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公开(公告)号:US20060178370A1
公开(公告)日:2006-08-10
申请号:US10548155
申请日:2004-03-15
申请人: Mark Bock , Bruce Dorsey , Dai-Shi Su , Wei Han , Michael Wood
发明人: Mark Bock , Bruce Dorsey , Dai-Shi Su , Wei Han , Michael Wood
IPC分类号: A61K31/496 , A61K31/495 , C07D403/02 , C07D241/06 , C07D241/08
CPC分类号: C07D403/12 , C07D241/08 , C07D401/12 , C07D401/14 , C07D403/14 , C07D413/12
摘要: Ketopiperazine derivatives are bradykinin B1 antagonists or inverse agonists useful in the treatment or prevention of symptoms such as pain and inflammation associated with the bradykinin B1 pathway.
摘要翻译: 酮哌嗪衍生物是可用于治疗或预防与缓激肽B1途径相关的疼痛和炎症等症状的缓激肽B1拮抗剂或反向激动剂。
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公开(公告)号:US20050085667A1
公开(公告)日:2005-04-21
申请号:US10503502
申请日:2003-02-04
申请人: Michael Wood , Neville Anthony , Mark Bock , Dong-Mei Feng , Scott Kuduk , Dai-Shi Su , Jenny Wai
发明人: Michael Wood , Neville Anthony , Mark Bock , Dong-Mei Feng , Scott Kuduk , Dai-Shi Su , Jenny Wai
IPC分类号: C07D249/08 , A61K31/235 , A61K31/341 , A61K31/343 , A61K31/352 , A61K31/36 , A61K31/381 , A61K31/4035 , A61K31/41 , A61K31/415 , A61K31/4164 , A61K31/4196 , A61K31/42 , A61K31/421 , A61K31/4245 , A61K31/426 , A61K31/44 , A61K31/4406 , A61K31/498 , A61K31/50 , A61K31/505 , A61P1/02 , A61P19/02 , A61P29/00 , A61P29/02 , A61P43/00 , C07C233/50 , C07C237/24 , C07D209/48 , C07D213/81 , C07D213/82 , C07D213/89 , C07D231/12 , C07D231/14 , C07D233/64 , C07D233/90 , C07D237/24 , C07D239/28 , C07D241/44 , C07D257/04 , C07D261/18 , C07D263/34 , C07D271/06 , C07D271/08 , C07D277/20 , C07D277/56 , C07D307/33 , C07D307/56 , C07D307/68 , C07D309/30 , C07D317/68 , C07D333/24 , C07D333/40 , C07D333/70 , C07D403/12 , C07D413/12
CPC分类号: C07C237/24 , C07C237/22 , C07C2601/02 , C07D209/48 , C07D213/81 , C07D213/82 , C07D231/12 , C07D237/24 , C07D239/28 , C07D241/44 , C07D249/08 , C07D249/10 , C07D257/04 , C07D261/18 , C07D263/34 , C07D271/06 , C07D307/68 , C07D317/68 , C07D333/38 , C07D333/70 , C07D403/12 , C07D413/12
摘要: N-Biphenyl(substituted methyl) aminocycloalkanecarboxamide derivatives are bradykinin B1 antagonists or inverse agonists useful in the treatment or prevention of symptoms such as pain and inflammation associated with the bradykinin B1 pathway.
摘要翻译: N-联苯(取代的甲基)氨基环烷基甲酰胺衍生物是缓激肽B1拮抗剂或反向激动剂,其可用于治疗或预防与缓激肽B1途径相关的疼痛和炎症等症状。
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3.2-(Bicyclo)alkylamino-derivatives as mediatores of chronic pain and inflammation 审中-公开
标题翻译: 2-(双环)烷基氨基衍生物作为慢性疼痛和炎症的介质公开(公告)号:US20050261327A1
公开(公告)日:2005-11-24
申请号:US11131642
申请日:2005-05-18
申请人: Mark Bock , Scott Kuduk , Dai-Shi Su , Michael Wood
发明人: Mark Bock , Scott Kuduk , Dai-Shi Su , Michael Wood
IPC分类号: A61K31/4747 , C07D487/10
CPC分类号: C07D239/42 , C07D213/75 , C07D401/12 , C07D405/12 , C07D405/14 , C07D413/12
摘要: Compounds disclosed herein are bradykinin B1 antagonist compounds useful in the treatment or prevention of symptoms such as pain and inflammation associated with the bradykinin B1 pathway.
