利索-全球专利检索

  1. 登录
  2. 注册

搜索结果

37 条记录 (耗时 0.036 秒)

    Inhibitors, obtained from bacilli, for glycoside hydrolases
    5.
    发明授权
    Inhibitors, obtained from bacilli, for glycoside hydrolases 失效
    抑制剂，从杆菌获得，用于糖苷水解酶

    公开(公告)号：US4307194A

    公开(公告)日：1981-12-22

    申请号：US858036

    申请日：1977-12-06

    申请人： Werner Frommer ,  Lutz Muller ,  Delf Schmidt ,  Walter Puls ,  Hans-Peter Krause ,  Ulrich Heber

    发明人： Werner Frommer ,  Lutz Muller ,  Delf Schmidt ,  Walter Puls ,  Hans-Peter Krause ,  Ulrich Heber

    IPC分类号： C12P17/12 ,  A23K1/17 ,  A23K1/18 ,  A61K31/445 ,  A61K35/74 ,  C07D211/46 ,  C12N1/20 ,  C12N9/99 ,  C12P1/04 ,  C12P19/26 ,  C12R1/07 ,  C12R1/12 ,  C12R1/125

    CPC分类号： C12R1/07 ,  A23K20/195 ,  A23K50/30 ,  A61K31/445 ,  C12N1/20 ,  C12P1/04 ,  Y10S435/832 ,  Y10S435/839

    摘要： According to the present invention inhibitors for glycoside hydrolases, and in particular glucosidase inhibitors especially saccharase inhibitors, which are active in the digestive tract are formed by culturing organisms of the family Bacillaceae, particularly by strains of the genus Bacillus.It has also been found that certain strains of organisms of the family Bacillaceae, especially strains DSM 7, DSM 704 and DSM 675 produce the antibiotic known as 1-desoxynojirimycin. The invention therefore provides a method of producing 1-desoxynojirimycin which comprises culturing a 1-desoxynojirimycin producing organism of the genus Bacillus. Inhibitors for glycoside hydrolases and the invention includes methods for producing such inhibitors, pharmaceutical compositions containing the inhibitors and methods of treatment involving the use of the inhibitors.

    摘要翻译： 根据本发明，通过培养家蚕科的生物体，特别是通过芽孢杆菌属的菌株形成糖苷水解酶抑制剂，特别是在消化道中有活性的葡糖苷酶抑制剂，特别是糖酶抑制剂。 还已经发现，芽孢杆菌科的特定菌株DSM 7，DSM 704和DSM 675的生物体产生称为1-脱氧野尻霉素的抗生素。 因此，本发明提供了一种生产1-脱氧野尻霉素的方法，该方法包括培养产生芽孢杆菌属的1-脱氧诺伊霉素生物的生物。 糖苷水解酶和本发明的抑制剂包括制备这种抑制剂的方法，含有抑制剂的药物组合物和涉及使用抑制剂的治疗方法。

    Herbicidal compositions
    7.
    发明授权
    Herbicidal compositions 失效
    除草成分

    公开(公告)号：US06743754B2

    公开(公告)日：2004-06-01

    申请号：US09882441

    申请日：2001-06-15

    申请人： Jochen Würtz ,  Jean Kocur ,  Hans-Peter Krause ,  Julio Martinez de Una ,  Detlev Haase ,  Udo Bickers ,  Gerhard Schnabel

    发明人： Jochen Würtz ,  Jean Kocur ,  Hans-Peter Krause ,  Julio Martinez de Una ,  Detlev Haase ,  Udo Bickers ,  Gerhard Schnabel

    IPC分类号： A01N2530

    CPC分类号： A01N25/30 ,  A01N47/36 ,  A01N25/32 ,  A01N2300/00

    摘要： The present invention relates to a herbicidal composition comprising A) one or more sulfonylureas of the formula (I) and/or their salts in which R1 is C2-C4-alkoxy or CO—Ra, where Ra is OH, C1-C6-alkoxy or NRbRc, where Rb and Rc independently of one another are identical or different and are H or C1-C6-alkyl, R2 is halogen or (A)n—NRdRe, where n is zero or 1, A is a group CRfRg, where Rf and Rg independently of one another are identical or different and are H or C1-C6-alkyl, Rd is H or C1-C6-alkyl and Re is H, C1-C6-alkyl or an acyl radical, where Rd and Re may also form a heterocyclic ring and where, if R1 is C2-C4-alkoxy, R2 may also be H, R3 is H or C1-C6-alkyl, m is zero or 1, X and Y independently of one another are identical or different and are C1-C6-alkyl, C1-C6-alkoxy or C1-C6-alkylthio, where each of the three radicals mentioned is unsubstituted or substituted by one or more radicals selected from the group consisting of halogen, C1-C4-alkoxy and C1-C4-alkylthio, or are C3-C6-cycloalkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C6-alkenyloxy or C3-C6-alkynyloxy, preferably C1-C4-alkyl or C1-C4-alkoxy, Z is CH or N, and B) one or more surfactants comprising as structural element at least 10 alkylene oxide units.

