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136 条记录 (耗时 0.038 秒)

    Benzylidenepyrazolones, their preparation and use
    52.
    发明授权
    Benzylidenepyrazolones, their preparation and use 失效
    亚苄基吡唑啉酮，其制备和用途

    公开(公告)号：US06500950B1

    公开(公告)日：2002-12-31

    申请号：US09765626

    申请日：2001-01-22

    申请人： Joachim Rheinheimer ,  Matthias Witschel ,  Stefan Engel ,  Ernst Baumann ,  Wolfgang von Deyn ,  Regina Luise Hill ,  Guido Mayer ,  Ulf Misslitz ,  Oliver Wagner ,  Martina Otten ,  Karl-Otto Westphalen ,  Helmut Walter

    发明人： Joachim Rheinheimer ,  Matthias Witschel ,  Stefan Engel ,  Ernst Baumann ,  Wolfgang von Deyn ,  Regina Luise Hill ,  Guido Mayer ,  Ulf Misslitz ,  Oliver Wagner ,  Martina Otten ,  Karl-Otto Westphalen ,  Helmut Walter

    IPC分类号： C07D41310

    CPC分类号： C07D413/06 ,  A01N43/56 ,  A01N43/78 ,  A01N43/80 ,  C07D231/16 ,  C07D231/20

    摘要： Benzylidenepyrazolones of the formula I, where the substituents and the index n have the following meanings: R1 is unsubstituted or substituted C1-C6-alkyl; R2 is unsubstituted or substituted C1-C6-alkyl, unsubstituted or substituted C1-C6-alkoxy, halogen, nitro, cyano; R3 is hydrogen, halogen, nitro, cyano, a group NR5R6, OCOR5, NR5COR6, CO2R5, —COSR5, —CONR5R6, C1-C4-alkoxyiminoalkyl, C1-C6-alkylcarbonyl, unsubstituted or substituted C1-C6-alkyl, unsubstituted or substituted C1-C6-alkoxy, unsubstituted or substituted C1-C6-alkylthio, unsubstituted or substituted C2-C6-alkenyl, unsubstituted or substituted C2-C6-alkynyl, unsubstituted or substituted phenyl, unsubstituted or substituted phenoxy, an unsubstituted or substituted 5- or 6-membered saturated or unsaturated heterocycle which may contain up to 4 nitrogen atoms and/or up to 2 oxygen or sulfur atoms as ring members; R4 is C1-C6-alkyl, C1-C4-haloalkyl; R3 and R4 form an optionally substituted saturated or unsaturated 2- or 3-membered bridge which may contain a sulfur atom which may be oxidized to the sulfoxide or sulfone; R5 is hydrogen or unsubstituted or substituted C1-C6-alkyl; R6 is unsubstituted or substituted C1-C6-alkyl; R7 is hydrogen, C1-C6-alkyl or C1-C4-haloalkyl; n is 0,1 or 2, X is hydrogen, chlorine or bromine; where the compounds claimed may be present both in the trans and in the cis form or as a mixture of these isomers, are described.

    摘要翻译： 式I的亚苄基吡唑酮，其中取代基和指数n具有以下含义：R 1是未取代的或取代的C 1 -C 6 - 烷基; R 2是未取代的或取代的C 1 -C 6 - 烷基，未取代或取代的C 1 -C 6 - 烷氧基，卤素 硝基，氰基; R 3是氢，卤素，硝基，氰基，NR 5 R 6，OCOR 5，NR 5 COR 6，CO 2 R 5，-COSR 5，-CONR 5 R 6，C 1 -C 4烷氧基亚氨基烷基，C 1 -C 6烷基羰基，未取代或取代的C 1 -C 6 - 未取代或取代的C 1 -C 6 - 烷硫基，未取代或取代的C 2 -C 6 - 烯基，未取代或取代的C 2 -C 6 - 炔基，未取代或取代的苯基，未取代或取代的苯氧基，未取代的 或可以含有至多4个氮原子和/或至多2个氧或硫原子作为环成员的取代的5或6元饱和或不饱和杂环; R 4是C 1 -C 6烷基，C 1 -C 4卤代烷基; R 3和 R4形成任选取代的饱和或不饱和的2-或3-元 桥可以含有可被氧化成亚砜或砜的硫原子; R5是氢或未取代或取代的C1-C6-烷基; R6是未取代的或取代的C1-C6-烷基; R7是氢，C1-C6-烷基 或C 1 -C 4卤代烷基; n为0,1或2，X为氢，氯或溴;其中要求保护的化合物可以以反式和顺式形式存在，或以这些异构体的混合物存在。

    Quinoline-3-carboxamides, their manufacture and use
    58.
    发明授权
    Quinoline-3-carboxamides, their manufacture and use 失效
    喹啉-3-甲酰胺，其制造和使用

    公开(公告)号：US5972841A

    公开(公告)日：1999-10-26

    申请号：US988765

    申请日：1997-12-11

    申请人： Wolfgang von Deyn ,  Hans Theobald ,  Christoph Nuebling ,  Uwe Kardorff ,  Helmut Walter ,  Karl-Otto Westphalen ,  Thomas Kappe ,  Matthias Gerber

    发明人： Wolfgang von Deyn ,  Hans Theobald ,  Christoph Nuebling ,  Uwe Kardorff ,  Helmut Walter ,  Karl-Otto Westphalen ,  Thomas Kappe ,  Matthias Gerber

