摘要:
7-(R)-Aminotriazolopyrimidines of the formula I where the substituents and the index are as defined below: R1 is hydrogen or methyl; R2 is methyl; R3 is C2-C1o-alkyl, C1-C4-alkoxymethyl, C3-C1o-cycloalkyl; R4 is halogen, Cl-C4-alkyl, C1-C4-haloalkyl or Cl-C4-alkoxy; n is a number from 1 to 5; Y is halogen, cyano, Cl-C4-alkyl or Cl-C4-alkoxy; where * is a center of chirality in the R configuration, processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.
摘要:
The invention relates to 7-amino triazolopyrimidines of formula (I), in which the substituents have the following meanings: R1, R2 represent hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, phenyl, naphthyl; or 5-membered or 6-membered heterocyclyl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or 5-membered or 6-membered heteroaryl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or R1 and R2 can, together with the nitrogen atom, which binds them, form a 5-membered or 6-membered ring containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R3 represents alkyl, alkenyl, alkynyl, cycloalkyl, phenylalkyl and alkyl halide; whereby R3 and R2 can be unsubstituted or partially or completely substituted according to the description; X represents halogen, cyano, alkoxy, alkyl halide, phenyl or phenyl that is substituted by Ra. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the same, and to their use.
摘要:
Triazolopyrimidines of formula (I), wherein the index and substituents have the following meaning: n=0 or a whole number of 1-5; R=halogen, cyano, hydroxy, cyanate, alkyl, alkenyl, alkinyl, halogenalkyl, halogenalkenyl, alkoxy, alkenyloxy, alkinyloxy, halogenalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkinyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, cycloalkylcarbonyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R1=alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S, R and/or R1 being able to be substituted according to the description; R2=alkyl, alkenyl or alkinyl which can be substituted by halogen, cyano, nitro, alkoxy or alkoxycarbonyl. The invention also relates to a method for the production of said compounds, agents containing same, and the use thereof in controlling noxious fungi.
摘要:
.beta.-Substituted cinnamic acid derivatives of the formula 1, ##STR1## where R.sup.1 is substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkyl or cycloalkenyl, and R.sup.1 can also be chlorine or bromine,--X-- is --O--, --S--, ##STR2## m is 0 or 1, --Y is --OR.sup.4, --O--N.dbd.CR.sup.5 R.sup.6, --NR.sup.7 R.sup.8, --NR.sup.7 R.sup.8, --N(OR.sup.9)R.sup.10 or SR.sup.11, where the abovementioned substitutes R.sup.2 to R.sup.11 are substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkyl or cycloalkenyl, and R.sup.2, R.sup.3 and R.sup.5 to R.sup.11 can be hydrogen and Z, U, V, W are defined in the specification.
摘要翻译:式1的β取代肉桂酸衍生物,其中R 1是取代或未取代的烷基,烯基,炔基,环烷基或环烯基,R 1也可以是氯或溴,-X-是-O-,-S - , - Y是-OR 4,-ON = CR 5 R 6,-NR 7 R 8,-NR 7 R 8,-N(OR 9)R 10或SR 11,其中上述取代基R 2至R 11是取代或未取代的烷基, 烯基,炔基,环烷基或环烯基,R2,R3和R5至R11可以是氢,Z,U,V,W在说明书中定义。
摘要:
2-[1′,2′,4′-Triazol-3′-yloxymethylene]anilides of the formula I where the index and the substituents have the following meanings: n is 0, 1, 2, 3, or 4; X is a direct bond, O or NRa; Ra is hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl or cycloalkenyl; R1 is nitro, cyano, halogen, unsubstituted or substituted alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy or alkynyloxy; R2 is hydrogen, nitro, cyano, halogen, alkyl, haloalkyl, alkoxy, alkylthio or alkoxycarbonyl; R3 is unsubstituted or substituted alkyl, alkenyl, alkynyl, cycloalkyl, heteocyclyl, aryl or heteroaryl; R4 is hydrogen, unsubstituted or substituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, alkylcarbonyl or alkoxycarbonyl; R5 is hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl or cycloalkenyl, processes and intermediates for their preparation and their use are described.
摘要:
5-Phenylpyrimidines of the formula I in which the substituents and the index are as defined below: R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl, and R1 and R2 together with the nitrogen atom to which they are attached may also form a saturated or unsaturated ring which may be interrupted by an ether, thio, sulfoxyl or sulfonyl group and may be substituted by one to four groups Ra and/or Rb; R3 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy or alkenyloxy; R4 is hydrogen, halogen, cyano, hydroxyl, mercapto, azido, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, —ON═CRaRb, —CRc═NORa, —NRcN═CRaRb, —NRaRb, —NRcNRaRb, —NORa, —NRcC(═NRc′)NRaRb, —NRcC(═O)NRaRb, —NRaC(═O)Rc, —NRaC(═NORc)Rc′, —OC(═O)Rc, —C(═NORc)NRaRb, —CRc(═NNRaRb), —C (═O)NRaRb or —C(═O)Rc; in which Ra, Rb and Rc are as defined in the description; X is halogen, alkyl, alkoxy or haloalkyl; and m is an integer from 1 to 5 ; processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.
