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64 条记录 (耗时 0.022 秒)

    N-VINYLFORMAMIDE DERIVATIVES, POLYMERS FORMED THEREFROM AND SYNTHESIS THEREOF
    4.
    发明申请
    N-VINYLFORMAMIDE DERIVATIVES, POLYMERS FORMED THEREFROM AND SYNTHESIS THEREOF 审中-公开
    N-乙烯基甲酰胺衍生物，由其形成的聚合物及其合成

    公开(公告)号：WO2004022524A2

    公开(公告)日：2004-03-18

    申请号：PCT/US0327732

    申请日：2003-09-05

    申请人： UNIV PITTSBURGH

    发明人： BECKMAN ERIC J ,  CHAPMAN TOBY M ,  SHI LIANJUN

    IPC分类号： C07C233/03 ,  C07C233/13 ,  C07D209/48 ,  C08F26/02 ,  C07C231/00

    CPC分类号： C07C233/03 ,  C07C233/13 ,  C07D209/48 ,  C08F26/02

    摘要： A method of synthesizing a compound having the formula (I), comprising the step of: reacting a N-vinylformamide salt having the formula (II), with a compound having the formula XRR ; wherein X is Br, CI or I, M is an alkali metal or an alkali earth metal, R is a C0-C25 alkylene group, a C0-C25 fluroalkylene group or a C0-C25 perfluoro alkylene group, R is H, provided R is not absent, an alkyl group, a fluroalkyl group, a perfluoroalkyl group, an aryl group, a hydroxy group, a polyether group, a heterocyclic group of 5 or 6 atoms wherein at least one of the atoms is not a carbon and is N, O, or S, -OR , wherein, R is an alkyl group, a fluoroalkyl group, a perfluoroalkyl group, or an aryl group, -C(O)R , -C(O)OR , -OC(O)R , wherein R is an H, an alkyl group, a fluoroalkyl group, a perfluoroalkyl group, or an aryl group, a phthalimide group or NR R wherein R and R are independently H, -C(O)R , an alkyl, a fluoroalkyl group, a perfluoroalkyl group or an aryl group.

    摘要翻译： 合成具有式（I）的化合物的方法，包括以下步骤：使具有式（II）的N-乙烯基甲酰胺盐与具有式XRR 1的化合物反应; 其中X是Br，Cl或I，M是碱金属或碱土金属，R 1是C 0 -C 25亚烷基，C 0 -C 25氟亚烷基或C 0 -C 25全氟亚烷基，R 2 如果R 1不存在则为H，烷基，氟代烷基，全氟烷基，芳基，羟基，聚醚基，5或6个原子的杂环基，其中至少一个 该原子不是碳并且是N，O或S，-OR 3，其中，R 3是烷基，氟烷基，全氟烷基或芳基，-C（O） R 4，-C（O）OR 4，-OC（O）R 4，其中R 4是H，烷基，氟烷基，全氟烷基或芳基 ，邻苯二甲酰亚胺基或NR 5 R 5，其中R 5和R 5独立地为H，-C（O）R 4，烷基，氟烷基，全氟烷基或芳基 组。

    NEW FUNCTIONALIZED POLYMERIC REAGENTS
    6.
    发明申请
    NEW FUNCTIONALIZED POLYMERIC REAGENTS 审中-公开
    新功能聚合物试剂

    公开(公告)号：WO01037983A1

    公开(公告)日：2001-05-31

    申请号：PCT/SE2000/002263

    申请日：2000-11-16

    IPC分类号： C07B61/00 ,  C07C233/13 ,  C07C233/18 ,  C07C291/10 ,  C07D311/88 ,  C08F8/30 ,  B01J19/00 ,  C07C265/08

    CPC分类号： C40B40/04 ,  C07B2200/11 ,  C07C291/10 ,  C07D311/88 ,  C08F8/30 ,  C40B20/04 ,  C40B30/04 ,  C40B50/14

    摘要： The present invention relates to functionalized polymeric reagents useful in solution and solid-phase synthesis. It relates more specifically to functionlized polymeric reagent, comprising an acid labile isonitrile moiety. In further aspects the present invention also relates to use of such functionalized polymeric reagent in solution and solid-phase synthesis, a method for preparing an organic compound by solution and solid-phase synthesis using such functionalized polymeric reagent, a method for preparing such functionalized polymeric reagent and to kits comprising the functionalized polymeric reagent of the invention. The present invention also relates to new intermediates for use in the preparation of the novel functionalized polymeric reagent. In one aspect, the present invention provides a functionalized polymeric reagent for use in solution and solid-phase synthesis, e.g. multicomponent reactions. The functionalized polymeric reagent comprises a linker, and said linker comprises an acid labile isonitrile moiety. The linker is covalently attached to the polymeric support.

