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    Insecticidal compounds
    15.
    发明授权
    Insecticidal compounds 有权
    杀虫化合物

    公开(公告)号：US08623896B2

    公开(公告)日：2014-01-07

    申请号：US12810478

    申请日：2008-12-16

    Applicant: Peter Renold ,  Werner Zambach ,  Peter Maienfisch ,  Michel Muehlebach

    Inventor： Peter Renold ,  Werner Zambach ,  Peter Maienfisch ,  Michel Muehlebach

    IPC: A61K31/42 ,  A61K31/38 ,  C07D261/02 ,  C07D331/04 ,  A01N31/00 ,  A01N33/00

    CPC classification number: A01N43/80 ,  C07D413/12

    Abstract: A compound of formula (I), wherein A1, A2, A3, A4, G1, L, R1, R2, R3, R4, Y1, Y2 and Y3 are as defined in claim 1; or a salt or N-oxide thereof. Furthermore, the present invention relates to processes and intermediates for preparing compounds of formula (I), to insecticidal, acaricidal, molluscicidal and nematicidal compositions comprising them and to methods of using them to combat and control insect, acarine, mollusc and nematode pests.

    Abstract translation: 式（I）化合物，其中A1，A2，A3，A4，G1，L，R1，R2，R3，R4，Y1，Y2和Y3如权利要求1所定义; 或其盐或N-氧化物。 此外，本发明涉及制备式（I）化合物的方法和中间体，其包含它们的杀虫，杀螨，杀软体动物和杀线虫组合物以及使用它们来对抗和控制昆虫，螨虫，软体动物和线虫的害虫的方法。

    Cyclic lipid derivatives as potent PAF antagonists
    18.
    发明授权
    Cyclic lipid derivatives as potent PAF antagonists 失效
    循环脂质衍生物作为有效的PAF拮抗剂

    公开(公告)号：US5610310A

    公开(公告)日：1997-03-11

    申请号：US476642

    申请日：1995-06-07

    Applicant: Soon H. Woo ,  Sung K. Chung ,  Soo H. Ban ,  Byoung E. Kim ,  Si H. Kim

    Inventor： Soon H. Woo ,  Sung K. Chung ,  Soo H. Ban ,  Byoung E. Kim ,  Si H. Kim

    IPC: A61K31/44 ,  A61K31/4418 ,  A61K31/4425 ,  A61K31/4427 ,  A61K31/443 ,  A61K31/4433 ,  A61K31/4436 ,  A61K31/47 ,  A61K31/4709 ,  A61P7/02 ,  C07D213/40 ,  C07D213/56 ,  C07D215/10 ,  C07D215/14 ,  C07D277/22 ,  C07D277/30 ,  C07D331/04 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12 ,  C07D491/113 ,  C07F9/09 ,  C07F9/58 ,  C07F9/60 ,  C07F9/6539 ,  C07D213/20

    CPC classification number: C07D401/12 ,  C07D409/12 ,  C07F9/581 ,  C07F9/582 ,  C07F9/60 ,  C07F9/6539

    Abstract: The present invention describes novel cyclic diol derivatives represented by formula I and II: ##STR1## in which Y represents O, S, SO, SO.sub.2, (CH.sub.2).sub.m wherein m is zero or an integer of 1 to 5, or NR.sup.a group wherein R.sup.a is hydrogen, lower alkyl, lower alkoxycarbonyl, aryl, arylalkyl or acyl;R.sup.1 represents an alkyl or alkylcarbamoyl group;R.sup.2 represents a group having formula T--(CH.sub.2).sub.n --V (X.sup.-)q, wherein T refers to a simple covalent bond, a CO, PO.sub.3.sup.-, C(O)O, or CONR.sup.b group wherein R.sup.b is hydrogen, lower alkyl or acyl;n refers to an integer of from 1 to 10;V represents either (i) the group indicated by formula --.sup.+ NR.sup.5 R.sup.6 R.sup.7 wherein R.sup.5, R.sup.6 and R.sup.7 stands for identical or different lower alkyl group, or two or three of R.sup.5, R.sup.6 and R.sup.7 taken together with the adjacent nitrogen form heterocyclic ammonio group, or (ii) the group indicated by the formula ##STR2## wherein R.sup.8 represents lower alkyl group;q is one or zero;X.sup.- represents a pharmaceutically acceptable anion.These compounds are potent PAF antagonists and thus useful for the treatment of the diseases in which PAF is involved.