摘要:
Disclosed are a method for producing fungicidal triazolopyrimidine compounds, agents containing said compounds, and the use thereof for controlling harmful fungi. Also disclosed are triazolopyrimidines of formula (I), in which the substituents have the following meaning: L1 represents alkyl; L2 represents halogen; L3represents hydrogen or halogen; X represents halogen, cyano, alkyl, alkoxy, or haloalkoxy; R1, R2 represent hydrogen, alkyl, haloalkyl, cycloalkyl, alkenyl, alkadienyl, alkinyl, or cycloalkinyl, phenyl, naphthyl, or a five-unit to ten-unit saturated, partially unsaturated, or aromatic heterocycle containing one to four heteroatoms from the group O, N, or S, R1 and R2 can also form a five-unit or six-unit ring along with the nitrogen atom to which they are linked. Said ring can be interrupted and/or substituted by an atom from the group O, N, and S while R1 and/or R2 can be substituted according to the description. The invention also relates to methods and intermediate products for producing said compounds, agents containing said compounds, and the use thereof for controlling harmful fungi
摘要翻译:公开了生产杀真菌三唑并嘧啶化合物的方法,含有所述化合物的试剂及其用于控制有害真菌的用途。 还公开了式(I)的三唑并嘧啶,其中取代基具有以下含义:L 1表示烷基; L 2表示卤素; L 3表示氢或卤素; X表示卤素,氰基,烷基,烷氧基或卤代烷氧基; R 1,R 2代表氢,烷基,卤代烷基,环烷基,烯基,链二烯基,炔基或环炔基,苯基,萘基或五个单元至十个单元 饱和的,部分不饱和的或含有一至四个O,N或S杂原子的杂环,R 1和R 2也可以形成五单元或 六单元环与它们所连接的氮原子一起。 所述环可以被O,N和S基团的原子中断和/或取代,而R 1和/或R 2可以根据描述被取代 。 本发明还涉及用于生产所述化合物的方法和中间产物,含有所述化合物的试剂及其用于控制有害真菌的用途
摘要:
5-Phenylpyrimidines, their preparation, compositions comprising them and their use 5-Phenylpyrimidines of the formula I in which the substituents and the index are as defined below: R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl, and R1 and R2 together with the nitrogen atom to which they are attached may also form a saturated or unsaturated ring which may be interrupted by an ether, thio, sulfoxyl or sulfonyl group and may be substituted by one to four groups Ra and/or Rb; R3 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy or alkenyloxy; R4 is hydrogen, halogen, cyano, hydroxyl, mercapto, azido, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, —ON═CRaRb, —CRc═NORa, —NRcN═CRaRb, —NRaRb, —NRcNRaRb, —NORa, —NRcC(═NRc′)NRaRb, —NRcC(═O)NRaRb, —NRaC(═O)Rc, —NRaC(═NORc)Rc′, —OC(═O)Rc, —C(═NORc)NRaRb, —CRc(═NNRaRb), —C(═O)NRaRb or —C(═O)Rc; in which Ra, Rb and Rc are as defined in the description; X is halogen, alkyl, alkoxy or haloalkyl; and m is an integer from 1 to 5; processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.
摘要翻译:其中取代基和指数如下定义的式I的5-苯基嘧啶:R1,R2是氢,烷基,卤代烷基,环烷基,卤代环烷基,烯基,卤代烯基,炔基或卤代炔基,R1和R2与氮原子一起 它们所连接的也可以形成可被醚,硫代,亚砜基或磺酰基中断的饱和或不饱和环,并且可以被一至四个基团R a和/或R b取代; R3是氢,卤素,氰基,烷基,卤代烷基,烷氧基,卤代烷氧基或烯氧基; R4是氢,卤素,氰基,羟基,巯基,叠氮基,烷基,烯基,炔基,卤代烷基,烷氧基,烯氧基,炔氧基,卤代烷氧基,烷硫基,烯硫基,炔硫基,卤代烷硫基,-ON-CRaRb,-CRc-NORa,-NRcN -CRaRb,-NRaRb,-NRcNRaRb,-NORa,-NRcC(-NRc')NRaRb,-NRcC(-O)NRaRb,-NRaC(-O)Rc,-NRaC(-NORc)Rc',-OC( - O)R c,-C(-NOR c)NR a R b,-CR c(-NNR a R b), - C(-O)NR a R b或-C(-O)R c; 其中Ra,Rb和Rc如说明书中所定义; X是卤素,烷基,烷氧基或卤代烷基; m为1〜5的整数。 描述了制备这些化合物的方法,包含它们的组合物及其用于控制有害真菌的用途。
摘要:
