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    HERBICIDAL BENZOYL DERIVATIVES
    32.
    发明申请
    HERBICIDAL BENZOYL DERIVATIVES 审中-公开
    除草剂苯甲酰

    公开(公告)号：WO1996026200A1

    公开(公告)日：1996-08-29

    申请号：PCT/EP1996000593

    申请日：1996-02-13

    Applicant: BASF AKTIENGESELLSCHAFT ,  VON DEYN, Wolfgang ,  HILL, Regina, Luise ,  KARDORFF, Uwe ,  ENGEL, Stefan ,  OTTEN, Martina ,  VOSSEN, Marcus ,  PLATH, Peter ,  RANG, Harald ,  HARREUS, Albrecht ,  RÖHL, Franz ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto ,  MISSLITZ, Ulf

    Inventor： BASF AKTIENGESELLSCHAFT

    IPC: C07D307/54

    CPC classification number: C07D271/06 ,  A01N43/08 ,  A01N43/10 ,  A01N43/74 ,  A01N43/80 ,  C07D261/04 ,  C07D261/08 ,  C07D263/14 ,  C07D263/32 ,  C07D277/26 ,  C07D307/46 ,  C07D333/22

    Abstract: The invention concerns benzoyl derivatives of formula (I) in which the substituents have the following meanings: L and M represent hydrogen, C1-C6 alkyl, C2-C6 alkenyl, C2-C6 alkinyl, C1-C4 alkoxy (these groups being optionally substituted by one to five halogen atoms or C1-C4 alkoxy), halogen, cyano, nitro, a -(Y)n-S(O)mR or -(Y)n-CO-R group; Z represents a five to six-membered heterocyclic saturated or unsaturated group containing one to three heteroatoms selected from the group comprising oxygen, sulphur and nitrogen and which can optionally be substituted by halogen, cyano, nitro, a -CO-R group, C1-C4 alkyl, C1-C4 alkyl halide, C3-C8 cycloalkyl, C1-C4 alkoxy, C1-C4 alkoxy halide, C1-C4 alkyl thio, C1-C4 alkyl thio halide, di-C1-C4 alkyl amino, phenyl optionally substituted by halogen, cyano, nitro, C1-C4 alkyl or C1-C4 alkyl halide, or an oxo group which can be present in the tautomeric form as a hydroxy group, is substituted or, together with a condensation-bound phenyl ring which is optionally substituted by halogen or, cyano, nitro, C1-C4 alkyl or C1-C4 alkyl halide, with a condensation-bound carbocycle or with a condensation-bound second heterocycle which can optionally be substituted by halogen, cyano, nitro, C1-C4 alkyl, di-C1-C4 alkyl amino, C1-C4 alkoxy, C1-C4 alkoxy halide or a C1-C4 alkyl halide, forms a bicyclic system; Y represents O or NR ; n is 0 or 1; m is 0, 1 or 2; R represents C1-C4 alkyl, C1-C4 alkyl halide or NR R ; R represents C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy or NR R ; R represents hydrogen or C1-C4 alkyl; R represents C1-C4 alkyl; Q represents a cyclohexane-1,2-dione ring connected at position 2 and of formula (II) in which R , R , R and R represent hydrogen or C1-C4 alkyl, R represents hydrogen, C1-C4 alkyl or a -COOR group, R represents hydrogen, C1-C4 alkyl, C3-C6 cycloalkyl, these groups optionally including one to three of the following substituents: halogen, C1-C4 alkyl thio, C1-C4 alkoxy, or R represents tetrahydropropanyl-3, tetrahydropropanyl-4 or tetrahydrothiopyranyl-3, or R and R together form a bond or a three to six-membered carbocyclic ring. The invention also concerns standard agricultural salts of compounds of formula (I) usually utilized in agriculture.