    摘要翻译： 本发明涉及可用于溶液和固相合成的官能化聚合物试剂。 它更具体地涉及功能化的聚合物试剂，其包含酸不稳定的异腈部分。 在另外的方面，本发明还涉及这样的官能化聚合物试剂在溶液和固相合成中的用途，通过使用这种官能化聚合物试剂的溶液和固相合成制备有机化合物的方法，制备这种官能化聚合物的方法 试剂和包含本发明的官能化聚合物试剂的试剂盒。 本发明还涉及用于制备新型官能化聚合物试剂的新中间体。 在一个方面，本发明提供了用于溶液和固相合成的官能化聚合物试剂，例如。 多组分反应。 官能化聚合试剂包含接头，所述接头包含酸不稳定的异腈部分。 连接体共价连接到聚合物载体上。

    PLANT GROWTH REGULATING AGENTS
    8.
    发明申请
    PLANT GROWTH REGULATING AGENTS 审中-公开
    植物生长调节剂

    公开(公告)号：WO99045774A1

    公开(公告)日：1999-09-16

    申请号：PCT/JP1999/001181

    申请日：1999-03-11

    IPC分类号： C07C233/05 ,  A01N25/02 ,  A01N37/30 ,  C07C233/09 ,  C07C233/11 ,  C07C233/13 ,  C07C233/18 ,  A01N37/18

    CPC分类号： A01N37/30 ,  C07C233/11 ,  C07C233/13 ,  C07C233/18

    摘要： Plant growth regulating agents containing as the active ingredient compounds represented by general formula (1) or salt thereof; plant growth regulating compositions containing the above compounds or salts thereof and pesticide carriers or fertilizer carriers; and utilization of the above compounds or salts thereof in the production of plant growth regulating agents. The plant growth regulating agents, etc. have a high activity of promoting rooting and scarcely show any side effects such as leaf epinasty. Thus, they are useful particularly in raising of seedlings and production of seeds and seedlings of agricultural products, fixation of turf plants, etc. and tissue culture. In said formula, Ar represents optionally substituted phenyl; A represents lower alkylene; B represents lower alkylene, etc.; and R represents hydroxy, etc.

    摘要翻译： 含有通式（1）表示的活性成分化合物或其盐的植物生长调节剂; 含有上述化合物或其盐和农药载体或肥料载体的植物生长调节组合物; 以及上述化合物或其盐在生产植物生长调节剂中的应用。 植物生长调节剂等具有促进生根的高活性，并且几乎不显示任何副作用如叶上皮。 因此，它们特别有利于提高幼苗的种子和种子，农产品的种子，草坪植物的固定等以及组织培养。 在所述式中，Ar表示任意取代的苯基; A表示低级亚烷基; B代表低级亚烷基等; R 1表示羟基等。

    N,N-DISUBSTITUTED AMIC ACID DERIVATIVE
    9.
    发明申请
    N,N-DISUBSTITUTED AMIC ACID DERIVATIVE 审中-公开
    N，N-取代的氨基酸衍生物

    公开(公告)号：WO1996005169A1

    公开(公告)日：1996-02-22

    申请号：PCT/JP1995001589

    申请日：1995-08-10

    申请人： BANYU PHARMACEUTICAL CO., LTD. ,  IWASAWA, Yoshikazu ,  AOYAMA, Tetsuya ,  KAWAKAMI, Kumiko ,  ARAI, Sachie ,  SATOH, Toshihiko ,  MONDEN, Yoshiaki

    发明人： BANYU PHARMACEUTICAL CO., LTD.

    IPC分类号： C07C233/13

    CPC分类号： C07D213/81 ,  C07C233/13 ,  C07C233/25 ,  C07C233/47 ,  C07D261/18 ,  C07D271/06 ,  C07D307/42 ,  C07D307/68 ,  C07D405/12 ,  C07D407/06 ,  C07D409/14 ,  C07D417/12

    摘要： A compound represented by general formula (I), a medicinally acceptable salt or ester thereof, and an antineoplastic containing the same as the active ingredient, wherein Ar , Ar , Ar and Ar represent each aryl or heteroaryl, A represents an optionally substituted hydrocarbon group; X and Y represent each oxygen, sulfur, carbonyl, -CHR - (R being hydrogen or lower alkyl) or -NR - (R being hydrogen or lower alkyl), or X and Y are combined together to represent vinylene or ethynylene; R , R , R , R and R represent each hydrogen, halogeno, hydroxy, lower alkyl or lower alkoxy; R and R represent each hydrogen, halogeno, hydroxy, amino, nitro, cyano, carboxy, lower alkoxycarbonyl, carbamoyl, lower alkylcarbamoyl, lower alkyl, lower hydroxyalkyl, lower fluoroalkyl or lower alkoxy; R represents lower alkyl; and R represents hydrogen or lower alkyl; provided when one of X and Y represents oxygen, sulfur or -NR -, the other of them represents carbonyl or -CHR -.

    摘要翻译： 由通式（I）表示的化合物，其药学上可接受的盐或酯，和含有该活性成分的抗肿瘤剂，其中Ar 1，Ar 2，Ar 3和Ar 4表示 每个芳基或杂芳基，A表示任选取代的烃基; X和Y表示各自的氧，硫，羰基，-CHR a - （R a为氢或低级烷基）或-NR b - （R b为氢或低级烷基），或X和 Y组合在一起代表亚乙烯基或亚乙炔基; R 1，R 2，R 3，R 8和R 9分别代表氢，卤代，羟基，低级烷基或低级烷氧基; R 4和R 5各自表示氢，卤代，羟基，氨基，硝基，氰基，羧基，低级烷氧基羰基，氨基甲酰基，低级烷基氨基甲酰基，低级烷基，低级羟烷基，低级氟烷基或低级烷氧基。 R 6表示低级烷基; R 7表示氢或低级烷基; 当X和Y中的一个表示氧，硫或-NR b时，其它的表示羰基或-CHR a - 。