公开(公告)号：US6117870A

公开(公告)日：2000-09-12

申请号：US437438

申请日：1999-11-10

申请人： Akihiko Hosoda ,  Nobuo Kobayashi ,  Naoko Tanabe ,  Tsuneo Koji ,  Masahiro Shibata ,  Akihiro Sekine ,  Masaharu Dozen

发明人： Akihiko Hosoda ,  Nobuo Kobayashi ,  Naoko Tanabe ,  Tsuneo Koji ,  Masahiro Shibata ,  Akihiro Sekine ,  Masaharu Dozen

IPC分类号： C07C211/00 ,  A61P19/02 ,  C07C271/24 ,  C07C275/26 ,  C07C311/20 ,  C07C311/29 ,  C07C311/46 ,  C07C317/44 ,  C07C323/60 ,  C07D213/71 ,  C07D213/75 ,  C07D223/12 ,  C07D231/40 ,  C07D243/08 ,  C07D277/48 ,  C07D277/68 ,  C07D295/215 ,  C07D295/26 ,  C07D295/32 ,  C07D307/14 ,  C07D307/33 ,  C07D307/52 ,  C07D309/20 ,  C07D317/28 ,  C07D317/46 ,  C07D317/58 ,  C07D317/66 ,  C07D317/68 ,  C07D317/72 ,  C07D319/06 ,  A61K31/5375

CPC分类号： C07D213/71 ,  C07C271/24 ,  C07C275/26 ,  C07C311/20 ,  C07C311/29 ,  C07C311/43 ,  C07C311/46 ,  C07C317/44 ,  C07C323/60 ,  C07D211/46 ,  C07D211/58 ,  C07D213/75 ,  C07D223/10 ,  C07D223/12 ,  C07D231/40 ,  C07D243/08 ,  C07D277/48 ,  C07D277/68 ,  C07D277/82 ,  C07D295/215 ,  C07D307/14 ,  C07D307/33 ,  C07D307/52 ,  C07D309/20 ,  C07D317/28 ,  C07D317/46 ,  C07D317/58 ,  C07D317/66 ,  C07D317/68 ,  C07D317/72 ,  C07D319/06 ,  C07C2101/14

摘要： A cyclic amide derivative of formula (I): ##STR1## wherein R.sup.1 represents a substituted alkyl group, a substituted alkenyl group, a substituted amino group, a substituted alkoxyl group, a substituted alkylthio group, a substituted carbamoyl group, a substituted sulfonamide group or a substituted amide group; the ring A represents a saturated cyclic alkyl group with 5 to 7 carbon atoms or a hetero-atom-containing saturated heterocyclic group with 3 to 6 carbon atoms; R.sup.2 represents a hydrogen atom, a substituted or unsubstituted alkyl group, a substituted or unsubstituted aromatic hydrocarbon group or a substituted or unsubstituted heterocyclic group; R.sup.3 represents a hydrogen atom, a group represented by the general formula R.sup.4 O-- or a group represented by the general formula R.sup.5 (R.sup.6)N-- wherein R.sup.4 represents hydrogen atom, a substituted or unsubstituted alkyl group, a substituted or unsubstituted aromatic hydrocarbon group or a substituted or unsubstituted heterocyclic group; R.sup.5 and R.sup.6 may be the same or different and each represents a hydrogen atom, a substituted or unsubstituted alkyl group, a substituted or unsubstituted aromatic hydrocarbon group or a substituted or unsubstituted heterocyclic group.The cyclic amide derivative of formula (I) have a strong and selective inhibitory action of a cathepsin K and a clinical efficacy when administered orally.