    Abstract translation: 式（I），其中取代基具有以下含义的苯甲酰衍生物：L，M是氢，C1-C6烷基，C2-C6链烯基，C2-C6炔基，C1-C4烷氧基，这些基团任选地被一个取代 可被取代到5个卤素原子或C1-C4烷氧基，卤素，氰基，硝基，基团 - （Y）N S（O）MR <7>或基团 - （Y）N-CO-R <8>，一个 5-或6-元杂环的饱和或含有选自氧，硫或氮中选择的一至三个杂原子的不饱和基团，其任选被卤素，氰基，硝基，基团-CO-R取代的<8>，C1- C4烷基，C1-C4卤代烷基，C3-C8环烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4烷硫基，C1-C4卤代烷硫基，二-C 1 -C 4 - 烷基氨基，任选地被取代的 卤素，氰基，硝基，C1-C4烷基或C1-C4卤代烷基取代的苯基或氧代基团，其也可以任选地以互变异构形式作为羟基存在，或在一个被取代的 稠合的，任选地被卤素，氰基，硝基，C1-C4烷基或C1-C4卤代烷基的苯环，稠合碳环或稠合的，任选被卤素取代，氰基，硝基，C1-C4烷基，二C1-C4取代的 烷基氨基，C1-C4烷氧基，C1-C4卤代烷氧基，或C1-C4卤代烷基取代的杂环第二形成双环体系; Y是O，NR <9>; n是0或1; m是零，1或2; [R <7> C1-C4烷基，C1-C4卤代烷基，或NR <9> - [R <10>; [R <8> C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，或NR <9> - [R <10>; [R <9>是氢或C1-C4烷基; [R <10> C1-C4烷基; Q，R <4>和R <6>表示一个在式环己烷-1,3-二酮环的2位连接（II）其中R <1>，R <2>是氢或C1-C4烷基， [R <5>是氢，C1-C4烷基或基团-COOR <10>，R <3>为氢，C1-C4烷基，C3-C6环烷基，这些基团任选地具有1至3个如下取代基取代的 可以：卤素，C1-C4烷硫基或C1-C4烷氧基，或R <3>为四氢吡喃基-3，四氢吡喃基-4或四氢噻喃基-3，或R <3>和R <5>一起代表一个键或 形成三至六元碳环，和化合物（I）的可农用常用盐。

    ANTIINFLAMMATORY AND ANTITUMOR 2-OXOTHIAZOLES AND 2-OXOTHIOPHENES COMPOUNDS
    35.
    发明申请
    ANTIINFLAMMATORY AND ANTITUMOR 2-OXOTHIAZOLES AND 2-OXOTHIOPHENES COMPOUNDS 审中-公开
    抗氧化剂和抗氧化剂2-氧杂环丙烷和2-氧杂环戊烯化合物

    公开(公告)号：WO2014118195A1

    公开(公告)日：2014-08-07

    申请号：PCT/EP2014/051655

    申请日：2014-01-28

    Applicant: AVEXXIN AS

    Inventor： JOHANSEN, Berit ,  SANDBERG, Marcel ,  AUKRUST, Inger-Reidun ,  KOKOTOS, George ,  BARBAYIANNI, Efrosini

    IPC: C07D277/24 ,  C07D277/56 ,  A61K31/426 ,  A61P1/00

    CPC classification number: C07D333/38 ,  A61K31/381 ,  A61K31/426 ,  A61K31/428 ,  A61K45/06 ,  C07D277/24 ,  C07D277/26 ,  C07D277/56 ,  C07D277/64

    Abstract: A compound of formula (I) wherein X is O, C O or S; Y is N or CH; R 2 and R 4 are each independently H, -(CH 2 ) p COOH, -(CH 2 ) p CON(R 5 ) 2 or - (CH 2 ) p COOC 1-6 alkyI; or R 2 and R 4 together form a 6-membered phenyl ring fused to the five membered ring; each R 1 is independently selected from H, halo (e.g. fluoro or chloro), C 6-10 aryl, C 7-12 arylalkyl, C 2-12 alkenyl; OC 1-2 alkyl, OC 2-12 aikenyl or a C 1-12 alkyl group; each R 5 is H or C 1-6 alkyl; each p is 0 to 3; n is 1 to 4; or a salt, ester, solvate, N-oxide, or prodrug thereof, e.g. a salt thereof.

    Abstract translation: 式（I）化合物，其中X为O，C O或S; Y为N或CH; R2和R4各自独立地为H， - （CH2）pCOOH， - （CH2）pCON（R5）2或 - （CH2）pOCOC 1-6烷基; 或者R 2和R 4一起形成与五元环稠合的6元苯环; 每个R 1独立地选自H，卤素（例如氟或氯），C 6-10芳基，C 7-12芳基烷基，C 2-12烯基; OC1-2烷基，OC2-12亚基或C1-12烷基; 每个R 5是H或C 1-6烷基; 每个p为0至3; n为1至4; 或其盐，酯，溶剂化物，N-氧化物或前药，例如。 其盐。

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