The invention relates to 2-(2-pyridyl)-5-phenyl-6-aminopyrimidines of formula I, wherein the substitutes and the index have the following meaning: R1 represents halogen, hydroxy, hyano, hxo, nitro, amino, mercapto, alkyl, halogenalkyl, alkenyl, alkinyl, cycloalkyl, alkoxy, halogenalkoxy, carboxyl, alkoxycarbonyl, carbamoyl, alkylaminocarbonyl, dialkylamincarbonyl, morpholinocarbonyl, pyrrolidinocarbonyl, alkylcarbonylamino, alkylamino. dialkylamino, alkylthio, alkylsulfinyl, alkylsulfonyl, hydroxysulfonyl, aminosulfonyl, alkylaminosulfonyl, dialkylaminosulfonyl; m=0 or 1-4; R2 represents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R3, R4 represents hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl, R3 and R4 together with the nitrogen atom to which they are connected, form a five or six-membered ring which is interrupted by an atom from the group O, N or S and/or can be substituted according to the description; R5 represents halogen, alkyl or halogenalkyl; R6 represents hydrogen or one of the known groups in R5; R7, R8 represent hydrogen, halogen, alkyl or halogenalkyl; R9 represents hydrogen, halogen, hydroxy, cyano, alkyl, alkoxy, cycloalkoxy, halogenalkoxy, alkoxycarbonyl or alkylaminocarbonyl. The invention also relates to a method and intermediate product for the production of said compound in addition to the use thereof for combating undesirable plants
摘要翻译:本发明涉及式I的2-(2-吡啶基)-5-苯基-6-氨基嘧啶,其中取代基和指数具有以下含义:R 1表示卤素,羟基,杂环基, 烷氧基,烷氧基羰基,氨基甲酰基,烷基氨基羰基,二烷基氨基羰基,吗啉代羰基,吡咯烷基羰基,烷基羰基氨基,烷基氨基。 二烷基氨基,烷硫基,烷基亚磺酰基,烷基磺酰基,羟基磺酰基,氨基磺酰基,烷基氨基磺酰基,二烷基氨基磺酰基; m = 0或1-4; R 2表示氢,卤素,氰基,烷基,卤代烷基或烷氧基; R 3,R 4表示氢,烷基,卤代烷基,环烷基,卤代烷基,烯基,卤代烯基,环烯基,炔基,卤代炔基或环炔基,R 3 O 和R 4与它们连接的氮原子一起形成5或6元环,其被来自基团O,N或S的原子和/或可被取代 根据说明; R 5表示卤素,烷基或卤代烷基; R 6表示氢或R 5中的已知基团之一; R 7,R 8表示氢,卤素,烷基或卤代烷基; R 9表示氢,卤素,羟基,氰基,烷基,烷氧基,环烷氧基,卤代烷氧基,烷氧基羰基或烷基氨基羰基。 本发明还涉及用于生产所述化合物的方法和中间产物,除了其用于对抗不期望的植物之外
摘要:
The invention relates to triazolopyrimidines of formula (I), in which the substituents are defined as follows: L1 represents cyano, S(═O)nA1 or C(═O)A2, wherein A1 stands for hydrogen, hydroxy, alkyl, alkylamino or dialkylamino; A2 stands for C1–C8 alkoxy, C1–C6 haloalkoxy or one of the groups named in A1; and n stands for 0, 1 or 2; L2, L3 represent hydrogen or halogen; L4, L5 represent hydrogen, halogen or alkyl; X represents halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1 represents alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl, or a five to ten-membered saturated, partially unsaturated or aromatic heterocyclus containing between one and four heteroatoms from the group containing O, N or S; R2 represents hydrogen or R1; R1 and R2 can form, together with the nitrogen atom to which they are bonded, a five or six-membered ring, which can be interrupted and/or substituted by an atom from the group O, N and S; whereby R1 and/or R2 can be substituted in accordance with the description. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the latter and to the use of said compounds for combating harmful fungi.
摘要翻译:本发明涉及式(I)的三唑并嘧啶,其中取代基定义如下:L 1表示氰基,S(-O)n A 1 或其中A 1代表氢,羟基,烷基,烷基氨基或二烷基氨基;或C(= O) A u> 2代表C 1 -C 8烷氧基,C 1 -C 6烷基,C 1 -C 6 - >卤代烷氧基或在A O>中命名的基团之一; 而n代表0,1或2; L 2,L 3表示氢或卤素; L 4,L 5代表氢,卤素或烷基; X表示卤素,氰基,烷基,卤代烷基,烷氧基或卤代烷氧基; R 1表示烷基,卤代烷基,环烷基,卤代环烷基,烯基,链烯基,卤代烯基,环烯基,炔基,卤代炔基或环炔基,苯基,萘基或五至十元饱和,部分不饱和或芳族杂环 含有一个至四个来自含有O,N或S的基团的杂原子; R 2表示氢或R 1; R 1和R 2可以与它们所键合的氮原子一起形成五元或六元环,其可被中断和/或被 来自O,N和S族的原子; 其中R 1和/或R 2可以根据描述被取代。 本发明还涉及用于生产所述化合物的方法和中间产物,含有后者的试剂和所述化合物用于防治有害真菌的用途。