摘要翻译： 式（I）的环状酰胺衍生物：其中R1表示取代的烷基，取代的烯基，取代的氨基，取代的烷氧基，取代的烷硫基，取代的氨基甲酰基，取代的磺酰胺基或取代的 酰胺基; 环A表示碳原子数5〜7的饱和环状烷基或碳原子数3〜6的含杂原子的饱和杂环基; R 2表示氢原子，取代或未取代的烷基，取代或未取代的芳香族烃基或取代或未取代的杂环基; R3表示氢原子，由通式R4O表示的基团或由通式R5（R6）表示的基团N-，其中R4表示氢原子，取代或未取代的烷基，取代或未取代的芳族烃基或 取代或未取代的杂环基; R 5和R 6可以相同或不同，各自表示氢原子，取代或未取代的烷基，取代或未取代的芳香族烃基或取代或未取代的杂环基。 式（I）的环状酰胺衍生物在口服给药时具有组织蛋白酶K的强烈和选择性抑制作用和临床疗效。

公开(公告)号：US5988486A

公开(公告)日：1999-11-23

申请号：US28459

申请日：1998-02-24

申请人： Nobuo Kobayashi ,  Toshiaki Nagasawa ,  Hisaya Watanabe ,  Kouji Oda ,  Isao Bundou

发明人： Nobuo Kobayashi ,  Toshiaki Nagasawa ,  Hisaya Watanabe ,  Kouji Oda ,  Isao Bundou

IPC分类号： B23K11/25 ,  B23K11/31 ,  B23K5/22 ,  B23K1/00 ,  B23K9/12 ,  B23K37/02

CPC分类号： B23K11/315 ,  B23K11/255 ,  B23K11/311 ,  B23K11/317

摘要： In a spot welding gun which is made up of a gun main body which is operated for equalization by a driving source, a stationary electrode tip which is immovable relative to the gun main body, and a movable electrode tip which is connected to a pressing source, both electrode tips are pressed to a workpiece with an even force, to thereby perform a high quality spot welding. The driving source is controlled such that the electrode force of the stationary electrode tip, by the driving source, to the workpiece becomes substantially zero. In this manner, there occurs no difference in the electrode forces by both the electrode tips to the workpiece.

摘要翻译： 在由用于由驱动源均衡的枪主体构成的点焊枪中，相对于枪主体不动的固定电极头和与压力源连接的可动电极头 两个电极头以均匀的力压在工件上，从而进行高质量的点焊。 驱动源受到控制，使得固定电极头的驱动源对工件的电极力基本上为零。 以这种方式，电极尖端与工件的电极力没有差别。

公开(公告)号：US5977505A

公开(公告)日：1999-11-02

申请号：US034009

申请日：1998-03-02

申请人： Nobuo Kobayashi ,  Isao Bundou ,  Toshihiro Murakawa ,  Kouji Oda ,  Toshiaki Nagasawa

发明人： Nobuo Kobayashi ,  Isao Bundou ,  Toshihiro Murakawa ,  Kouji Oda ,  Toshiaki Nagasawa

IPC分类号： B23K11/24 ,  B23K11/11 ,  B23K11/16 ,  B23K11/31 ,  B23K11/10

CPC分类号： B23K11/317 ,  B23K11/16 ,  B23K11/31 ,  B23K11/311 ,  B23K11/315

摘要： When a workpiece which is made up by laminating a plurality of plates of different thicknesses is welded by using a spot welding gun having a pair of electrode tips, the electrode force to the workpiece by one of the electrode tips, which is positioned on the side of a thinner plate, is made larger that the electrode force to the workpiece by the other of the electrode tips. The contact pressure on the side of the thinner plate becomes larger with the result that the contact resistance decreases. Therefore, the nugget on the side of the thinner plate becomes smaller than the nugget on the side of the thicker plate.

摘要翻译： 通过使用具有一对电极头的点焊枪对通过层叠多个不同厚度的板构成的工件进行焊接时，通过位于一侧的电极头之一对工件施加电极力 更薄的板，使得电极通过另一个电极尖端对工件的力较大。 更薄板侧面的接触压力变大，接触电阻降低。 因此，较薄板侧面的熔核变得比厚板侧面的熔核小。

公开(公告)号：US5742052A

公开(公告)日：1998-04-21

申请号：US676295

申请日：1996-07-18

申请人： Toshihiro Noguchi ,  Nobuo Kobayashi ,  Yukitoshi Tamura ,  Toshiei Matsuzaki

发明人： Toshihiro Noguchi ,  Nobuo Kobayashi ,  Yukitoshi Tamura ,  Toshiei Matsuzaki

