Abstract:
The present invention relates to a process for the preparation of a compound of formula (I), wherein R 1 is selected from C 1-6 -alkyl, C 3-6 -cycloalkyl and aralkyl, and wherein R 2 at each occurrence independently is halogen or C 1-6 -alkyl, and m is an integer from 0 to 4, Q is selected from halogen, -NO 2 and -NR 3 R 4 , wherein R 3 and R 4 are independently selected from hydrogen, C 1-6 -alkyl, C 3-6 -cycloalkyl, aryl, aralkyl, mesyl and tosyl, or wherein R 3 and R 4 together form a C 4-6 -alkylene group, Y at each occurrence is hydrogen or a hydroxy protection group W that can be hydrolytically cleaved under acidic conditions, and n is an integer from 1 to 3, and n is an integer from 1 to 3, with the proviso that n and m together are not greater than 5.
Abstract:
Die Erfindung betrifft ein Verfahren zur (2E)-2-(Hydroxyphenyl)-2-(alkoxyimino)-N-methylacetamiden der Formel (I) in welcher R für einfach bis dreifach durch Fluor subsituiertes oder unsubstituiertes C 1 -C 6 -Alkyl steht, durch Umsetzung von Benzofuran-2,3-dion-3-oxim mit Methylamin and anschliessender Alkylierung.
Abstract:
A medicine containing as the active ingredient a novel carboxylic acid derivative useful as an insulin resistance ameliorant. The carboxylic acid derivative is represented by the following general formula (I). Also provided are a salt or ester of the derivative and a hydrate of either. (I) In the formula, R 1 represents carboxyl, alkyl, alkoxy, etc.; L and T each represents a single bond, alkylene, alkynylene, etc.; M represents alkylene, etc.; W represents carboxyl; X represents oxygen, −NR X1 CQ 1 O−, −OCQ 1 NR X1 −, −CQ 1 NR X1 O− (wherein Q 1 represents oxygen, etc. and R X1 represents hydrogen, alkyl, etc.), etc.; and Y and Z each represents an optionally substituted 5− to 14−membered aromatic group, etc.
Abstract:
The present invention provides an ester compound encompassed by formula (I) wherein R represents a hydrogen atom, a C1 to C5 alkyl group which may be substituted with at least one halogen atom, a C4 to C5 cycloalkyl group which may be substituted with at least one halogen atom, a C3 to C5 alkenyl group which may be substituted with at least one halogen atom, a C3 to C5 alkynyl group which may be substituted with at least one halogen atom, a (C3 to C5 cycloalkyl)methyl group which may be substituted with at least one halogen atom or a C2 to C5 (alkoxyalkyl) group which may be substituted with at least one halogen atom. Further, the present invention provides an aldehyde compound encompassed by formula (II) Furthermore, the present invention provides pesticidal methods.
Abstract:
The invention relates to novel fluoromethoximino compounds, methods for producing the same and their use as pest-control agents, as well as to new intermediate products and several methods for producing said products.
Abstract:
Compounds of formula (I) and possible isomers and isomeric mixtures thereof, wherein: a) X is CH2F or CHF2; Y is CH and Z is OMe, or b) X is CH2F or CHF2; Y is a nitrogen atom and Z is OMe or NHCH3, and wherein also m is 0, 1, 2, 3, 4 or 5 and U represents identical or different substituents selected from halogen, cyano, nitro, C1-C12alkyl, C3-C8cycloalkyl, C3-C6alkenyl, C3-C6alkenyloxyiminomethyl, C1-C4alkoxy, C1-C4alkoxyiminomethyl, C1-C2haloalkyl, C1-C2haloalkoxy, unsubstituted or substituted phenyl, unsubstituted or substituted phenoxy and unsubstituted or substituted benzyl or represents substituents at two adjacent positions of the phenyl ring of formula (I) that define a fused hydrocarbon bridge so as to form a larger hydrocarbon ring having up to 14 carbon atoms, are suitable for controlling and preventing microorganisms, insects and Acarina on plants. They can be used in the form of commercially customary formulated compositions.
Abstract:
Cyclohexenone derivates have the formula (I), in which R1 stands for alkyl, alkenyl, alkinyl, cycloalkyl, aloxyalkyl, alkylthioalkyl, possibly substituted phenyl, possibly substituted benzyl, possibly substituted 5-/6-membered heteroaryl; W stands for 0, =N-OR2 or =N-R3; R2 stands for possibly substituted alkyl, alkenyl or alkinyl residue, possibly substituted 3- to 6-membered alkyl chain or 4- to 6-membered alkenyl or alkinyl chain, a chain link in each of the chains being substituted by -0-, -S-, -S0-, -S0¿2?- or -N(R?8)-; R8¿ stands for H, alkyl, alkenyl, alkinyl, alkylcarbonyl, benzoyl; R3 stands for H, alkyl hydroxyakyl, alkoxyalkyl or alkylthioalkyl, possibly substituted phenyl, possibly substituted benzyl; X, Y stand for -OR?4 or -NR5 R6; R4¿ stands for H, alkyl, akenyl, alkinyl, alkoxyalkyl, alkylthioalkyl; R5 stands for H, alkyl, alkenyl, alkinyl, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl and R6 stands for H, alkyl, alkenyl, alkinyl, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkylcarbonyl, possibly substituted benzoyl or R5-R6 form together with the shared N atom a 5-/6-membered heterocycle that may contain -O-, -S- or -N(R7)- as ring element; R7 stands for H, alkyl, alkenyl, alkinyl, alkylcarbonyl, benzoyl. Also disclosed are the agriculturally useful salts and esters of C¿1?-C10-carboxylic acids and anorganic acids of the compounds having the formula (I). These cyclohexenone derivates (I) are useful as herbicides and plant growth regulators.
Abstract:
The invention relates to novel compounds of formula (I), in which R1, R2, R3, R4, R5, Y, Q and G are defined as indicated above, to several methods and intermediate products for the production thereof and use thereof as herbicides and/or pesticides. The invention also relates to selective herbicidal agents which contain phenyl-substituted bicyclooctane-1,3-dione-derivatives and a compound which improves crop plant compatibility. The invention further relates to increasing the effect of plant protection agents containing, in particular, phenyl-substituted bicyclooctane-1,3-dione derivatives, by adding ammonium or phosphonium salts and optionally penetration enhancers, to the corresponding products, to methods for producing the same and use thereof in plant protection as pesticides and/or for preventing undesired plant growth.
Abstract:
The present invention relates to non-steroidal compounds useful in the treatment of inflammatory conditions and pharmaceutical compositions comprising them. A representative example of these compounds is formula (III).