    Abstract translation: 本发明描述了由式I和II表示的新型环状二醇衍生物：其中Y表示O，S，SO，SO 2，（CH 2）m，其中m为0或1至5的整数，或NR a基团，其中 R a是氢，低级烷基，低级烷氧基羰基，芳基，芳烷基或酰基; R1表示烷基或烷基氨基甲酰基; R2表示具有式T-（CH2）nV（X-q）的基团，其中T表示简单共价键，CO，PO 3 - ，C（O）O或CONR b基团，其中R b是氢，低级烷基或 酰基; n表示1〜10的整数， V表示（i）由式 - + NR5R6R7表示的基团，其中R5，R6和R7表示相同或不同的低级烷基，或者R5，R6和R7中的两个或三个与相邻的氮形式杂环基团一起， 或者（ⅱ）由下式表示的基团：其中R 8表示低级烷基; q是1或0; X-表示药学上可接受的阴离子。 这些化合物是有效的PAF拮抗剂，因此可用于治疗涉及PAF的疾病。

    Sulfonylureas
    19.
    发明授权
    Sulfonylureas 失效
    SULFONYLUREAS

    公开(公告)号：US5209771A

    公开(公告)日：1993-05-11

    申请号：US823515

    申请日：1992-01-21

    Applicant: Willy Meyer

    Inventor： Willy Meyer

    IPC: A01N43/66 ,  A01N47/36 ,  A01N47/46 ,  A01P13/00 ,  C07C275/28 ,  C07C335/42 ,  C07D20060101 ,  C07D239/42 ,  C07D249/14 ,  C07D251/12 ,  C07D305/08 ,  C07D331/04 ,  C07D405/12 ,  C07D409/12 ,  C07D521/00

    CPC classification number: C07D521/00 ,  A01N47/36 ,  C07D305/08 ,  C07D331/04

    Abstract: N-Phenylsulfonyl N'-triazinylureas and -thioureas of formula I ##STR1## in which X is oxygen, sulfur, SO or SO.sub.2 ; W is oxygen or sulfur; R.sub.1 is hydrogen or methyl; R.sub.2 is hydrogen, fluorine, chlorine, bromine, iodine, (X).sub.n R.sub.3, NO.sub.2, NR.sub.4 R.sub.5, --C.tbd.CR.sub.6, ##STR2## or cyano; n is the number 0 or 1; R.sub.3 is C.sub.1 -C.sub.4 alkyl or C.sub.1 -C.sub.4 alkyl which is substituted by 1-4 halogen atoms, C.sub.1 -C.sub.3 alkoxy or C.sub.1 -C.sub.3 alkylthio; or C.sub.2 -C.sub.4 alkenyl or C.sub.2 -C.sub.4 alkenyl which is substituted by 1-4 halogen atoms; R.sub.4 is hydrogen, CH.sub.3 O, CH.sub.3 CH.sub.2 O or C.sub.1 -C.sub.3 alkyl; R.sub.5 is hydrogen or C.sub.1 -C.sub.3 alkyl; R.sub.6 is hydrogen, methyl or ethyl; R.sub.7 is hydrogen or methyl; Z is ##STR3## E is nitrogen; R.sub.8 is C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 haloalkylthio, C.sub.1 -C.sub.4 alkylthio, halogen, C.sub.2 -C.sub.5 alkoxyalkyl, C.sub.2 -C.sub.5 alkoxyalkoxy, amino, C.sub.1 -C.sub.3 alkylamino or di(C.sub.1 -C.sub.3 alkyl)amino and R.sub.9 is C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, C.sub.1 -C.sub.4 haloalkylthio, C.sub.1 -C.sub.4 alkylthio, C.sub.2 -C.sub.5 alkoxyalkyl, C.sub.2 -C.sub.5 alkoxyalkoxy, C.sub.2 -C.sub.5 alkylthioalkyl or cyclopropyl, and the salts of these compounds with amines, alkali metal or alkaline earth metal bases or quaternary ammonium bases have good pre- and postemergence selective herbicidal and growth-regulating properties.

    Abstract translation: 式I的N-苯基磺酰基N'-三嗪基脲和硫脲其中X是氧，硫，SO或SO 2; W是氧或硫; R1是氢或甲基; R2是氢，氟，氯，溴，碘，（X）nR3，NO2，NR4R5，-C3OND CR6， n是数字0或1; R3是被1-4个卤素原子取代的C1-C4烷基或C1-C4烷基，C1-C3烷氧基或C1-C3烷硫基; 或被1-4个卤素原子取代的C 2 -C 4烯基或C 2 -C 4烯基; R4是氢，CH3O，CH3CH2O或C1-C3烷基; R5是氢或C1-C3烷基; R6是氢，甲基或乙基; R7是氢或甲基; Z是氮; R8是C1-C4烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基，C1-C4卤代烷硫基，C1-C4烷硫基，卤素，C2-C5烷氧基烷基，C2-C5烷氧基烷氧基，氨基，C1-C3烷基氨基或二（C1-C3烷基）氨基和 R9是C1-C4烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷硫基，C1-C4烷硫基，C2-C5烷氧基烷基，C2-C5烷氧基烷氧基，C2-C5烷硫基烷基或环丙基，这些化合物与胺，碱金属或碱土 金属碱基或季铵碱基具有良好的芽前和芽后选择性除草和生长调节性质。