    IPC分类号： A01N43/42 ,  C07D215/56

    CPC分类号： A01N43/42 ,  C07D215/56

    摘要： Quinoline-3-carboxamides I ##STR1## where R.sup.1 is hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, and the organic radicals may be substituted or unsubstituted;R.sup.2 is hydrogen, hydroxyl, alkoxy, alkenyloxy, dialkylamino, alkyl, alkenyl, alkynyl, cycloalkyl, and the organic radicals may be substituted or unsubstituted;orR.sup.1, R.sup.2 together denote an alkylene chain of 4 to 7 members and which may be interrupted by oxygen, sulfur or N-methyl;R.sup.3 -R.sup.6 are hydrogen, alkyl, alkoxy, haloalkyl, haloalkoxy, alkylthio, haloalkylthio, halogen, cyano or nitro;X is oxygen or sulfur;with the proviso that R.sup.2 is not hydrogen, C.sub.1 -C.sub.3 -alkyl, n-butyl, 3-methylbutyl, cyclohexyl, hexyl, heptyl, octyl, 2-chlorobenzyl, 3-(dimethylamino)propyl, 3-(diethylamino)propyl, 2-morpholinoethyl or 2-(3,4-dimethoxyphenyl)ethyl when R.sup.1 and R.sup.3 to R.sup.6 are hydrogen and X is oxygen, and that R.sup.2 is not benzyl when R.sup.1 is methyl, R.sup.3 to R.sup.6 are hydrogen and X is oxygen, and that R.sup.1 and R.sup.2 do not jointly denote morpholino when R.sup.3 to R.sup.6 are hydrogen and X is oxygen.

    摘要翻译： 其中R 1是氢，烷基，烯基，炔基，环烷基和有机基团的喹啉-3-甲酰胺I可以是取代或未取代的; R2是氢，羟基，烷氧基，烯氧基，二烷基氨基，烷基，烯基，炔基，环烷基，有机基可以是取代或未取代的; 或R 1，R 2一起表示4至7个成员的亚烷基链，并且可被氧，硫或N-甲基中断; R3-R6是氢，烷基，烷氧基，卤代烷基，卤代烷氧基，烷硫基，卤代烷硫基，卤素，氰基或硝基; X是氧或硫; 条件是R2不是氢，C1-C3-烷基，正丁基，3-甲基丁基，环己基，己基，庚基，辛基，2-氯苄基，3-（二甲基氨基）丙基，3-（二乙基氨基）丙基， 当R 1和R 3至R 6为氢且X为氧时，R 2为苄基，R 3为R 6为氢，X为氧时，R 2为苄基， 当R 3至R 6为氢且X为氧时，R 2不共同表示吗啉代。

    Saccharin derivatives
    60.
    发明授权
    Saccharin derivatives 失效
    糖精衍生物

    公开(公告)号：US5716905A

    公开(公告)日：1998-02-10

    申请号：US776568

    申请日：1997-02-03

    申请人： Peter Plath ,  Wolfgang von Deyn ,  Stefan Engel ,  Uwe Kardorff ,  Christoph Nubling ,  Hartmann Konig ,  Harald Rang ,  Matthias Gerber ,  Helmut Walter ,  Karl-Otto Westphalen

    发明人： Peter Plath ,  Wolfgang von Deyn ,  Stefan Engel ,  Uwe Kardorff ,  Christoph Nubling ,  Hartmann Konig ,  Harald Rang ,  Matthias Gerber ,  Helmut Walter ,  Karl-Otto Westphalen

    IPC分类号： C07D275/04 ,  A01N43/80 ,  C07D275/06

    CPC分类号： C07D275/06 ,  A01N43/80

    摘要： Saccharin derivatives of the formula I ##STR1## where the substituents have the following meanings: L and M are hydrogen, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -alkylthio, chlorine, cyano, methylsulfonyl, nitro or trifluoromethyl; Z is hydrogen, C.sub.1 -C.sub.4 -alkyl, C.sub.3 -C.sub.8 -cycloalkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.5 -alkynyl, C.sub.1 -C.sub.4 -acyl, benzyl or phenyl, the phenyl rings being unsubstituted or substituted by halogen or C.sub.1 -C.sub.4 -alkyl; R.sup.1 is cyclopropyl, 1-methylcyclopropyl, 1-methylthiocyclopropyl or tert-butyl; and agriculturally customary salts of the compounds I are described.

    摘要翻译： PCT No.PCT / EP95 / 02977。 371日期1997年2月3日 102（e）日期1997年2月3日PCT提交1995年7月27日PCT公布。 出版物WO96 / 05183 日期：1996年2月22日式Ⅰ的糖精衍生物其中取代基具有下列含义：L和M是氢，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基，C 1 -C 4 - 烷硫基，氯，氰基 ，甲基磺酰基，硝基或三氟甲基; Z是氢，C 1 -C 4 - 烷基，C 3 -C 8 - 环烷基，C 3 -C 6 - 烯基，C 3 -C 5炔基，C 1 -C 4酰基，苄基或苯基，苯环是未取代的或被卤素或C1- C4-烷基; R1是环丙基，1-甲基环丙基，1-甲硫基环丙基或叔丁基; 并描述了化合物I的农业常规盐。