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    Benzothiophene derivatives, their preparation and use as urokinase inhibitors
    1.
    发明授权
    Benzothiophene derivatives, their preparation and use as urokinase inhibitors 失效
    苯并噻吩衍生物，其制备和用作尿激酶抑制剂

    公开(公告)号：US6093710A

    公开(公告)日：2000-07-25

    申请号：US147812

    申请日：1999-03-12

    Applicant: Akito Tanaka ,  Hiroaki Mizuno ,  Minoru Sakurai

    Inventor： Akito Tanaka ,  Hiroaki Mizuno ,  Minoru Sakurai

    IPC: C07D333/24 ,  A61K31/343 ,  A61K31/381 ,  A61K31/542 ,  A61P9/00 ,  A61P15/18 ,  A61P19/02 ,  A61P19/10 ,  A61P27/02 ,  A61P35/00 ,  C07D307/82 ,  C07D307/85 ,  C07D333/70 ,  C07D333/80 ,  C07D513/04 ,  C07D493/04 ,  C07D495/04

    CPC classification number: C07D513/04 ,  C07D307/85 ,  C07D333/70 ,  C07D333/80 ,  Y02P20/55

    Abstract: A compound of the formula ##STR1## in which R.sup.1 is hydrogen, lower alkyl, optionally substituted ar(lower)alkyl, cyclo(lower)alkyl(lower)alkyl, protected carboxy)lower)alkyl, carboxy)lower)alkyl, hydroxy(lower)alkyl, optionally substituted lower alkylcarbamoyl(lower)alkyl, lower alkylthio(lower)alkyl, carboxy(lower)alkanoyl, protected carboxy(lower)alkanoyl, aroyl, lower alkanoyl, or optionally substituted arylcarbamoyl(lower)alkyl,R.sup.2 is hydrogen, carboxy, protected carboxy, formyl or N-(lower)alkyl-N-(lower)alkoxycarbamoyl,R.sup.3 is hydrogen or amidino-protective group,A is lower alkylene or carbonyl,X is ##STR2## Y is --S-- or --SO.sub.2 --, Z is --S-- or --O--,or pharmaceutically acceptable salts thereofwhich is useful as a medicament.

    Abstract translation: PCT No.PCT / JP97 / 03215 Sec。 371 1999年3月12日 102（e）1999年3月12日PCT PCT 1997年9月12日PCT公布。 出版物WO98 / 11089 日本公开的化合物，其中R 1为氢，低级烷基，任选取代的芳（低级）烷基，环（低级）烷基（低级）烷基，被保护的羧基）低级烷基，羧基）低级）烷基， 羟基（低级）烷基，任选取代的低级烷基氨基甲酰基（低级）烷基，低级烷硫基（低级）烷基，羧基（低级）烷酰基，受保护的羧基（低级）烷酰基，芳酰基，低级烷酰基或任选取代的芳基氨基甲酰基 （低级）烷基-N-（低级）烷氧基氨基甲酰基，R3是氢或脒基保护基，A是低级亚烷基或羰基，X是Y是-S-或-SO2 - ，Z是-S-或-O-，或其药学上可接受的盐，其可用作药物。

    Amidino substituted tetrahydrobenzo thiophene or furan derivatives and their use as urokinase inhibitors
    2.
    发明授权
    Amidino substituted tetrahydrobenzo thiophene or furan derivatives and their use as urokinase inhibitors 失效
    脒基取代的四氢苯并噻吩或呋喃衍生物及其用作尿激酶抑制剂

    公开(公告)号：US06274619B1

    公开(公告)日：2001-08-14

    申请号：US09584136

    申请日：2000-05-31

    Applicant: Akito Tanaka ,  Hiroaki Mizuno ,  Minoru Sakurai

    Inventor： Akito Tanaka ,  Hiroaki Mizuno ,  Minoru Sakurai

    IPC: C07D30785

    CPC classification number: C07D513/04 ,  C07D307/85 ,  C07D333/70 ,  C07D333/80 ,  Y02P20/55

    Abstract: A compound of the formula: in which R1 is hydrogen, optionally substituted lower alkylcarbamoyl(lower)alkylidene, lower alkylidene, lower alkyl, optionally substituted ar(lower)alkyl, cyclo(lower)alkyl(lower)alkyl, protected carboxy(lower)alkyl, carboxy(lower)alkyl, hydroxy(lower)alkyl, optionally substituted lower alkylcarbamoyl(lower)alkyl, lower alkylthio(lower)alkyl, carboxy(lower)alkanoyl, protected carboxy(lower)alkanoyl, aroyl, lower alkanoyl, or optionally substituted arylcarbamoyl(lower)alkyl, R2 is hydrogen, carboxy, protected carboxy, formyl or N-(lower)alkyl-N-(lower)alkoxycarbamoyl, R3 is hydrogen or amidino-protective group, A is lower alkylene or carbonyl, X is Y is lower alkylene, —S— or —SO2—, Z is —S— or —O—, and the line: is a single bond or a double bond, or pharmaceutically acceptable salts thereof, which is useful as a medicament.

