NOVEL PROPARGYLETHER DERIVATIVES FOR CONTROLLING PHYTOPATHOGENIC MICROORGANISMS
    61.
    发明申请
    NOVEL PROPARGYLETHER DERIVATIVES FOR CONTROLLING PHYTOPATHOGENIC MICROORGANISMS 审中-公开
    用于控制致病性微生物的新型衍生物衍生物

    公开(公告)号:WO2004033413A2

    公开(公告)日:2004-04-22

    申请号:PCT/EP2003/011218

    申请日:2003-10-09

    IPC分类号: C07C235/00

    摘要: The invention relates to 4-propargyloxy-benzyl dervatives of the general formula (I ) including the optical isomers thereof and mixtures of such isomers, wherein R 1 is hydrogen, optionally substituted alkyl, optionally substituted cycloalkyl or optionally substituted aryl; R 2 , R 3 , R 5 , R 6 , and R 7 are each independently of each other hydrogen or optionally substituted alkyl; R 4 is optionally substituted alkyl; X is O or N-R 7 ; and R 8 is a group R 9 is optionally substituted aryl or optionally substituted heteroaryl; R 10 and R 11 are each independently hydrogen, optionally substituted alkyl, optionally substituted alkenyl or optionally substituted alkynyl; R 12 is optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted aryl or optionally substituted heteroaryl; R 13 is hydrogen or optionally substituted alkyl, alkenyl or alkynyl; and R 14 is optionally substituted alkyl or optionally substituted amino. These compounds possess useful plant protecting properties and may advantageously be employed in agricultural practice for controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi.

    摘要翻译: 本发明涉及通式(I)的4-炔丙氧基 - 苄基衍生物,包括其旋光异构体和这些异构体的混合物,其中R 1是氢,任选取代的烷基,任选取代的环烷基或任选取代的芳基; R2,R3,R5,R6和R7各自独立地为氢或任选取代的烷基; R4是任选取代的烷基; X为O或N-R7; 并且R 8为基团R 9为任选取代的芳基或任选取代的杂芳基; R 10和R 11各自独立地为氢,任选取代的烷基,任选取代的烯基或任选取代的炔基; R12是任选取代的烷基,任选取代的环烷基,任选取代的芳基或任选取代的杂芳基; R13是氢或任选取代的烷基,烯基或炔基; 并且R 14是任选取代的烷基或任选取代的氨基。 这些化合物具有有用的植物保护性质,并且可有利地用于农业实践中以控制或防止植物病原微生物特别是真菌侵染植物。

    UNIVERSAL SUPPORTS FOR OLIGONUCLEOTIDE SYNTHESIS
    62.
    发明申请
    UNIVERSAL SUPPORTS FOR OLIGONUCLEOTIDE SYNTHESIS 审中-公开
    用于寡核苷酸合成的通用支持

    公开(公告)号:WO02044398A2

    公开(公告)日:2002-06-06

    申请号:PCT/US2001/044326

    申请日:2001-11-29

    摘要: Universal supports for oligonucleotide synthesis include a support material represented by the formula (I). In this formula, substituent A is selected from H, alkyl, aryl, or a polymeric or silica base material; substituent B is selected from acyl, aroyl or a polymeric or silica base material; and substituent C is selected from a dimethoxytrityl group or a protecting group removable under acidic or neutral conditions. For the supports, one of substituents A or B constitutes the polymeric or silica base material. In use, an oligonucleotide is attached to the support at substituent C.

    摘要翻译: 寡核苷酸合成的通用载体包括由式(I)表示的载体材料。 在该式中,取代基A选自H,烷基,芳基或聚合物或二氧化硅基材; 取代基B选自酰基,芳酰基或聚合物或二氧化硅基材; 取代基C选自二甲氧基三苯甲基或在酸性或中性条件下可除去的保护基。 对于载体,取代基A或B之一构成聚合物或二氧化硅基材。 在使用中,寡核苷酸与取代基C的载体连接。