    Branched amides of L-aspartyl-D-amino acid dipeptides
    20.
    发明授权
    Branched amides of L-aspartyl-D-amino acid dipeptides 失效

    公开(公告)号：US4804782A

    公开(公告)日：1989-02-14

    申请号：US796173

    申请日：1985-11-08

    Applicant: Thomas M. Brennan ,  Michael E. Hendrick

    Inventor： Thomas M. Brennan ,  Michael E. Hendrick

    IPC: A23L27/30 ,  C07C45/00 ,  C07C45/29 ,  C07C45/61 ,  C07C45/63 ,  C07C45/64 ,  C07C45/68 ,  C07C45/75 ,  C07C233/00 ,  C07C323/25 ,  C07D307/22 ,  C07D307/32 ,  C07D331/04 ,  C07D333/32 ,  C07D333/36 ,  C07D335/02 ,  C07K5/072 ,  C07C103/37 ,  A23L1/236 ,  C07C103/52

    CPC classification number: C07D307/32 ,  A23L27/32 ,  C07C323/00 ,  C07C323/25 ,  C07C45/004 ,  C07C45/292 ,  C07C45/61 ,  C07C45/63 ,  C07C45/64 ,  C07C45/68 ,  C07C45/75 ,  C07D307/22 ,  C07D331/04 ,  C07D333/32 ,  C07D333/36 ,  C07D335/02 ,  C07K5/06113

    Abstract: Amides of L-aspartyl-D-amino acid dipeptides of the formula ##STR1## and physiologically acceptable cationic and acid addition salts thereof wherein R.sup.a is methyl, ethyl, n-propyl or isopropyl; R is a branched member selected from the group consisting of fenchyl, diisopropylcarbinyl, d-methyl-t-butylcarbinyl, d-ethyl-t-butylcarbinyl, di-t-butylcarbinyl, 2-methylthio-2,4-dimethylpentan-3-yl, ##STR2## where at least one of R.sup.3, R.sup.4, R.sup.5, R.sup.6 is alkyl having from one to four carbon atoms and the remainder are hydrogen or alkyl having from one to four carbon atoms, X is O, S, SO, SO.sub.2, C.dbd.O or CHOH; m is zero or 1-4, n and p are each zero, 1, 2 or 3 where the sum of n+p is not greater than 3 and the sum of the carbon atoms in R.sup.3, R.sup.4, R.sup.5 and R.sup.6 is not greater than six, and when both of R.sup.3 and R.sup.4 or R.sup.5 and R.sup.6 are alkyl they are methyl or ethyl, ##STR3## where one of R.sup.7, R.sup.8, R.sup.9 is alkyl having from one to four carbon atoms and the remainder are hydrogen or alkyl having from one to four carbon atoms and the sum of the carbon atoms in R.sup.7, R.sup.8 and R.sup.9 is not greater than six, m and q are the same or different and each have the values previously defined for m; ##STR4## where each of R.sup.12 and R.sup.13 are methyl or ethyl, or R.sup.12 is hydrogen and R.sup.13 is alkyl having from one to four carbon atoms, Z is O or NH and t is 1 or 2, ##STR5## where w is 1-4, R.sup.14 and R.sup.16 are each alkyl having from one to four carbon atoms, R.sup.15 is H, OH, methyl or ethyl and the sum of the carbon atoms in R.sup.14, R.sup.15 and R.sup.16 is not greater than six and when both of R.sup.14 and R.sup.15 are alkyl they are methyl or ethyl, and where R.sup.17 and R.sup.19 are alkyl having from one to four carbon atoms, R.sup.18 and R.sup.20 are H or alkyl having one to two carbon atoms, A is OH and B is H, OH or CH.sub.3 and taken together A and B are ##STR6## where the sum of the carbon atoms in R.sup.17, R.sup.18, R.sup.19 and R.sup.20 is not greater than six and when both of R.sup.17 and R.sup.18 or R.sup.19 and R.sup.20 are alkyl they are methyl or ethyl;said amides are potent sweetners having advantages over the prior art, edible compositions containing them, methods for their use in edible compositions and novel amine and amide intermediates useful in their production.

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