摘要翻译: 本文公开的化合物是缓激肽B1拮抗剂化合物,其可用于治疗或预防与缓激肽B1途径相关的疼痛和炎症等症状。
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4.N-biphenylmethyl aminocycloalkanecarboxamide derivatives with a substiituent on the methyl useful as bradykinin antagonists 审中-公开
标题翻译: 用作缓激肽拮抗剂的甲基上的取代基的N-联苯甲基氨基环烷甲酰胺衍生物公开(公告)号:US20050084463A1
公开(公告)日:2005-04-21
申请号:US10503501
申请日:2003-02-04
申请人: Michael Wood , Neville Anthony , Marg Bock , Dong-Mei Feng , Scott Kuduk , Dai-Shi Su , Jenny Wau
发明人: Michael Wood , Neville Anthony , Marg Bock , Dong-Mei Feng , Scott Kuduk , Dai-Shi Su , Jenny Wau
IPC分类号: A61K31/166 , A61K31/24 , A61K31/41 , A61K31/42 , A61K31/4245 , A61K31/505 , A61P1/02 , A61P1/04 , A61P1/16 , A61P1/18 , A61P9/10 , A61P11/00 , A61P11/06 , A61P11/08 , A61P13/10 , A61P13/12 , A61P17/02 , A61P17/06 , A61P19/02 , A61P19/08 , A61P21/00 , A61P25/04 , A61P25/06 , A61P25/28 , A61P27/16 , A61P29/00 , A61P31/04 , A61P35/00 , A61P37/08 , C07C237/24 , C07D213/82 , C07D239/28 , C07D257/04 , C07D261/18 , C07D271/06 , C07D403/12 , C07D413/12 , A61K7/025
CPC分类号: C07D257/04 , C07D213/82 , C07D239/28 , C07D261/18 , C07D271/06 , C07D403/12 , C07D413/12
摘要: N-Biphenyl(substituted methyl)aminocycloalkanecarboxamide derivatives are bradykinin B1 antagonists or inverse agonists useful in the treatment or prevention of symptoms such as pain and inflammation associated with the bradykinin B1 pathway.
摘要翻译: N-联苯(取代的甲基)氨基环烷基甲酰胺衍生物是缓激肽B1拮抗剂或反向激动剂,其可用于治疗或预防与缓激肽B1途径相关的疼痛和炎症等症状。
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公开(公告)号:US20060173023A1
公开(公告)日:2006-08-03
申请号:US11334931
申请日:2006-01-19
申请人: Michael Wood , Dai-Shi Su , Jenny Wai
发明人: Michael Wood , Dai-Shi Su , Jenny Wai
IPC分类号: A61K31/506 , A61K31/454 , A61K31/42 , A61K31/401
CPC分类号: A61K31/401 , A61K31/42 , A61K31/454 , A61K31/506 , C07C237/22 , C07D205/04 , C07D207/22 , C07D209/20 , C07D211/60 , C07D239/28 , C07D261/18 , C07D413/06
摘要: Compounds disclosed herein are bradykinin B1 antagonist compounds useful in the treatment or prevention of symptoms such as pain and inflammation associated with the bradykinin B1 pathway.
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公开(公告)号:US20060142612A1
公开(公告)日:2006-06-29
申请号:US10561319
申请日:2004-06-30
申请人: Neville Anthony , Jon Lim , Dai-shi Su , Michael Wood
发明人: Neville Anthony , Jon Lim , Dai-shi Su , Michael Wood
IPC分类号: C07C311/29
CPC分类号: C07D207/27 , C07C311/46 , C07C311/47 , C07C323/62 , C07C2601/02 , C07C2601/08 , C07C2601/14 , C07D207/14 , C07D207/28 , C07D211/38 , C07D211/42 , C07D211/46 , C07D211/56 , C07D211/74 , C07D211/76 , C07D213/50 , C07D213/643 , C07D213/65 , C07D213/75 , C07D213/84 , C07D213/89 , C07D215/14 , C07D231/12 , C07D233/32 , C07D235/16 , C07D239/10 , C07D239/28 , C07D241/12 , C07D249/08 , C07D261/08 , C07D261/20 , C07D263/22 , C07D265/30 , C07D277/64 , C07D295/13 , C07D295/15 , C07D295/192 , C07D307/12 , C07D307/16 , C07D307/24 , C07D307/33 , C07D309/12 , C07D401/04 , C07D401/12 , C07D405/14 , C07D413/12 , C07D471/04 , C07D487/04 , C07D513/04
摘要: N-aryl arylsulfonamide derivatives are bradykinin B1 antagonists or inverse agonists useful in the treatment or prevention of symptoms such as pain and inflammation associated with the bradykinin B1 pathway.
摘要翻译: N-芳基芳基磺酰胺衍生物是可用于治疗或预防与缓激肽B1途径相关的疼痛和炎症等症状的缓激肽B1拮抗剂或反向激动剂。
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公开(公告)号:US20050288305A1
公开(公告)日:2005-12-29
申请号:US10523911
申请日:2003-08-25
申请人: Scott Kuduk , Michael Wood , Mark Bock
发明人: Scott Kuduk , Michael Wood , Mark Bock
IPC分类号: C07D213/24 , A61K31/44 , A61K31/4439 , A61K31/505 , A61K31/506 , A61P1/04 , A61P1/16 , A61P1/18 , A61P3/10 , A61P7/10 , A61P9/00 , A61P9/10 , A61P11/00 , A61P11/02 , A61P11/06 , A61P13/10 , A61P13/12 , A61P17/00 , A61P17/02 , A61P17/06 , A61P19/02 , A61P19/06 , A61P21/00 , A61P25/00 , A61P25/04 , A61P25/06 , A61P25/28 , A61P27/02 , A61P29/00 , A61P31/04 , A61P37/08 , C07D213/40 , C07D213/56 , C07D213/61 , C07D239/02 , C07D239/28 , C07D239/42 , C07D401/10 , C07D401/12 , C07D401/14 , C07D413/10 , C07D413/12 , C07D417/12
CPC分类号: C07D417/12 , C07D213/40 , C07D213/61 , C07D239/28 , C07D239/42 , C07D401/10 , C07D401/12 , C07D401/14 , C07D413/10 , C07D413/12
摘要: N-Biarylmethylainocycloalkanecarboxamide derivatives are bradykinin B1 antagonists or inverse agonists useful in the treatment or prevention of symptoms such as pain and inflammation associated with the bradykinin B1 pathway.