    摘要翻译： 本发明涉及一种除草组合物，其包含A）一种或多种式（I）的磺酰脲和/或其盐，其中R 1是C 2 -C 4 - 烷氧基或CO-R a，其中R 5'是OH ，C 1 -C 6烷氧基或NR c R c，其中R b和R c彼此独立地相同或不同，为H或C 1 -C 6 - 烷基，R 2为卤素 或（A）n-NR d R e，其中n为零或1，A为基团CR ，其中R f和R g彼此独立地为 相同或不同的是H或C 1 -C 6烷基，R d是H或C 1 -C 6烷基，R e是H，C 1 -C 6烷基或酰基，其中R d和R 也可以形成杂环，其中如果R 1是C 2 -C 4 - 烷氧基，则R 2也可以是H，R 3是H或C 1 -C 6 - 烷基，m是0或 1，X和Y彼此独立地相同或不同，并且是C 1 -C 6 - 烷基，C 1 -C 6 - 烷氧基或C 1 -C 6 - 烷硫基，其中所提及的三个基团中的每一个是未取代的或被一个或多个选自 由卤素，C 1 -C 4烷氧基组成 y和C 1 -C 4 - 烷硫基，或者是C 3 -C 6 - 环烷基，C 2 -C 6 - 烯基，C 2 -C 6 - 炔基，C 3 -C 6 - 烯氧基或C 3 -C 6 - 炔氧基，优选C 1 -C 4烷基或C 1 -C 4 - 烷氧基，Z是CH或N，和B）一种或多种表面活性剂，其包含至少10个环氧烷单元作为结构元素。

    Azaneophyl sulfides, and their use as pesticides
    9.
    发明授权
    Azaneophyl sulfides, and their use as pesticides 失效
    硫唑烷酮和它们作为农药的用途

    公开(公告)号：US5002957A

    公开(公告)日：1991-03-26

    申请号：US327971

    申请日：1989-03-23

    申请人： Hans H. Schubert ,  Gerhard Salbeck ,  Hans-Peter Krause ,  Werner Knauf ,  Anna Waltersdorfer ,  Manfred Kern

    发明人： Hans H. Schubert ,  Gerhard Salbeck ,  Hans-Peter Krause ,  Werner Knauf ,  Anna Waltersdorfer ,  Manfred Kern

    IPC分类号： C07D253/06 ,  A01N43/40 ,  A01N55/00 ,  A01N55/10 ,  C07D213/32 ,  C07D213/61 ,  C07D213/64 ,  C07D213/643 ,  C07D213/70 ,  C07D237/12 ,  C07D237/14 ,  C07D237/18 ,  C07D239/26 ,  C07D239/32 ,  C07D239/34 ,  C07D241/16 ,  C07D241/18 ,  C07D257/08 ,  C07D401/12 ,  C07D409/12 ,  C07D491/056 ,  C07F7/10

    CPC分类号： C07D213/64 ,  A01N43/40 ,  A01N55/00 ,  C07D213/643 ,  C07D213/70 ,  C07D409/12

    摘要： Azaneophyl and silazaneophyl sulfides, processes for their preparation, agents containing them, and their use as pesticides.Compounds of the formula I, their optical isomers and mixtures thereof ##STR1## where M denotes C or Si,R.sup.1 denotes unsubstituted or substituted pyridyl, unsubstituted or substituted pyrimidyl, andwhen M=C- denotes unsubstituted or substituted pyridazinyl, unsubstituted or substituted pyrazinyl, unsubstituted or substituted 1,2,4-triazinyl, unsubstituted or substituted 1,2,4,5-tetrazinyl, R.sup.2, R.sup.3 independently or one another denote alkyl, alkenyl, haloalkyl, phenyl, or R.sup.2 and R.sup.3 denote an alkylene chain which - together with the quaternary central atom (M) - form an unsubstituted or fluorine-substituted ring having four to six ring members (when M=Si) or having three to six ring members (when M=C),R.sup.4 denotes H, F, --CN, --CCl.sub.3, --C.dbd.CH, (C.sub.1 -C.sub.4)alkyl, ##STR2## R.sup.5 denotes pyridyl, furyl, thienyl, all of which can be substituted, phthalimidyl, dialkylmaleinimidyl, thiophthalimidyl, dihydrophthalimidyl, tetrahydrophthalimidyl, substituted phenylor R.sup.4 and R.sup.5 - together with the carbon atom bridging them denote an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical,and to their salts and quaternization products for advantageous insecticidal, acaricidal or nematocidal properties.

    摘要翻译： Azaneophyl和silazaneophyl硫化物，它们的制备方法，含有它们的试剂，以及它们作为农药的用途。 式I化合物，其旋光异构体及其混合物，其中M表示C或Si，R1表示未取代或取代的吡啶基，未取代或取代的嘧啶基，当M = C-表示未取代或取代的哒嗪基时，未取代的 或取代的吡嗪基，未取代或取代的1,2,4-三嗪基，未取代或取代的1,2,4,5-四嗪基，R2，R3独立地或者彼此表示烷基，烯基，卤代烷基，苯基或R2和R3表示 亚烷基链与四元中心原子（M）一起形成具有四至六个环成员（当M = Si）或具有三至六个环成员（当M = C时）的未取代或氟取代的环，R4表示 H，F，-CN，-CCl 3，-C = CH，（C 1 -C 4）烷基，R 5表示吡啶基，呋喃基，噻吩基，它们都可被取代，苯二酰亚氨基，二烷基马来酰亚胺基，硫代邻苯二甲酰亚胺基，二氢邻苯二甲酰亚氨基，四氢邻苯二甲酰亚胺基， 取代的苯基或R 4和R 5 - 与碳原子一起 桥接它们表示任选取代的茚满基，环戊烯基或环戊烯基，以及它们的盐和季铵化产物，用于有利的杀虫，杀螨或杀线虫性质。