IPC分类号： H01L31/02 ,  G01J5/02 ,  H01L23/14

CPC分类号： H01L31/02002 ,  H01L2224/45144 ,  H01L2224/48091 ,  H01L2924/3011 ,  H01L2924/3025

摘要： An infrared detector comprising an infrared detector element for generating an electrical signal, a support for the infrared detector element, and a circuit board for receiving the electrical signal from the infrared detector element. The support is formed integrally with the circuit board. The support comprises a matrix of composite material essentially consisting of one of thermosetting resins and thermoplastic resins having a thermal deformation temperature of at least 100.degree. C. and a tensile elastic modulus of at least 100 kgf/mm.sup.2, and of carbon fibers contained in the range of 10 to 40% by weight and dispersed in the matrix. The circuit board is formed with a through-hole having an inner surface processed so as to be electrically conductive.

摘要翻译： PCT No.PCT / JP95 / 02367 Sec。 371日期：1996年7月18日 102（e）日期1996年7月18日PCT提交1995年11月20日PCT公布。 WO96 / 16441 PCT出版物 日期：1996年5月30日包括用于产生电信号的红外检测器元件，红外线检测器元件的支撑件和用于从红外线检测器元件接收电信号的电路板的红外检测器。 支撑件与电路板一体形成。 载体包括基本上由热固性树脂和热变形温度至少为100℃，拉伸弹性模量为至少100kgf / mm 2的热塑性树脂之一的复合材料基体和包含在 范围为10〜40重量％，分散在基质中。 电路板形成有具有被处理为导电的内表面的通孔。

公开(公告)号：US5276150A

公开(公告)日：1994-01-04

申请号：US850201

申请日：1992-03-12

申请人： Hiroshi Ikawa ,  Akiyoshi Kadoiri ,  Nobuo Kobayashi ,  Yasuko Konagai ,  Yasuo Sekine

发明人： Hiroshi Ikawa ,  Akiyoshi Kadoiri ,  Nobuo Kobayashi ,  Yasuko Konagai ,  Yasuo Sekine

IPC分类号： C07D211/90 ,  C07D401/04 ,  C07D401/14 ,  C07D405/04 ,  C07D405/14 ,  C07D409/04 ,  C07D409/14 ,  C07D473/04 ,  C07D473/08 ,  C07D521/00 ,  C07D217/18 ,  C07D417/04 ,  C07D419/04

CPC分类号： C07D231/12 ,  C07D211/90 ,  C07D233/56 ,  C07D249/08 ,  C07D401/04 ,  C07D401/14 ,  C07D405/04 ,  C07D405/14 ,  C07D409/04 ,  C07D409/14 ,  C07D473/04 ,  C07D473/08

摘要： 1,4-dihydropyridine derivatives of formula (I): ##STR1## wherein Ar.sup.1 and Ar.sup.2 each represent an unsubstituted or substituted aromatic hydrocarbon or aromatic heterocyclic group; and R.sup.1 represents --CO.sub.2 R.sup.2, --SO.sub.2 R.sup.3, --COR.sup.4, --CON(R.sup.5).sub.2, --CH--or --NO.sub.2 in which R.sup.2 is hydrogen, a straight chain, branched chain or cyclic saturated hydrocarbon group, which may have a substituent or a straight chain, branched chain or cyclic unsaturated hydrocarbon group having 2 to 10 carbon atoms, which may have a substituent, R.sup.3 is an alkyl group having 1 to 4 carbon atoms, R.sup.4 is an alkyl group having 1 to 4 carbon atoms or a phenyl group; and R.sup.5 is an alkyl group having 1 to 4 carbon atoms.