摘要翻译: N-双芳基甲酰基环烷酰胺衍生物是缓激肽B1拮抗剂或反激动剂,其可用于治疗或预防与缓激肽B1途径相关的疼痛和炎症等症状。
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8.2-(Bicyclo)alkylamino-derivatives as mediators of chronic pain and inflammation 审中-公开
标题翻译: 2-(双环)烷基氨基衍生物作为慢性疼痛和炎症的介质公开(公告)号:US20060128765A1
公开(公告)日:2006-06-15
申请号:US11297005
申请日:2005-12-08
申请人: Michael Wood , Scott Kuduk , Mark Bock , Ronald Chang
发明人: Michael Wood , Scott Kuduk , Mark Bock , Ronald Chang
IPC分类号: A61K31/44 , A61K31/195 , A61K31/165 , A61K31/16 , C07D213/56
CPC分类号: C07D213/56 , C07C235/34 , C07C235/40 , C07C237/24 , C07C271/22 , C07C309/17 , C07C311/03 , C07C311/08 , C07C311/09 , C07C317/44 , C07C323/60 , C07C2601/02 , C07D207/08 , C07D207/12 , C07D207/16 , C07D207/452 , C07D209/08 , C07D209/18 , C07D209/48 , C07D211/22 , C07D211/26 , C07D211/42 , C07D211/44 , C07D211/58 , C07D211/60 , C07D211/62 , C07D213/38 , C07D213/42 , C07D213/70 , C07D213/73 , C07D213/74 , C07D213/75 , C07D215/06 , C07D217/04 , C07D233/22 , C07D233/24 , C07D233/64 , C07D235/16 , C07D239/28 , C07D295/096 , C07D295/13 , C07D295/135 , C07D295/15 , C07D295/155 , C07D295/205 , C07D333/24 , C07D471/04
摘要: Compounds disclosed herein are bradykinin B1 antagonist compounds useful in the treatment or prevention of symptoms such as pain and inflammation associated with the bradykinin B1 pathway.
摘要翻译: 本文公开的化合物是缓激肽B1拮抗剂化合物,其可用于治疗或预防与缓激肽B1途径相关的疼痛和炎症等症状。
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公开(公告)号:US20060122236A1
公开(公告)日:2006-06-08
申请号:US11291560
申请日:2005-12-01
申请人: Michael Wood , Mark Bock , Kathy Books , Roger Freidinger , June Kim
发明人: Michael Wood , Mark Bock , Kathy Books , Roger Freidinger , June Kim
IPC分类号: A61K31/44 , A61K31/195 , A61K31/24 , C07D213/72
CPC分类号: C07D213/82 , C07D213/74 , C07D213/75 , C07D213/76 , C07D213/80 , C07D213/85 , C07D295/13 , C07D401/04 , C07D401/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D471/04 , C07D487/04 , C07D487/10
摘要: Substituted biaryl carboxylate derivatives are bradykinin B1 antagonists or inverse agonists useful in the treatment or prevention of symptoms such as pain and inflammation associated with the bradykinin B1 pathway.
摘要翻译: 取代的联芳基羧酸酯衍生物是缓激肽B1拮抗剂或反激动剂,其可用于治疗或预防与缓激肽B1途径相关的疼痛和炎症等症状。
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公开(公告)号:US20060111392A1
公开(公告)日:2006-05-25
申请号:US11284740
申请日:2005-11-22
申请人: Michael Wood , Mark Bock , Kathy Books , Roger Freidinger , June Kim
发明人: Michael Wood , Mark Bock , Kathy Books , Roger Freidinger , June Kim
IPC分类号: A61K31/4745 , A61K31/4545 , C07D401/04 , C07D471/02
CPC分类号: C07D401/04 , C07C275/24 , C07D211/58 , C07D213/40 , C07D213/74 , C07D233/24 , C07D295/13 , C07D295/135 , C07D471/04
摘要: Substituted biaryl-carboyxlate derivatives are bradykinin B1 antagonists or inverse agonists useful in the treatment or prevention of symptoms such as pain and inflammation associated with the bradykinin B1 pathway.
摘要翻译: 取代的联芳基 - 羧甲基化衍生物是缓激肽B1拮抗剂或反激动剂,其可用于治疗或预防与缓激肽B1途径相关的疼痛和炎症等症状。
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