    Abstract translation: 下式化合物：其中R 1为氢，任选取代的低级烷基氨基甲酰基（低级）亚烷基，低级亚烷基，低级烷基，任选取代的芳（低级）烷基，环（低级）烷基（低级）烷基，被保护的羧基 ，羧基（低级）烷基，羟基（低级）烷基，任选取代的低级烷基氨基甲酰基（低级）烷基，低级烷硫基（低级）烷基，羧基（低级）烷酰基，受保护羧基（低级）烷酰基，芳酰基，低级烷酰基或任选取代 芳基氨基甲酰基（低级）烷基，R2是氢，羧基，保护的羧基，甲酰基或N-（低级）烷基-N-（低级）烷氧基氨基甲酰基，R3是氢或脒基保护基，A是低级亚烷基或羰基，X是Y 低级亚烷基，-S-或-SO 2 - ，Z是-S-或-O-，并且行：是 单键或双键，或其药学上可接受的盐，其可用作药物。

    Electronic apparatus
    4.
    发明申请
    Electronic apparatus 有权
    电子仪器

    公开(公告)号：US20080150811A1

    公开(公告)日：2008-06-26

    申请号：US11902448

    申请日：2007-09-21

    Applicant: Tomoko Honda ,  Nobuyoshi Kuroiwa ,  Masaomi Nakahata ,  Jun Morimoto ,  Satoru Honda ,  Yoshikazu Hata ,  Koichi Sato ,  Akihiro Tsujimura ,  Makoto Tabata ,  Minoru Sakurai ,  Shoji Kato

    Inventor： Tomoko Honda ,  Nobuyoshi Kuroiwa ,  Masaomi Nakahata ,  Jun Morimoto ,  Satoru Honda ,  Yoshikazu Hata ,  Koichi Sato ,  Akihiro Tsujimura ,  Makoto Tabata ,  Minoru Sakurai ,  Shoji Kato

    IPC: H01Q1/22

    CPC classification number: H01Q9/40 ,  H01Q9/42 ,  H01Q21/28 ,  H05K1/0284 ,  H05K1/144 ,  H05K3/325 ,  H05K2201/048 ,  H05K2201/0999 ,  H05K2203/167

    Abstract: An electronic apparatus includes: a housing provided with a first conductive pattern; a substrate provided with a first wiring layer in a surface thereof and fixed to the housing; and a first conductive member connecting the first conductive pattern and the first wiring layer. The first conductive pattern extends onto an outer surface and an inner surface of the housing. The first conductive member is in contact with each of at least a part of the first conductive pattern extending onto the inner surface and an end of the first wiring layer. Alternatively, an electronic apparatus includes: a housing provided with a conductive pattern and having a through part in a frame portion thereof; and a substrate provided with a wiring layer on a surface thereof and having a protruding part and fixed to the housing. The protruding part and the through part are fit. The conductive pattern extends onto an outer surface of the housing and onto an inner surface of the through part. At least some of the conductive pattern extending onto the inner surface is in contact with an end of the wiring layer.

    Abstract translation: 电子设备包括：具有第一导电图案的壳体; 基板，其在其表面上设置有第一布线层并固定到所述壳体; 以及连接第一导电图案和第一布线层的第一导电构件。 第一导电图案延伸到壳体的外表面和内表面上。 第一导电构件与延伸到第一布线层的内表面和端部的第一导电图案的至少一部分中的每一个接触。 或者，电子设备包括：壳体，设置有导电图案，并且在其框架部分中具有通孔部分; 以及在其表面上设置有布线层并且具有突出部并固定到壳体的基板。 突出部分和贯穿部分是合适的。 导电图案延伸到壳体的外表面上并延伸到通孔的内表面上。 延伸到内表面上的至少一些导电图案与布线层的端部接触。

    Aminoalcohol derivatives
    5.
    发明申请
    Aminoalcohol derivatives 失效
    氨基醇衍生物