摘要翻译： 式（I）的1,4-二氢吡啶衍生物：其中Ar 1和Ar 2各自表示未取代或取代的芳族烃或芳族杂环基; 和R 1表示可以具有取代基的直链，支链或环状饱和烃基的-CO 2 R 2，-SO 2 R 3，-COR 4，-CON（R 5）2，-CH或-NO 2， 可以具有取代基的碳原子数为2〜10的直链，支链或支链或环状不饱和烃基，R3为碳原子数1〜4的烷基，R4为碳原子数1〜4的烷基或苯基 ; R5为碳原子数为1〜4的烷基。

公开(公告)号：US5218641A

公开(公告)日：1993-06-08

申请号：US739237

申请日：1991-08-01

申请人： Kensaku Abe ,  Nobuo Kobayashi

发明人： Kensaku Abe ,  Nobuo Kobayashi

IPC分类号： H04B1/16 ,  H04B10/07 ,  H04B10/11 ,  H04B10/112 ,  H04B10/548 ,  H04B10/80 ,  H04R3/00

CPC分类号： H04B10/114 ,  H04R3/00 ,  H04R2400/00 ,  H04R2420/07

摘要： A wireless receiver has an FM receiver for receiving an infrared radiation modulated by an audio signal. The received infrared radiation is demodulated into the audio signal, which is then supplied through a power amplifier to a loudspeaker unit or a headphone unit. The wireless receiver includes a detector for detecting whether or not the infrared radiation is received. An output signal from the detector is used to turn the power supply of the FM receiver and the power amplifier on or off. The user of the wireless receiver is not required to turn the receiver on and off manually.

公开(公告)号：US5171960A

公开(公告)日：1992-12-15

申请号：US785261

申请日：1991-10-30

申请人： Fumitomo Takano ,  Nobuo Kobayashi ,  Kazuo Isogai ,  Hitoshi Saito ,  Kenji Miyanaga

发明人： Fumitomo Takano ,  Nobuo Kobayashi ,  Kazuo Isogai ,  Hitoshi Saito ,  Kenji Miyanaga

IPC分类号： B23K11/25

CPC分类号： B23K11/252

摘要： A direct-current resistance welding apparatus includes pneumatic actuators for pressurizing welding guns, respectively, to grip respective workpieces, an inverter composed of a plurality of parallel-connected switching device units each comprising a pair of series-connected switching devices, and a plurality of welding transformers connected to the welding guns, respectively, and also connected between the switching device units. A timer circuit applies an energization signal to energize the switching device units. The pneumatic actuators are actuated by a control circuit to pressurize the welding guns and successively energize the switching device units according to s sequence read from a sequence memory circuit.

摘要翻译： 直流电阻焊接装置包括用于分别对焊枪进行加压以夹紧各个工件的气动致动器，由多个并联的开关装置单元组成的逆变器，每个并联的开关装置单元包括一对串联的开关装置，以及多个 焊接变压器分别连接到焊枪，并且还连接在开关装置单元之间。 定时器电路施加通电信号以激励开关装置单元。 气动致动器由控制电路致动，以对焊接枪进行加压，并根据从序列存储器电路读取的序列连续激励开关装置单元。

公开(公告)号：US5003008A

公开(公告)日：1991-03-26

申请号：US427017

申请日：1989-10-25

申请人： Nobuo Kobayashi

发明人： Nobuo Kobayashi

IPC分类号： C08J3/24 ,  C08F259/08

CPC分类号： C08F259/08

摘要： Shaped articles of a crosslinked poly(vinylidene fluoride) resin can be prepared in a relatively simple process to be imparted with greatly improved resistance against heat, water, and chemicals in a much higher productivity than in the conventional electron-beam irradiation method. The method comprises the steps of (a) compounding the resin with an organosilane compound having an ethylenically unsaturated group, e.g., vinyl, and at least one alkoxy group in a molecule and a free-radical generator, e.g., organic peroxides, (b) heating the resin compound to effect graft-polymerization of the organosilane compound to the polymer molecules, (c) shaping the resin compound into a desired form, and (d) heating the shaped body in water containing a silanol-condensation catalyst dissolved or dispersed therein.

