Morpholinothio oxamides
    54.
    发明授权
    Morpholinothio oxamides 失效
    吗啉代氧酰胺

    公开(公告)号:US4006140A

    公开(公告)日:1977-02-01

    申请号:US588310

    申请日:1975-06-19

    申请人: Pyong-Nae Son

    发明人: Pyong-Nae Son

    CPC分类号: C07D295/26 C08K5/43

    摘要: Vulcanizable rubber compositions comprising a sulfur vulcanizable rubber, sulfur, a thiazole sulfenamide accelerator, a morpholinothio amide compound, and optionally a benzothiazole or thiuram accelerator exhibit good scorch safety and yield vulcanizates having excellent original and heat aged properties.

    摘要翻译: 包含硫硫化橡胶,硫,噻唑亚磺酰胺促进剂,吗啉代硫代酰胺化合物和任选的苯并噻唑或秋兰姆加速剂的可硫化橡胶组合物表现出良好的焦烧安全性,并且具有优异的原始和热老化性能的硫化胶。

    Formamidine insecticides
    55.
    发明授权
    Formamidine insecticides 失效
    甲脒杀虫剂

    公开(公告)号:US3998969A

    公开(公告)日:1976-12-21

    申请号:US575247

    申请日:1975-05-07

    申请人: Victor L. Rizzo

    发明人: Victor L. Rizzo

    摘要: Novel pesticidal compounds of the formula: ##STR1## wherein R.sub.1 is lower alkyl of from 1 to 4 carbon atoms; R.sub.2 is hydrogen, halogen or lower alkyl of from 1 to 4 carbon atoms; R.sub.3 and R.sub.4 are the same or different and are hydrogen, alkyl of 1 to 8 carbon atoms, inclusive; haloalkyl, arylalkyl and ##STR2## WHEREIN ALKYL IS FROM 1 TO 4 CARBON ATOMS, CYCLOALKYL OF FROM 3 TO 6 CARBON ATOMS, ARYL AND R.sub.3 and R.sub.4 taken together are a member selected from the group piperidine, morpholine, pyrazole, tribromopyrazole, N-methylpiperazine, pyrrole, pyrrolidine, pyrrolidone.The compounds are combined with carriers to prepare compositions and are useful in controlling insect pests either as an insecticide or behavioral modifier and are particularly effective as miticides.

    摘要翻译: 下式的新型杀虫化合物:其中R 1是1至4个碳原子的低级烷基; R 2是氢,卤素或具有1至4个碳原子的低级烷基; R3和R4相同或不同,为氢,1〜8个碳原子的烷基,包括端值; 卤代烷基,芳基烷基和其中亚烷基是1至4个碳原子,3至6个碳原子的环烷基,芳基和R3和R4一起是选自哌啶,吗啉,吡唑,三溴吡唑, 甲基哌嗪,吡咯,吡咯烷,吡咯烷酮。

    3-(4-Acylaminopiperazin-1-yl alkyl)indoles, precursors and processes for
the preparation thereof
    57.
    发明授权
    3-(4-Acylaminopiperazin-1-yl alkyl)indoles, precursors and processes for the preparation thereof 失效
    3-(4-酰氨基哌嗪-1-基烷基)吲哚,其前体及其制备方法

    公开(公告)号:US3997539A

    公开(公告)日:1976-12-14

    申请号:US475315

    申请日:1974-05-31

    CPC分类号: C07D403/06

    摘要: New 3-(4-acylaminopiperazin-1-ylalkyl)indole compounds, and their immediate precursors possessing antihypertensive and tranquilizing properties, their physiologically acceptable salts and a process for the preparation thereof are described; said compounds are of the general formula: ##STR1## wherein X represents hydrogen or hydroxy, n can vary from 0-1, R.sub.1 and R.sub.2 each represents hydrogen or alkoxy of 1-2 carbon atoms; R.sub.3 represents hydrogen or alkyl of 1-3 carbon atoms and Z represents hydrogen or ##STR2## and R.sub.4 is selected from a member of the group consisting of alkyl of 1-4 carbon atoms, benzhydryl, cycloalkyl of 6-10 carbon atoms; bridged cycloalkyl of 6-10 carbon atoms, phenyl, mono, di or tri substituted phenyl, and heterocyclic moieties such as pyridyl, furyl, pyrrolyl, thienyl, pyrazinyl.

