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    Imino oxyphenyl acetic acid derivatives, methods and intermediates for their preparation and use thereof
    32.
    发明授权
    Imino oxyphenyl acetic acid derivatives, methods and intermediates for their preparation and use thereof 失效
    亚氨基氧苯乙酸衍生物，其制备方法和中间体及其用途

    公开(公告)号：US5994359A

    公开(公告)日：1999-11-30

    申请号：US91921

    申请日：1998-06-25

    申请人： Thomas Grote ,  Hubert Sauter ,  Reinhard Kirstgen ,  Herbert Bayer ,  Ruth Muller ,  Bernd Muller ,  Klaus Oberdorf ,  Wassilios Grammenos ,  Norbert Gotz ,  Michael Rack ,  Albrecht Harreus ,  Franz Rohl ,  Eberhard Ammermann ,  Volker Harries ,  Gisela Lorenz ,  Siegfried Strathmann

    发明人： Thomas Grote ,  Hubert Sauter ,  Reinhard Kirstgen ,  Herbert Bayer ,  Ruth Muller ,  Bernd Muller ,  Klaus Oberdorf ,  Wassilios Grammenos ,  Norbert Gotz ,  Michael Rack ,  Albrecht Harreus ,  Franz Rohl ,  Eberhard Ammermann ,  Volker Harries ,  Gisela Lorenz ,  Siegfried Strathmann

    IPC分类号： A01N37/38 ,  A01N37/50 ,  C07C251/60

    CPC分类号： C07C251/60 ,  A01N37/38 ,  A01N37/50 ,  C07C2101/10 ,  C07C2101/14

    摘要： 2-Iminooxyphenylacetic acid derivatives ##STR1## where the substituents and the index have the following meanings: R.sup.1 is C(CO.sub.2 CH.sub.3).dbd.NOCH.sub.3 (Ia), C(CONHCH.sub.3).dbd.NOCH.sub.3 (Ib), C(CONH.sub.2).dbd.NOCH.sub.3 (Ic), C(CO.sub.2 CH.sub.3).dbd.CHOCH.sub.3 (Id) or C(CO.sub.2 CH.sub.3).dbd.CHCH.sub.3 (Ie);R.sup.2 is cyano, nitro, halogen, alkyl, haloalkyl or alkoxy;m is 0, 1 or 2;R.sup.3 is hydrogen, cyano, hydroxyl, halogen,alkyl, haloalkyl, alkoxyalkyl, alkoxy, haloalkoxy, alkylthio, cyclopropyl, alkenyl,unsubstituted or substituted aryloxyalkyl, benzyl or benzyloxy,R.sup.4 is hydrogen, cyano,unsubstituted or substituted alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl and hetaryl;unsubstituted or substituted alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, heterocyclyloxy, aryloxy and hetaryloxy;unsubstituted or substituted arylthio and hetarylthio;--Q--C(R.sup.5).dbd.N--Y.sup.1 --R.sup.6 or --Q--O--N.dbd.CR.sup.7 R.sup.8,R.sup.3 and R.sup.4 together with the carbon atom to which they are bonded are an unsubstituted or substituted four- to eight-membered ring which, besides carbon atoms, may contain one or two oxygen and/or sulfur atoms and/or NH and/or N(C.sub.1 -C.sub.4 -alkyl) groups;R.sup.3 and R.sup.4 not simultaneously being bonded to the carbon atom via hetero atoms;their salts, processes and intermediates for their preparation, and their use.

    摘要翻译： PCT No.PCT / EP96 / 05642 Sec。 371日期：1998年6月25日第 102（e）日期1998年6月25日PCT 1996年12月16日PCT PCT。 出版物WO97 / 24317 日期：1992年7月10日 - 亚氨基氧苯基乙酸衍生物，其中取代基和指数具有以下含义：R 1为C（CO 2 CH 3）= NOCH 3（Ia），C（CONHCH 3）= NOCH 3（Ib），C（CONH 2）= NOCH 3 Ic），C（CO 2 CH 3）= CHOCH 3（Id）或C（CO 2 CH 3）= CHCH 3（Ie）; R2是氰基，硝基，卤素，烷基，卤代烷基或烷氧基; m为0,1或2; R3是氢，氰基，羟基，卤素，烷基，卤代烷基，烷氧基烷基，烷氧基，卤代烷氧基，烷硫基，环丙基，烯基，未取代或取代的芳氧基烷基，苄基或苄氧基，R4是氢，氰基，未取代或取代的烷基，烯基，炔基， 环烷基，杂环基，芳基和杂芳基; 未取代或取代的烷氧基，烯氧基，炔氧基，环烷氧基，杂环氧基，芳氧基和芳氧基; 未取代或取代的芳硫基和杂芳硫基; -QC（R5）= N-Y1-R6或-QON = CR7R8，R3和R4与它们所键合的碳原子一起是未取代或取代的四至八元环，除碳原子外， 一个或两个氧和/或硫原子和/或NH和/或N（C 1 -C 4 - 烷基）基团; R3和R4不同时通过杂原子键合到碳原子上; 它们的盐，其制备方法和中间体及其用途。

