Fungicidal substituted 3-amino-2-pyrazolin-5-ones, compositions and use
    5.
    发明授权
    Fungicidal substituted 3-amino-2-pyrazolin-5-ones, compositions and use 失效
    杀真菌剂取代的3-氨基-2-吡唑啉-5-酮,组合物和用途

    公开(公告)号:US4968714A

    公开(公告)日:1990-11-06

    申请号:US481487

    申请日:1990-02-16

    摘要: Fungicidal substituted 3-amino-2-pyrazolin-5-ones of the formula ##STR1## in which R.sup.1 represents unsubstituted or substituted alkyl, unsubstituted or substituted alkenyl or alkinyl, or unsubstituted or substituted cycloalkyl or cycloalkenyl,R.sup.2 represents hydrogen, unsubstituted or substituted alkyl, unsubstituted or substituted alkenyl or alkinyl, unsubstituted or substituted cycloalky or cycloalkenyl, unsubstituted or substituted aryl or unsubstituted or substituted heterocyclyl, or represents one of the radicals --CX--YR.sup.3, --CXNR.sup.4 R.sup.5, ##STR2## --SO.sub.2 NR.sup.4 R.sup.5 or --SO.sub.2 R.sup.7, R.sup.3 represents unsubstituted or substituted alkyl or unsubstituted or substituted alkenyl or alkinyl,R.sup.4 and R.sup.5 are identical or different and represent hydrogen, unsubstituted or substituted alkyl, unsubstituted or substituted alkenyl or alkinyl or unsubstituted or substituted aryl or heterocyclyl, or together with the nitrogen atom to which they are bonded represent an unsubstituted or substituted heterocyclic ring which can contain further hetero atoms,R.sup.6 represents hydrogen, unsubstituted or substituted alkyl, unsubstituted or substituted alkenyl or alkinyl, unsubstituted or substituted cycloalkyl or cycloalkenyl, unsubstituted or substituted aryl or unsubstituted or substituted heterocyclyl alkoxycarbonyl or phenylcarbonyl,R.sup.7 represents unsubstituted or substituted alkyl or unsubstituted or substituted aryl andX and Y are identical or different and represent oxygen or sulphur.

    摘要翻译: R 1表示未取代或取代的烷基,未取代或取代的烯基或炔基,或未取代或取代的环烷基或环烯基的式(I)的杀真菌剂取代的3-氨基-2-吡唑啉-5-酮,R 2表示氢, 未取代或取代的烷基,未取代或取代的烯基或炔基,未取代或取代的环烷基或环烯基,未取代或取代的芳基或未取代或取代的杂环基,或代表基团-CX-YR3,-CXNR4R5,-SO2NR4R5或 - SO 2 R 7,R 3表示未取代或取代的烷基或未取代或取代的烯基或炔基,R 4和R 5相同或不同,表示氢,未取代或取代的烷基,未取代或取代的烯基或炔基或未取代或取代的芳基或杂环基, 它们所键合的氮原子表示未取代或取代的杂环, 未取代或取代的烯基或炔基,未取代或取代的环烷基或环烯基,未取代或取代的芳基或未取代或取代的杂环基烷氧基羰基或苯基羰基,R7代表未取代或取代的烷基或未取代的烷基 或取代的芳基,X和Y相同或不同,代表氧或硫。

    Combating fungi with trisubstituted cyanoguanidines
    10.
    发明授权
    Combating fungi with trisubstituted cyanoguanidines 失效
    抗真菌与三取代的氰基胍

    公开(公告)号:US4491595A

    公开(公告)日:1985-01-01

    申请号:US249249

    申请日:1981-03-30

    CPC分类号: C07D295/215 C07C279/28

    摘要: Trisubstituted cyanoguanidines of the formula ##STR1## in which R.sup.1 represents an optionally substituted phenyl or phenylalkyl radical, an alkyl radical with more than 1 carbon atom, a substituted alkyl radical, an alkenyl or alkinyl radical or an optionally substituted cycloalkyl radical,R.sup.2 represents an optionally substituted alkyl radical or an alkenyl or alkinyl radical andR.sup.3 represents an optionally substituted alkyl radical, an alkenyl or alkinyl radical, an optionally substituted cycloalkyl radical or an optionally substituted phenyl or phenylalkyl radical, orR.sup.2 and R.sup.3, together with the nitrogen atom to which they are bonded, represent an optionally substituted heterocyclic radical, which optionally contains an oxygen atom as a further hetero-atom,or a physiologically acceptable acid addition salt thereof, which possess fungicidal properties. Processes for their preparation are also taught.

    摘要翻译: 其中R 1表示任选取代的苯基或苯基烷基,具有多于1个碳原子的烷基,取代的烷基,链烯基或炔基或任选取代的环烷基,其中R 3代表下式的三取代的氰基胍: 任选取代的烷基或烯基或炔基,R 3表示任选取代的烷基,烯基或炔基,任选取代的环烷基或任选取代的苯基或苯基烷基,或R 2和R 3与氮原子一起 它们是键合的,表示任选地含有氧原子作为另外的杂原子的任选取代的杂环基,或其生理上可接受的酸加成盐,其具有杀真菌性。 还介绍了其准备过程。