    摘要翻译: 描述了新的3-(4-酰氨基哌嗪-1-基烷基)吲哚化合物及其具有抗高血压和镇静特性的其直接前体,其生理学上可接受的盐及其制备方法; 所述化合物具有以下通式:其中X表示氢或羟基,n可以为0-1,R1和R2各自表示氢或1-2个碳原子的烷氧基; R 3表示氢或1-3个碳原子的烷基,Z表示氢或者R 4选自1-4个碳原子的烷基,二苯甲基,6-10个碳原子的环烷基; 6-10个碳原子的桥连环烷基,苯基,单或二取代的苯基,以及杂环部分如吡啶基,呋喃基,吡咯基,噻吩基,吡嗪基。

    1-(ARYLTHIO, ARYLSULFINYL AND ARYLSULFONYL)-1,1-DIHALOMETHANESULFONAMIDES
    58.
    发明授权
    1-(ARYLTHIO, ARYLSULFINYL AND ARYLSULFONYL)-1,1-DIHALOMETHANESULFONAMIDES 失效
    1-(ARYLTHIO,ARYLSULFINYL和ARYLSULFONYL)-1,1-二缩水甘油醚

    公开(公告)号:US3946007A

    公开(公告)日:1976-03-23

    申请号:US554953

    申请日:1975-03-03

    CPC分类号: C07D295/26 C07D211/10

    摘要: The compounds of the formula ##SPC1##In which R is lower alkyl, lower alkoxy or halo, x is an integer from 0 to 2, n is an integer from 0 to 3, Y is halo and R.sub.1 and R.sub.2 independently are hydrogen, lower alkyl, phenyl or substituted phenyl, or, together with the nitrogen atom, form a heterocyclic ring also containing up to one oxygen atom in the heterocycle. The compounds in which x is 0 are prepared by adding chlorine or bromine to a 1-arylthiomethanesulfonamide in the presence of pyridine to form the 1-arylthio-1, 1-dihalomethanesulfonamide. The compounds in which x is 1 or 2 is prepared by adding sodium hypochlorite or sodium hypobromite to a 1-(arylsulfinyl)methane-sulfonamide or a 1-(arylsulfonyl)methanesulfonamide to form the 1-(arylsulfinyl)-1,1-dihalomethanesulfonamide or 1-(arylsulfonyl)-1,1-dihalomethanesulfonamide, respectively. The compounds are useful as antimicrobial agents.

    摘要翻译: 式中R为低级烷基,低级烷氧基或卤素的化合物,x为0至2的整数,n为0至3的整数,Y为卤素,R 1和R 2各为氢,低级烷基,苯基 或取代的苯基,或者与氮原子一起形成在该杂环中也含有至多一个氧原子的杂环。 在吡啶存在下,通过在1-芳基硫代甲磺酰胺中加入氯或溴来制备x为0的化合物,形成1-芳硫基-1,1-二卤代甲磺酰胺。 通过向1-(芳基亚磺酰基)甲磺酰胺或1-(芳基磺酰基)甲磺酰胺中加入次氯酸钠或次溴酸钠,形成1-(芳基亚磺酰基)-1,1-二卤代甲磺酰胺制备x为1或2的化合物 或1-(芳基磺酰基)-1,1-二卤代甲磺酰胺。 这些化合物可用作抗微生物剂。

    N,N'-bisimidothio-diamines
    59.
    发明授权
    N,N'-bisimidothio-diamines 失效
    N,N {40-双嘧啶硫代二胺

    公开(公告)号:US3944552A

    公开(公告)日:1976-03-16

    申请号:US448858

    申请日:1974-03-07

    申请人: John P. Lawrence

    发明人: John P. Lawrence

    IPC分类号: C08K5/43 C07D295/22

    CPC分类号: C08K5/43 C08K5/44

    摘要: Imides such as N-(morpholinothio)phthalimide are used to affect the vulcanization characteristics of sulfur vulcanizable polymers by increasing the state of vulcanization and/or improving scorch resistance and/or increasing the rate of vulcanization.

    摘要翻译: 通过增加硫化状态和/或改善抗焦烧性和/或提高硫化速率,使用N-(吗啉代硫代)邻苯二甲酰亚胺等酰亚胺来影响硫可硫化聚合物的硫化特性。