    Phenylacetic acid derivatives, preparation thereof and intermediates therefor, and compositions containing them
    37.
    发明授权
    Phenylacetic acid derivatives, preparation thereof and intermediates therefor, and compositions containing them 失效
    苯乙酸衍生物，其制备方法及其中间体，以及含有它们的组合物

    公开(公告)号：US06187812B1

    公开(公告)日：2001-02-13

    申请号：US09497152

    申请日：2000-02-03

    申请人： Herbert Bayer ,  Hubert Sauter ,  Ruth Müller ,  Wassilios Grammenos ,  Albrecht Harreus ,  Reinhard Kirstgen ,  Franz Röhl ,  Eberhard Ammermann ,  Gisela Lorenz

    发明人： Herbert Bayer ,  Hubert Sauter ,  Ruth Müller ,  Wassilios Grammenos ,  Albrecht Harreus ,  Reinhard Kirstgen ,  Franz Röhl ,  Eberhard Ammermann ,  Gisela Lorenz

    IPC分类号： A01N3718

    CPC分类号： C07D207/333 ,  A01N37/50 ,  A01N37/52 ,  A01N43/06 ,  A01N43/36 ,  A01N43/40 ,  A01N43/54 ,  A01N43/80 ,  A01N43/82 ,  C07C251/58 ,  C07C255/11 ,  C07C327/48 ,  C07C327/58 ,  C07D213/53 ,  C07D213/64 ,  C07D239/34 ,  C07D261/08 ,  C07D263/32 ,  C07D271/06 ,  C07D277/24 ,  C07D307/42

    摘要： Phenylacetic acid derivatives of the formula I where the substituents and the index have the following meanings: X is oxygen or sulfur; R is hydrogen or alkyl; R1 is hydrogen or alkyl; R2 is cyano, nitro, trifluoromethyl, halogen, alkyl or alkoxy; m is 0, 1 or 2, it being possible for the R2 radicals to be different if m is 2; R3 is hydrogen, cyano, nitro, hydroxyl, amino, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, alkylamino or dialkylamino; R4 is hydrogen, cyano, nitro, hydroxyl, amino, halogen, unsubstituted or substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, alkenyl, alkenyloxy, alkenylthio, alkenylamino, N-alkenyl-N-alkylamino, alkynyl, alkynyloxy, alkynylthio, alkynylamino, N-alkynyl-N-alkylamino; unsubstituted or substituted cycloalkyl, cycloalkoxy, cycloalkylthio, cycloalkylamino, N-cycloalkyl-N-alkylamino, cycloalkenyl, cycloalkenyloxy, cycloalkenylthio, cycloalkenylamino, N-cycloalkenyl-N-alkylamino, heterocyclyl, heterocyclyloxy, heterocyclylthio, heterocyclylamino, N-heterocyclyl-N-alkylamino, aryl, aryloxy, arylthio, arylamino, N-aryl-N-alkylamino, hetaryl, hetaryloxy, hetarylthio, hetaryl amino, N-hetaryl-N-alkylamino; R5 is hydrogen, unsubstituted or substituted alkyl, cycloalkyl, alkenyl, alkynyl, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl or alkylsulfonyl; unsubstituted or substituted aryl, arylcarbonyl, arylsulfonyl; hetaryl, hetarylcarbonyl or hetarylsulfonyl, and their salts, processes and intermediates for their preparation, and their use are described.

    摘要翻译： 式I的苯乙酸衍生物，其中取代基和指数具有以下含义：X是氧或硫; R是氢或烷基; R 1是氢或烷基; R 2是氰基，硝基，三氟甲基，卤素，烷基或烷氧基; m 如果m是2，则R2基团可能不同; R3是氢，氰基，硝基，羟基，氨基，卤素，烷基，卤代烷基，烷氧基，卤代烷氧基，烷硫基，烷基氨基或二烷基氨基; R4是氢，氰基，硝基，羟基，氨基，卤素，未取代或取代的烷基，烷氧基，烷硫基，烷基氨基，二烷基氨基，烯基，烯氧基，烯硫基，烯基氨基，N-烯基-N-烷基氨基，炔基，炔氧基，炔硫基，炔基氨基 ，N-炔基-N-烷基氨基，未取代或取代的环烷基，环烷氧基，环烷硫基，环烷基氨基，N-环烷基-N-烷基氨基，环烯基，环烯基氧基，环烯基硫基，环烯基氨基，N-环烯基-N-烷基氨基，杂环基，杂环氧基，杂环基硫基， 杂种 N-烷基氨基，N-杂环基-N-烷基氨基，芳基，芳氧基，芳硫基，芳基氨基，N-芳基-N-烷基氨基，杂芳基，杂芳氧基，杂芳硫基，杂芳基氨基，N-芳基-N-烷基氨基; R 5为氢，未取代或取代 烷基，环烷基，烯基，炔基，烷基羰基，烯基羰基，炔基羰基或烷基磺酰基;未取代或取代的芳基，芳基羰基，芳基磺酰基; 杂芳基，杂芳基羰基或杂芳基磺酰基及其盐，其制备方法和中间体及其用途。