)将天然产物中的现有官能团上的氟化亲电体(例如五氟苯基磺酰胺基,2-氟吡啶基或3,5-二硝基-4-氟苯基) 具有氟化亲电体的天然产物中的芳香环,或iii)在分子的一部分中将氟化亲电体连接至开放价态,其不会干扰识别和结合微管蛋白位点。 衍生物基于秋水仙碱,steganacin,鬼臼毒素,诺考达唑,考布他汀,curacin A,长春花碱,长春新碱,多卡他汀,2-甲氧基雌二醇,二羟基 - 五甲氧基黄酮等。