    公开(公告)号：US20050137236A1

    公开(公告)日：2005-06-23

    申请号：US11016886

    申请日：2004-12-21

    Applicant: Kouji Hattori ,  Susumu Toda ,  Masashi Imanishi ,  Shinji Ito ,  Kenichi Washizuka ,  Takanobu Araki ,  Minoru Sakurai ,  Daisuke Tanabe

    Inventor： Kouji Hattori ,  Susumu Toda ,  Masashi Imanishi ,  Shinji Ito ,  Kenichi Washizuka ,  Takanobu Araki ,  Minoru Sakurai ,  Daisuke Tanabe

    IPC: C07C229/38 ,  C07C229/56 ,  C07C271/16 ,  C07C311/51 ,  C07C323/63 ,  C07D213/38 ,  C07D213/61 ,  A61K31/44 ,  A61K31/195

    CPC classification number: C07C229/56 ,  C07C229/38 ,  C07C271/16 ,  C07C311/51 ,  C07C323/63 ,  Y02P20/55

    Abstract: The present invention relates to a compound formula[I]: wherein X is bond, —CH2—, —O— or —NH—, R1 and R12 are each independently hydrogen, halogen, lower alkyl, etc., R2 is hydrogen or optionally substituted lower alkyl, R3 is hydrogen or an amino protective group, R4, R5 and R6 are each independently hydrogen or optionally substituted lower alkyl, R7 is -Z-R13, in which Z is bond, etc., and R13 is carboxy, lower alkoxycarbonyl, (lower alkylsulfonyl)carbamoyl or lower alkanoylsulfamoyl, R8 is —Y—R9, in which Y is bond, —CH2—, —O—, —S—, etc., and R9 is hydrogen, lower alkyl, cyclo(lower)alkyl, etc., and R11 is hydrogen, lower alkyl, lower alkoxy, etc., or a salt thereof. The compound [I] of the present invention and pharmaceutically acceptable salts thereof are useful for the prophylactic and/or the therapeutic treatment of pollakiurea or urinary incontinence.

    Abstract translation: 本发明涉及化合物式[I]：其中X是键，-CH 2 - ， - O-或-NH-，R 1和R 2 > 12个各自独立地为氢，卤素，低级烷基等，R 2为氢或任选取代的低级烷基，R 3为氢或氨基 保护基，R 4，R 5和R 6各自独立地为氢或任选取代的低级烷基，R 7 O 其中Z为键，等等，R 13为羧基，低级烷氧基羰基，（低级烷基磺酰基）氨基甲酰基或低级烷酰基氨磺酰基，R 0为 其中Y为键，-CH 2 - ， - O - ， - S-等，其中R为 - 低级烷基，环（低级）烷基等，R 11是氢，低级烷基，低级烷氧基等，或其盐。 本发明的化合物[I]及其药学上可接受的盐可用于预防和/或治疗呼吸窘迫症或尿失禁。

    Helical antenna and portable communication terminal
    10.
    发明授权
    Helical antenna and portable communication terminal 失效
    螺旋天线和便携式通讯终端

    公开(公告)号：US06661383B2

    公开(公告)日：2003-12-09

    申请号：US10201929

    申请日：2002-07-25

    Applicant: Minoru Sakurai ,  Masanobu Shimanuki

    Inventor： Minoru Sakurai ,  Masanobu Shimanuki

    IPC: H01Q124

    CPC classification number: H01Q1/244 ,  H01Q1/362 ,  H01Q11/08

    Abstract: In a helical antenna for use in a portable communication terminal containing a radio unit which transmits and receives a radio signal, an antenna element is connectable to the radio unit, and contains a bottom portion formed into a helical portion and a top portion formed into a linear portion, the linear portion being positioned along a screw axis of the helical portion. A cap houses the antenna element if the cap covers the antenna element from a top end of the antenna element. A position portion is provided in the cap and positions the linear portion of the antenna element along the screw axis of the helical portion. By virtue of this structure, an appropriate distance can be reliably secured between the antenna element and a human body, thereby maintaining a good characteristic of the antenna.

    Abstract translation: 在用于携带无线电信号的无线电单元的便携式通信终端中使用的螺旋天线中，天线元件可连接到无线电单元，并且包含形成为螺旋部分的底部和形成为 线性部分沿着螺旋部分的螺旋轴线定位。 如果盖子从天线元件的顶端覆盖天线元件，则盖子容纳天线元件。 一个位置部分设置在盖中，并将天线元件的直线部分沿着螺旋部分的螺旋轴线定位。 通过这种结构，能够可靠地确保天线元件与人体之间的适当距离，从而保持天线的良好特性。

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