摘要翻译： 交联聚（偏二氟乙烯）树脂的成型制品可以以相对简单的方法制备，以比常规电子束照射方法更高的生产率赋予大大提高的抗热，水和化学品的耐受性。 该方法包括以下步骤：（a）将树脂与分子中具有乙烯基和至少一个烷氧基的有机硅烷化合物和自由基发生剂（例如有机过氧化物）混合，（b） 加热树脂化合物以使有机硅烷化合物与聚合物分子接枝，（c）将树脂化合物成型为所需形式，和（d）在含有溶解或分散在其中的硅烷醇缩合催化剂的水中加热成型体 。

公开(公告)号：US4839099A

公开(公告)日：1989-06-13

申请号：US147018

申请日：1988-01-15

申请人： Kiyoshi Umehara ,  Hisaomi Yamamoto ,  Nobuo Kobayashi ,  Tsutomu Imai

发明人： Kiyoshi Umehara ,  Hisaomi Yamamoto ,  Nobuo Kobayashi ,  Tsutomu Imai

IPC分类号： B27K3/36 ,  B27K3/16 ,  B27K3/50 ,  B27K5/00 ,  C09K21/12 ,  C09K21/14

CPC分类号： C09K21/12 ,  B27K2240/30 ,  B27K3/50 ,  Y10S428/92 ,  Y10S428/921 ,  Y10T428/31989 ,  Y10T428/662

摘要： A fire retardent for woody materials, which is an aqueous solution comprising 100 parts by weight as solids content of a water-soluble 3-(dialkylphosphonopropionamide) represented by the following general formula ##STR1## wherein each of R.sub.1 and R.sub.2 represents an alkyl group having 1 to 3 carbon atoms, and R.sub.3 represents a hyrogen atom or a methyl group, and at least 100 parts by weight as solids of a water-soluble melamine resin as essential ingredients and having a pH of not more than 3.

摘要翻译： 木质材料的阻燃剂，其为包含100重量份作为固体含量的由下列通式（IMAGE）表示的水溶性3-（二烷基膦酰丙酰胺）的水溶液，其中R1和R2各自表示具有 1〜3个碳原子，R3表示氢原子或甲基，至少100重量份作为固体的水溶性三聚氰胺树脂作为必要成分，pH值不大于3。

公开(公告)号：US4785685A

公开(公告)日：1988-11-22

申请号：US36451

申请日：1987-04-09

申请人： Nobuo Kobayashi ,  Shigeo Aiba ,  Shigetoshi Miyoshi ,  Takahiro Iwase ,  Tsutomu Sugiura ,  Takeshi Onogi ,  Taisuke Nakamura

发明人： Nobuo Kobayashi ,  Shigeo Aiba ,  Shigetoshi Miyoshi ,  Takahiro Iwase ,  Tsutomu Sugiura ,  Takeshi Onogi ,  Taisuke Nakamura

IPC分类号： B62D3/12 ,  F16H55/28 ,  F16H57/12 ,  F16H19/04

CPC分类号： B62D3/123 ,  F16H55/283 ,  Y10T74/1967 ,  Y10T74/19819

摘要： The synthetic resin rack guide to be housed in a gear box of a rack and pinion type steering device for a vehicle. The rack guide includes a generally semi-cylindrical head, an outer cylinder and an inner cylinder. The generally semi-cylindrical head includes a semi-cylindrical concave surface which slidably contacts a back surface of a rack bar. The outer cylinder is separated from the inner cylinder by a circumferentially extending space and is divided into a plurality of sections in the circumferential direction by a plurality of slits which extend in parallel with an axis of the rack guide. Due to the provision of the slits, the outer cylinder can shrink radially inward when it is inserted into a rack housing with no clearance between them and when an interference between them is increased in proportion to an increase in ambient temperature. Thus, a locking of the rack guide with the rack housing is prevented and a smooth sliding is obtained even with the increase in ambient temperature.

摘要翻译： 合成树脂齿条引导件被容纳在用于车辆的齿条和小齿轮型转向装置的齿轮箱中。 齿条引导件包括大致半圆柱形的头部，外部圆柱体和内部圆柱体。 大致半圆柱形头部包括可滑动地接触齿条的后表面的半圆柱形凹面。 外筒通过周向延伸的空间与内筒隔开，并且通过与齿条引导件的轴线平行地延伸的多个狭缝在圆周方向上分成多个部分。 由于设置狭缝，当外筒在插入到机架壳体中时，径向向内收缩，其间没有间隙，并且当它们之间的干扰与环境温度的增加成比例地增加时。 因此，防止了齿条引导件与齿条壳体的锁定，并且即使随着环境温度的增加也获得平滑的滑动。